Herbicidal sulfonamides

ABSTRACT

Tetrazole-substituted benzenesulfonamides are useful as agricultural chemicals and, in particular, as growth regulants and herbicides.

RELATED APPLICATION

This application is a division of application Ser. No. 114,584 filed on Oct. 30, 1987 now U.S. Pat. No. 4,786,311, which in turn is a continuation-in-part of copending application U.S. Ser. No. 934,118, filed Nov. 24, 1986, now U.S. Pat. No. 4,746,353, which in turn is a continuation-in-part of copending application U.S. Ser. No. 849,618, filed Apr. 11, 1986, now abandoned, which in turn is a continuation-in-part of copending application U.S. Ser. No. 739,214, filed May 30, 1985, now abandoned.

BACKGROUND OF THE INVENTION

This invention relates to tetrazole-substituted benzene sulfonamides which are useful as agricultural chemicals such as growth regulants and herbicides.

U.S. Pat. No. 4,127,405 and U.S. Pat. No. 4,169,719 disclose herbicidal benzenesulfonylureas.

EP-A-165,753, published Dec. 27, 1985, discloses herbicidal thiophenesulfonamides of formula ##STR1## wherein Q is optionally substituted phenyl or an optionally substituted saturated or unsaturated 5- or 6-membered heterocyclic ring containing one to three heteroatoms.

EP-A-83,975 (published July 20, 1983) discloses herbicidal benzenesulfonamides of formula ##STR2## wherein Q is selected from various five or six-membered aromatic or partially unsaturated heterocyclic rings containing 2 or 3 heteroatoms selected from O, S or NR.

EP-A-85,476 (published Aug. 10, 1983) discloses herbicidal benzenesulfonamides of formulae ##STR3## wherein Q is selected from various 5-membered aromatic heterocycles, and their dihydro and tetrahydro analogs, which contain one heteroatom selected from O, S or NR, or Q is a saturated or partially unsaturated 6-membered ring containing one heteroatom selected from O or S; and

Q¹ is a 6-membered aromatic heterocycle containing one to three N atoms.

South African Patent Application 83/8416 (published May 12, 1984) discloses herbicidal benzenesulfonamides of formula ##STR4## wherein A is an unsaturated or only partially saturated 5- or 6-membered heterocyclic ring system which is bonded through a carbon atom and contains 1, 2 or 3 heteroatoms.

EP-A-116,518, published Aug. 22, 1984, discloses herbicidal sulfonamides of formula ##STR5## wherein X is NR₆ R₇, N(SO₂ R₉)₂ or ##STR6## A is CO, SO₂, CONR₂₃ or CO₂ ; B is C₁ -C₄ alkyl or C₂ -C₄ alkenyl; and

C is CO, CR₂₁ R₂₂ or SO₂.

U.S. Pat. No. 4,475,944 discloses herbicidal sulfamates, possessing an ortho-heterocyclic ring, such as those of formula ##STR7## wherein W is O, S or NR₁.

EP-A-164,268, published Dec. 11, 1985, discloses herbicidal benzylsulfonamides of formula ##STR8## wherein Q is a saturated, 5- or 6-membered ring containing 1 to 2 heteroatoms selected from 0-2 S or 0-2 O or an unsaturated 5- or 6-membered ring containing 1 to 3 heteroatoms selected from 0-1 S, 0-1 O or 0-3 N and Q may optionally be substituted by one or more groups selected from C₁ -C₄ alkyl, halogen, C₁ -C₃ alkoxy, C₁ -C₃ alkylthio, C₁ -C₂ haloalkoxy, C₃ -C₄ alkenylthio, C₁ -C₂ haloalkylthio or SCH₂ CN.

EP-A-165,753, published Dec. 27, 1985, discloses herbicidal pyridinesulfonamides of formula ##STR9## wherein Q is phenyl optionally substituted with Cl, CH₃ O or CH₃, a saturated 5-membered ring containing 1 heteroatom selected from O or S, or an unsaturated 5- or 6-membered ring containing 1 to 3 heteroatoms selected from 0-1 S, 0-1 O or 0-3 N and when Q is an unsaturated 5- or 6-membered ring, it may optionally be substituted by one or more groups selected from C₁ -C₄ alkyl, halogen, C₁ -C₃ alkoxy, C₁ -C₃ alkylthio, C₃ -C₄ alkenylthio, C₁ -C₂ haloalkoxy or C₁ -C₂ haloalkylthio.

EP-A-176,304, published Apr. 11, 1986, discloses herbicidal pyrazolesulfonamides such as those of formula ##STR10## wherein Q is a saturated 5- or 6-membered ring containing 1 heteroatom selected from 0-1 S or 0-1 O or an unsaturated 5- or 6-membered ring containing 1-3 heteroatoms selected from 0-1 S, 0-1 O or 0-3 N and Q may optionally be substituted by one or more groups selected from C₁ -C₄ alkyl, C₁ -C₄ haloalkyl, halogen, C₁ -C₃ alkoxy, C₁ -C₃ alkylthio, C₃ -C₄ alkenylthio, C₃ -C₄ alkenyloxy, C₁ -C₂ haloalkoxy, C₁ -C₂ haloalkylthio, C₂ -C₄ cyanoalkylthio or C₁ -C₂ alkoxycarbonylmethylthio.

EP-A-141,777, published May 15, 1985, discloses ortho-benzyl-substituted sulfonylureas of the formula ##STR11## wherein Y is O or S; and

R¹⁷ is a 5- to 6-membered unsaturated heterocyclic radical including ##STR12##

U.S. Pat. No. 4,602,936 carrying part of this disclosure, issued July 29, 1986.

South African Patent Application 83/0441, published July 25, 1983, discloses herbicidal benzenesulfonamides of formula ##STR13## wherein R₁ is H, halogen, NO₂, C₁ -C₄ alkyl, C₁ -C₄ alkoxy, C₂ -C₅ alkenyl or C₁ -C₄ alkoxycarbonyl;

R₂ is C₁ -C₃ alkyl or C₁ -C₃ alkoxy, each unsubstituted or substituted by 1 to 3 halogen atoms;

R₃ is halogen, H, NR₄ R₅, C₁ -C₃ alkyl, unsubstituted or substituted by 1 to 3 alkoxy, unsubstituted or substituted by methoxy, ethoxy, or 1 to 3 halogen atoms;

A is C₁ -C₄ alkylene or C₂ -C₄ alkenylene, each unsubstituted or substituted by C₁ -C₄ alkyl;

m is 0 or 1;

E is N or CH;

X is oxygen, sulfur, SO or SO₂ ; and

Q is, in part, a 5- or 6-membered heterocyclic ring bound through carbon or nitrogen, such heterocycles including furan, pyrane, thiophene, triazole, pyridine, pyrroline, oxaxole, isooxazole, thiazole, isothiazole, thiadiaxole, oxathiole, pyrrole, imidazole, pyrazole, pyrazine, pyrimidine, pyridazine, symmetrical and assymetrical triazines, oxdiazole, oxazine, furazane, pyridine-N-oxide, thiophene-S-oxide, benzthiophene, benzofuran, isobenzofuran, chromene, chromane, indole, isoindole, indazole, quinoline, isoquinoline, phthalazine, quinoxaline, quinazoline, quinoline, benzthiazole and benzimidiazole, and partially or completely hydrogenated and fused homoglogues thereof.

South African Patent Application 85/2646, published Oct. 11, 1985, discloses herbicidal benzenesulfonamides of formula ##STR14## wherein R₁ is H, halogen, NO₂, alkyl, alkoxy, alkoxycarbonyl or haloalkyl;

X is O, S, SO or SO₂ ;

Y is O or S;

E is CH or N;

R₂ and R₃ are independently alkyl, alkoxy or alkoxyalkyl;

A is alkylene or alkenylene;

m is 0 or 1;

Q is, in part, ##STR15## each of which is optionally substituted and/or optionally partially hydrogenated; and

X' is O, S or NR.

The presence of undesired vegetation causes substantial damage to useful crops, especially agricultural products that satisfy man's basic food needs, such as corn, soybeans, wheat and the like. The current population explosion and concomitant world food shortage demand improvements in the efficiency of producing these crops. Prevention or minimization of the loss of a portion of valuable crops by killing or inhibiting the growth of undesired vegetation is one way of improving this efficiency.

A wide variety of materials, useful for killing, or inhibiting (controlling) the growth of undesired vegetation is available. Such materials are commonly referred to as herbicides. The need exists, however, for still more effective herbicides that destroy or retard weeds without causing signficant damage to useful crops.

SUMMARY OF THE INVENTION

This invention relates to novel compounds of Formula I, agriculturally suitable compositions containing them, and their method-of-use as preemergent or postemergent herbicides or as plant growth regulants. ##STR16## wherein J is ##STR17## W is O, S or NR_(X) ; R_(X) is H, OH, C₁ -C₃ alkyl, C₁ -C₃ alkoxy, allyloxy, propargyloxy, C₁ -C₃ haloalkyl, C₁ -C₃ haloalkoxy or NR_(Y) R_(Z) ;

R_(Y) is H or C₁ -C₃ alkyl;

R_(Z) is C₁ -C₃ alkyl;

G is O, S, SO or SO₂ ;

m is 0 or 1;

n is 0, 1 or 2;

R is H or CH₃ ;

E is a single bond, CH₂ or O;

Q is ##STR18## R₁ is H, C₁ -C₃ alkyl, C₁ -C₃ haloalkyl, halogen, nitro, C₁ -C₃ alkoxy, SO₂ NR_(a) R_(b), C₁ -C₃ alkylthio, C₁ -C₃ alkylsulfinyl, C₁ -C₃ alkylsulfonyl, CN, SCN, CO₂ R_(c), C₁ -C₃ haloalkoxy, C₁ -C₃ haloalkylthio, amino, C₁ -C₃ alkylamino, di(C₁ -C₃ alkyl)amino or C₁ -C₂ alkyl substituted with C₁ -C₂ alkoxy, C₁ -C₂ haloalkoxy, C₁ -C₂ alkylthio, C₁ -C₂ haloalkylthio or CN;

R₂ is H, C₁ -C₃ alkyl, allyl or phenyl;

R₃ is H, C₁ -C₆ alkyl, C₃ -C₆ cycloalkyl, C₁ -C₆ haloalkyl, CH₂ -(C₂ -C₅ alkenyl), CH₂ (C₂ -C₅ haloalkenyl), CH₂ (C₂ -C₅ alkynyl), CH₂ (C₂ -C₅ haloalkynyl), C₆ H₅ or C₁ -C₄ alkyl substituted with C₁ -C₂ alkoxy, C₁ -C₂ alkylthio, C₁ -C₂ alkylsulfinyl or C₁ -C₂ alkylsulfonyl;

R₄ is H, halogen, C₁ -C₆ alkyl, C₃ -C₆ cycloalkyl, C₁ -C₆ haloalkyl, C₂ -C₆ alkenyl, C₂ -C₆ haloalkenyl, C₂ -C₆ alkynyl, C₃ -C₆ haloalkynyl, C₆ H₅, C₁ -C₄ alkoxy, C₁ -C₄ haloalkoxy, C₁ -C₄ alkylthio, C₁ -C₄ alkylsulfinyl, C₁ -C₄ alkylsulfonyl, OCH₂ CH₂ O-(C₁ -C₂ alkyl) or di(C₁ -C₃ alkyl)amino;

R₅ is H, C₁ -C₃ alkyl, C₁ -C₃ haloalkyl, allyl or propargyl;

R_(a) is H, C₁ -C₄ alkyl, C₂ -C₃ cyanoalkyl, methoxy or ethoxy;

R_(b) is H, C₁ -C₄ alkyl or C₃ -C₄ alkenyl; or

R_(a) and R_(b) may be taken together as --(CH₂)₃ --, --(CH₂)₄ --, --(CH₂)₅ -- or --CH₂ CH₂ OCH₂ CH₂ --;

R_(c) is C₁ -C₄ alkyl, C₃ -C₄ alkenyl, C₃ -C₄ alkynyl, C₂ -C₄ haloalkyl, C₁ -C₂ cyanoalkyl, C₅ -C₆ cycloalkyl, C₄ -C₇ cycloalkylalkyl or C₂ -C₄ alkoxyalkyl;

A is ##STR19## X is H, C₁ -C₄ alkyl, C₁ -C₄ alkoxy, C₁ -C₄ haloalkoxy, C₁ -C₄ haloalkyl, C₁ -C₄ haloalkylthio, C₁ -C₄ alkylthio, halogen, C₂ -C₅ alkoxyalkyl, C₂ -C₅ alkoxyalkoxy, amino, C₁ -C₃ alkylamino, di(C₁ -C₃ alkyl)amino or C₃ -C₅ cycloalkyl;

Y is H, C₁ -C₄ alkyl, C₁ -C₄ alkoxy, C₁ -C₄ haloalkoxy, C₁ -C₄ haloalkylthio, C₁ -C₄ alkylthio, C₂ -C₅ alkoxyalkyl, C₂ -C₅ alkoxyalkoxy, amino, C₁ -C₃ alkylamino, di(C₁ -C₃ alkyl)amino, C₃ -C₄ alkenyloxy, C₃ -C₄ alkynyloxy, C₂ -C₅ alkylthioalkyl, C₂ -C₅ alkylsulfinylalkyl, C₂ -C₅ alkylsulfonylalkyl, C₁ -C₄ haloalkyl, C₂ -C₄ alkynyl, azido, cyano, ##STR20## p is 2 or 3; L₁ and L₂ are independently O or S;

R₆ is H or CH₃ ;

R₇ and R₈ are independently C₁ -C₃ alkyl;

Z is CH, N, CCH₃, CC₂ H₅, CCl or CBr;

Y₁ is O or CH₂ ;

X₁ is CH₃, OCH₃, OC₂ H₅ or OCF₂ H;

X₂ is CH₃, C₂ H₅ or CH₂ CF₃ ;

Y₂ is OCH₃, OC₂ H₅, SCH₃, SC₂ H₅, CH₃ or CH₂ CH₃ ;

X₃ is CH₃ or OCH₃ ;

Y₃ is H or CH₃ ;

X₄ is CH₃, OCH₃, OC₂ H₅, CH₂ OCH₃ or Cl;

Y₄ is CH₃, OCH₃, OC₂ H₅ or Cl; and

Z¹ is CH or N;

and their agriculturally suitable salts; provided that

(a) when X is Cl, F, Br or I, then Z is CH and Y is OCH₃, OC₂ H₅, N(OCH₃)CH₃, NHCH₃, N(CH₃)₂ or OCF₂ H;

(b) when X or Y is C₁ haloalkoxy, then Z is CH;

(c) when J is J-9 and n is O, then Q is Q-1 or Q-2;

(d) when E is O, then J is J-1;

(e) when W is S, then A is A-1, R is H, and Y is CH₃, OCH₃, OC₂ H₅, CH₂ OCH₃, C₂ H₅, CF₃, SCH₃, OCH₂ CH═CH₂, OCH₂ C.tbd.CH, OCH₂ CH₂ OCH₃, CH(OCH₃)₂ or ##STR21## (f) when the total number of carbon atoms in X and Y is greater than 4, then the carbon content of R₁, R₃, R₄ and R₅ must each be less than or equal to 2;

(g) X₄ and Y₄ cannot simultaneously be Cl;

(h) when J is J-1 and m is 0, then n is 0; and

(i) when n is 0 and m is 1, then Q is Q-1 or Q-2.

In the above definitions, the term "alkyl" used either alone or in compound words such as "alkylthio" or "haloalkyl", denotes straight chain or branched alkyl, e.g., methyl, ethyl, n-propyl, isopropyl or the different butyl, pentyl or hexyl isomers.

Alkoxy denotes methoxy, ethoxy, n-propoxy, isopropoxy and the different butyl isomers.

Alkenyl denotes straight chain or branched alkenes, e.g., vinyl, 1-propenyl, 2-propenyl, 3-propenyl and the different butenyl, pentenyl or hexenyl isomers.

Alkynyl denotes straight chain or branched alkynes, e.g., ethynyl, 1-propynyl, 2-propynyl and the different butynyl, pentynyl and hexynyl isomers.

Alkylsulfonyl denotes methylsulfonyl, ethylsulfonyl or the different propylsulfonyl isomers.

Alkylthio, alkylsulfinyl, alkylamino, etc. are defined in an analogous manner.

Cycloalkyl denotes cyclopropyl, cyclobutyl, cyclopentyl and cyclohexyl.

The term "halogen", either alone or in compound words such as "haloalkyl", denotes fluorine, chlorine, bromine or iodine.

In terms such as C₂ -C₃ alkylthioalkyl, the specified number of carbon atoms is meant to define the total number of carbon atoms in that substituent group. For example, C₂ -C₃ alkylthioalkyl would designate CH₂ SCH₃, CH₂ SC₂ H₅, CH₂ CH₂ SCH₃ or CH(CH₃)SCH₃, and C₂ -C₅ alkoxyalkoxy would represent OCH₂ OCH₃ through O(CH₂)₄ OCH₃ or OCH₂ O(CH₂)₃ CH₃ and the various structural isomers embraced therein.

Preferred for reasons of increased ease of synthesis and/or greater herbicidal efficacy are:

(1) Compounds of Formula I where E is a single bond.

(2) Compounds of Formula I where E is CH₂.

(3) Compounds of Formula I where E is O.

(4) Compounds of Preferred 1 were

m is O; and

W is O.

(5) Compounds of Preferred 4 where

X is C₁ -C₂ alkyl, C₁ -C₂ alkoxy, cyclopropyl, Cl, F, Br, I, OCF₂ H, CH₂ F, CF₃, OCH₂ CH₂ F, OCH₂ CHF₂, OCH₂ CF₃, CH₂ Cl or CH₂ Br; and

Y is H, C₁ -C₂ alkyl, C₁ -C₂ alkoxy, CH₂ OCH₃, CH₂ OCH₂ CH₃, NHCH₃, N(OCH₃)CH₃, N(CH₃)₂, CF₃, SCH₃, OCH₂ CH.tbd.CH₂, OCH₂ C.tbd.CH, OCH₂ CH₂ OCH₃, CH₂ SCH₃, ##STR22## OCF₂ H, SCF₂ H, OCF₂ Br, C.tbd.CH or C.tbd.CCH₃. (6) Compounds of Preferred 5 where

R₁ is H, CH₃, F, Cl, Br, OCH₃, SCH₃, CH₂ CN, CH₂ OCH₃, CF₃ or OCF₂ H; and

n is O.

(7) Compounds of Preferred 6 where

R₃ is H, C₁ -C₃ alkyl, C₁ -C₂ alkyl substituted with C₁ -C₂ alkoxy, CH₂ CH₂ Cl, CH₂ CH₂ F, CH₂ CHF₂, CH₂ CF₃, allyl or propargyl; and

R₄ is H, C₁ -C₃ alkyl, C₁ -C₂ alkoxy, C₁ -C₂ alkylthio, N(CH₃)₂, allyl, propargyl or C₁ -C₂ alkyl substituted with 1-3 atoms of F, Cl or Br.

(8) Compounds of Preferred 7 where J is J-1.

(9) Compounds of Preferred 8 where

A is A-1;

Z is CH or N;

X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H;

Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.

(10) Compounds of Preferred 9 where Q is Q₁.

(11) Compounds of Preferred 9 where Q is Q₂.

(12) Compounds of Preferred 9 where Q is Q₃.

(13) Compounds of Preferred 9 where Q is Q₄.

(14) Compounds of Preferred 9 where Q is Q₅.

(15) Compounds of Preferred 9 where Q is Q₆.

(16) Compounds of Preferred 9 where Q is Q₇.

(17) Compounds of Preferred 7 where J is J-2.

(18) Compounds of Preferred 17 where

A is A-1;

Z is CH or N;

X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H;

Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.

(19) Compounds of Preferred 18 where Q is Q₁.

(20) Compounds of Preferred 18 where Q is Q₂.

(21) Compounds of Preferred 18 where Q is Q₃.

(22) Compounds of Preferred 18 where Q is Q₄.

(23) Compounds of Preferred 18 where Q is Q₅.

(24) Compounds of Preferred 18 where Q is Q₆.

(25) Compounds of Preferred 18 where Q is Q₇.

(26) Compounds of Preferred 7 where J is J-3.

(27) Compounds of Preferred 26 where

A is A-1;

Z is CH or N;

X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H;

Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.

(28) Compounds of Preferred 27 where Q is Q₁.

(29) Compounds of Preferred 27 where Q is Q₂.

(30) Compounds of Preferred 27 where Q is Q₃.

(31) Compounds of Preferred 27 where Q is Q₄.

(32) Compounds of Preferred 27 where Q is Q₅.

(33) Compounds of Preferred 27 where Q is Q₆.

(34) Compounds of Preferred 27 where Q is Q₇.

(35) Compounds of Preferred 7 where J is J-4.

(36) Compounds of Preferred 35 where

A is A-1;

Z is CH or N;

X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H;

Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.

(37) Compounds of Preferred 36 where Q is Q₁.

(38) Compounds of Preferred 36 where Q is Q₂.

(39) Compounds of Preferred 36 where Q is Q₃.

(40) Compounds of Preferred 36 where Q is Q₄.

(41) Compounds of Preferred 36 where Q is Q₅.

(42) Compounds of Preferred 36 where Q is Q₆.

(43) Compounds of Preferred 36 where Q is Q₇.

(44) Compounds of Preferred 7 where J is J-5.

(45) Compounds of Preferred 44 where

A is A-1;

Z is CH or N;

X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H;

Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.

(46) Compounds of Preferred 45 where Q is Q₁.

(47) Compounds of Preferred 45 where Q is Q₂.

(48) Compounds of Preferred 45 where Q is Q₃.

(49) Compounds of Preferred 45 where Q is Q₄.

(50) Compounds of Preferred 45 where Q is Q₅.

(51) Compounds of Preferred 45 where Q is Q₆.

(52) Compounds of Preferred 45 where Q is Q₇.

(53) Compounds of Preferred 7 where J is J-6.

(54) Compounds of Preferred 53 where

A is A-1;

Z is CH or N;

X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H;

Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.

(55) Compounds of Preferred 54 where Q is Q₁.

(56) Compounds of Preferred 54 where Q is Q₂.

(57) Compounds of Preferred 54 where Q is Q₃.

(58) Compounds of Preferred 54 where Q is Q₄.

(59) Compounds of Preferred 54 where Q is Q₅.

(60) Compounds of Preferred 54 where Q is Q₆.

(61) Compounds of Preferred 54 where Q is Q₇.

(62) Compounds of Preferred 7 where J is J-7.

(63) Compounds of Preferred 62 where

A is A-1;

Z is CH or N;

X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H;

Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.

(64) Compounds of Preferred 63 where Q is Q₁.

(65) Compounds of Preferred 63 where Q is Q₂.

(66) Compounds of Preferred 63 where Q is Q₃.

(67) Compounds of Preferred 63 where Q is Q₄.

(68) Compounds of Preferred 63 where Q is Q₅.

(69) Compounds of Preferred 63 where Q is Q₆.

(70) Compounds of Preferred 63 where Q is Q₇.

(71) Compounds of Preferred 7 where J is J-8.

(72) Compounds of Preferred 71 where

A is A-1;

Z is CH or N;

X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H;

Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.

(73) Compounds of Preferred 72 where Q is Q₁.

(74) Compounds of Preferred 72 where Q is Q₂.

(75) Compounds of Preferred 72 where Q is Q₃.

(76) Compounds of Preferred 72 where Q is Q₄.

(77) Compounds of Preferred 72 where Q is Q₅.

(78) Compounds of Preferred 72 where Q is Q₆.

(79) Compounds of Preferred 72 where Q is Q₇.

(80) Compounds of Preferred 7 where J is J-9.

(81) Compounds of Preferred 80 where

A is A-1;

Z is CH or N;

X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H;

Y is CH₃, OCH₃, C₂ H₅, CH₅ OCH₃, NHCH₃ or CH(OCH₃)₂.

(82) Compounds of Preferred 81 where Q is Q₁.

(83) Compounds of Preferred 81 where Q is Q₂.

(84) Compounds of Preferred 81 where Q is Q₃.

(85) Compounds of Preferred 81 where Q is Q₄.

(86) Compounds of Preferred 81 where Q is Q₅.

(87) Compounds of Preferred 81 where Q is Q₆.

(88) Compounds of Preferred 81 where Q is Q₇.

(89) Compounds of Preferred 7 where J is J-10.

(90) Compounds of Preferred 89 where

A is A-1;

Z is CH or N;

X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H;

Y is CH₃, OCH₃, C₂ h₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.

(91) Compounds of Preferred 90 where Q is Q₁.

(92) Compounds of Preferred 90 where Q is Q₂.

(93) Compounds of Preferred 90 where Q is Q₃.

(94) Compounds of Preferred 90 where Q is Q₄.

(95) Compounds of Preferred 90 where Q is Q₅.

(96) Compounds of Preferred 90 where Q is Q₆.

(97) Compounds of Preferred 90 where Q is Q₇.

(98) Compounds of Preferred 7 where J is J-11.

(99) Compounds of Preferred 98 where

A is A-1;

Z is CH or N;

X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H;

Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.

(100) Compounds of Preferred 99 where Q is Q₁.

(101) Compounds of Preferred 99 where Q is Q₂.

(102) Compounds of Preferred 99 where Q is Q₃.

(103) Compounds of Preferred 99 where Q is Q₄.

(104) Compounds of Preferred 99 where Q is Q₅.

(105) Compounds of Preferred 99 where Q is Q₆.

(106) Compounds of Preferred 99 where Q is Q₇.

(107) Compounds of Preferred 7 where J is J-12.

(108) Compounds of Preferred 107 where

A is A-1;

Z is CH or N;

X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H;

Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.

(109) Compounds of Preferred 108 where Q is Q₁.

(110) Compounds of Preferred 108 where Q is Q₂.

(111) Compounds of Preferred 108 where Q is Q₃.

(112) Compounds of Preferred 108 where Q is Q₄.

(113) Compounds of Preferred 108 where Q is Q₅.

(114) Compounds of Preferred 108 where Q is Q₆.

(115) Compounds of Preferred 108 where Q is Q₇.

(116) Compounds of Preferred 7 where J is J-13.

(117) Compounds of Preferred 116 where

A is A-1;

Z is CH or N;

X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H;

Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.

(118) Compounds of Preferred 117 where Q is Q₁.

(119) Compounds of Preferred 117 where Q is Q₂.

(120) Compounds of Preferred 117 wherein Q is Q₃.

(121) Compounds of Preferred 117 where Q is Q₄.

(122) Compounds of Preferred 117 where Q is Q₅.

(123) Compounds of Preferred 117 where Q is Q₆.

(124) Compounds of Preferred 117 where Q is Q₇.

(125) Compounds of Preferred 2 where

m is O;

n is O;

J is J-1, J-2, J-3, J-8, J-10 or J-11;

W is O;

R is H;

R₁ is H, CH₃, F, Cl, Br, OCH₃, SCH₃, CH₂ CN, CH₂ OCH₃, CF₃ or OCF₂ H;

R₃ is H, C₁ -C₃ alkyl, CH₂ CH₂ OCH₃, CH₂ CH₂ Cl, CH₂ CH₂ F, CH₂ CHF₂, CH₂ CF₃, allyl or propargyl;

R₄ is H or C₁ -C₃ alkyl;

A is A-1;

Z is CH or N;

X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H; and

Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.

(126) Compounds of Preferred 3 where

m is O;

R is H;

R₁ is H;

R₃ is H or C₁ -C₃ alkyl;

R₄ is H or C₁ -C₃ alkyl;

A is A-1;

Z is CH or N;

X is CH₃, OCH₃, OCH₂ CH₃, cyclopropyl, Cl or OCF₂ H; and

Y is CH₃, OCH₃, C₂ H₅, CH₂ OCH₃, NHCH₃ or CH(OCH₃)₂.

Specifically preferred for reasons of greatest ease of synthesis and/or greatest herbicidal efficacy are:

N-[(4-chloro-6-methoxypyrimidin-2-yl)aminocarbonyl]-2-(1-ethyl-1H-tetrazol-5-yl)benzenesulfonamide, m.p. 223°-225° C.;

N-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-methyl-6-(1-methyl-1H-tetrazol-5-yl)benzenesulfonamide, m.p. 178°-189° C.;

N-[(4-chloro-6-methoxypyrimidin-2-yl)aminocarbonyl]-2-(1-methyl-1H-tetrazol-5-yl)benzenesulfonamide, m.p. 225°-227° C.;

N-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(1-methyl-1H-tetrazol-5-yl)benzenesulfonamide, m.p. 207°-210° C.;

N-[(4,6-dimethylpyrimidin-2-yl)aminocarbonyl]-2-(1-methyl-1H-tetrazol-5-yl)benzenesulfonamide, m.p. 224°-226° C.;

N-[(4-methoxy-6-methylpyrimidin-2-yl)aminocarbonyl]-1-methyl-4-(2-methyl-2H-tetrazol-5-yl)-1H-pyrazole-5-sulfonamide, m.p. 181°-183° C.;

N-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-1-methyl-4-(2-methyl-2H-tetrazol-5-yl)-1H-pyrazole-5-sulfonamide, m.p. 171°-173° C.

N-[[N-4,6-dimethoxy-1,3,5-triazin-2-yl)-N-methylamino]carbonyl]-2-(5-methyl-1H-tetrazol-1-yl)benzenesulfonamide, m.p. 180°-182° C.; and

N-[[N-(4,6-dimethoxy-1,3,5-triazin-2-yl)-N-methylamino]carbonyl]-2-(5-methyl-1H-tetrazol-1-yl)benzenesulfonamide, sodium salt, NMR (CDCl₃) δ 8.4-8.13 (m, 1H), 7.70-7.40 (m, 1H), 7.25-7.00 (m, 1H), 3.85 (s, 6H), 3.19 (s, 3H), 2.32 (s, 3H).

DETAILED DESCRIPTION OF THE INVENTION

Synthesis

Compounds of Formula I can be synthesized by one or both of the methods known below in Equation 1 and 2.

Equation 1 illustrates the reaction of sulfonyl isocyanates and isothiocyanates of Formula II with the appropriate heterocyclic amines of Formula III to give the desired sulfonylureas and sulfonylthioureas of Formula I.

Equation 1 ##STR23## wherein J, W, R, and A are as previously defined.

The reaction of Equation 1 is best carried out in an inert aprotic solvent such as methylene chloride, tetrahydrofuran or acetonitrile at a temperature between 0° and 82° C. A catalytic amount of 1,4-diazabicyclo[2,2,2]octane (DABCO®) may be used to accelerate the reaction. In cases in which the products are insoluble in the reaction solvent, they may be isolated by simple filtration. When the products are soluble, they can be isolated by evaporation of the solvent and trituration of the residue with solvents such as 1-chlorobutane, diethyl ether or ethyl acetate, and filtration.

Compounds of Formula I can be prepared as shown below in Equation 2 by the reaction of sulfonamides IV with the phenyl ester of the appropriate carbamic acid or thiocarbamic acid of Formula V, in the presence of an equimolar quantity of a tertiary amine base such as 1,8-diazabicyclo[5,4,0]undec-7-ene (DBU).

Equation 2 ##STR24## wherein

J, R, W and A are as previously defined.

The reaction shown in Equation 2 is best carried out at 25° C. in a solvent such as dioxane or acetonitrile for 1-2 hours under an inert atmosphere as described in European Patent Application No. 70,804 (published Jan. 26, 1983). The desired products of Formula I can be coveniently isolated by acidifying the reaction solution with aqueous hydrochloric acid. Alternatively, the aqueous layer can be extracted with a solvent such as methylene chloride or ethyl acetate. Drying and evaporation of the solvent affords the desired products.

The phenylcarbamates and phenylthiocarbamates of Formula V can be prepared by methods, or modifications thereof known to those skilled in the art, described in South African Patent Application 82/5671 and South African Patent Application 82/5045.

A judicious choice of the appropriate methods for preparing compounds of Formula I must take into account the nature of the substituents contained within the J values (J₁ -J₆), namely Q and R₁, and their chemical compatibility with the reaction conditions of Equations 1 and 2.

Sulfonyl isocyanates of Formula II can be prepared as shown in Equation 3 by the reaction of sulfonamides of the general structure IV with phosgene in the presence of n-butyl isocyanate and a catalytic amount of 1,4-diazabicyclo[2.2.2]octane (DABCO).

Equation 3 ##STR25## wherein

J is as previously defined, provided E is not oxygen.

The reaction depicted in Equation 3 is best carried out according to the procedure described in U.S. Pat. No. 4,238,621.

Alternatively, sulfonyl isocyanates II can be prepared via phosgenation of the preformed n-butylureas of Formula VI as represented in Equation 4.

Equation 4 ##STR26## wherein

J is as previously defined, provided E is not oxygen.

The compounds of Formula VI are conveniently prepared by stirring a mixture of the appropriate sulfonamide IV, anhydrous potassium carbonate, and n-butyl isocyanate in a suitable solvent such as acetone or methyl ethyl ketone at 25° to 80° C. until all of the isocyanate has reacted. The products are isolated by quenching in dilute aqueous acid and recrystallizing the insoluble solid. The n-butylureas VI are then treated with phosgene and a catalytic amount of DABCO in refluxing xylenes or chlorobenzene in a manner analogous to that described in the reference cited for Equation 3.

Alternatively, treatment of the sulfonamides of Formula IV with thionyl chloride gives intermediate N-sulfinylsulfonamides VII, which afford sulfonylisocyanates II (where W is O) upon exposure to phosgene in the presence of a catalytic amount of pyridine.

Equation 5 ##STR27##

The reaction of Equation 5 can best be performed according to the procedure of H. Ulrich, B. Tucker and A. Sayigh, J. Org. Chem., 34, 3200 (1969).

Sulfonyl isothiocyanates II (where W is S) are known in the art and are prepared from the corresponding sulfonamides (IV) by reaction with carbon disulfide and potassium hydroxide followed by treatment of the resulting dipotassium salt with phosgene. Such a procedure is described in Arch. Pharm. 299, 174 (1966).

A judicious choice of the appropriate method for preparing compounds of Formula II must take into account the nature of the substituents contained within the J values (J₁ -J₆), namely Q and R₁, and their chemical compatibility with reaction conditions of Equations 3-5.

The required sulfonamides of Formula IV can be synthesized by one or more of the methods shown below.

Equation 6 depicts the reaction of sulfonyl chlorides of Formula VIII with ammonia to give sulfonamides of Formula IVa.

Equation 6 ##STR28## wherein

J is as previously defined, provided E is not oxygen.

The amination of Equation 6 can be effected by adding at least two molar equivalents of either anhydrous ammonia or concentrated ammonium hydroxide to a solution of the sulfonyl chloride VIII in a solvent such as diethyl ether, methylene chloride, or tetrahydrofuran at temperatures between -30° and 25° C. The sulfonamides of Formula IVa are isolated either by filtration, in which case the ammonium chloride by-product is removed by washing with water, or extraction into an organic solvent such as methylene chloride. Drying and evaporation of the solvent affords the sulfonamides IVa, which are usually sufficiently pure to be carried directly on to the next step.

Sulfonyl chlorides of Formula VIII can be prepared by one or more of the methods shown below in Equations 7, 8 and 9.

The reaction of an appropriately substituted N-arylhydroxylamine of Formula IX, as shown in Equation 7, and subsequent displacement with sulfur dioxide in the presence of cupric or cuprous chloride yields the desired sulfonyl chloride of Formula VIII.

Equation 7 ##STR29##

The reaction of Equation 7 can be carried out by combining the appropriate arylhydroxylamine with aqueous concentrated hydrochloric acid and acetic acid and adding an aqueous solution of sodium nitrite at -10° to 10° C. After being stirred for 10 minutes to two hours the reaction mixture is added to a mixture of acetic acid, a catalytic amount of cuprous or cupric chloride and excess sulfur dioxide at -5° to 20° C. After being stirred for 0.5 to 24 hours the mixture is diluted with cold water and the product is extracted into a solvent such as methylene chloride or ethyl ether.

The solution of sulfonyl chloride thus obtained can be treated as in Equation 6 to prepare the desired sulfonamide IVa.

Diazotization of appropriately substituted amine derivatives of Formula X, as shown in Equation 8, and subsequent reaction with sulfur dioxide in the presence of either cupric or cuprous chloride gives the desired products of Formula VIII.

Equation 8 ##STR30##

The reaction of Equation 8 can be effected by methods analogous to those described in EP-A Nos. 83,975 and 85,476 (published Aug. 10, 1983). In Equation 8, a substituted amine X, in concentrated hydrochloric acid is treated with a solution of sodium nitrite in water at -5° to 5° C. After being stirred for 10 minutes to one hour at about 0° C., the solution is added to a mixture of excess sulfur dioxide and a catalytic amount of cupric or cuprous chloride in acetic acid at about 10° C. After being stirred for 0.25 to 24 hours at temperatures between 10° to 25° C., the solution is poured into a large excess of ice water. The sulfonyl chloride VIII can be isolated by filtration, or by extraction into a solvent such as methylene chloride or ether, followed by drying and evaporation of the solvent.

Alternatively, diazotization of appropriately substituted amine hydrochloride salts of Formula Xa can be effected under anhydrous conditions, as shown in Equation 8a, and subsequent reaction with sulfur dioxide and cupric chloride gives the desired products of Formula VIII.

Equation 8a ##STR31##

The amine hydrochloride salts Xa are diazotized with an alkylnitrite in a suitable solvent such as acetonitrile or acetone, and the resulting diazonium salts are reacted with sulfur dioxide and cupric chloride to give sulfonyl chlorides VIII. M. Doyle, in J. Org. Chem. 42, 2426, 2431 (1977), describes conditions for conducting similar Meerwein reactions.

Sulfonyl chlorides can also be prepared as shown below in Equation 9 by metal halogen exchange or directed lithiation of appropriately substituted aryl or heterocyclic substrates XI, and trapping with sulfuryl chloride.

Equation 9 ##STR32## wherein

J is as previously described provided that R₁ is not CO₂ R_(c), C₁ -C₃ haloalkyl, Br, nitro, C₁ -C₃ alkylsulfonyl or CN.

The lithiation shown in Equation 9 can be performed according to the procedure of S. H. Bhattacharya, et al., J. Chem. Soc. (C), 1265 (1968) or by procedures reviewed by H. Gschwind and H. Rodriquez in Organic Reactions, Vol. 26, Wiley, New York, 1979, and references cited within.

Compounds of Formula VIII can be prepared via oxidative chlorination of the appropriate thioethers or mercaptans of Formula XII as represented in Equation 10.

Equation 10 ##STR33## wherein

J is as previously defined, R₁₅ is H, C₂ -C₄ alkyl or benzyl, R₁ is not C₁ -C₃ alkylthio or C₁ -C₃ alkylsulfinyl, and R₄ is not C₁ -C₄ alkylthio or C₁ -C₄ alkylsulfinyl.

The reaction of Equation 10 can be carried out by treating a solution of the thioether XII in a solvent such as acetic acid in the presence of at least 2.5 equivalents of water and at least 3.0 equivalents of chlorine at 0°-30° C. for 0.25 to 5 hours. The reaction is poured into ice-water and the product is isolated by extraction with a suitable solvent such as methylene chloride, dried, and the solvent evaporated to yield a product sufficiently pure to be carried directly on to the next step.

Arylmethanesulfonyl chlorides of Formula VIIIb can be prepared from appropriately substituted benzyl chlorides or bromides of Formula XIII by a simple two-step procedure outlined in Equation 11.

Equation 11 ##STR34## wherein J'CH₂ is defined as for J-1 through J-6 where E is CH₂ ;

R₁, R₄ and Q are as previously defined except R₁ is not C₁ -C₃ alkylthio or C₁ -C₃ alkylsulfinyl, and R₄ is not C₁ -C₄ alkylthio or C₁ -C₄ alkylsulfinyl; and

M is Cl or Br.

The conversion of alkyl halides of Formula XIII to isothiouronium salts of Formula XIV can be carried out by the procedure or T. B. Johnson and J. M. Sprague, J. Am. Chem. Soc., 58, 1348 (1936); 59 1837 and 2439 (1937); 61 176 (1939). Oxidative chlorination of isothouronium salts such as XIV to afford sulfonyl chlorides of Formula VIIIb is best carried out according to the procedure of Johnson as described in J. Am. Chem. Soc. 61, 2548 (1939).

The requisite tetrazole substituted intermediates can be prepared by various methods depending on the nature of the aromatic ring in J (J-1 to J-6) systems on which the tetrazole is substituted and the nature of the other substituents present on J (J-1 to J-6). These intermediates can be prepared by one skilled in the art by the methods referred to in the following reviews on tetrazole chemistry: F. R. Benson, "Heterocyclic Compounds" (R. C. Elderfield, Ed.) 8, 1-104, John Wiley and Sons, New York, (1967); R. N. Butler, "Advances in Heterocyclic Chem.", 21, 323-436, Academic Press (1977); R N. Butler, "Comprehensive Heterocyclic Chem.", (K. T. Potts, Ed.) 5, 791-838, Pergamon Press (1984) and F. R. Benson, "High Nitrogen Compounds", John Wiley and Sons, New York (1983).

The heterocyclic amines of Formula III in Equation 1 above can be prepared by methods known in the literature, or simple modifications thereof, by those skilled in the art. For instance, EP-A No. 84,224 (published July 27, 1983) and W. Braker et al., J. Am. Chem. Soc., 69, 3072 (1947) describes methods for preparing aminopyridines and triazines substituted by acetal groups such as dialkoxymethyl or 1,3-dioxolan-2-yl, among other groups. Also, for example, South African patent application Nos. 82/5045 and 82/5671 describe methods for preparing aminopyrimidines and triazines substituted by haloalkyl or haloalkylthio groups such as OCH₂ CH₂ F, OCH₂ CF₃, SCF₂ H, or OCF₂ H, among other groups. South African patent application No. 83/7434 (published Oct. 5, 1983) describes methods for the synthesis of cycopropylpyrimidines and triazines substituted by such groups as alkyl, haloalkyl, alkoxy, haloalkoxy, alkylamino, dialkylamino or alkoxyalkyl.

The 5,6-dihydrofuro[2,3-d]pyrimidine-2-amines, the cyclopenta[d]pyrimidin-2-amines (III, A is A-2) and the 6,7-dihydro-5H-pyrano[2,3-d]pyrimidin-2-amines (III, A is A-3) can be prepared as described in EP-A No. 15,683. The furo[2,3-d]pyrimidin-2-amines (III, A is A-4) are described in EP-A No. 46,677.

Compounds of Formula III, where A is A-5, are described in EP-A-73,562. Compounds of Formula III, where A is A-6 are described in EP-A-94,260.

In addition, general methods for preparing aminopyrimidines and triazines have been reviewed in the following publications:

"The Chemistry of Heterocyclic Compounds", a series published by Interscience Publishers, Inc., New York and London;

"Pyrimidines", Vol. 16 of the same series by D. J. Brown;

"s-Triazines and Derivatives", Vol. 13 of the same series by E. M. Smolin and L. Rappoport; and

F. C. Schaefer, U.S. Pat. No. 3,154,547 and K. R. Huffman and F. C. Schaefer, J. Org. Chem., 28, 1812 (1963), which describes the synthesis of triazines.

Agriculturally suitable salts of compounds of Formula I are also useful herbicides and can be prepared in a number of ways known to the art. For example, metal salts can be made by contacting compounds of Formula I with a solution of an alkali or alkaline earth metal salt having a sufficiently basic anion (e.g., hydroxide, alkoxide or carbonate). Quaternary amine salts can be made by similar techniques.

A particularly useful process for preparing salts of compounds of Formula I involves reaction of a solution of the sulfonylurea in a water-immiscible halogenated hydrocarbon solvent with the appropriate alkali or alkaline earth metal hydroxide as described in copending application, U.S. Ser. No. 086,867 filed on Aug. 19, 1987.

Salts of compounds of Formula I can also be prepared by exchange of one cation for another. Cationic exchange can be effected by direct contact of an aqueous solution of a salt of a compound of Formula I (e.g. alkali or quaternary amine salt) with a solution containing the cation to be exchanged. This method is most effective when the desired salt containing the exchange cation is insoluble in water and can be separated by filtration.

Exchange may also be effected by passing an aqueous solution of a salt of a compound of Formula I (e.g., an alkali metal or quaternary amine salt) through a column packed with a cation exchange resin containing the cation to be exchanged for that of the original salt and the desired product is eluted from the column. This method is particularly useful when the desired salt is water-soluble, e.g., a potassium, sodium or calcium salt.

Acid addition salts, useful in this invention, can be obtained by reacting a compound of Formula I with a suitable acid, e.g., p-toluenesulfonic acid, trichloroacetic acid or the like.

The preparation of the compounds of this invention is further illustrated by the following specific examples.

EXAMPLE 1 1-(2-Chlorosulfonylphenyl)-5-methyl-1H-tetrazole

To 5 g of 1-(2-hydroxylaminophenyl)-5-methyl-1H-tetrazole in 12 mL of 37% hydrochloric acid and 5 mL of acetic acid at 0°-5° C. was added 2.3 g of sodium nitrite in 10 mL of water. The resultant solution was stirred at -5° to +5° C. for one hour and then added portionwise, with stirring, to a mixture of 25 mL of acetic acid, 0.5 g of cupric chloride and 5 mL of liquified sulfur dioxide at below 5° C. After stirring for two hours, during which time the mixture was allowed to warm to room temperature, it was poured into 150 mL of ice and water and extracted twice with 150 mL of methylene chloride. The methylene chloride solution was washed three times with 100 mL portions of water, two times with 100 mL of saturated aqueous sodium bicarbonate followed by single washes with 100 mL of saturated aqueous sodium chloride and 100 mL of water. The methylene chloride solution was then dried over magnesium sulfate and filtered to yield a solution containing the desired sulfonylchloride. This solution was used without further work-up to prepare the sulfonamide of Example 2.

EXAMPLE 2 1-(2-Aminosulfonylphenyl)-5-methyl-1H-tetrazole

Twenty-five mL of 28% ammonium hydroxide was added to the methylene chloride solution obtained from Example 2 and the mixture was stirred for two hours and concentrated in vacuo to yield a mixture of an oil and a solid. The solid product was separated by filtration and washed with water to yield 2.2 g of the desired product, which melted at 141°-148° C. Infrared absorption peaks at 3260 and 3360 cm⁻¹ were consistent for NH₂ and 1160 and 1350 cm⁻¹ consistent for the SO₂ of the desired product. Elem. anal. calc'd for C₈ H₉ N₅ O₂ S:C, 40.15; H, 3.79; N, 29.26, S. 13.39. Found: C, 40.43; H, 3.84; N, 29.61; S, 13.04.

EXAMPLE 4 5-(2-Chlorosulfonylphenyl)-2-methyl-2H-tetrazole and 5-(2-chlorosulfonylphenyl)-1-methyl-1H-tetrazole

To 5 g of a mixture of 5-(2-hydroxylaminophenyl)-2-methyl-2H-tetrazole and 5-(2-hydroxyaminophenyl)-1-methyl-1H-tetrazole dissolved in 12 mL of 37% hydrochloric acid and 5 mL of acetic acid was added with stirring 2.3 g of sodium nitrite dissolved in 10 mL of water at -5° to 5° C. After one hour this solution was added, at 0°-5° C., portionwise to a mixture of 25 mL of acetic acid, 0.5 g of cupric chloride and 5 mL of liquified sulfur dioxide. After the addition was completed the cooling bath was removed and the reaction mixture was allowed to warm to 31° C. whereupon the cooling bath was reapplied and the stirring was continued until two and one half hours after completion of the addition. The mixture was then poured into ice and worked up as described in Example 1 except that the desired methylene chloride solution was concentrated in vacuo to yield an oil which solidified. This product, (3.28 g) which was a mixture of the desired sulfonylchlorides, was of sufficient purity for the preparation of the sulfonamides of Example 4.

EXAMPLE 4 5-(2-Aminosulfonylphenyl)-2-methyl-2H-tetrazole and 5-(2-aminosulfonylphenyl)-1-methyl-1H-tetrazole

The solid product obtained in Example 3 was dissolved in 50 mL of tetrahydrofuran and added portionwise to 20 mL of 28% ammonium hydroxide. The mixture was stirred for one hour and concentrated in vacuo. Water was added to the residue, the mixture filtered and the solid washed with a small amount of cold water to yield 1.3 g of the isomer mixture. Infrared absorption spectra showed peaks at 3260 and 3360 cm⁻¹ consistent for NH₂ and 1160 and 1330 consistent for the SO₂ group of the desired product. Elem. anal. calc'd. for C₈ H₉ N₅ O₂ S:C, 40.15; H, 3.79; N, 29.26; S, 13.39. Found: C, 40.49; H, 3.86; N, 29.99; S, 13.75.

EXAMPLE 5 5-(2-Aminosulfonylphenyl)-1-methyl-1H-tetrazole

To 4.4 g of 5-(2-ethylthiophenyl)-1-methyl-1H-tetrazole in 40 mL of propionic acid and 1.08 g of water at -10° C. was added slowly, dropwise, 5.2 mL, of liquid chlorine (1.367 g/mL). After the addition the mixture was allowed to warm to room temperature, and was then poured into approximately 100 g of ice. The resultant sulfonyl chloride was extracted with methylene chloride, washed with water and the methylene chloride solution added to 45 mL of concentrated aqueous ammonium hydroxide while maintaining the reaction temperature below 25° C. with ice bath cooling. Evaporation of the methylene chloride yielded a solid product which was removed by filtration from the aqueous residue and washed with water. The product, 3.72 g, melted at 176°-179° C. and showed absorption peaks by infrared spectroscopy at 3210 and 3300 cm⁻¹, consistent for the desired sulfonamide.

EXAMPLE 6 5-(2-Aminosulfonyl-4-methylphenyl)-1-methyl-1H-tetrazole

To a mixture of 4.68 g of 5-(4-methyl-2-propylthiophenyl)-1-methyl-1H-tetrazole, 40 mL of propionic acid and 1.08 g of water cooled to -10° C. was added dropwise 5.2 mL (liquified) of chlorine while maintaining the reaction temperature at -10° to 0° C. After one-half hour the reaction mixture was allowed to warm to room temperature and stirred for one hour. It was then poured into 200 mL of ice and water and extracted with methylene chloride. The methylene chloride solution was added to 45 mL of concentrated ammonium hydroxide at 10° C. and stirred overnight. The mixture was concentrated in vacuo to an oil residue which was taken up in 100 mL of methylene chloride washed with three 100 mL portions of water and 100 mL of saturated aqueous sodium hydroxide. The methylene chloride solution was then dried over magnesium sulfate, filtered, and the filtrate evaporated to yield 4.1 g of the desired product melting at 161°-171° C.

NMR (CDCl₃): δ 2.56 (s, CH₃ on phenyl); 3.99 (s, CH₃ on tetrazole); 5.6 (s, w, NH₂); and 7.3-8.1 (m, 3 CH on phenyl).

EXAMPLE 7 5-(2-Aminosulfonyl-3-methylphenyl)-1-methyl-1H-tetrazole

To a mixture of 14.6 mL of concentrated (12M) hydrochloric acid, 6.1 mL of acetic acid, 25 mL of ethyl ether and 6.91 g of 5-(2-amino-3-methylphenyl)-1-methyl-1H-tetrazole at 0° C. was added dropwise 2.8 g of sodium nitrite dissolved in 12.2 mL of water while maintaining the reaction temperature at below 10° C. Stirring was continued for one hour after the addition was completed. This mixture was then added slowly to 30.5 mL of acetic acid containing 0.6 g of cupric chloride and 6.1 mL of liquified sulfur dioxide.

After stirring for two hours at ambient temperature, the mixture was poured into 200 mL of ice-water and extracted twice with 125 mL of methylene chloride. The organic phase was then washed twice with 200 ml of water, once with 200 mL saturated aqueous sodium chloride, once with 200 mL aqueous sodium bicarbonate followed by 200 mL of water and 200 mL saturated aqueous sodium chloride. The organic phase was then added dropwise to 25 mL of concentrated aqueous ammonium hydroxide and the mixture stirred overnight and evaporated to a solid, which was washed with water and dried. The crude product thus obtained melted at 140°-161° C., yield 6.26 g. Mass spectral analysis showed a molecular weight of 253 (calc. 253) for the product.

EXAMPLE 8 N-[(4,6-Dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(2-methyl-2H-tetrazol-5-yl)benzenesulfonamide

To 25 mL of acetonitrile was added at ambient temperature and pressure 0.48 g of 5-(2-aminosulfonylphenyl)-2-methyl-2H-tetrazole and 0.54 g of phenyl N-(4,6-dimethoxypyrimidin-2-yl)carbamate followed by 0.3 mL of DBU. After being stirred for three hours the reaction mixture was added to 25 g of ice and acidified to pH 3 with hydrochloric acid. The precipitate thus obtained was filtered, washed with water and dried to yield 0.66 g of the desired product, m.p. 214°-222° C. Infrared absorptions at 1720, 1600 and 1580 cm⁻¹ were consistent with the desired structure.

NMR(CDCl₃):δ 3.91 (s, 2 X CH₃ O), 5.82 (s, CH, pyrimidin), 4.43 (s, CH₃ on N-2 of tetrazole), 4.38 (s, CH₃ on N-1 of tetrazole).

Integration of the peaks at 4.43 d and 4.38 d total one CH₃ indicating a ratio of 2-methyl-2H-tetrazole to 1-methyl-1H-tetrazole of 2:1. This mixture is suitable for purposes of this invention. If desired, the isomer mixture obtained in Example 6 can be separated by chromatography into its component parts.

EXAMPLE 9 N-[(4,6-Dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(5-methyl-1H-tetrazol-1-yl)benzenesulfonamide

To 0.48 g of 1-(2-aminosulfonylphenyl)-5-methyl 1H-tetrazole in 25 mL of acetonitrile was added at ambient temperature and pressure 0.54 g of phenyl N-(4,6-dimethoxypyrimidin-2-yl)carbamate and 0.3 mL of DBU. The reaction mixture was stirred for three hours, added to 25 g of ice and acidified to pH 3 with hydrochloric acid. The precipitate thus obtained was filtered, washed with water and dried to yield 0.74 g of the desired product, melting point at 213°-216° C. Infrared absorption spectra showed peaks at 1710, 1605 and 1570 cm⁻¹, consistent for the desired product.

NMR(CDCl₃): δ2.48 (s, CH₃ on tetrazole), 3.82 (s, 2XCH₃ O), 5.81 (s, CH-pyrimidin).

EXAMPLE 10 N-[(4-Methoxy-6-methyl-1,3,5-triazin-2-yl)aminocarbonyl]-2-(5-methyl-1H-tetrazol-1-yl)benzenesulfonamide

To 0.48 g of 1-(2-aminosulfonylphenyl)-5-methyl-1H-tetrazole and 0.52 g of phenyl N-(4-methoxy-6-methyl-1,3,5-triazin-2-yl)carbamate in 25 mL of acetonitrile at ambient temperature and pressure was added 0.3 mL of DBU. The mixture was stirred for three hours and then added to 25 g of ice and acidified with hydrochloric acid. The precipitate thus obtained was filtered, washed with water and dried in vacuo to yield 0.65 g of the desired product melting at 207°-209° C. Infrared absorption spectra showed absorption at 1700, 1600 and 1550 cm⁻¹, consistent for the desired structure.

EXAMPLE 11 N-[(4-Chloro-6-methoxypyrimidine-2-yl)aminocarbonyl]-2-(1-methyl-1H-tetrazol-5-yl)benzenesulfonamide

To 0.48 g of 5-(2-aminosulfonylphenyl)-1-methyl-1H-tetrazole and 0.56 g of phenyl N-(4-chloro-6-methoxypyrimidine-2-yl)carbamate in 20 mL of dry acetonitrile at ambient temperature was added, with stirring, 0.3 mL of DBU. After stirring 16 hours the mixture was then poured into 25 g of ice followed by the addition of 10 mL of 2N hydrochloric acid. The precipitate thus formed was removed by filtration, washed with water and dried to yield 0.74 g of the desired product, m.p. 225°-227° C.

NMR (CDCl₃): δ 3.88 (s, CH₃ on tetrazole); 3.95 (s, CH₃ O); 6.52 (s, CH of pyrimidine); 7.2-7.5 (m, CH of phenyl and NH); 7.84 (m, 2 CH of phenyl); 8.6 (m, CH of phenyl); and 11.96 (s, NH).

EXAMPLE 12 N-[(4,6-Dimethoxypyrimidin-2-yl)aminocarbonyl]-5-chloro-2-(4-methyl-5-oxo-1H,4H-tetrazol-5-yl)-benzenesulfonamide

To a stirred solution of 0.29 g of 1-(2-aminosulfonyl-5-chlorophenyl)-4-methyl-1H-tetrazol-5[4H]-one and 0.27 g of phenyl N-(4,6-dimethoxypyrimidin-2-yl)carbamate in 10 mL of acetonitrile at ambient temperature was added 0.1 mL of DBU. The mixture was stirred for two hours, poured into 20 g of ice and acidified with 2N hydrochloric acid. The precipitate was removed by filtration, washed with water and dried to yield 0.37 g of product, m.p. 178°-180° C.

NMR (CDCl₃ 0: δ 3.63 (s, CH₃ on tetrazole); 3.92 (s, 2 X CH₃ O); 5.81 (s, CH or pyrimidine); 7.4-8.6 (m, 3 CH of phenyl); and 12.6 (s, w, NH).

EXAMPLE 13 3-(2-Methyl-2H-tetrazole-5-yl)-1-phenyl-1H-pyrazole-5-sulfonamide

To a mixture of 3.1 mL of 12N hydrochloric acid, 12.5 mL of acetic acid, 3.7 mL of formic acid and 4.5 g of 5-amino-1-phenyl-3-(2-methyl-2H-tetrazol-5-yl)-1H-pyrazole was added dropwise 1.4 g of sodium nitrite in 2.5 mL of water at -8° to -6° C. The mixture was stirred for 15 minutes and then added to 20 mL of acetic acid containing 3.7 mL (liquid) of sulfur dioxide and 0.75 g of cupric chloride dihydrate. After stirring for thirty minutes and allowing to warm to room temperature, the mixture was poured into an ice and water mixture and the precipitate removed by filtration. After washing with water the solid was dissolved in tetrahydrofuran, cooled to -78° C., and ammonia (liquified, 1.0 mL) was added dropwise. The mixture was allowed to stand overnight at ambient temperature and filtered to yield a brown solid. This solid showed peaks at 3300 and 3200 cm⁻¹, consistent for NH₂, and 1370, 1185 and 1170 cm⁻¹, consistent for SO₂.

EXAMPLE 14 N-[[N-(4,6-Dimethoxy-1,3,5-triazin-2-yl)-N-methylamino]carbonyl]-2-(5-methyl-1H-tetrazol-1-yl)benzenesulfonamide

To 0.22 g of 2-(5-methyl-1H-tetrazol-1-yl)benzenesulfonamide (compound of Example 2, 0.32 g) and 0.32 g of phenyl (4,6-dimethoxy-1,3,5-triazin-2-yl)-(methyl)-carbamate in 4 ml of dry acetonitrile was added at room temperature 0.2 ml of DBU. The reaction mixture was allowed to stand for four days, then diluted with 4 ml of water, several ice chips and 4 ml of diethyl ether. After stirring this solution for one minute, the ether layer was removed by pipet and the remaining mixture was acidified by dropwise addition of 1N HCl. The resulting precipitate was filtered, washed with water and dried to give 0.32 g of a white solid, m.p. 180°-182° C. (d).

EXAMPLE 15 Preparation of the sodium salt of N-[[N-(4,6-Dimethoxy-1,3,5-triazin-2-yl)-N-methylamino]carbonyl]-2-(5-methyl-1H-tetrazol-1-yl)-benzenesulfonamide

To a stirred suspension of the compound of Example 14 (16.87 g, 38.7 mmol) and sodium carbonate (36 g) in methylene chloride (400 g), was added 1.79 g of sodium hydroxide (powder, 44.7 mmol). The suspension was allowed to stir at ambient temperature (20°-25° C.) for 16 hours before it was filtered. The filtrate was evaporated under reduced pressure using a rotary evaporator. A colorless solid (17.8 g, 38.7 mmol, 100% yield) was isolated;

NMR (90 MHz, CDCl₃): δ 8.4-8.13 (m, 1H); 7.70-7.40 (m, 1H); 7.25-7.00 (m, 1H); 3.85 (s, 6H); 3.19 (s, 3H); 2.32 (s, 3H).

By using the procedures described in the foregoing equations and examples of modifications thereof, one skilled in the art can prepare the compounds shown in the following tables.

    ______________________________________                                         Compounds                                                                      ______________________________________                                          ##STR35##                                                                     In General Structure 1, A is A-1                                               In General Structure 2, A is A-2                                               In General Structure 3, A is A-3                                               In General Structure 4, A is A-4                                               In General Structure 5, A is A-5                                               In General Structure 6, A is A-6                                               In General Structure 7, A is A-7                                               General Structure 8                                                                        ##STR36##                                                          General Structure 9                                                                        ##STR37##                                                          General Structure 10                                                                       ##STR38##                                                          General Structure 11                                                                       ##STR39##                                                          General Structure 12                                                                       ##STR40##                                                          General Structure 13                                                                       ##STR41##                                                          General Structure 14                                                                       ##STR42##                                                          General Structure 15                                                                       ##STR43##                                                          General Structure 16                                                                       ##STR44##                                                          General Structure 17                                                                       ##STR45##                                                          General Structure 18                                                                       ##STR46##                                                          General Structure 19                                                                       ##STR47##                                                          General Structure 20                                                                       ##STR48##                                                          ______________________________________                                    

                                      TABLE I                                      __________________________________________________________________________     General Structure 1                                                            R.sub.1  E  Q  R.sub.3    W     R  X       Y         Z  m.p.                   __________________________________________________________________________                                                             (°C.)           H        -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             CH.sub.3  CH 224-226                H        -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             OCH.sub.3 CH 222-224                H        -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 CH 207-210                H        -- Q-1                                                                               CH.sub.3   O     H    Cl    OCH.sub.3 CH 225-227                H        -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             OCH.sub.3 N  196-198                H        -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 N  172-187                H        -- Q-1                                                                               C.sub.2 H.sub.5                                                                           O     H    CH.sub.3                                                                             CH.sub.3  CH 200-207                H        -- Q-1                                                                               C.sub.2 H.sub.5                                                                           O     H    CH.sub.3                                                                             OCH.sub.3 CH 203-205                H        -- Q-1                                                                               C.sub.2 H.sub.5                                                                           O     H    OCH.sub.3                                                                            OCH.sub.3 CH 214-217                H        -- Q-1                                                                               C.sub.2 H.sub.5                                                                           O     H    Cl    OCH.sub.3 CH 223-225                H        -- Q-1                                                                               C.sub.2 H.sub.5                                                                           O     H    OC.sub.2 H.sub.5                                                                     NHCH.sub.3                                                                               N  193-200                H        -- Q-1                                                                               C.sub.2 H.sub.5                                                                           O     H    CH.sub.3                                                                             OCH.sub.3 N  192-196                H        -- Q-1                                                                               C.sub.2 H.sub.5                                                                           O     H    OCH.sub.3                                                                            OCH.sub.3 N  192-195                H        -- Q-1                                                                               CH(CH.sub.3).sub.2                                                                        O     H    CH.sub.3                                                                             CH.sub.3  CH                        H        -- Q-1                                                                               CH(CH.sub.3).sub.2                                                                        O     H    CH.sub.3                                                                             OCH.sub.3 CH                        H        -- Q-1                                                                               CH(CH.sub.3).sub.2                                                                        O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        H        -- Q-1                                                                               CH(CH.sub.3).sub.2                                                                        O     H    Cl    OCH.sub.3 CH                        H        -- Q-1                                                                               CH(CH.sub.3).sub.2                                                                        O     H    CH.sub.3                                                                             OCH.sub.3 N                         H        -- Q-1                                                                               CH(CH.sub.3).sub.2                                                                        O     H    OCH.sub.3                                                                            OCH.sub.3 N                         H        -- Q-1                                                                               (CH.sub.2).sub.4 CH.sub.3                                                                 O     H    CH.sub.3                                                                             CH.sub.3  CH                        H        -- Q-1                                                                               (CH.sub.2).sub.4 CH.sub.3                                                                 O     H    CH.sub.3                                                                             OCH.sub.3 CH                        H        -- Q-1                                                                               (CH.sub.2).sub.4 CH.sub.3                                                                 O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        H        -- Q-1                                                                               (CH.sub.2).sub.4 CH.sub.3                                                                 O     H    Cl    OCH.sub.3 CH                        H        -- Q-1                                                                               (CH.sub.2).sub.4 CH.sub.3                                                                 O     H    CH.sub.3                                                                             OCH.sub.3 N                         H        -- Q-1                                                                               (CH.sub.2).sub.4 CH.sub.3                                                                 O     H    OCH.sub.3                                                                            OCH.sub.3 N                         H        -- Q-1                                                                               cyclopentyl                                                                               O     H    CH.sub.3                                                                             CH.sub.3  CH                        H        -- Q-1                                                                               cyclopentyl                                                                               O     H    CH.sub.3                                                                             OCH.sub.3 CH                        H        -- Q-1                                                                               cyclopentyl                                                                               O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        H        -- Q-1                                                                               cyclopentyl                                                                               O     H    Cl    OCH.sub.3 CH                        H        -- Q-1                                                                               cyclopentyl                                                                               O     H    CH.sub.3                                                                             OCH.sub.3 N                         H        -- Q-1                                                                               cyclopentyl                                                                               O     H    OCH.sub.3                                                                            OCH.sub.3 N                         H        -- Q-1                                                                               CH.sub.2 Cl                                                                               O     H    CH.sub.3                                                                             CH.sub.3  CH                        H        -- Q-1                                                                               CH.sub.2 Cl                                                                               O     H    CH.sub.3                                                                             OCH.sub.3 CH                        H        -- Q-1                                                                               CH.sub.2 Cl                                                                               O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        H        -- Q-1                                                                               CH.sub.2 Cl                                                                               O     H    Cl    OCH.sub.3 CH                        H        -- Q-1                                                                               CH.sub.2 Cl                                                                               O     H    CH.sub.3                                                                             OCH.sub.3 N                         H        -- Q-1                                                                               CH.sub.2 Cl                                                                               O     H    OCH.sub.3                                                                            OCH.sub.3 N                         H        -- Q-1                                                                               (CH.sub.2).sub.2 F                                                                        O     H    CH.sub.3                                                                             CH.sub.3  CH                        H        -- Q-1                                                                               (CH.sub.2).sub.2 F                                                                        O     H    CH.sub.3                                                                             OCH.sub.3 CH                        H        -- Q-1                                                                               (CH.sub.2).sub.2 F                                                                        O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        H        -- Q-1                                                                               (CH.sub.2).sub.2 F                                                                        O     H    Cl    OCH.sub.3 CH                        H        -- Q-1                                                                               (CH.sub.2).sub.2 F                                                                        O     H    CH.sub.3                                                                             OCH.sub.3 N                         H        -- Q-1                                                                               (CH.sub.2).sub.2 F                                                                        O     H    OCH.sub.3                                                                            OCH.sub.3 N                         H        -- Q-1                                                                               --CH.sub.2 CH═CH.sub.2                                                                O     H    CH.sub.3                                                                             CH.sub.3  CH                        H        -- Q-1                                                                               --CH.sub.2 CH═CH.sub.2                                                                O     H    CH.sub.3                                                                             OCH.sub.3 CH                        H        -- Q-1                                                                               --CH.sub.2 CH═CH.sub.2                                                                O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        H        -- Q-1                                                                               --CH.sub.2 CH═CH.sub.2                                                                O     H    Cl    OCH.sub.3 CH                        H        -- Q-1                                                                               --CH.sub.2 CH═CH.sub.2                                                                O     H    CH.sub.3                                                                             OCH.sub.3 N                         H        -- Q-1                                                                               --CH.sub.2 CH═CH.sub.2                                                                O     H    OCH.sub.3                                                                            OCH.sub.3 N                         H        -- Q-1                                                                               CH.sub.2 CH═CHCH.sub. 2 Cl                                                            O     H    CH.sub.3                                                                             CH.sub.3  CH                        H        -- Q-1                                                                               CH.sub.2 CH═CHCH.sub.2 Cl                                                             O     H    CH.sub.3                                                                             OCH.sub.3 CH                        H        -- Q-1                                                                               CH.sub.2 CH═CHCH.sub.2 Cl                                                             O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        H        -- Q-1                                                                               CH.sub.2 CH═CHCH.sub.2 Cl                                                             O     H    Cl    OCH.sub.3 CH                        H        -- Q-1                                                                               CH.sub.2 CH═CHCH.sub.2 Cl                                                             O     H    CH.sub.3                                                                             OCH.sub.3 N                         H        -- Q-1                                                                               CH.sub.2 CH═CHCH.sub.2 Cl                                                             O     H    OCH.sub.3                                                                            OCH.sub.3 N                         H        -- Q-1                                                                               CH.sub.2 --C.tbd.C--CH.sub.3                                                              O     H    CH.sub.3                                                                             CH.sub.3  CH                        H        -- Q-1                                                                               CH.sub.2 --C.tbd.C--CH.sub.3                                                              O     H    CH.sub.3                                                                             OCH.sub.3 CH                        H        -- Q-1                                                                               CH.sub.2 --C.tbd.C--CH.sub.3                                                              O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        H        -- Q-1                                                                               CH.sub.2 --C.tbd.C--CH.sub.3                                                              O     H    Cl    OCH.sub.3 CH                        H        -- Q-1                                                                               CH.sub.2 --C.tbd.C--CH.sub.3                                                              O     H    CH.sub.3                                                                             OCH.sub.3 N                         H        -- Q-1                                                                               CH.sub.2 --C.tbd.C--CH.sub.3                                                              O     H    OCH.sub.3                                                                            OCH.sub.3 N                         H        -- Q-1                                                                               C.sub.6 H.sub.5                                                                           O     H    CH.sub.3                                                                             CH.sub.3  CH                        H        -- Q-1                                                                               C.sub.6 H.sub.5                                                                           O     H    CH.sub.3                                                                             OCH.sub.3 CH                        H        -- Q-1                                                                               C.sub.6 H.sub.5                                                                           O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        H        -- Q-1                                                                               C.sub.6 H.sub.5                                                                           O     H    Cl    OCH.sub.3 CH                        H        -- Q-1                                                                               C.sub.6 H.sub.5                                                                           O     H    CH.sub.3                                                                             OCH.sub.3 N                         H        -- Q-1                                                                               C.sub.6 H.sub.5                                                                           O     H    OCH.sub.3                                                                            OCH.sub.3 N                         H        -- Q-1                                                                               (CH.sub.2).sub.4 OCH.sub.3                                                                O     H    CH.sub.3                                                                             CH.sub.3  CH                        H        -- Q-1                                                                               (CH.sub.2).sub.4 OCH.sub.3                                                                O     H    CH.sub.3                                                                             OCH.sub.3 CH                        H        -- Q-1                                                                               (CH.sub.2).sub.4 OCH.sub.3                                                                O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        H        -- Q-1                                                                               (CH.sub.2).sub.4 OCH.sub.3                                                                O     H    Cl    OCH.sub.3 CH                        H        -- Q-1                                                                               (CH.sub.2).sub.4 OCH.sub.3                                                                O     H    CH.sub.3                                                                             OCH.sub.3 N                         H        -- Q-1                                                                               (CH.sub.2).sub.4 OCH.sub.3                                                                O     H    OCH.sub.3                                                                            OCH.sub.3 N                         H        -- Q-1                                                                               (CH.sub.2).sub.2 SCH.sub.2 CH.sub.3                                                       O     H    CH.sub.3                                                                             CH.sub.3  CH                        H        -- Q-1                                                                               (CH.sub.2).sub.2 SCH.sub.2 CH.sub.3                                                       O     H    CH.sub.3                                                                             OCH.sub.3 CH                        H        -- Q-1                                                                               (CH.sub.2).sub.2 SCH.sub.2 CH.sub.3                                                       O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        H        -- Q-1                                                                               (CH.sub.2).sub.2 SCH.sub.2 CH.sub.3                                                       O     H    Cl    OCH.sub.3 CH                        H        -- Q-1                                                                               (CH.sub.2).sub.2 SCH.sub.2 CH.sub.3                                                       O     H    CH.sub.3                                                                             OCH.sub.3 N                         H        -- Q-1                                                                               (CH.sub.2).sub.2 SCH.sub.2 CH.sub.3                                                       O     H    OCH.sub.3                                                                            OCH.sub.3 N                         5-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             CH.sub.3  CH 235-238                5-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             OCH.sub.3 CH 233-234                5-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 CH 213-216                5-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H    Cl    OCH.sub.3 CH 217-219                5-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             OCH.sub.3 N  200-205                5-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 N  195-198                3-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 CH 192-197                3-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 N  201-206                3-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            CH.sub.3  N  159-173                3-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            CH.sub.3  CH 219-222                3-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             CH.sub.3  CH 223-226                3-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H    Cl    OCH.sub.3 CH 181-186                3-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H    OC.sub.2 H.sub.5                                                                     NHCH.sub.3                                                                               N  187-190                4-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            CH.sub.3  N  179-186                4-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 CH 214-218                4-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            CH.sub.3  CH 225-229                4-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 N  191-196                4-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             CH.sub.3  CH 182-196                4-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H    Cl    OCH.sub.3 CH 140-150                4-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H    OC.sub.2 H.sub.5                                                                     NHCH.sub.3                                                                               N  152-160                6-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 N  197-200                6-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            CH.sub.3  N  198-202                6-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 CH 178-180                6-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            CH.sub.3  CH 180-183                6-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             CH.sub.3  CH 213-215                6-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H    Cl    OCH.sub.3 CH 196-199                5-Cl     -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             CH.sub.3  CH 221-223                5-Cl     -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             OCH.sub.3 CH 207-210                5-Cl     -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 CH 214-216                5-Cl     -- Q-1                                                                               CH.sub.3   O     H    Cl    OCH.sub.3 CH 203-205                5-Cl     -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             OCH.sub.3 N  191-193                5-Cl     -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 N  175-180                5-Cl     -- Q-1                                                                               CH.sub.3   O     H    OC.sub.2 H.sub.5                                                                     NHCH.sub.3                                                                               N  144-158                5-Cl     -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            CH(OCH.sub.3).sub.2                                                                      CH 180-183                5-Br     -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             CH.sub.3  CH                        5-Br     -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             OCH.sub.3 CH                        5-Br     -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        5-Br     -- Q-1                                                                               CH.sub.3   O     H    Cl    OCH.sub.3 CH                        5-Br     -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             OCH.sub.3 N                         5-Br     -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 N                         5-OCF.sub.2 H                                                                           -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             CH.sub.3  CH                        5-OCF.sub.2 H                                                                           -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             OCH.sub.3 CH                        5-OCF.sub.2 H                                                                           -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        5-OCF.sub.2 H                                                                           -- Q-1                                                                               CH.sub.3   O     H    Cl    OCH.sub.3 CH                        5-OCF.sub.2 H                                                                           -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             OCH.sub.3 N                         5-OCF.sub.2 H                                                                           -- Q-1                                                                               CH.sub. 3  O     H    OCH.sub.3                                                                            OCH.sub.3 N                         5-OCH.sub.3                                                                             -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             CH.sub.3  CH 198-200                5-OCH.sub.3                                                                             -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             OCH.sub.3 CH 218-219                5-OCH.sub.3                                                                             -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 CH 205-207                5-OCH.sub.3                                                                             -- Q-1                                                                               CH.sub.3   O     H    Cl    OCH.sub.3 CH 185-188                5-OCH.sub.3                                                                             -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             OCH.sub.3 N                         5-OCH.sub.3                                                                             -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 N                         5-CF.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             CH.sub.3  CH                        5-CF.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             OCH.sub.3 CH                        5-CF.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        5-CF.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H    Cl    OCH.sub.3 CH                        5-CF.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             OCH.sub.3 N                         5-CF.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 N                         5-CH.sub.2 OCH.sub.3                                                                    -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             CH.sub.3  CH                        5-CH.sub.2 OCH.sub.3                                                                    -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             OCH.sub.3 CH                        5-CH.sub.2 OCH.sub.3                                                                    -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        5-CH.sub.2 OCH.sub.3                                                                    -- Q-1                                                                               CH.sub.3   O     H    Cl    OCH.sub.3 CH                        5-CH.sub.2 OCH.sub.3                                                                    -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             OCH.sub.3 N                         5-CH.sub.2 OCH.sub.3                                                                    -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 N                         6-Cl     -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             CH.sub.3  CH 159-164                6-Cl     -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            CH.sub.3  CH 196-199                6-Cl     -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 CH 153-156                6-Cl     -- Q-1                                                                               CH.sub.3   O     H    Cl    OCH.sub.3 CH 166-170                6-Cl     -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             OCH.sub.3 N  187-189                6-Cl     -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 N  202-205                6-OCH.sub.3                                                                             -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             CH.sub.3  CH 181-186                6-OCH.sub.3                                                                             -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            CH.sub.3  CH 205-209                6-OCH.sub.3                                                                             -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 CH 174-181                5-SCH.sub.3                                                                             -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             CH.sub.3  CH                        5-SCH.sub.3                                                                             -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             OCH.sub.3 CH                        5-SCH.sub.3                                                                             -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        5-SCH.sub.3                                                                             -- Q-1                                                                               CH.sub.3   O     H    Cl    OCH.sub.3 CH                        5-SCH.sub.3                                                                             -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             OCH.sub.3 N                         5-SCH.sub.3                                                                             -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 N                         5-SCH.sub.3                                                                             -- Q-1                                                                               C.sub.2 H.sub.5                                                                           O     H    CH.sub.3                                                                             CH.sub.3  CH                        5-SCH.sub.3                                                                             -- Q-1                                                                               C.sub.2 H.sub.5                                                                           O     H    CH.sub.3                                                                             OCH.sub.3 CH                        5-SCH.sub.3                                                                             -- Q-1                                                                               C.sub.2 H.sub.5                                                                           O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        5-SCH.sub.3                                                                             -- Q-1                                                                               C.sub.2 H.sub.5                                                                           O     H    Cl    OCH.sub.3 CH                        5-SCH.sub.3                                                                             -- Q-1                                                                               C.sub.2 H.sub.5                                                                           O     H    CH.sub.3                                                                             OCH.sub.3 N                         5-SCH.sub.3                                                                             -- Q-1                                                                               C.sub.2 H.sub.5                                                                           O     H    OCH.sub.3                                                                            OCH.sub.3 N                         H        -- Q-1                                                                               CH.sub.3   O     CH.sub. 3                                                                           CH.sub.3                                                                             CH.sub.3  CH                        H        -- Q-1                                                                               CH.sub.3   O     CH.sub.3                                                                            CH.sub.3                                                                             OCH.sub.3 CH                        H        -- Q-1                                                                               CH.sub.3   O     CH.sub.3                                                                            OCH.sub.3                                                                            OCH.sub.3 CH                        H        -- Q-1                                                                               CH.sub.3   O     CH.sub.3                                                                            Cl    OCH.sub.3 CH                        H        -- Q-1                                                                               CH.sub.3   O     CH.sub.3                                                                            CH.sub.3                                                                             OCH.sub.3 N                         H        -- Q-1                                                                               CH.sub.3   O     CH.sub.3                                                                            OCH.sub.3                                                                            OCH.sub.3 N                         H        -- Q-1                                                                               CH.sub.3   S     H    CH.sub.3                                                                             CH.sub.3  CH                        H        -- Q-1                                                                               CH.sub.3   S     H    CH.sub.3                                                                             OCH.sub.3 CH                        H        -- Q-1                                                                               CH.sub.3   S     H    OCH.sub.3                                                                            OCH.sub.3 CH                        H        -- Q-1                                                                               CH.sub.3   S     H    Cl    OCH.sub.3 CH                        H        -- Q-1                                                                               CH.sub.3   S     H    CH.sub.3                                                                             OCH.sub.3 N                         H        -- Q-1                                                                               CH.sub.3   S     H    OCH.sub.3                                                                            OCH.sub.3 N                         H        -- Q-1                                                                               CH.sub.3   O     H    H     OCH.sub.3 CH                        H        -- Q-1                                                                               CH.sub.3   O     H    H     OC.sub.2 H.sub.5                                                                         CH                        H        -- Q-1                                                                               CH.sub.3   O     H    H     OCF.sub.2 H                                                                              CH                        H        -- Q-1                                                                               CH.sub.3   O     H    CH.sub. 3                                                                            CF.sub.3  CH                        H        -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             SCH.sub.3 CH                        H        -- Q-1                                                                               CH.sub.3   O     H    Cl    OCH.sub.3 CH                        H        -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             CH.sub.2 OCH.sub.3                                                                       CH                        H        -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             OCH.sub.2 OCH.sub.3                                                                      CH                        H        -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             NHCH.sub.3                                                                               CH                        H        -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             N(CH.sub.3).sub.2                                                                        CH                        H        CH.sub.2                                                                          Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             CH.sub.3  CH                        H        CH.sub.2                                                                          Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             OCH.sub.3 CH                        H        CH.sub.2                                                                          Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        H        CH.sub.2                                                                          Q-1                                                                               CH.sub.3   O     H    Cl    OCH.sub.3 CH                        H        CH.sub.2                                                                          Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             OCH.sub.3 N                         H        CH.sub.2                                                                          Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 N                         H        O  Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             CH.sub.3  CH                        H        O  Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             OCH.sub.3 CH                        H        O  Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        H        O  Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             OCH.sub.3 N                         H        O  Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             CH.sub.3  CH                        H        O  Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             OCH.sub.3 CH                        H        O  Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        H        O  Q-1                                                                               CH.sub.3   O     H    Cl    OCH.sub.3 CH                        H        O  Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             OCH.sub.3 N                         H        O  Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 N                         H        -- Q-1                                                                               CH.sub.3   O     H    OC.sub.2 H.sub.5                                                                     NHCH.sub.3                                                                               CH                        H        -- Q-1                                                                               CH.sub.3   O     H    H     OCH.sub.3 CH                        H        -- Q-1                                                                               CH.sub.3   O     H    H     OC.sub.2 H.sub.5                                                                         CH                        H        -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             CF.sub.3  CH                        H        -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             SCH.sub.3 CH                        H        -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             CH.sub.2 OCH.sub.3                                                                       CH                        H        -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             NHCH.sub.3                                                                               CH                        H        -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             N(CH.sub.3).sub.2                                                                        CH                        H        -- Q-1                                                                               CH.sub.3   O     H    H     OCH.sub.3 N                         H        -- Q-1                                                                               CH.sub.3   O     H    H     OC.sub.2 H.sub.5                                                                         N                         H        -- Q-1                                                                               CH.sub.3   O     H    H     OCF.sub.2 H                                                                              N                         H        -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             CH.sub.2 OCH.sub.3                                                                       N                         H        -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             NHCH.sub.3                                                                               N                         H        -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             N(CH.sub.3).sub.2                                                                        N                         3-( -n-C.sub.3 H.sub.7)                                                                 -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             CH.sub.3  CH                        3-( -n-C.sub.3 H.sub.7)                                                                 -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        3-( -n-C.sub.3 H.sub.7)                                                                 -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            CH.sub.3  CH                        5-CH.sub.2 CH.sub.2 Cl                                                                  -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            CH.sub.3  CH                        5-CH.sub.2 CH.sub.2 Cl                                                                  -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        5-OCH.sub.2 CH.sub.2 CH.sub.3                                                           -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        5-OCH.sub.2 CH.sub.2 CH.sub.3                                                           -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            CH.sub.3  CH                        6-SO.sub.2 N(CH.sub.3).sub.2                                                            -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        6-SO.sub.2 N(CH.sub.3).sub.2                                                            -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            CH.sub.3  CH                        6-OCH.sub.2 CH.sub.2 CH.sub.3                                                           -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            CH.sub.3  CH                        6-OCH.sub.2 CH.sub.2 CH.sub.3                                                           -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        6-SCH.sub.2 CH.sub.2 CH.sub.3                                                           -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        6-SCH.sub.2 CH.sub.2 CH.sub.3                                                           -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            CH.sub.3  CH                        6-SOCH.sub.3                                                                            -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        6-SOCH.sub.3                                                                            -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            CH.sub.3  CH                        6-SO.sub.2 CH.sub.3                                                                     -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            CH.sub.3  CH                        6-SO.sub.2 CH.sub.3                                                                     -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        5-CN     -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        5-CN     -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            CH.sub.3  CH                        5-CO.sub.2 CH.sub.3                                                                     -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            CH.sub.3  CH                        5-CO.sub.2 CH.sub.3                                                                     -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        5-OCH.sub.2 CH.sub.2 Cl                                                                 -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        5-OCH.sub.2 CH.sub.2 Cl                                                                 -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            CH.sub.3  CH                        5-OCH.sub.2 CF.sub.3                                                                    -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            CH.sub.3  CH                        5-OCH.sub.2 CF.sub.3                                                                    -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        5-SCH.sub.2 CF.sub.3                                                                    -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            CH.sub.3  CH                        5-SCH.sub.2 CF.sub.3                                                                    -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        5-NH.sub.2                                                                              -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        5-NH.sub.2                                                                              -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            CH.sub.3  CH                        5-NHC.sub.2 H.sub.5                                                                     -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            CH.sub.3  CH                        5-NHC.sub.2 H.sub.5                                                                     -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        5-N(CH.sub.3).sub.2                                                                     -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        5-N(CH.sub.3).sub.2                                                                     -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            CH.sub.3  CH                        5-CH.sub.2 OCH.sub.3                                                                    -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            CH.sub.3  CH                        5-CH.sub.2 OCH.sub.3                                                                    -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        5-C.sub.2 H.sub.4 OCH.sub.3                                                             -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        5-C.sub.2 H.sub.4 OCH.sub.3                                                             -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            CH.sub.3  CH                        5-C.sub.2 H.sub.4 OC.sub.2 H.sub.5                                                      -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            CH.sub.3  CH                        5-C.sub.2 H.sub.4 OC.sub.2 H.sub.5                                                      -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        5-CH.sub.2 OC.sub.2 H.sub.4 Cl                                                          -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        5-CH.sub.2 OC.sub.2 H.sub.4 Cl                                                          -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            CH.sub.3  CH                        5-CH.sub.2 OCH.sub.2 CF.sub.3                                                           -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            CH.sub.3  CH                        5-CH.sub.2 OCH.sub.2 CF.sub.3                                                           -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        5-CH.sub.2 SCH.sub.3                                                                    -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        5-CH.sub.2 SCH.sub.3                                                                    -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            CH.sub.3  CH                        5-CH.sub.2 SC.sub.2 H.sub.4 Cl                                                          -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            CH.sub.3  CH                        5-CH.sub.2 SC.sub.2 H.sub.4 Cl                                                          -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        5-CH.sub.2 CN                                                                           -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        5-CH.sub.2 CN                                                                           -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            CH.sub.3  CH                        H        -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.2 CH.sub.2 CH.sub.2                                                    CH.sub.3  CH                        H        -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.2 CH.sub.2 Cl                                                                    CH                        H        -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.2 CH.sub.2 CH.sub.2                                                              CH                        H        -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            SCH.sub.2 CH.sub.2 Cl                                                                    CH                        H        -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            SCHF.sub.2                                                                               CH                        H        -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            SCH.sub.2 CH.sub.                                                                        CH                        H        -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            CH.sub.2 OCH.sub.3                                                                       CH                        H        -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            C.sub.2 H.sub.4 OC.sub.2                                                       H.sub.5   CH                        H        -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OC.sub.2 H.sub.4 OC.sub.2                                                      H.sub.5   CH                        H        -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.2 CH═CH.sub.2                                                                CH                        H        -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.2 C.tbd.CH                                                                       CH                        H        -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            CH.sub.2 SCH.sub.3                                                                       CH                        H        -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            C.sub.2 H.sub.4 SCH.sub.3                                                                CH                        H        -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            C.sub.2 H.sub.4 SC.sub.2                                                       H.sub.5   CH                        H        -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            CH.sub.2 SO.sub.2 CH.sub.3                                                               CH                        H        -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            C.sub.2 H.sub.4 SO.sub.2                                                       CH.sub.3  CH                        H        -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            C.sub.2 H.sub.4 SOCH.sub.3                                                               CH                        H        -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            CH.sub.2 CH.sub.2 CH.sub.2                                                               CH                        H        -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            CH.sub.2 C.tbd.CH                                                                        CH                        H        -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            N.sub.3   CH                        H        -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            CN        CH                        H        -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            COCH.sub.3                                                                               CH                        H        -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            C(CH.sub.3)(OCH.sub.3).sub.2                                                             CH                        H        -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            2-methyldi-                                                                              CH                                                                   oxolan-2-yl                         H        -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            N(OCH.sub.3)CH.sub.3                                                                     CH                        H        -- Q-1                                                                               CH.sub.3   O     H    OC.sub.2 H.sub.5                                                                     NHCH.sub.3                                                                               N  204-208                H        -- Q-2                                                                               CH.sub.3   O     H    CH.sub.3                                                                             CH.sub.3  CH                        H        -- Q-2                                                                               CH.sub.3   O     H    CH.sub.3                                                                             OCH.sub.3 CH                        H        -- Q-2                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 CH 214-222                H        -- Q-2                                                                               CH.sub.3   O     H    Cl    OCH.sub.3 CH                        H        -- Q-2                                                                               CH.sub.3   O     H    CH.sub.3                                                                             OCH.sub.3 N                         H        -- Q-2                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 N                         H        -- Q-2                                                                               C.sub.2 H.sub.5                                                                           O     H    CH.sub.3                                                                             CH.sub.3  CH                        H        -- Q-2                                                                               C.sub.2 H.sub.5                                                                           O     H    CH.sub.3                                                                             OCH.sub.3 CH                        H        -- Q-2                                                                               C.sub.2 H.sub.5                                                                           O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        H        -- Q-2                                                                               C.sub.2 H.sub.5                                                                           O     H    Cl    OCH.sub.3 CH                        H        -- Q-2                                                                               C.sub.2 H.sub.5                                                                           O     H    CH.sub.3                                                                             OCH.sub.3 N                         H        -- Q-2                                                                               C.sub.2 H.sub.5                                                                           O     H    OCH.sub.3                                                                            OCH.sub.3 N                         H        -- Q-2                                                                               CH(CH.sub.3).sub.2                                                                        O     H    CH.sub.3                                                                             CH.sub.3  CH                        H        -- Q-2                                                                               CH(CH.sub.3).sub.2                                                                        O     H    CH.sub.3                                                                             OCH.sub.3 CH                        H        -- Q-2                                                                               CH(CH.sub.3).sub.2                                                                        O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        H        -- Q-2                                                                               CH(CH.sub.3).sub.2                                                                        O     H    Cl    OCH.sub.3 CH                        H        -- Q-2                                                                               CH(CH.sub.3).sub.2                                                                        O     H    CH.sub.3                                                                             OCH.sub.3 N                         H        -- Q-2                                                                               CH(CH.sub.3).sub.2                                                                        O     H    OCH.sub.3                                                                            OCH.sub.3 N                         H        -- Q-2                                                                               (CH.sub.2).sub.2 CH.sub.3                                                                 O     H    CH.sub. 3                                                                            CH.sub.3  CH                        H        -- Q-2                                                                               (CH.sub.2).sub.2 CH.sub.3                                                                 O     H    CH.sub.3                                                                             OCH.sub.3 CH                        H        -- Q-2                                                                               (CH.sub.2).sub.2 CH.sub.3                                                                 O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        H        -- Q-2                                                                               (CH.sub.2).sub.2 CH.sub.3                                                                 O     H    Cl    OCH.sub.3 CH                        H        -- Q-2                                                                               (CH.sub.2).sub.2 CH.sub.3                                                                 O     H    CH.sub.3                                                                             OCH.sub.3 N                         H        -- Q-2                                                                               (CH.sub.2).sub.2 CH.sub.3                                                                 O     H    OCH.sub.3                                                                            OCH.sub.3 N                         H        -- Q-1                                                                               CH.sub.2 C.tbd.CH                                                                         O     H    CH.sub.3                                                                             CH.sub.3  CH                        H        -- Q-1                                                                               CH.sub.2 C.tbd.CH                                                                         O     H    CH.sub.3                                                                             OCH.sub.3 CH                        H        -- Q-1                                                                               CH.sub.2 C.tbd.CH                                                                         O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        H        -- Q-1                                                                               CH.sub.2 C.tbd.CH                                                                         O     H    Cl    OCH.sub.3 CH                        H        -- Q-1                                                                               CH.sub.2 C.tbd.CH                                                                         O     H    CH.sub.3                                                                             OCH.sub.3 N                         H        -- Q-1                                                                               CH.sub.2 C.tbd.CH                                                                         O     H    OCH.sub.3                                                                            OCH.sub.3 N                         H        -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCF.sub.2 H                                                                              CH 160-165                H        -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             OCF.sub.2 H                                                                              CH 195-198                5-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCF.sub.2 H                                                                              CH 168-172                5-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             OCF.sub.2 H                                                                              CH 90-93                  H        -- Q-2                                                                               CH.sub.2 OCH.sub.3                                                                        O     H    CH.sub.3                                                                             CH.sub.3  CH                        H        -- Q-2                                                                               CH.sub.2 OCH.sub.3                                                                        O     H    CH.sub.3                                                                             OCH.sub.3 CH                        H        -- Q-2                                                                               CH.sub.2 OCH.sub.3                                                                        O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        H        -- Q-2                                                                               CH.sub.2 OCH.sub.3                                                                        O     H    Cl    OCH.sub.3 CH                        H        -- Q-2                                                                               CH.sub.2 OCH.sub.3                                                                        O     H    CH.sub.3                                                                             OCH.sub.3 N                         H        -- Q-2                                                                               CH.sub.2 OCH.sub.3                                                                        O     H    OCH.sub.3                                                                            OCH.sub.3 N                         5-OCF.sub.2 H                                                                           -- Q-2                                                                               CH.sub.3   O     H    CH.sub.3                                                                             CH.sub.3  CH                        5-OCF.sub.2 H                                                                           -- Q-2                                                                               CH.sub.3   O     H    CH.sub.3                                                                             OCH.sub.3 CH                        5-OCF.sub.2 H                                                                           -- Q-2                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        5-OCF.sub.2 H                                                                           -- Q-2                                                                               CH.sub.3   O     H    Cl    OCH.sub.3 CH                        5-OCF.sub.2 H                                                                           -- Q-2                                                                               CH.sub.3   O     H    CH.sub.3                                                                             OCH.sub.3 N                         5-OCF.sub.2 H                                                                           -- Q-2                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 N                         5-OCH.sub.3                                                                             -- Q-2                                                                               CH.sub.3   O     H    CH.sub.3                                                                             CH.sub.3  CH                        5-OCH.sub.3                                                                             -- Q-2                                                                               CH.sub.3   O     H    CH.sub.3                                                                             OCH.sub.3 CH                        5-OCH.sub.3                                                                             -- Q-2                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        5-OCH.sub.3                                                                             -- Q-2                                                                               CH.sub.3   O     H    Cl    OCH.sub.3 CH                        5-OCH.sub.3                                                                             -- Q-2                                                                               CH.sub.3   O     H    CH.sub.3                                                                             OCH.sub.3 N                         5-OCH.sub.3                                                                             -- Q-2                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 N                         6-Cl     -- Q-2                                                                               CH.sub.3   O     H    CH.sub.3                                                                             CH.sub.3  CH                        6-Cl     -- Q-2                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            CH.sub.3  CH                        6-Cl     -- Q-2                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        6-OCH.sub.3                                                                             -- Q-2                                                                               CH.sub.3   O     H    CH.sub.3                                                                             CH.sub.3  CH                        6-OCH.sub.3                                                                             -- Q-2                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            CH.sub.3  CH                        6-OCH.sub.3                                                                             -- Q-2                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        5-SCH.sub.3                                                                             -- Q-2                                                                               CH.sub.3   O     H    CH.sub.3                                                                             CH.sub.3  CH                        5-SCH.sub. 3                                                                            -- Q-2                                                                               CH.sub.3   O     H    CH.sub.3                                                                             OCH.sub.3 CH                        5-SCH.sub.3                                                                             -- Q-2                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        5-SCH.sub.3                                                                             -- Q-2                                                                               CH.sub.3   O     H    Cl    OCH.sub.3 CH                        5-SCH.sub.3                                                                             -- Q-2                                                                               CH.sub.3   O     H    CH.sub.3                                                                             OCH.sub.3 N                         5-SCH.sub.3                                                                             -- Q-2                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 N                         5-SCH.sub.3                                                                             -- Q-2                                                                               C.sub.2 H.sub.5                                                                           O     H    CH.sub.3                                                                             CH.sub.3  CH                        5-SCH.sub.3                                                                             -- Q-2                                                                               C.sub.2 H.sub.5                                                                           O     H    CH.sub.3                                                                             OCH.sub.3 CH                        5-SCH.sub.3                                                                             -- Q-2                                                                               C.sub.2 H.sub.5                                                                           O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        5-SCH.sub.3                                                                             -- Q-2                                                                               C.sub.2 H.sub.5                                                                           O     H    Cl    OCH.sub.3 CH                        5-SCH.sub.3                                                                             -- Q-2                                                                               C.sub.2 H.sub.5                                                                           O     H    CH.sub.3                                                                             OCH.sub.3 N                         5-SCH.sub.3                                                                             -- Q-2                                                                               C.sub.2 H.sub.5                                                                           O     H    OCH.sub.3                                                                            OCH.sub.3 N                         H        -- Q-2                                                                               CH.sub.3   O     CH.sub.3                                                                            CH.sub.3                                                                             CH.sub.3  CH                        H        -- Q-2                                                                               CH.sub.3   O     CH.sub.3                                                                            CH.sub.3                                                                             OCH.sub.3 CH                        H        -- Q-2                                                                               CH.sub.3   O     CH.sub.3                                                                            OCH.sub.3                                                                            OCH.sub.3 CH                        H        -- Q-2                                                                               CH.sub.3   O     CH.sub.3                                                                            Cl    OCH.sub.3 CH                        H        -- Q-2                                                                               CH.sub.3   O     CH.sub.3                                                                            CH.sub.3                                                                             OCH.sub.3 N                         H        -- Q-2                                                                               CH.sub.3   O     CH.sub.3                                                                            OCH.sub.3                                                                            OCH.sub.3 N                         H        -- Q-2                                                                               CH.sub.3   S     H    CH.sub.3                                                                             CH.sub.3  CH                        H        -- Q-2                                                                               CH.sub.3   S     H    CH.sub.3                                                                             OCH.sub.3 CH                        H        -- Q-2                                                                               CH.sub.3   S     H    OCH.sub.3                                                                            OCH.sub.3 CH                        H        -- Q-2                                                                               CH.sub.3   S     H    Cl    OCH.sub.3 CH                        H        -- Q-2                                                                               CH.sub.3   S     H    CH.sub.3                                                                             OCH.sub.3 N                         H        -- Q-2                                                                               CH.sub.3   S     H    OCH.sub.3                                                                            OCH.sub.3 N                         H        -- Q-2                                                                               CH.sub.3   O     H    OC.sub.2 H.sub.5                                                                     NHCH.sub.3                                                                               N                         H        -- Q-2                                                                               CH.sub.3   O     H    H     OCH.sub.3 CH                        H        -- Q-2                                                                               CH.sub.3   O     H    H     OC.sub.2 H.sub.5                                                                         CH                        H        -- Q-2                                                                               CH.sub.3   O     H    H     OCF.sub.2 H                                                                              CH                        H        -- Q-2                                                                               CH.sub.3   O     H    CH.sub.3                                                                             SCF.sub.2 H                                                                              CH                        H        -- Q-2                                                                               CH.sub.3   O     H    Cl    OCH.sub.3 CH                        H        -- Q-2                                                                               CH.sub.3   O     H    CH.sub.3                                                                             CH.sub.2 OCH.sub.3                                                                       CH                        H        -- Q-2                                                                               CH.sub.3   O     H    CH.sub.3                                                                             OCH.sub.2 OCH.sub.3                                                                      CH                        H        -- Q-2                                                                               CH.sub.3   O     H    OC.sub.2 H.sub.5                                                                     NHCH.sub.3                                                                               N                         H        -- Q-2                                                                               CH.sub.3   O     H    H     OCH.sub.3 CH                        H        -- Q-2                                                                               CH.sub.3   O     H    H     OC.sub.2 H.sub.5                                                                         CH                        H        -- Q-2                                                                               CH.sub.3   O     H    CH.sub.3                                                                             CF.sub.3  CH                        H        -- Q-2                                                                               CH.sub.3   O     H    CH.sub.3                                                                             SCH.sub.3 CH                        H        -- Q-2                                                                               CH.sub.3   O     H    Cl    OCH.sub.3 CH                        H        -- Q-2                                                                               CH.sub.3   O     H    CH.sub.3                                                                             CH.sub.2 OCH.sub.3                                                                       CH                        H        -- Q-2                                                                               CH.sub.3   O     H    CH.sub.3                                                                             OCH.sub.2 OCH.sub.3                                                                      CH                        H        -- Q-2                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OC.sub.2 H.sub.5                                                                         N                         H        -- Q-2                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH(CH.sub.3).sub.2                                                                      N                         H        -- Q-2                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.2 CF.sub.3                                                                       N                         H        -- Q-2                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            CF.sub.3  N                         H        -- Q-2                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            O(CH.sub.2).sub.2 OCH.sub.3                                                              N                         H        -- Q-2                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            C.tbd.C--CH.sub.3                                                                        N                         H        -- Q-2                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            N(CH.sub.3)OCH.sub.3                                                                     N                         H        -- Q-2                                                                               C.sub.2 H.sub.5                                                                           S     H    CH.sub.3                                                                             CH.sub.3  CH                        H        -- Q-2                                                                               C.sub.2 H.sub.5                                                                           S     H    CH.sub.3                                                                             OCH.sub.3 CH                        H        -- Q-2                                                                               C.sub.2 H.sub.5                                                                           S     H    OCH.sub.3                                                                            OCH.sub.3 CH                        H        -- Q-2                                                                               C.sub.2 H.sub.5                                                                           S     H    Cl    OCH.sub.3 CH                        H        -- Q-2                                                                               C.sub.2 H.sub.5                                                                           S     H    CH.sub.3                                                                             OCH.sub.3 N                         6-CH.sub.3                                                                              -- Q-2                                                                               CH.sub.3   O     H    CH.sub.3                                                                             CH.sub.3  CH                        6-CH.sub.3                                                                              -- Q-2                                                                               CH.sub.3   O     H    CH.sub.3                                                                             OCH.sub.3 CH                        6-CH.sub.3                                                                              -- Q-2                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 CH                        6-CH.sub.3                                                                              -- Q-2                                                                               CH.sub.3   O     H    Cl    OCH.sub.3 CH                        6-CH.sub.3                                                                              -- Q-2                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            CH.sub.3  N                         6-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H    Br    OCH.sub. 3                                                                               CH 196-198 dec.           6-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     CH.sub.3                                                                            CH.sub.3                                                                             OCH.sub.3 CH 199-200 dec.           6-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     CH.sub.3                                                                            CH.sub.3                                                                             OCH.sub.3 N  49-56                  6-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H    H     CH.sub.3  CH 196-199 dec.           6-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H    H     OCH.sub.3 CH 163-166 dec.           6-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H    C.sub.2 H.sub.5                                                                      OCH.sub.3 CH 160-164                6-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H    C.sub.2 H.sub.5                                                                      OCH.sub.3 N  179-180 dec.           6-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     CH.sub.3                                                                            OCH.sub.3                                                                            OCH.sub.3 N                         6-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H    cyclopropyl                                                                          OCH.sub.3 N  222-223 dec.           6-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             OC.sub.2 H.sub.5                                                                         CH                        6-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            CH.sub.2 OC.sub.2 H.sub.5                                                                CH 189-190 dec.           6-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.2 CF.sub.3                                                                       CH 140-145 dec.           6-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OC.sub.2 H.sub.5                                                                         N  159-164 dec.           6-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCF.sub.2 H                                                                              CH 168-172                6-CH.sub.3                                                                              -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             OCF.sub.2 H                                                                              CH 90-93                  H        -- Q-1                                                                               CH.sub.3   NH    H    OCH.sub.3                                                                            OCH.sub.3 CH                        H        -- Q-1                                                                               CH.sub.3   NOCH.sub.3                                                                           H    CH.sub.3                                                                             OCH.sub.3 CH                        H        -- Q-2                                                                               CH.sub.3   NOH   H    CH.sub.3                                                                             OCH.sub.3 CH                        H        -- Q-2                                                                               C.sub.2 H.sub.5                                                                           NNHCH.sub.3                                                                          H    OCH.sub.3                                                                            OCH.sub.3 CH                        3-Cl     -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 N  199-202                3-Cl     -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             OCH.sub.3 N  206-209                3-Cl     -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 CH 143-162                3-Cl     -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             OCH.sub.3 CH 226-227                3-Cl     -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             CH.sub.3  CH 221-223 dec.           3-Cl     -- Q-1                                                                               CH.sub.3   O     H    Cl    OCH.sub.3 CH 189-192                5-F      -- Q-1                                                                               CH.sub. 3  O     H    OCH.sub.3                                                                            OCH.sub.3 CH 209-212                5-F      -- Q-1                                                                               CH.sub.3   O     H    Cl    OCH.sub.3 CH 199-201                5-F      -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 N  187-190                5-F      -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             OCH.sub.3 N  196-201                5-F      -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             CH.sub.3  CH 233-236                5-F      -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             OCH.sub.3 CH 164-168                H        -- Q-1                                                                               C.sub.2 H.sub.5                                                                           O     H    OCH.sub.3                                                                            OCF.sub.2 H                                                                              CH 87-94                  6-Cl     -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCF.sub.2 H                                                                              CH 93-95                  6-Cl     -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             OCF.sub.2 H                                                                              CH 118-120                6-OCH.sub.3                                                                             -- Q-1                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 N  194-197                6-OCH.sub.3                                                                             -- Q-1                                                                               CH.sub.3   O     H    CH.sub.3                                                                             OCH.sub.3 N  172-182                6-OCH.sub.3                                                                             -- Q-1                                                                               CH.sub.3   O     H    Cl    OCH.sub.3 CH 206-209                6-Cl     -- Q-2                                                                               CH.sub.3   O     H    Cl    OCH.sub.3 CH                        6-Cl     -- Q-2                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 N                         6-Cl     -- Q-2                                                                               CH.sub.3   O     H    CH.sub.3                                                                             OCH.sub.3 N                         6-OCH.sub.3                                                                             -- Q-2                                                                               CH.sub.3   O     H    Cl    OCH.sub.3 CH                        6-OCH.sub.3                                                                             -- Q-2                                                                               CH.sub.3   O     H    OCH.sub.3                                                                            OCH.sub.3 N                         6-OCH.sub.3                                                                             -- Q-2                                                                               CH.sub.3   O     H    CH.sub.3                                                                             OCH.sub.3 N                         __________________________________________________________________________

                                      TABLE Ia                                     __________________________________________________________________________     General Structure 1                                                            R.sub.1                                                                               E   Q    R.sub.4 W  R  X       Y        Z  m.p. (°C.)            __________________________________________________________________________     H      --  Q-3  H       O  H  CH.sub.3                                                                               CH.sub.3 CH 214 dec.                     H      --  Q-3  H       O  H  CH.sub.3                                                                               OCH.sub.3                                                                               CH 204-205                      H      --  Q-3  H       O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               CH 187-188                      H      --  Q-3  H       O  H  Cl      OCH.sub.3                                                                               CH 195-196                      H      --  Q-3  H       O  H  CH.sub.3                                                                               OCH.sub.3                                                                               N  199-202                      H      --  Q-3  H       O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               N  191-192                      H      --  Q-3  CH.sub.3                                                                               O  H  CH.sub.3                                                                               CH.sub.3 CH                              H      --  Q-3  CH.sub.3                                                                               O  H  OC.sub.2 H.sub.5                                                                       NHCH.sub.3                                                                              N  167-200 dec.                 H      --  Q-3  CH.sub.3                                                                               O  H  CH.sub.3                                                                               OCH.sub.3                                                                               CH 221-223                      H      --  Q-3  CH.sub.3                                                                               O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               CH 213-216                      H      --  Q-3  CH.sub.3                                                                               O  H  Cl      OCH.sub.3                                                                               CH 208-210                      H      --  Q-3  CH.sub.3                                                                               O  H  CH.sub.3                                                                               OCH.sub.3                                                                               N  207-209                      H      --  Q-3  CH.sub.3                                                                               O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               N  209-216                      H      --  Q-3  C.sub.2 H.sub.5                                                                        O  H  CH.sub.3                                                                               CH.sub.3 CH 217-220                      H      --  Q-3  C.sub.2 H.sub.5                                                                        O  H  CH.sub.3                                                                               OCH.sub.3                                                                               CH 224-228                      H      --  Q-3  C.sub.2 H.sub.5                                                                        O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               CH 193-196                      H      --  Q-3  C.sub.2 H.sub.5                                                                        O  H  Cl      OCH.sub.3                                                                               CH 200-204                      H      --  Q-3  C.sub.2 H.sub.5                                                                        O  H  CH.sub.3                                                                               OCH.sub.3                                                                               N  174-179                      H      --  Q-3  C.sub.2 H.sub.5                                                                        O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               N  194-197                      H      --  Q-3  CH(CH.sub.3).sub.2                                                                     O  H  CH.sub.3                                                                               CH.sub.3 CH                              H      --  Q-3  CH(CH.sub.3).sub.2                                                                     O  H  CH.sub.3                                                                               OCH.sub.3                                                                               CH                              H      --  Q-3  CH(CH.sub.3).sub.2                                                                     O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               CH                              H      --  Q-3  CH(CH.sub.3).sub.2                                                                     O  H  Cl      OCH.sub.3                                                                               CH                              H      --  Q-3  CH(CH.sub.3).sub.2                                                                     O  H  CH.sub.3                                                                               OCH.sub.3                                                                               N                               H      --  Q-3  CH(CH.sub.3).sub.2                                                                     O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               N                               H      --  Q-3  cyclopropyl                                                                            O  H  CH.sub.3                                                                               CH.sub.3 CH                              H      --  Q-3  cyclopropyl                                                                            O  H  CH.sub.3                                                                               OCH.sub.3                                                                               CH                              H      --  Q-3  cyclopropyl                                                                            O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               CH                              H      --  Q-3  cyclopropyl                                                                            O  H  Cl      OCH.sub.3                                                                               CH                              H      --  Q-3  cyclopropyl                                                                            O  H  CH.sub.3                                                                               OCH.sub.3                                                                               N                               H      --  Q-3  cyclopropyl                                                                            O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               N                               H      --  Q-3  CH.sub.2 Cl                                                                            O  H  CH.sub.3                                                                               CH.sub.3 CH                              H      --  Q-3  CH.sub.2 Cl                                                                            O  H  CH.sub.3                                                                               OCH.sub.3                                                                               CH                              H      --  Q-3  CH.sub.2 Cl                                                                            O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               CH                              H      --  Q-3  CH.sub.2 Cl                                                                            O  H  Cl      OCH.sub.3                                                                               CH                              H      --  Q-3  CH.sub.2 Cl                                                                            O  H  CH.sub.3                                                                               OCH.sub.3                                                                               N                               H      --  Q-3  CH.sub.2 Cl                                                                            O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               N                               H      --  Q-3  CF.sub.3                                                                               O  H  CH.sub.3                                                                               CH.sub.3 CH                              H      --  Q-3  CF.sub.3                                                                               O  H  CH.sub.3                                                                               OCH.sub.3                                                                               CH                              H      --  Q-3  CF.sub.3                                                                               O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               CH                              H      --  Q-3  CF.sub.3                                                                               O  H  Cl      OCH.sub.3                                                                               CH                              H      --  Q-3  CF.sub.3                                                                               O  H  CH.sub.3                                                                               OCH.sub.3                                                                               N                               H      --  Q-3  CF.sub.3                                                                               O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               N                               H      --  Q-3  OCH.sub.3                                                                              O  H  CH.sub.3                                                                               CH.sub.3 CH 195-196                      H      --  Q-3  OCH.sub.3                                                                              O  H  CH.sub.3                                                                               OCH.sub.3                                                                               CH 175-177                      H      --  Q-3  OCH.sub.3                                                                              O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               CH 188-189                      H      --  Q-3  OCH.sub.3                                                                              O  H  Cl      OCH.sub.3                                                                               CH 200-201                      H      --  Q-3  OCH.sub.3                                                                              O  H  CH.sub.3                                                                               OCH.sub.3                                                                               N  189-190                      H      --  Q-3  OCH.sub.3                                                                              O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               N  180                          H      --  Q-3  OC.sub.2 H.sub.5                                                                       O  H  CH.sub.3                                                                               CH.sub.3 CH 199-200 dec.                 H      --  Q-3  OC.sub.2 H.sub.5                                                                       O  H  CH.sub.3                                                                               OCH.sub.3                                                                               CH 197-198 dec.                 H      --  Q-3  OC.sub.2 H.sub.5                                                                       O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               CH 200-201 dec.                 H      --  Q-3  OC.sub.2 H.sub.5                                                                       O  H  Cl      OCH.sub.3                                                                               CH 184-185 dec.                 H      --  Q-3  OC.sub.2 H.sub.5                                                                       O  H  CH.sub.3                                                                               OCH.sub.3                                                                               N  170-173 dec.                 H      --  Q-3  OC.sub.2 H.sub.5                                                                       O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               N  178-180 dec.                 H      --  Q-3  SCH.sub.3                                                                              O  H  CH.sub.3                                                                               CH.sub.3 CH                              H      --  Q-3  SCH.sub.3                                                                              O  H  CH.sub.3                                                                               OCH.sub.3                                                                               CH                              H      --  Q-3  SCH.sub.3                                                                              O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               CH                              H      --  Q-3  SCH.sub.3                                                                              O  H  Cl      OCH.sub.3                                                                               CH                              H      --  Q-3  SCH.sub.3                                                                              O  H  CH.sub.3                                                                               OCH.sub.3                                                                               N                               H      --  Q-3  SCH.sub.3                                                                              O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               N                               H      --  Q-3  N(CH.sub.3).sub.2                                                                      O  H  CH.sub.3                                                                               CH.sub.3 CH                              H      --  Q-3  N(CH.sub.3).sub.2                                                                      O  H  CH.sub.3                                                                               OCH.sub.3                                                                               CH                              H      --  Q-3  N(CH.sub.3).sub.2                                                                      O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               CH                              H      --  Q-3  N(CH.sub.3 ).sub.2                                                                     O  H  Cl      OCH.sub.3                                                                               CH                              H      --  Q-3  N(CH.sub.3).sub.2                                                                      O  H  CH.sub.3                                                                               OCH.sub.3                                                                               N                               H      --  Q-3  N(CH.sub.3).sub.2                                                                      O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               N                               5-CH.sub.3                                                                            --  Q-3  CH.sub.3                                                                               O  H  CH.sub.3                                                                               CH.sub.3 CH                              5-CH.sub.3                                                                            --  Q-3  CH.sub.3                                                                               O  H  CH.sub.3                                                                               OCH.sub.3                                                                               CH                              5-CH.sub.3                                                                            --  Q-3  CH.sub.3                                                                               O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               CH 177-186                      5-CH.sub.3                                                                            --  Q-3  CH.sub.3                                                                               O  H  Cl      OCH.sub.3                                                                               CH 207-208                      5-CH.sub.3                                                                            --  Q-3  CH.sub.3                                                                               O  H  CH.sub.3                                                                               OCH.sub.3                                                                               N  200-202                      5-CH.sub.3                                                                            --  Q-3  CH.sub.3                                                                               O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               N                               5-Cl   --  Q-3  CH.sub.3                                                                               O  H  CH.sub.3                                                                               CH.sub.3 CH 227-230                      5-Cl   --  Q-3  CH.sub.3                                                                               O  H  CH.sub.3                                                                               OCH.sub.3                                                                               CH 173-180                      5-Cl   --  Q-3  CH.sub.3                                                                               O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               CH 216-220                      5-Cl   --  Q-3  CH.sub.3                                                                               O  H  Cl      OCH.sub.3                                                                               CH 227-230                      5-Cl   --  Q-3  CH.sub.3                                                                               O  H  CH.sub.3                                                                               OCH.sub.3                                                                               N  188- 195                     5-Cl   --  Q-3  CH.sub.3                                                                               O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               N  192-194                      5-Cl   --  Q-3  CH.sub.3                                                                               O  H  OC.sub.2 H.sub.5                                                                       NHCH.sub.3                                                                              N  181-185                      5-Br   --  Q-3  CH.sub.3                                                                               O  H  CH.sub.3                                                                               CH.sub.3 CH                              5-Br   --  Q-3  CH.sub.3                                                                               O  H  CH.sub.3                                                                               OCH.sub.3                                                                               CH                              5-Br   --  Q-3  CH.sub.3                                                                               O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               CH                              5-Br   --  Q-3  CH.sub.3                                                                               O  H  Cl      OCH.sub.3                                                                               CH                              5-Br   --  Q-3  CH.sub.3                                                                               O  H  CH.sub.3                                                                               OCH.sub.3                                                                               N                               5-Br   --  Q-3  CH.sub.3                                                                               O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               H                               5-OCF.sub.2 H                                                                         --  Q-3  CH.sub.3                                                                               O  H  CH.sub.3                                                                               CH.sub.3 CH                              5-OCF.sub.2 H                                                                         --  Q-3  CH.sub.3                                                                               O  H  CH.sub.3                                                                               OCH.sub.3                                                                               CH                              5-OCF.sub.2 H                                                                         --  Q-3  CH.sub.3                                                                               O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               CH                              5-OCF.sub.2 H                                                                         --  Q-3  CH.sub.3                                                                               O  H  Cl      OCH.sub.3                                                                               CH                              5-OCF.sub.2 H                                                                         --  Q-3  CH.sub.3                                                                               O  H  CH.sub.3                                                                               OCH.sub.3                                                                               N                               5-OCF.sub.2 H                                                                         --  Q-3  CH.sub.3                                                                               O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               N                               5-OCH.sub. 3                                                                          --  Q-3  CH.sub.3                                                                               O  H  CH.sub.3                                                                               CH.sub.3 CH                              5-OCH.sub.3                                                                           --  Q-3  CH.sub.3                                                                               O  H  CH.sub.3                                                                               OCH.sub.3                                                                               CH                              5-OCH.sub.3                                                                           --  Q-3  CH.sub.3                                                                               O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               CH                              5-OCH.sub.3                                                                           --  Q-3  CH.sub.3                                                                               O  H  Cl      OCH.sub.3                                                                               CH                              5-OCH.sub.3                                                                           --  Q-3  CH.sub.3                                                                               O  H  CH.sub.3                                                                               OCH.sub.3                                                                               N                               5-OCH.sub.3                                                                           --  Q-3  CH.sub.3                                                                               O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               N                               5-CF.sub.3                                                                            --  Q-3  CH.sub.3                                                                               O  H  CH.sub.3                                                                               CH.sub.3 CH                              5-CF.sub.3                                                                            --  Q-3  CH.sub.3                                                                               O  H  CH.sub.3                                                                               OCH.sub.3                                                                               CH                              5-CF.sub.3                                                                            --  Q-3  CH.sub.3                                                                               O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               CH                              5-CF.sub.3                                                                            --  Q-3  CH.sub.3                                                                               O  H  Cl      OCH.sub.3                                                                               CH                              5-CF.sub.3                                                                            --  Q-3  CH.sub.3                                                                               O  H  CH.sub.3                                                                               OCH.sub.3                                                                               N                               5-CF.sub.3                                                                            --  Q-3  CH.sub.3                                                                               O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               N                               5-SCH.sub.3                                                                           --  Q-3  CH.sub.3                                                                               O  H  CH.sub.3                                                                               CH.sub.3 CH                              5-SCH.sub.3                                                                           --  Q-3  CH.sub.3                                                                               O  H  CH.sub.3                                                                               OCH.sub.3                                                                               CH                              5-SCH.sub.3                                                                           --  Q-3  CH.sub.3                                                                               O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               CH                              5-SCH.sub.3                                                                           --  Q-3  CH.sub.3                                                                               O  H  Cl      OCH.sub.3                                                                               CH                              5-SCH.sub.3                                                                           --  Q-3  CH.sub.3                                                                               O  H  CH.sub.3                                                                               OCH.sub.3                                                                               N                               5-SCH.sub.3                                                                           --  Q-3  CH.sub.3                                                                               O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               N                               5-CH.sub.2 OCH.sub.3                                                                  --  Q-3  CH.sub.3                                                                               O  H  CH.sub.3                                                                               CH.sub.3 CH                              5-CH.sub.2 OCH.sub.3                                                                  --  Q-3  CH.sub.3                                                                               O  H  CH.sub.3                                                                               OCH.sub.3                                                                               CH                              5-CH.sub.2 OCH.sub.3                                                                  --  Q-3  CH.sub.3                                                                               O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               CH                              5-CH.sub.2 OCH.sub.3                                                                  --  Q-3  CH.sub.3                                                                               O  H  Cl      OCH.sub.3                                                                               CH                              5-CH.sub.2 OCH.sub.3                                                                  --  Q-3  CH.sub.3                                                                               O  H  CH.sub.3                                                                               OCH.sub.3                                                                               N                               5-CH.sub.2 OCH.sub.3                                                                  --  Q-3  CH.sub.3                                                                               O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               N                               5-OCH.sub.2 CH.sub.3                                                                  --  Q-3  CH.sub.3                                                                               O  H  CH.sub.3                                                                               CH.sub.3 CH                              5-OCH.sub.2 CH.sub.3                                                                  --  Q-3  CH.sub.3                                                                               O  H  CH.sub.3                                                                               OCH.sub.3                                                                               CH                              5-OCH.sub.2 CH.sub.3                                                                  --  Q-3  CH.sub.3                                                                               O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               CH                              5-OCH.sub.2 CH.sub.3                                                                  --  Q-3  CH.sub.3                                                                               O  H  Cl      OCH.sub.3                                                                               CH                              5-OCH.sub.2 CH.sub.3                                                                  --  Q-3  CH.sub.3                                                                               O  H  CH.sub.3                                                                               OCH.sub.3                                                                               N                               5-OCH.sub.2 CH.sub.3                                                                  --  Q-3  CH.sub.3                                                                               O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               N                               H      --  Q-3  CH.sub.2 OCH.sub.3                                                                     O  H  CH.sub.3                                                                               CH.sub.3 CH                              H      --  Q-3  CH.sub.2 OCH.sub.3                                                                     O  H  CH.sub.3                                                                               OCH.sub.3                                                                               CH                              H      --  Q-3  CH.sub.2 OCH.sub.3                                                                     O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               CH                              H      --  Q-3  CH.sub.2 OCH.sub.3                                                                     O  H  Cl      OCH.sub.3                                                                               CH                              H      --  Q-3  CH.sub.3 OCH.sub.3                                                                     O  H  OCH.sub.3                                                                              CH.sub.3 N                               H      --  Q-3  CH.sub.3 OCH.sub.3                                                                     O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               N                               H      --  Q-3  CH.sub.3                                                                               O  H  cyclopropyl                                                                            OCH.sub.3                                                                               CH                              H      --  Q-3  CH.sub.3                                                                               O  H  OCH.sub.3                                                                              N.sub.3  CH                              H      --  Q-3  CH.sub.3                                                                               O  H  OCH.sub.3                                                                              CN       CH                              H      --  Q-3  CH.sub.3                                                                               O  H  OCH.sub.3                                                                              C(O)CH.sub.3                                                                            CH                              H      --  Q-3  CH.sub.3                                                                               O  H  OCH.sub.3                                                                              CH(OCH.sub.3).sub.2                                                                     CH                              H      --  Q-3  CH.sub.3                                                                               O  H  OCH.sub.3                                                                              1,3-dioxo-                                                                              CH                                                                    lan-2-yl                                 H      --  Q-3  CH.sub.3                                                                               O  H  OCH.sub.3                                                                              1,3-diox-                                                                               CH                                                                    an-2-yl                                  H      CH.sub.2                                                                           Q-3  CH.sub.3                                                                               O  H  CH.sub.3                                                                               CH.sub.3 CH                              H      CH.sub.2                                                                           Q-3  CH.sub.3                                                                               O  H  CH.sub.3                                                                               OCH.sub.3                                                                               CH                              H      CH.sub.2                                                                           Q-3  CH.sub.3                                                                               O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               CH                              H      CH.sub.2                                                                           Q-3  CH.sub.3                                                                               O  H  Cl      OCH.sub.3                                                                               CH                              H      CH.sub.2                                                                           Q-3  CH.sub.3                                                                               O  H  CH.sub.3                                                                               OCH.sub.3                                                                               N                               H      CH.sub.2                                                                           Q-3  CH.sub.3                                                                               O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               N                               H      O   Q-3  CH.sub.3                                                                               O  H  CH.sub.3                                                                               CH.sub.3 CH                              H      O   Q-3  CH.sub.3                                                                               O  H  CH.sub.3                                                                               OCH.sub.3                                                                               CH                              H      O   Q-3  CH.sub.3                                                                               O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               CH                              H      O   Q-3  CH.sub.3                                                                               O  H  Cl      OCH.sub.3                                                                               CH                              H      O   Q-3  CH.sub.3                                                                               O  H  CH.sub.3                                                                               OCH.sub.3                                                                               N                               H      O   Q-3  CH.sub.3                                                                               O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               N                               H      --  Q-3  CH.sub.3                                                                               S  H  CH.sub.3                                                                               CH.sub.3 CH                              H      --  Q-3  CH.sub.3                                                                               S  H  CH.sub.3                                                                               OCH.sub.3                                                                               CH                              H      --  Q-3  CH.sub.3                                                                               S  H  OCH.sub.3                                                                              OCH.sub.3                                                                               CH                              H      --  Q-3  CH.sub.3                                                                               S  H  Cl      OCH.sub.3                                                                               CH                              H      --  Q-3  CH.sub.3                                                                               S  H  CH.sub.3                                                                               OCH.sub.3                                                                               N                               H      --  Q-3  CH.sub.3                                                                               S  H  OCH.sub.3                                                                              OCH.sub.3                                                                               N                               H      --  Q-3  CH.sub.3                                                                               O  CH.sub.3                                                                          CH.sub.3                                                                               CH.sub.3 CH                              H      --  Q-3  CH.sub.3                                                                               O  CH.sub.3                                                                          CH.sub.3                                                                               OCH.sub.3                                                                               CH                              H      --  Q-3  CH.sub.3                                                                               O  CH.sub.3                                                                          OCH.sub.3                                                                              OCH.sub.3                                                                               CH                              H      --  Q-3  CH.sub.3                                                                               O  CH.sub.3                                                                          Cl      OCH.sub.3                                                                               CH                              H      --  Q-3  CH.sub.3                                                                               O  CH.sub.3                                                                          CH.sub.3                                                                               OCH.sub.3                                                                               N                               H      --  Q-3  CH.sub.3                                                                               O  CH.sub.3                                                                          OCH.sub.3                                                                              OCH.sub.3                                                                               N  180-182(d)                   H      --  Q-3  CH.sub.3                                                                               O  H  OC.sub.2 H.sub.5                                                                       NHCH.sub.3                                                                              CH                              H      --  Q-3  CH.sub.3                                                                               O  H  H       OCH.sub.3                                                                               CH                              H      --  Q-3  CH.sub.3                                                                               O  H  H       OC.sub.2 H.sub.5                                                                        CH                              H      --  Q-3  CH.sub.3                                                                               O  H  H       OCF.sub.2 H                                                                             CH                              H      --  Q-3  CH.sub.3                                                                               O  H  CH.sub.3                                                                               SCF.sub.2 H                                                                             CH                              H      --  Q-3  CH.sub.3                                                                               O  H  CH.sub.3                                                                               CH.sub.2 OCH.sub.3                                                                      CH                              H      --  Q-3  CH.sub.3                                                                               O  H  OCH.sub.3                                                                              OC.sub.2 H.sub.5                                                                        CH                              H      --  Q-3  CH.sub.3                                                                               O  H  OCH.sub.3                                                                              CF.sub.3 CH                              H      --  Q-3  CH.sub.3                                                                               O  H  OCH.sub.3                                                                              O(CH.sub.2).sub.2 OCH.sub.3                                                             CH                              H      --  Q-3  CH.sub.3                                                                               O  H  OCH.sub.3                                                                              SCF.sub.2 H                                                                             CH                              H      --  Q-3  CH.sub.3                                                                               O  H  OCH.sub.3                                                                              C.tbd.CH CH                              H      --  Q-3  CH.sub.3                                                                               O  H  OCH.sub.3                                                                              C.tbd.C--CH.sub.3                                                                       CH                              H      --  Q-3  CH.sub.3                                                                               O  H  OCH.sub.3                                                                              N(OCH.sub.3)CH.sub.3                                                                    CH                              H      --  Q-4  CH.sub.3                                                                               O  H  CH.sub.3                                                                               CH.sub.3 CH                              H      --  Q-4  CH.sub.3                                                                               O  H  CH.sub.3                                                                               OCH.sub.3                                                                               CH                              H      --  Q-4  CH.sub.3                                                                               O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               CH                              H      --  Q-4  CH.sub.3                                                                               O  H  Cl      OCH.sub.3                                                                               CH                              H      --  Q-4  CH.sub.3                                                                               O  H  CH.sub.3                                                                               OCH.sub.3                                                                               N                               H      --  Q-4  CH.sub.3                                                                               O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               N                               H      --  Q-4  OCH.sub.3                                                                              O  H  CH.sub.3                                                                               CH.sub.3 CH                              H      --  Q-4  OCH.sub.3                                                                              O  H  CH.sub.3                                                                               OCH.sub.3                                                                               CH                              H      --  Q-4  OCH.sub.3                                                                              O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               CH                              H      --  Q-4  OCH.sub.3                                                                              O  H  Cl      OCH.sub.3                                                                               CH                              H      --  Q-4  OCH.sub.3                                                                              O  H  CH.sub.3                                                                               OCH.sub.3                                                                               N                               H      --  Q-4  OCH.sub.3                                                                              O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               N                               H      --  Q-4  SCH.sub.3                                                                              O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               N                               H      --  Q-4  SCH.sub.3                                                                              O  H  CH.sub.3                                                                               OCH.sub.3                                                                               CH                              H      --  Q-4  SCH.sub.3                                                                              O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               CH                              H      --  Q-4  SCH.sub.3                                                                              O  H  Cl      OCH.sub.3                                                                               CH                              H      --  Q-4  SCH.sub.3                                                                              O  H  CH.sub.3                                                                               OCH.sub.3                                                                               N                               H      --  Q-4  SCH.sub.3                                                                              O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               N                               H      --  Q-4  N(CH.sub.2).sub.4                                                                      O  H  CH.sub.3                                                                               CH.sub.3 CH                              H      --  Q-4  N(CH.sub.2).sub.4                                                                      O  H  CH.sub.3                                                                               OCH.sub.3                                                                               CH                              H      --  Q-4  N(CH.sub.2).sub.4                                                                      O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               CH                              H      --  Q-4  N(CH.sub.2).sub.4                                                                      O  H  Cl      OCH.sub.3                                                                               CH                              H      --  Q-4  N(CH.sub.2).sub.4                                                                      O  H  CH.sub.3                                                                               OCH.sub.3                                                                               N                               H      --  Q-4  N(CH.sub.2).sub.4                                                                      O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               N                               H      --  Q-4  C.sub.6 H.sub.5                                                                        O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               CH                              H      --  Q-4  C.sub.6 H.sub.5                                                                        O  H  OCH.sub.3                                                                              CH.sub.3 CH                              H      --  Q-4  C.sub.6 H.sub.5                                                                        O  H  CH.sub.3                                                                               CH.sub.3 CH                              H      --  Q-4  C.sub.6 H.sub.5                                                                        O  H  Cl      OCH.sub.3                                                                               CH                              H      --  Q-4  C.sub.6 H.sub.5                                                                        O  H  CH.sub.3                                                                               OCH.sub.3                                                                               N                               H      --  Q-4  CF.sub.3                                                                               O  H  CH.sub.3                                                                               OCH.sub.3                                                                               CH                              H      --  Q-4  CF.sub.3                                                                               O  H  CH.sub.3                                                                               CH.sub.3 CH                              H      --  Q-4  CF.sub.3                                                                               O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               CH                              H      --  Q-4  CF.sub.3                                                                               O  H  Cl      OCH.sub.3                                                                               CH                              H      --  Q-4  CF.sub.3                                                                               O  H  OCH.sub.3                                                                              CH.sub.3 N                               H      --  Q-4  CF.sub.3                                                                               O  H  OC.sub.2 H.sub.5                                                                       NHCH.sub.3                                                                              N                               H      --  Q-4  CH.sub.2 CH═CH.sub.2                                                               O  H  CH.sub.3                                                                               CH.sub. 3                                                                               CH                              H      --  Q-4  CH.sub.2 CH═CH.sub.2                                                               O  H  CH.sub.3                                                                               OCH.sub.3                                                                               CH                              H      --  Q-4  CH.sub.2 CH═CH.sub.2                                                               O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               CH                              H      --  Q-4  CH.sub.2 CH═CH.sub.2                                                               O  H  OCH.sub.3                                                                              CH.sub.3 N                               6-CH.sub.3                                                                            --  Q-3  CH.sub.3                                                                               O  H  CH.sub.3                                                                               CH.sub.3 CH                              6-CH.sub.3                                                                            --  Q-3  CH.sub.3                                                                               O  H  OCH.sub.3                                                                              CH.sub.3 CH                              6-CH.sub.3                                                                            --  Q-3  CH.sub.3                                                                               O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               CH                              6-CH.sub.3                                                                            --  Q-3  CH.sub.3                                                                               O  H  Cl      OCH.sub.3                                                                               CH                              6-CH.sub.3                                                                            --  Q-3  CH.sub.3                                                                               O  H  OCH.sub.3                                                                              CH.sub.3 N                               6-Cl   --  Q-3  CH.sub.3                                                                               O  H  CH.sub.3                                                                               CH.sub.3 CH                              6-Cl   --  Q-3  CH.sub.3                                                                               O  H  OCH.sub.3                                                                              CH.sub.3 CH                              6-Cl   --  Q-3  CH.sub.3                                                                               O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               CH                              6-Cl   --  Q-3  CH.sub.3                                                                               O  H  Cl      OCH.sub.3                                                                               CH                              H      --  Q-3  OC.sub.3 H.sub.7                                                                       O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               CH 170-171                      H      --  Q-3  OC.sub.3 H.sub.7                                                                       O  H  CH.sub.3                                                                               OCH.sub. 3                                                                              CH 171-173                      H      --  Q-3  OC.sub.3 H.sub.7                                                                       O  H  CH.sub.3                                                                               CH.sub.3 CH 176-178                      H      --  Q-3  OC.sub.3 H.sub.7                                                                       O  H  Cl      OCH.sub.3                                                                               CH 163-167                      H      --  Q-3  OC.sub.3 H.sub.7                                                                       O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               N  148-152                      H      --  Q-3  OC.sub.3 H.sub.7                                                                       O  H  CH.sub.3                                                                               OCH.sub.3                                                                               N  158-160                      5-CH.sub.3                                                                            --  Q-3  OCH.sub.3                                                                              O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               CH 181-184                      5-CH.sub.3                                                                            --  Q-3  OCH.sub.3                                                                              O  H  CH.sub.3                                                                               OCH.sub.3                                                                               CH 188-190                      5-CH.sub.3                                                                            --  Q-3  OCH.sub.3                                                                              O  H  CH.sub.3                                                                               CH.sub.3 CH 166-168                      5-CH.sub.3                                                                            --  Q-3  OCH.sub.3                                                                              O  H  Cl      OCH.sub.3                                                                               CH 182-184                      5-CH.sub.3                                                                            --  Q-3  OCH.sub.3                                                                              O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               N  184-186                      5-CH.sub.3                                                                            --  Q-3  OCH.sub.3                                                                              O  H  CH.sub.3                                                                               OCH.sub.3                                                                               N  175-178                      5-CH.sub.3                                                                            --  Q-3  OC.sub.2 H.sub.5                                                                       O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               CH 180-181                      5-CH.sub.3                                                                            --  Q-3  OC.sub.2 H.sub.5                                                                       O  H  CH.sub.3                                                                               OCH.sub.3                                                                               CH 188-191                      5-CH.sub.3                                                                            --  Q-3  OC.sub.2 H.sub.5                                                                       O  H  CH.sub.3                                                                               CH.sub.3 CH 198-199                      5-CH.sub.3                                                                            --  Q-3  OC.sub.2 H.sub.5                                                                       O  H  Cl      OCH.sub.3                                                                               CH 184-186                      5-CH.sub.3                                                                            --  Q-3  OC.sub.2 H.sub.5                                                                       O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               N  204-206                      5-CH.sub.3                                                                            --  Q-3  OC.sub.2 H.sub.5                                                                       O  H  CH.sub.3                                                                               OCH.sub.3                                                                               N  175-179                      5-OCH.sub.3                                                                           --  Q-3  OCH.sub.3                                                                              O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               CH 192-193                      5-OCH.sub.3                                                                           --  Q-3  OCH.sub.3                                                                              O  H  CH.sub.3                                                                               OCH.sub.3                                                                               CH 182-184                      5-OCH.sub.3                                                                           --  Q-3  OCH.sub.3                                                                              O  H  CH.sub.3                                                                               CH.sub.3 CH 181-183                      5-OCH.sub.3                                                                           --  Q-3  OCH.sub.3                                                                              O  H  Cl      OCH.sub.3                                                                               CH 172-175                      5-OCH.sub.3                                                                           --  Q-3  OCH.sub.3                                                                              O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               N  167-170                      5-OCH.sub.3                                                                           --  Q-3  OCH.sub.3                                                                              O  H  CH.sub.3                                                                               OCH.sub.3                                                                               N  174-176                      H      --  Q-3  OCF.sub.2 H                                                                            O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               CH                              H      --  Q-3  OCF.sub.2 H                                                                            O  H  CH.sub.3                                                                               OCH.sub.3                                                                               CH                              H      --  Q-3  OCF.sub.2 H                                                                            O  H  CH.sub.3                                                                               CH.sub.3 CH                              H      --  Q-3  OCF.sub.2 H                                                                            O  H  Cl      OCH.sub.3                                                                               CH                              H      --  Q-3  OCF.sub.2 H                                                                            O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               N                               H      --  Q-3  OCF.sub.2 H                                                                            O  H  CH.sub.3                                                                               OCH.sub.3                                                                               N                               3-CH.sub.3                                                                            --  Q-3  OC.sub.2 H.sub.5                                                                       O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               CH                              3-CH.sub.3                                                                            --  Q-3  OC.sub.2 H.sub.5                                                                       O  H  CH.sub.3                                                                               OCH.sub.3                                                                               CH                              3-CH.sub.3                                                                            --  Q-3  OC.sub.2 H.sub.5                                                                       O  H  CH.sub.3                                                                               CH.sub.3 CH                              3-CH.sub.3                                                                            --  Q-3  OC.sub.2 H.sub.5                                                                       O  H  Cl      OCH.sub.3                                                                               CH                              3-CH.sub.3                                                                            --  Q-3  OC.sub.2 H.sub.5                                                                       O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               N                               3-CH.sub.3                                                                            --  Q-3  OC.sub.2 H.sub.5                                                                       O  H  CH.sub.3                                                                               OCH.sub.3                                                                               N                               5-OC.sub.2 H.sub.5                                                                    --  Q-3  OCH.sub.3                                                                              O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               CH                              5-OC.sub.2 H.sub.5                                                                    --  Q-3  OCH.sub.3                                                                              O  H  CH.sub.3                                                                               OCH.sub.3                                                                               CH                              5-OC.sub.2 H.sub.5                                                                    --  Q-3  OCH.sub.3                                                                              O  H  CH.sub.3                                                                               CH.sub.3 CH                              5-OC.sub.2 H.sub.5                                                                    --  Q-3  OCH.sub.3                                                                              O  H  Cl      OCH.sub.3                                                                               CH                              5-OC.sub.2 H.sub.5                                                                    --  Q-3  OCH.sub.3                                                                              O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               N                               5-OC.sub.2 H.sub.5                                                                    --  Q-3  OCH.sub.3                                                                              O  H  CH.sub.3                                                                               OCH.sub.3                                                                               N                               5-OC.sub.2 H.sub.5                                                                    --  Q-3  OC.sub.2 H.sub.5                                                                       O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               CH                              5-OC.sub.2 H.sub.5                                                                    --  Q-3  OC.sub.2 H.sub.5                                                                       O  H  CH.sub.3                                                                               OCH.sub.3                                                                               CH                              5-OC.sub.2 H.sub.5                                                                    --  Q-3  OC.sub.2 H.sub.5                                                                       O  H  CH.sub.3                                                                               CH.sub.3 CH                              5-OC.sub.2 H.sub.5                                                                    --  Q-3  OC.sub.2 H.sub.5                                                                       O  H  Cl      OCH.sub.3                                                                               CH                              5-OC.sub.2 H.sub.5                                                                    --  Q-3  OC.sub.2 H.sub.5                                                                       O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               N                               5-OC.sub.2 H.sub.5                                                                    --  Q-3  OC.sub.2 H.sub.5                                                                       O  H  CH.sub.3                                                                               OCH.sub.3                                                                               N                               5-Br   --  Q-3  OCH.sub.3                                                                              O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               CH                              5-Br   --  Q-3  OCH.sub.3                                                                              O  H  CH.sub.3                                                                               OCH.sub.3                                                                               CH                              5-Br   --  Q-3  OCH.sub.3                                                                              O  H  CH.sub.3                                                                               CH.sub.3 CH                              5-Br   --  Q-3  OCH.sub.3                                                                              O  H  Cl      OCH.sub.3                                                                               CH                              5-Br   --  Q-3  OCH.sub.3                                                                              O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               N                               5-Br   --  Q-3  OCH.sub.3                                                                              O  H  CH.sub.3                                                                               OCH.sub.3                                                                               N                               5-Br   --  Q-3  OC.sub.2 H.sub.5                                                                       O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               CH                              5-Br   --  Q-3  OC.sub.2 H.sub.5                                                                       O  H  CH.sub.3                                                                               OCH.sub.3                                                                               CH                              5-Br   --  Q-3  OC.sub.2 H.sub.5                                                                       O  H  CH.sub.3                                                                               CH.sub.3 CH                              5-Br   --  Q-3  OC.sub.2 H.sub.5                                                                       O  H  Cl      OCH.sub.3                                                                               CH                              5-Br   --  Q-3  OC.sub.2 H.sub.5                                                                       O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               N                               5-Br   --  Q-3  OC.sub.2 H.sub.5                                                                       O  H  CH.sub.3                                                                               OCH.sub.3                                                                               N                               H      --  Q-3  SOCH.sub.3                                                                             O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               CH                              H      --  Q-3  SOCH.sub.3                                                                             O  H  CH.sub.3                                                                               OCH.sub.3                                                                               CH                              H      --  Q-3  SOCH.sub.3                                                                             O  H  CH.sub.3                                                                               CH.sub.3 CH                              H      --  Q-3  SOCH.sub.3                                                                             O  H  Cl      OCH.sub.3                                                                               CH                              H      --  Q-3  SOCH.sub.3                                                                             O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               N                               H      --  Q-3  SOCH.sub.3                                                                             O  H  CH.sub.3                                                                               OCH.sub.3                                                                               N                               H      --  Q-3  SO.sub.2 CH.sub.3                                                                      O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               CH                              H      --  Q-3  SO.sub.2 CH.sub.3                                                                      O  H  CH.sub.3                                                                               OCH.sub.3                                                                               CH                              H      --  Q-3  SO.sub.2 CH.sub.3                                                                      O  H  CH.sub.3                                                                               CH.sub.3 CH                              H      --  Q-3  SO.sub.2 CH.sub.3                                                                      O  H  Cl      OCH.sub.3                                                                               CH                              H      --  Q-3  SO.sub.2 CH.sub.3                                                                      O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               N                               H      --  Q-3  SO.sub.2 CH.sub.3                                                                      O  H  CH.sub.3                                                                               OCH.sub.3                                                                               N                               H      --  Q-3  CH.sub.2 CH═CH.sub.2                                                               O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               CH                              H      --  Q-3  CH.sub.2 CH═CH.sub.2                                                               O  H  CH.sub.3                                                                               OCH.sub.3                                                                               CH                              H      --  Q-3  CH.sub.2 CH═CH.sub.2                                                               O  H  CH.sub.3                                                                               CH.sub.3 CH                              H      --  Q-3  CH.sub.2 CH═CH.sub.2                                                               O  H  Cl      OCH.sub.3                                                                               CH                              H      --  Q-3  CH.sub.2 CH═CH.sub.2                                                               O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               N                               H      --  Q-3  CH.sub.2 CH═CH.sub.2                                                               O  H  CH.sub.3                                                                               OCH.sub.3                                                                               N                               6-CH.sub.3                                                                            --  Q-3  OCH.sub.3                                                                              O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               CH                              6-CH.sub.3                                                                            --  Q-3  OCH.sub.3                                                                              O  H  CH.sub.3                                                                               OCH.sub.3                                                                               CH                              6-CH.sub.3                                                                            --  Q-3  OCH.sub.3                                                                              O  H  CH.sub.3                                                                               CH.sub.3 CH                              6-CH.sub.3                                                                            --  Q-3  OCH.sub.3                                                                              O  H  Cl      OCH.sub.3                                                                               CH                              6-CH.sub.3                                                                            --  Q-3  OCH.sub.3                                                                              O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               N                               6-CH.sub.3                                                                            --  Q-3  OCH.sub.3                                                                              O  H  CH.sub.3                                                                               OCH.sub.3                                                                               N                               6-Cl   --  Q-3  OCH.sub.3                                                                              O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               CH                              6-Cl   --  Q-3  OCH.sub.3                                                                              O  H  CH.sub.3                                                                               OCH.sub.3                                                                               CH                              6-Cl   --  Q-3  OCH.sub.3                                                                              O  H  CH.sub.3                                                                               CH.sub.3 CH                              6-Cl   --  Q-3  OCH.sub.3                                                                              O  H  Cl      OCH.sub.3                                                                               CH                              6-Cl   --  Q-3  OCH.sub.3                                                                              O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               N                               6-Cl   --  Q-3  OCH.sub.3                                                                              O  H  CH.sub.3                                                                               OCH.sub.3                                                                               N                               6-CH.sub.3                                                                            --  Q-3  CH.sub.3                                                                               O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               N                               6-Cl   --  Q-3  CH.sub.3                                                                               O  H  CH.sub.3                                                                               OCH.sub.3                                                                               N                               6-Cl   --  Q-3  CH.sub.3                                                                               O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               N                               H      --  Q-4  CH.sub.2 CH═CH.sub.2                                                               O  H  Cl      OCH.sub.3                                                                               CH                              H      --  Q-4  CH.sub.2 CH═CH.sub.2                                                               O  H  OCH.sub.3                                                                              OCH.sub.3                                                                               N                               __________________________________________________________________________

                                      TABLE Ib                                     __________________________________________________________________________     General Structure 1                                                            R.sub.1                                                                              E Q  R.sub.5 W R X   Y    Z  m.p. (°C.)                           __________________________________________________________________________     H     --                                                                               Q-5                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           CH.sub.3                                                                            CH                                             H     --                                                                               Q-5                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           OCH.sub.3                                                                           N  199-201                                     H     --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           CH 213-218                                     H     --                                                                               Q-5                                                                               CH.sub.3                                                                               O H Cl  OCH.sub.3                                                                           CH                                             H     --                                                                               Q-5                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           OCH.sub.3                                                                           N                                              H     --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           N                                              H     --                                                                               Q-5                                                                               CH.sub.2 CH.sub.3                                                                      O H CH.sub.3                                                                           CH.sub.3                                                                            CH 185-189                                     H     --                                                                               Q-5                                                                               CH.sub.2 CH.sub.3                                                                      O H CH.sub.3                                                                           OCH.sub.3                                                                           CH 201-206                                     H     --                                                                               Q-5                                                                               CH.sub.2 CH.sub.3                                                                      O H OCH.sub.3                                                                          OCH.sub.3                                                                           CH 191-209                                     H     --                                                                               Q-5                                                                               CH.sub.2 CH.sub.3                                                                      O H Cl  OCH.sub.3                                                                           CH 196-199                                     H     --                                                                               Q-5                                                                               CH.sub.2 CH.sub. 3                                                                     O H CH.sub.3                                                                           OCH.sub.3                                                                           N  194-198                                     H     --                                                                               Q-5                                                                               CH.sub.2 CH.sub.3                                                                      O H OCH.sub.3                                                                          OCH.sub.3                                                                           N  166-169                                     H     --                                                                               Q-6                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           CH.sub.3                                                                            CH                                             H     --                                                                               Q-6                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           OCH.sub.3                                                                           CH                                             H     --                                                                               Q-6                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                             H     --                                                                               Q-6                                                                               CH.sub.3                                                                               O H Cl  OCH.sub.3                                                                           CH                                             H     --                                                                               Q-6                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           OCH.sub.3                                                                           N                                              H     --                                                                               Q-6                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           N                                              H     --                                                                               Q-6                                                                               C.sub.2 H.sub.5                                                                        O H CH.sub.3                                                                           CH.sub.3                                                                            CH                                             H     --                                                                               Q-6                                                                               C.sub.2 H.sub.5                                                                        O H CH.sub.3                                                                           OCH.sub.3                                                                           CH                                             H     --                                                                               Q-6                                                                               C.sub.2 H.sub.5                                                                        O H OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                             H     --                                                                               Q-6                                                                               C.sub.2 H.sub.5                                                                        O H Cl  OCH.sub.3                                                                           CH                                             H     --                                                                               Q-6                                                                               C.sub.2 H.sub.5                                                                        O H CH.sub.3                                                                           OCH.sub.3                                                                           N                                              H     --                                                                               Q-6                                                                               C.sub.2 H.sub.5                                                                        O H OCH.sub.3                                                                          OCH.sub.3                                                                           N                                              H     --                                                                               Q-6                                                                               CH.sub.2 CH═ CH.sub.2                                                              O H CH.sub.3                                                                           CH.sub.3                                                                            CH                                             H     --                                                                               Q-6                                                                               CH.sub.2 CH═CH.sub.2                                                               O H CH.sub.3                                                                           OCH.sub.3                                                                           CH                                             H     --                                                                               Q-6                                                                               CH.sub.2 CH═CH.sub.2                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                             H     --                                                                               Q-6                                                                               CH.sub.2 CH═CH.sub.2                                                               O H Cl  OCH.sub.3                                                                           CH                                             H     --                                                                               Q-6                                                                               CH.sub.2 CH═CH.sub.2                                                               O H CH.sub.3                                                                           OCH.sub.3                                                                           N                                              H     --                                                                               Q-6                                                                               CH.sub.2 CH═CH.sub.2                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           N                                              H     --                                                                               Q-7                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           CH.sub.3                                                                            CH                                             H     --                                                                               Q-7                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           OCH.sub.3                                                                           CH                                             H     --                                                                               Q-7                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                             H     --                                                                               Q-7                                                                               CH.sub.3                                                                               O H Cl  OCH.sub.3                                                                           CH                                             H     --                                                                               Q-7                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           OCH.sub.3                                                                           N                                              H     --                                                                               Q-7                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           N                                              H     --                                                                               Q-7                                                                               C.sub.2 H.sub.5                                                                        O H CH.sub.3                                                                           CH.sub.3                                                                            CH                                             H     --                                                                               Q-7                                                                               C.sub.2 H.sub.5                                                                        O H CH.sub.3                                                                           OCH.sub.3                                                                           CH                                             H     --                                                                               Q-7                                                                               C.sub. 2 H.sub.5                                                                       O H OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                             H     --                                                                               Q-7                                                                               C.sub.2 H.sub.5                                                                        O H Cl  OCH.sub.3                                                                           CH                                             H     --                                                                               Q-7                                                                               C.sub.2 H.sub.5                                                                        O H CH.sub.3                                                                           OCH.sub.3                                                                           N                                              H     --                                                                               Q-7                                                                               C.sub.2 H.sub.5                                                                        O H OCH.sub.3                                                                          OCH.sub.3                                                                           N                                              H     --                                                                               Q-7                                                                               CH.sub.2 CH═CH.sub.2                                                               O H CH.sub.3                                                                           CH.sub.3                                                                            CH                                             H     --                                                                               Q-7                                                                               CH.sub.2 CH═CH.sub.2                                                               O H CH.sub.3                                                                           OCH.sub.3                                                                           CH                                             H     --                                                                               Q-7                                                                               CH.sub.2 CH═CH.sub.2                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                             H     --                                                                               Q-7                                                                               CH.sub.2 CH═CH.sub.2                                                               O H Cl  OCH.sub.3                                                                           CH                                             H     --                                                                               Q-7                                                                               CH.sub.2 CH═CH.sub.2                                                               O H CH.sub.3                                                                           OCH.sub.3                                                                           N  202                                         H     --                                                                               Q-7                                                                               CH.sub.2 CH═CH.sub.2                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           N                                              5-Cl  --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           CH 178-180                                     5-Cl  --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          CH.sub.3                                                                            CH 134-140                                     5-Cl  --                                                                               Q-5                                                                               CH.sub.3                                                                               O H Cl  OCH.sub.3                                                                           CH                                             5-Cl  --                                                                               Q-5                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           CH.sub.3                                                                            CH                                             5-Cl  --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          CH.sub.3                                                                            N  202                                         5-CH.sub.3                                                                           --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                             5-CH.sub.3                                                                           --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          CH.sub.3                                                                            CH                                             5-CH.sub.3                                                                           --                                                                               Q-5                                                                               CH.sub.3                                                                               O H Cl  OCH.sub.3                                                                           CH                                             5-CH.sub.3                                                                           --                                                                               Q-5                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           CH.sub.3                                                                            CH                                             5-CH.sub.3                                                                           --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          CH.sub.3                                                                            N                                              6-CH.sub.3                                                                           --                                                                               Q-5                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           CH.sub.3                                                                            CH                                             6-CH.sub.3                                                                           --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          CH.sub.3                                                                            CH                                             6-CH.sub.3                                                                           --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                             6-CH.sub.3                                                                           --                                                                               Q-5                                                                               CH.sub.3                                                                               O H Cl  OCH.sub.3                                                                           CH                                             6-CH.sub.3                                                                           --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          CH.sub.3                                                                            N                                              5-OCH.sub.3                                                                          --                                                                               Q-5                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           CH.sub.3                                                                            CH                                             5-OCH.sub.3                                                                          --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          CH.sub.3                                                                            CH                                             5-OCH.sub.3                                                                          --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                             5-OCH.sub. 3                                                                         --                                                                               Q-5                                                                               CH.sub.3                                                                               O H Cl  OCH.sub.3                                                                           CH                                             5-OCH.sub.3                                                                          --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          CH.sub.3                                                                            N                                              6-Cl  --                                                                               Q-5                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           CH.sub.3                                                                            CH                                             6-Cl  --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          CH.sub.3                                                                            CH                                             6-Cl  --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                             6-Cl  --                                                                               Q-5                                                                               CH.sub.3                                                                               O H Cl  OCH.sub.3                                                                           CH                                             6-Cl  --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          CH.sub.3                                                                            N                                              5-(CH.sub.3).sub.2 N                                                                 --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          CH.sub.3                                                                            CH                                             5-(CH.sub.3).sub.2 N                                                                 --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                             5-(CH.sub.3).sub.2 N                                                                 --                                                                               Q-5                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           CH.sub.3                                                                            CH                                             5-(CH.sub.3).sub.2 N                                                                 --                                                                               Q-5                                                                               CH.sub.3                                                                               O H Cl  OCH.sub.3                                                                           CH                                             5-(CH.sub.3).sub.2 N                                                                 --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          CH.sub.3                                                                            N                                              5-F   --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                             5-F   --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          CH.sub.3                                                                            CH                                             5-F   --                                                                               Q-5                                                                               CH.sub.3                                                                               O H Cl  OCH.sub.3                                                                           CH                                             5-F   --                                                                               Q-5                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           CH.sub.3                                                                            CH                                             H     --                                                                               Q-5                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           OCF.sub.2 H                                                                         CH 196-198                                     H     --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCF.sub.2 H                                                                         CH 162-166                                     5-CH.sub.3                                                                           --                                                                               Q-5                                                                               C.sub.2 H.sub.5                                                                        O H Cl  OCH.sub.3                                                                           CH 125-128                                     5-CH.sub.3                                                                           --                                                                               Q-5                                                                               C.sub.2 H.sub.5                                                                        O H OCH.sub.3                                                                          OCH.sub.3                                                                           N  70-112                                      5-CH.sub.3                                                                           --                                                                               Q-5                                                                               C.sub.2 H.sub.5                                                                        O H CH.sub.3                                                                           OCH.sub.3                                                                           N  190-194                                     5-CH.sub.3                                                                           --                                                                               Q-5                                                                               C.sub.2 H.sub.5                                                                        O H OCH.sub.3                                                                          OCH.sub.3                                                                           CH 153-157                                     5-CH.sub.3                                                                           --                                                                               Q-5                                                                               C.sub.2 H.sub.5                                                                        O H CH.sub.3                                                                           OCH.sub.3                                                                           CH 170-173                                     5-CH.sub.3                                                                           --                                                                               Q-5                                                                               C.sub.2 H.sub.5                                                                        O H CH.sub.3                                                                           CH.sub.3                                                                            CH 141-143                                     5-Cl  --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           N                                              5-CH.sub.3                                                                           --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           N                                              6-CH.sub.3                                                                           --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           N                                              5-OCH.sub.3                                                                          --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           N                                              6-Cl  --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           N                                              5-(CH.sub.3).sub.2 N                                                                 --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           N                                              5-F   --                                                                               Q-5                                                                               CH.sub.3                                                                               O H CH.sub.3                                                                           OCH.sub.3                                                                           N                                              5-F   --                                                                               Q-5                                                                               CH.sub.3                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                           N                                              __________________________________________________________________________

                                      TABLE II                                     __________________________________________________________________________     General Structure 2                                                            R.sub.1                                                                             E Q  R.sub.3    W R X.sub.1                                                                             Y.sub.1                                                                           m.p. (°C.)                             __________________________________________________________________________     H    --                                                                               Q-1                                                                               CH.sub.3   O H CH.sub.3                                                                            O                                                H    --                                                                               Q-1                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                H    --                                                                               Q-1                                                                               CH.sub.3   O H OC.sub.2 H.sub.5                                                                    O                                                H    --                                                                               Q-1                                                                               CH.sub.3   O H OCF.sub.2 H                                                                         O                                                H    --                                                                               Q-1                                                                               CH.sub.3   O H CH.sub.3                                                                            CH.sub.2                                         H    --                                                                               Q-1                                                                               CH.sub.3   O H OCH.sub.3                                                                           CH.sub.2                                         H    --                                                                               Q-1                                                                               CH.sub.3   O H OC.sub.2 H.sub.5                                                                    CH.sub.2                                         H    --                                                                               Q-1                                                                               CH.sub.3   O H OCF.sub.2 H                                                                         CH.sub.2                                         H    --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                           O H CH.sub.3                                                                            O                                                H    --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                           O H OCH.sub.3                                                                           O                                                H    --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                           O H OC.sub.2 H.sub.5                                                                    O                                                H    --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                           O H OCF.sub.2 H                                                                         O                                                H    --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                           O H CH.sub.3                                                                            CH.sub.2                                         H    --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                           O H OCH.sub.3                                                                           CH.sub.2                                         H    --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                           O H OC.sub.2 H.sub.5                                                                    CH.sub.2                                         H    --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                           O H OCF.sub.2 H                                                                         CH.sub.2                                         H    --                                                                               Q-1                                                                               (CH.sub.2).sub.5 CH.sub.3                                                                 O H OCH.sub.3                                                                           O                                                H    --                                                                               Q-1                                                                               CH.sub.2 CH═CH--CH.sub.2 Cl                                                           O H OCH.sub.3                                                                           O                                                H    --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                           O H OCH.sub.3                                                                           O                                                5-CH.sub.3                                                                          --                                                                               Q-1                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                5-CH.sub.3                                                                          --                                                                               Q-1                                                                               CH.sub.3   O H OCH.sub.3                                                                           CH.sub.2                                         5-CH.sub.3                                                                          --                                                                               Q-1                                                                               CH.sub.3   O H OCH.sub.3                                                                           CH.sub.2                                         5-CH.sub.3                                                                          --                                                                               Q-1                                                                               CH.sub.3   O H OCH.sub.3                                                                           CH.sub.2                                         5-Cl --                                                                               Q-1                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                5-OCH.sub.3                                                                         --                                                                               Q-1                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                5-OCH.sub.3                                                                         --                                                                               Q-1                                                                               CH.sub.3   O H CH.sub.3                                                                            O                                                5-OC.sub.2 H.sub.5                                                                  --                                                                               Q-1                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                5-OC.sub.2 H.sub.5                                                                  --                                                                               Q-1                                                                               CH.sub.3   O H CH.sub.3                                                                            O                                                5-SCH.sub.3                                                                         --                                                                               Q-1                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                5-SCH.sub.3                                                                         --                                                                               Q-1                                                                               CH.sub.3   O H CH.sub.3                                                                            O                                                5-SC.sub.2 H.sub.5                                                                  --                                                                               Q-1                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                5-SC.sub.2 H.sub.5                                                                  --                                                                               Q-1                                                                               CH.sub.3   O H CH.sub.3                                                                            O                                                5-CN --                                                                               Q-1                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                5-CN --                                                                               Q-1                                                                               CH.sub.3   O H CH.sub.3                                                                            O                                                5-OCF.sub.2 H                                                                       --                                                                               Q-1                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                5-OCF.sub.2 H                                                                       --                                                                               Q-1                                                                               CH.sub.3   O H CH.sub.3                                                                            O                                                H    --                                                                               Q-2                                                                               CH.sub.3   O H CH.sub.3                                                                            O                                                H    --                                                                               Q-2                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                H    --                                                                               Q-2                                                                               CH.sub.3   O H OC.sub.2 H.sub.5                                                                    O                                                H    --                                                                               Q-2                                                                               CH.sub.3   O H OCF.sub.2 H                                                                         O                                                H    --                                                                               Q-2                                                                               CH.sub.3   O H CH.sub.3                                                                            CH.sub.2                                         H    --                                                                               Q-2                                                                               CH.sub.3   O H OCH.sub.3                                                                           CH.sub.2                                         H    --                                                                               Q-2                                                                               CH.sub.3   O H OC.sub.2 H.sub. 5                                                                   CH.sub.2                                         H    --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                           O H CH.sub.3                                                                            O                                                H    --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                           O H OCH.sub.3                                                                           O                                                H    --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                           O H CH.sub.3                                                                            CH.sub.2                                         H    --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                           O H OCH.sub.3                                                                           CH.sub.2                                         5-CH.sub.3                                                                          --                                                                               Q-2                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                5-CH.sub.3                                                                          --                                                                               Q-2                                                                               CH.sub.3   O H OCH.sub.3                                                                           CH.sub.2                                         5-C.sub.2 H.sub.5                                                                   --                                                                               Q-2                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                5-OCH.sub.3                                                                         --                                                                               Q-2                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                5-OCH.sub.3                                                                         --                                                                               Q-2                                                                               CH.sub.3   O H CH.sub.3                                                                            O                                                5-OC.sub.2 H.sub.5                                                                  --                                                                               Q-2                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                5-OC.sub.2 H.sub.5                                                                  --                                                                               Q-2                                                                               CH.sub.3   O H CH.sub.3                                                                            O                                                5-SCH.sub.3                                                                         --                                                                               Q-2                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                5-SCH.sub.3                                                                         --                                                                               Q-2                                                                               CH.sub.3   O H CH.sub.3                                                                            O                                                5-SC.sub.2 H.sub.5                                                                  --                                                                               Q-2                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                5-OCF.sub.2 H                                                                       --                                                                               Q-2                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                6-CH.sub. 3                                                                         --                                                                               Q-1                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                6-CH.sub.3                                                                          --                                                                               Q-1                                                                               CH.sub.3   O H CH.sub.3                                                                            O                                                6-CH.sub.3                                                                          --                                                                               Q-1                                                                               CH.sub.3   O H OCH.sub.3                                                                           CH.sub.2                                         6-Cl --                                                                               Q-1                                                                               CH.sub.3   O H OCH.sub.3                                                                           O                                                6-Cl --                                                                               Q-1                                                                               CH.sub.3   O H CH.sub.3                                                                            O                                                6-Cl --                                                                               Q-1                                                                               CH.sub.3   O H OCH.sub.3                                                                           CH.sub.2                                         __________________________________________________________________________

                  TABLE IIa                                                        ______________________________________                                         General Structure 2                                                                                                            m.p.                           R.sub.1                                                                               E     Q      R.sub.4                                                                              W   R   X.sub.1                                                                               Y.sub.1                                                                               (°C.)                   ______________________________________                                         H      --    Q-3    CH.sub.3                                                                             O   H   CH.sub.3                                                                              O                                     H      --    Q-3    CH.sub.3                                                                             O   H   OCH.sub.3                                                                             O                                     H      --    Q-3    CH.sub.3                                                                             O   H   OC.sub.2 H.sub.5                                                                      O                                     H      --    Q-3    CH.sub.3                                                                             O   H   OCF.sub.2 H                                                                           O                                     H      --    Q-3    CH.sub.3                                                                             O   H   CH.sub.3                                                                              CH.sub.2                              H      --    Q-3    CH.sub.3                                                                             O   H   OCH.sub.3                                                                             CH.sub.2                              H      --    Q-3    CH.sub.3                                                                             O   H   OC.sub.2 H.sub.5                                                                      CH.sub.2                              H      --    Q-3    C.sub.2 H.sub.5                                                                      O   H   CH.sub.3                                                                              O                                     H      --    Q-3    C.sub.2 H.sub.5                                                                      O   H   OCH.sub.3                                                                             O                                     H      --    Q-3    C.sub.2 H.sub.5                                                                      O   H   OC.sub.2 H.sub.5                                                                      O                                     H      --    Q-3    C.sub.2 H.sub.5                                                                      O   H   CH.sub.3                                                                              CH.sub.2                              H      --    Q-3    C.sub.2 H.sub.5                                                                      O   H   OCH.sub.3                                                                             CH.sub.2                              H      --    Q-3    C.sub.2 H.sub.5                                                                      O   H   OC.sub.2 H.sub.5                                                                      CH.sub.2                              H      --    Q-3    C.sub.2 H.sub.5                                                                      O   H   OCF.sub.2 H                                                                           CH.sub.2                              H      --    Q-3    C.sub.2 H.sub.5                                                                      O   H   OCH.sub.3                                                                             O                                     H      --    Q-3    C.sub.2 H.sub.5                                                                      O   H   OCH.sub.3                                                                             O                                     5-CH.sub.3                                                                            --    Q-3    CH.sub.3                                                                             O   H   OCH.sub.3                                                                             O                                     5-CH.sub.3                                                                            --    Q-3    CH.sub.3                                                                             O   H   OCH.sub.3                                                                             CH.sub.2                              5-Cl   --    Q-3    CH.sub.3                                                                             O   H   OCH.sub.3                                                                             O                                     5-Cl   --    Q-3    CH.sub.3                                                                             O   H   OCH.sub.3                                                                             O                                     5-Cl   --    Q-3    CH.sub.3                                                                             O   H   CH.sub.3                                                                              O                                     5-OCH.sub.3                                                                           --    Q-3    CH.sub.3                                                                             O   H   OCH.sub.3                                                                             O                                     5-OCH.sub.3                                                                           --    Q-3    CH.sub.3                                                                             O   H   CH.sub.3                                                                              O                                     5-OC.sub.2 H.sub.5                                                                    --    Q-3    CH.sub.3                                                                             O   H   OCH.sub.3                                                                             O                                     5-OC.sub.2 H.sub.5                                                                    --    Q-3    CH.sub.3                                                                             O   H   CH.sub.3                                                                              O                                     5-SCH.sub.3                                                                           --    Q-3    CH.sub.3                                                                             O   H   OCH.sub.3                                                                             O                                     5-SCH.sub.3                                                                           --    Q-3    CH.sub.3                                                                             O   H   CH.sub.3                                                                              O                                     5-SC.sub.2 H.sub.5                                                                    --    Q-3    CH.sub.3                                                                             O   H   OCH.sub.3                                                                             O                                     5-SC.sub.2 H.sub.5                                                                    --    Q-3    CH.sub.3                                                                             O   H   CH.sub.3                                                                              O                                     5-OCF.sub.2 H                                                                         --    Q-3    CH.sub.3                                                                             O   H   OCH.sub.3                                                                             O                                     5-OCF.sub.2 H                                                                         --    Q-3    CH.sub.3                                                                             O   H   CH.sub.3                                                                              O                                     5-SCF.sub.2 H                                                                         --    Q-3    CH.sub.3                                                                             O   H   OCH.sub.3                                                                             O                                     5-SCF.sub.2 H                                                                         --    Q-3    CH.sub.3                                                                             O   H   CH.sub.3                                                                              O                                     H      --    Q-4    CH.sub.3                                                                             O   H   CH.sub.3                                                                              O                                     H      --    Q-4    CH.sub.3                                                                             O   H   OCH.sub.3                                                                             O                                     H      --    Q-4    CH.sub.3                                                                             O   H   OC.sub.2 H.sub.5                                                                      O                                     H      --    Q-4    CH.sub.3                                                                             O   H   OCF.sub.2 H                                                                           O                                     H      --    Q-4    CH.sub.3                                                                             O   H   CH.sub.3                                                                              CH.sub.2                              H      --    Q-4    CH.sub.3                                                                             O   H   OCH.sub.3                                                                             CH.sub.2                              H      --    Q-4    CH.sub.3                                                                             O   H   OC.sub.2 H.sub.5                                                                      CH.sub.2                              H      --    Q-4    CH.sub.3                                                                             O   H   OCF.sub. 2 H                                                                          CH.sub.2                              H      --    Q-4    C.sub.2 H.sub.5                                                                      O   H   CH.sub.3                                                                              O                                     H      --    Q-4    C.sub.2 H.sub.5                                                                      O   H   OCH.sub.3                                                                             O                                     H      --    Q-4    C.sub.2 H.sub.5                                                                      O   H   OC.sub.2 H.sub.5                                                                      O                                     H      --    Q-4    C.sub.2 H.sub.5                                                                      O   H   OCF.sub.2 H                                                                           O                                     H      --    Q-4    C.sub.2 H.sub.5                                                                      O   H   CH.sub.3                                                                              CH.sub.2                              H      --    Q-4    C.sub.2 H.sub.5                                                                      O   H   OCH.sub.3                                                                             CH.sub.2                              H      --    Q-4    C.sub.2 H.sub.5                                                                      O   H   OC.sub.2 H.sub.5                                                                      CH.sub.2                              H      --    Q-4    C.sub.2 H.sub.5                                                                      O   H   OCF.sub.2 H                                                                           CH.sub.2                              6-CH.sub.3                                                                            --    Q-3    CH.sub.3                                                                             O   H   OCH.sub.3                                                                             CH.sub.2                              6-CH.sub.3                                                                            --    Q-3    CH.sub.3                                                                             O   H   OCH.sub.3                                                                             O                                     6-CH.sub.3                                                                            --    Q-3    CH.sub.3                                                                             O   H   CH.sub.3                                                                              O                                     6-Cl   --    Q-3    CH.sub.3                                                                             O   H   OCH.sub.3                                                                             CH.sub.2                              6-Cl   --    Q-3    CH.sub.3                                                                             O   H   OCH.sub.3                                                                             O                                     6-Cl   --    Q-3    CH.sub.3                                                                             O   H   CH.sub.3                                                                              O                                     6-CH.sub.3                                                                            --    Q-4    CH.sub.3                                                                             O   H   OCH.sub.3                                                                             CH.sub.2                              6-CH.sub.3                                                                            --    Q-4    CH.sub.3                                                                             O   H   OCH.sub.3                                                                             O                                     6-CH.sub.3                                                                            --    Q-4    CH.sub.3                                                                             O   H   CH.sub.3                                                                              O                                     6-Cl   --    Q-4    CH.sub.3                                                                             O   H   OCH.sub.3                                                                             CH.sub.2                              6-Cl   --    Q-4    CH.sub.3                                                                             O   H   OCH.sub.3                                                                             O                                     6-Cl   --    Q-4    CH.sub.3                                                                             O   H   CH.sub.3                                                                              O                                     H      --    Q-3    H     O   H   OCH.sub.3                                                                             O                                     H      --    Q-3    H     O   H   CH.sub.3                                                                              O                                     H      --    Q-3    H     O   H   OCH.sub.3                                                                             CH.sub.2                              H      --    Q-3    H     O   H   CH.sub.3                                                                              CH.sub.2                              H      --    Q-3    OCH.sub.3                                                                            O   H   OCH.sub.3                                                                             O                                     H      --    Q-3    OCH.sub.3                                                                            O   H   CH.sub.3                                                                              O                                     H      --    Q-3    OCH.sub.3                                                                            O   H   OCH.sub.3                                                                             CH.sub.2                              H      --    Q-3    OCH.sub.3                                                                            O   H   CH.sub.3                                                                              CH.sub.2                              H      --    Q-3    OC.sub.2 H.sub.5                                                                     O   H   OCH.sub.3                                                                             O                                     H      --    Q-3    OC.sub.2 H.sub.5                                                                     O   H   CH.sub.3                                                                              O                                     H      --    Q-3    OC.sub.2 H.sub.5                                                                     O   H   OCH.sub.3                                                                             CH.sub.2                              H      --    Q-3    OC.sub.2 H.sub.5                                                                     O   H   CH.sub.3                                                                              CH.sub.2                              H      --    Q-3    SCH.sub.3                                                                            O   H   OCH.sub.3                                                                             O                                     H      --    Q-3    SCH.sub.3                                                                            O   H   CH.sub.3                                                                              O                                     H      --    Q-3    SCH.sub.3                                                                            O   H   OCH.sub.3                                                                             CH.sub.2                              H      --    Q-3    SCH.sub.3                                                                            O   H   CH.sub.3                                                                              CH.sub.2                              ______________________________________                                    

                  TABLE IIb                                                        ______________________________________                                         General Structure 2                                                            R.sub.1                                                                               E     Q      R.sub.5                                                                              W   R   X.sub.1                                                                              Y.sub.1                                                                             m.p. (°C.)                 ______________________________________                                         H      --    Q-5    CH.sub.3                                                                             O   H   OCH.sub.3                                                                            O                                      H      --    Q-5    CH.sub.3                                                                             O   H   OCH.sub.3                                                                            CH.sub.2                               H      --    Q-5    CH.sub.3                                                                             O   H   CH.sub.3                                                                             O                                      H      --    Q-5    C.sub.2 H.sub.5                                                                      O   H   OCH.sub.3                                                                            O                                      H      --    Q-5    C.sub.2 H.sub.5                                                                      O   H   OCH.sub.3                                                                            CH.sub.2                               H      --    Q-5    C.sub.2 H.sub.5                                                                      O   H   CH.sub.3                                                                             O                                      5-CH.sub.3                                                                            --    Q-5    CH.sub.3                                                                             O   H   OCH.sub.3                                                                            O                                      5-CH.sub.3                                                                            --    Q-5    CH.sub.3                                                                             O   H   OCH.sub.3                                                                            CH.sub.2                               5-CH.sub.3                                                                            --    Q-5    CH.sub.3                                                                             O   H   CH.sub.3                                                                             O                                      5-Cl   --    Q-5    CH.sub.3                                                                             O   H   OCH.sub.3                                                                            O                                      5-Cl   --    Q-5    CH.sub.3                                                                             O   H   OCH.sub.3                                                                            CH.sub.2                               5-Cl   --    Q-5    CH.sub.3                                                                             O   H   CH.sub.3                                                                             O                                      6-CH.sub.3                                                                            --    Q-5    CH.sub.3                                                                             O   H   OCH.sub.3                                                                            O                                      6-CH.sub.3                                                                            --    Q-5    CH.sub.3                                                                             O   H   OCH.sub.3                                                                            CH.sub.2                               6-CH.sub.3                                                                            --    Q-5    CH.sub.3                                                                             O   H   CH.sub.3                                                                             O                                      6-Cl   --    Q-5    CH.sub.3                                                                             O   H   OCH.sub.3                                                                            O                                      6-Cl   --    Q-5    CH.sub.3                                                                             O   H   OCH.sub.3                                                                            CH.sub.2                               6-Cl   --    Q-5    CH.sub.3                                                                             O   H   CH.sub.3                                                                             O                                      5-F    --    Q-5    CH.sub.3                                                                             O   H   OCH.sub.3                                                                            O                                      5-F    --    Q-5    CH.sub.3                                                                             O   H   OCH.sub.3                                                                            CH.sub.2                               5-F    --    Q-5    CH.sub.3                                                                             O   H   CH.sub.3                                                                             O                                      5-OCH.sub.3                                                                           --    Q-5    CH.sub.3                                                                             O   H   OCH.sub.3                                                                            O                                      5-OCH.sub.3                                                                           --    Q-5    CH.sub.3                                                                             O   H   OCH.sub.3                                                                            CH.sub.2                               5-OCH.sub.3                                                                           --    Q-5    CH.sub.3                                                                             O   H   CH.sub.3                                                                             O                                      ______________________________________                                    

                                      TABLE III                                    __________________________________________________________________________     General Structure 3                                                            R.sub.1                                                                             E Q  R.sub.3                                                                            R.sub.4                                                                            R.sub.5                                                                           W R X.sub.1                                                                             m.p. (°C.)                                __________________________________________________________________________     H    --                                                                               Q-1                                                                               CH.sub.3                                                                           --  -- O H CH.sub.3                                              H    --                                                                               Q-1                                                                               CH.sub.3                                                                           --  -- O H OCH.sub.3                                             H    --                                                                               Q-1                                                                               CH.sub.3                                                                           --  -- O H OC.sub.2 H.sub.5                                      H    --                                                                               Q-1                                                                               CH.sub.3                                                                           --  -- O H OCF.sub.2 H                                           H    --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                    --  -- O H CH.sub.3                                              H    --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                    --  -- O H OCH.sub.3                                             H    --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                    --  -- O H OC.sub.2 H.sub.5                                      H    --                                                                               Q-2                                                                               CH.sub.3                                                                           --  -- O H CH.sub.3                                              H    --                                                                               Q-2                                                                               CH.sub.3                                                                           --  -- O H OCH.sub.3                                             H    --                                                                               Q-2                                                                               CH.sub.3                                                                           --  -- O H OC.sub.2 H.sub.5                                      H    --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                    --  -- O H OCH.sub.3                                             H    --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                    --  -- O H CH.sub.3                                              H    --                                                                               Q-3                                                                               --  CH.sub.3                                                                           -- O H OC.sub.2 H.sub.5                                      H    --                                                                               Q-3                                                                               --  CH.sub.3                                                                           -- O H OCH.sub.3                                             H    --                                                                               Q-3                                                                               --  CH.sub.3                                                                           -- O H CH.sub.3                                              H    --                                                                               Q-3                                                                               --  C.sub.2 H.sub.5                                                                    -- O H CH.sub.3                                              H    --                                                                               Q-3                                                                               --  C.sub.2 H.sub.5                                                                    -- O H OCH.sub.3                                             6-CH.sub.3                                                                          --                                                                               Q-1                                                                               CH.sub.3                                                                           --  -- O H OCH.sub.3                                             6-CH.sub.3                                                                          --                                                                               Q-1                                                                               CH.sub.3                                                                           --  -- O H CH.sub.3                                              6-Cl --                                                                               Q-1                                                                               CH.sub.3                                                                           --  -- O H CH.sub.3                                              6-Cl --                                                                               Q-1                                                                               CH.sub.3                                                                           --  -- O H OCH.sub.3                                             H    --                                                                               Q-4                                                                               --  CH.sub.3                                                                           -- O H OCH.sub.3                                             H    --                                                                               Q-5                                                                               --  --  CH.sub.3                                                                          O H OCH.sub.3                                             H    --                                                                               Q-5                                                                               --  --  CH.sub.3                                                                          O H CH.sub.3                                              H    --                                                                               Q-6                                                                               --  --  CH.sub.3                                                                          O H OCH.sub.3                                             H    --                                                                               Q-7                                                                               --  --  CH.sub.3                                                                          O H OCH.sub.3                                             H    --                                                                               Q-3                                                                               --  H   -- O H OCH.sub.3                                             H    --                                                                               Q-3                                                                               --  H   -- O H CH.sub.3                                              H    --                                                                               Q-3                                                                               --  OCH.sub.3                                                                          -- O H OCH.sub.3                                             H    --                                                                               Q-3                                                                               --  OCH.sub.3                                                                          -- O H CH.sub.3                                              H    --                                                                               Q-3                                                                               --  OC.sub.2 H.sub.5                                                                   -- O H OCH.sub.3                                             H    --                                                                               Q-3                                                                               --  OC.sub.2 H.sub.5                                                                   -- O H CH.sub.3                                              H    --                                                                               Q-3                                                                               --  SCH.sub.3                                                                          -- O H OCH.sub.3                                             H    --                                                                               Q-3                                                                               --  SCH.sub.3                                                                          -- O H CH.sub.3                                              __________________________________________________________________________

                                      TABLE IV                                     __________________________________________________________________________     General Structure 4                                                            R.sub.1                                                                            E Q  R.sub.3                                                                           R.sub.4                                                                            R.sub.5                                                                           W R X.sub.1                                                                            Y.sub.3                                                                           m.p. (°C.)                                __________________________________________________________________________     H   --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                           H                                                   H   --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          H                                                   H   --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OC.sub.2 H.sub.5                                                                   H                                                   H   --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                           CH.sub.3                                            H   --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          CH.sub.3                                            H   --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCF.sub.2 H                                                                        CH.sub.3                                            H   --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --  -- O H CH.sub.3                                                                           H                                                   H   --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --  -- O H OCH.sub.3                                                                          H                                                   H   --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --  -- O H CH.sub.3                                                                           CH.sub.3                                            H   --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          CH.sub.3                                            H   --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          H                                                   H   --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                           H                                                   H   --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          CH.sub.3                                            H   --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                           CH.sub.3                                            H   --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                          CH.sub.3                                            H   --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                          CH.sub.3                                            H   --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                    -- O H CH.sub.3                                                                           CH.sub.3                                            H   --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                    -- O H OCH.sub.3                                                                          H                                                   H   --                                                                               Q-4                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                          H                                                   H   --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H OCH.sub.3                                                                          H                                                   H   --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H OCH.sub.3                                                                          CH.sub.3                                            H   --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H CH.sub.3                                                                           H                                                   5-Cl                                                                               --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H CH.sub.3                                                                           H                                                   6-CH.sub.3                                                                         --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H OCH.sub.3                                                                          H                                                   H   --                                                                               Q-3                                                                               -- H   -- O H CH.sub.3                                                                           H                                                   H   --                                                                               Q-3                                                                               -- H   -- O H OCH.sub.3                                                                          H                                                   H   --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H CH.sub.3                                                                           CH.sub.3                                            H   --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H OCH.sub.3                                                                          CH.sub.3                                            H   --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                   -- O H CH.sub.3                                                                           H                                                   H   --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                   -- O H OCH.sub.3                                                                          H                                                   H   --                                                                               Q-3                                                                               -- SCH.sub.3                                                                          -- O H CH.sub.3                                                                           CH.sub.3                                            H   --                                                                               Q-3                                                                               -- SCH.sub.3                                                                          -- O H OCH.sub.3                                                                          CH.sub.3                                            __________________________________________________________________________

                                      TABLE V                                      __________________________________________________________________________     General Structure 5                                                            R.sub.1                                                                            E Q  R.sub.3                                                                              R.sub.4                                                                            R.sub.5                                                                           W R X.sub.2                                                                             Y.sub.2                                                                            m.p. (°C.)                           __________________________________________________________________________     H   --                                                                               Q-1                                                                               CH.sub.3                                                                             --  -- O H CH.sub.3                                                                            OCH.sub.3                                       H   --                                                                               Q-1                                                                               CH.sub.3                                                                             --  -- O H CH.sub.2 CF.sub.3                                                                   OCH.sub.3                                       H   --                                                                               Q-1                                                                               CH.sub.3                                                                             --  -- O H CH.sub.3                                                                            SC.sub.2 H.sub.5                                H   --                                                                               Q-1                                                                               CH.sub.3                                                                             --  -- O H CH.sub.3                                                                            SCH.sub.3                                       H   --                                                                               Q-1                                                                               CH.sub.3                                                                             --  -- O H CH.sub.3                                                                            OC.sub.2 H.sub.5                                H   --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                      --  -- O H CH.sub.3                                                                            SCH.sub.3                                       H   --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                      --  -- O H CH.sub.3                                                                            OCH.sub.3                                       H   --                                                                               Q-2                                                                               CH.sub.3                                                                             --  -- O H CH.sub.3                                                                            OCH.sub.3                                       H   --                                                                               Q-2                                                                               CH(CH.sub.3).sub.2                                                                   --  -- O H CH.sub.3                                                                            OCH.sub.3                                       H   --                                                                               Q-3                                                                               --    CH.sub.3                                                                           -- O H CH.sub.3                                                                            SCH.sub.3                                       H   --                                                                               Q-3                                                                               --    CH.sub.3                                                                           -- O H CH.sub.3                                                                            SC.sub.2 H.sub.5                                H   --                                                                               Q-3                                                                               --    C.sub.2 H.sub.5                                                                    -- O H CH.sub.3                                                                            SCH.sub.3                                       H   --                                                                               Q-3                                                                               --    CF.sub.3                                                                           -- O H CH.sub.3                                                                            SCH.sub.3                                       H   --                                                                               Q-4                                                                               --    CH.sub.3                                                                           -- O H CH.sub.3                                                                            SCH.sub.3                                       6-CH.sub.3                                                                         --                                                                               Q-4                                                                               --    CH.sub.3                                                                           -- O H CH.sub.3                                                                            SCH.sub.3                                       6-Cl                                                                               --                                                                               Q-4                                                                               --    CH.sub.3                                                                           -- O H CH.sub.3                                                                            SCH.sub.3                                       H   --                                                                               Q-5                                                                               --    --  CH.sub.3                                                                          O H CH.sub.3                                                                            SCH.sub.3                                       H   --                                                                               Q-6                                                                               --    --  CH.sub.3                                                                          O H CH.sub.3                                                                            SCH.sub.3                                       H   --                                                                               Q-7                                                                               --    --  CH.sub.3                                                                          O H CH.sub.3                                                                            SCH.sub.3                                       6-CH.sub.3                                                                         --                                                                               Q-1                                                                               CH.sub.3                                                                             --  -- O H CH.sub.3                                                                            SCH.sub.3                                       5-Cl                                                                               --                                                                               Q-1                                                                               CH.sub.3                                                                             --  -- O H CH.sub. 3                                                                           SCH.sub.3                                       H   --                                                                               Q-3                                                                               --    H   -- O H CH.sub.3                                                                            SCH.sub.3                                       H   --                                                                               Q-3                                                                               --    H   -- O H C.sub.2 H.sub.5                                                                     OCH.sub.3                                       H   --                                                                               Q-3                                                                               --    OCH.sub.3                                                                          -- O H CH.sub.3                                                                            OCH.sub.3                                       H   --                                                                               Q-3                                                                               --    OCH.sub.3                                                                          -- O H CH.sub.3                                                                            OC.sub.2 H.sub.5                                H   --                                                                               Q-3                                                                               --    SCH.sub.3                                                                          -- O H CH.sub.3                                                                            OCH.sub.3                                       H   --                                                                               Q-3                                                                               --    SCH.sub.3                                                                          -- O H CH.sub.3                                                                            OC.sub.2 H.sub.5                                __________________________________________________________________________

                                      TABLE VI                                     __________________________________________________________________________     General Structure 6                                                            R.sub.1                                                                            E Q  R.sub.3                                                                           R.sub.4                                                                              R.sub.5                                                                           W R X.sub.3                                                                            m.p. (°C.)                                 __________________________________________________________________________     H   --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O H CH.sub.3                                              H   --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O H OCH.sub.3                                             H   --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O H CH.sub.3                                              H   --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O H OCH.sub.3                                             H   --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O H CH.sub.3                                              H   --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O H CH.sub.3                                              H   --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O H CH.sub.3                                              H   --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O H OCH.sub.3                                             H   --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O H CH.sub.3                                              H   --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O H OCH.sub.3                                             H   --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O H OCH.sub.3                                             H   --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O H OCH.sub.3                                             H   --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O H OCH.sub.3                                             H   --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O H OCH.sub.3                                             6-CH.sub.3                                                                         --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O H OCH.sub.3                                             6-Cl                                                                               --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O H OCH.sub.3                                             5-Cl                                                                               --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O H OCH.sub.3                                             H   --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O H OCH.sub.3                                             H   --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O H CH.sub.3                                              H   --                                                                               Q-6                                                                               -- --    CH.sub.3                                                                          O H OCH.sub.3                                             H   --                                                                               Q-6                                                                               -- --    CH.sub.3                                                                          O H CH.sub.3                                              H   --                                                                               Q-7                                                                               -- --    CH.sub.3                                                                          O H OCH.sub.3                                             H   --                                                                               Q-3                                                                               -- H     -- O H CH.sub.3                                              H   --                                                                               Q-3                                                                               -- H     -- O H OCH.sub.3                                             H   --                                                                               Q-3                                                                               -- OCH.sub. 3                                                                           -- O H CH.sub.3                                              H   --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O H OCH.sub.3                                             H   --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O H CH.sub.3                                              H   --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O H OCH.sub.3                                             H   --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O H CH.sub.3                                              H   --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O H OCH.sub.3                                             __________________________________________________________________________

                                      TABLE VII                                    __________________________________________________________________________     General Structure 7                                                            R.sub.1                                                                            E Q  R.sub.3                                                                           R.sub.4                                                                            R.sub.5                                                                           W R X.sub.4                                                                              Y.sub.4                                                                            Z.sup.1                                                                           m.p. (°C.)                          __________________________________________________________________________     H   --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                             CH.sub.3                                                                           N                                             H   --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                            CH.sub.3                                                                           N                                             H   --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OC.sub.2 H.sub.5                                                                     CH.sub.3                                                                           N                                             H   --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.2 OCH.sub.3                                                                   CH.sub.3                                                                           N                                             H   --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H Cl    CH.sub.3                                                                           N                                             H   --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                             OCH.sub.3                                                                          N                                             H   --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                            OCH.sub.3                                                                          N                                             H   --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OC.sub.2 H.sub.5                                                                     OCH.sub.3                                                                          N                                             H   --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.2 OCH.sub.3                                                                   OCH.sub.3                                                                          N                                             H   --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H Cl    OCH.sub.3                                                                          N                                             H   --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                             CH.sub.3                                                                           CH                                            H   --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                            CH.sub.3                                                                           CH                                            H   --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OC.sub.2 H.sub.5                                                                     CH.sub.3                                                                           CH                                            H   --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.2 OCH.sub.3                                                                   CH.sub.3                                                                           CH                                            H   --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H Cl    CH.sub.3                                                                           CH                                            H   --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                             OCH.sub.3                                                                          CH                                            H   --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                            OCH.sub.3                                                                          CH                                            H   --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OC.sub.2 H.sub.5                                                                     OCH.sub.3                                                                          CH                                            H   --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.2 OCH.sub.3                                                                   OCH.sub.3                                                                          CH                                            H   --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H Cl    OCH.sub.3                                                                          CH                                            H   --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                            OC.sub.2 H.sub.5                                                                   CH                                            H   --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                            Cl  CH                                            H   --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                             OC.sub.2 H.sub.5                                                                   CH                                            H   --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                             Cl  CH                                            6-CH.sub.3                                                                         --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                             CH.sub.3                                                                           CH                                            6-CH.sub.3                                                                         --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                            OCH.sub.3                                                                          CH                                            6-CH.sub.3                                                                         --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                             OCH.sub.3                                                                          CH                                            5-CH.sub.3                                                                         --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                             OCH.sub.3                                                                          CH                                            5-CH.sub.3                                                                         --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                            OCH.sub.3                                                                          CH                                            5-CH.sub.3                                                                         --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                             CH.sub.3                                                                           CH                                            5-OCH.sub.3                                                                        --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                             CH.sub.3                                                                           CH                                            5-OCH.sub.3                                                                        --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                            CH.sub.3                                                                           CH                                            5-OCH.sub.3                                                                        --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                            OCH.sub.3                                                                          CH                                            H   --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                             CH.sub.3                                                                           CH                                            H   --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                            OCH.sub.3                                                                          CH                                            H   --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                             OCH.sub.3                                                                          CH                                            H   --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                            CH.sub.3                                                                           CH                                            6-CH.sub.3                                                                         --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                            OCH.sub.3                                                                          CH                                            6-CH.sub.3                                                                         --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                            OCH.sub.3                                                                          N                                             5-Cl                                                                               --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                            OCH.sub.3                                                                          CH                                            5-Cl                                                                               --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                            CH.sub.3                                                                           CH                                            5-OCH.sub.3                                                                        --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                            OCH.sub.3                                                                          CH                                            5-OCH.sub.3                                                                        --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                             OCH.sub.3                                                                          CH                                            5-OCH.sub.3                                                                        --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                            CH.sub.3                                                                           CH                                            H   --                                                                               Q-4                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                            OCH.sub.3                                                                          CH                                            H   --                                                                               Q-4                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                             CH.sub.3                                                                           CH                                            H   --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H CH.sub.3                                                                             CH.sub.3                                                                           CH                                            H   --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H CH.sub.3                                                                             OCH.sub.3                                                                          CH                                            H   --                                                                               Q-6                                                                               -- --  CH.sub.3                                                                          O H CH.sub.3                                                                             OCH.sub.3                                                                          CH                                            H   --                                                                               Q-7                                                                               -- --  CH.sub.3                                                                          O H CH.sub.3                                                                             OCH.sub.3                                                                          CH                                            H   --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                             OCH.sub.3                                                                          N                                             H   --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                            OCH.sub.3                                                                          CH                                            H   --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --  -- O H CH.sub.3                                                                             CH.sub.3                                                                           CH                                            H   --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --  -- O H OCH.sub.3                                                                            CH.sub.3                                                                           CH                                            H   --                                                                               Q-3                                                                               -- H   -- O H CH.sub.3                                                                             OCH.sub.3                                                                          CH                                            H   --                                                                               Q-3                                                                               -- H   -- O H OCH.sub.3                                                                            OCH.sub.3                                                                          N                                             H   --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                             CH.sub.3                                                                           CH                                            H   --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                            CH.sub.3                                                                           N                                             H   --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H CH.sub.3                                                                             OCH.sub.3                                                                          CH                                            H   --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H OCH.sub.3                                                                            OCH.sub.3                                                                          N                                             H   --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                   -- O H CH.sub.3                                                                             CH.sub.3                                                                           CH                                            H   --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                   -- O H OCH.sub.3                                                                            CH.sub.3                                                                           N                                             H   --                                                                               Q-3                                                                               -- SCH.sub.3                                                                          -- O H CH.sub.3                                                                             OCH.sub.3                                                                          CH                                            H   --                                                                               Q-3                                                                               -- SCH.sub.3                                                                          -- O H OCH.sub.3                                                                            OCH.sub.3                                                                          N                                             __________________________________________________________________________

                                      TABLE VIII                                   __________________________________________________________________________     General Structure 8                                                            R.sub.1                                                                            n E Q  R.sub.3                                                                           R.sub.4                                                                              R.sub.5                                                                           W    R  X   Y    Z  m.p. (°C.)                   __________________________________________________________________________     H   0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O    H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                      H   0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O    H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O    H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                      H   0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O    H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O    H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-5                                                                               -- --    C.sub.2 H.sub.5                                                                   O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-5                                                                               -- --    C.sub.2 H.sub.5                                                                   O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-5                                                                               -- --    C.sub.2 H.sub.5                                                                   O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-5                                                                               -- --    C.sub.2 H.sub.5                                                                   O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-5                                                                               -- --    C.sub.2 H.sub.5                                                                   O    H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                      4-CH.sub.3                                                                         0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                     4-CH.sub.3                                                                         0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     4-CH.sub.3                                                                         0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  Cl  OCH.sub.3                                                                           CH                                     4-CH.sub.3                                                                         0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     4-CH.sub.3                                                                         0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                      4-Cl                                                                               0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          CH.sub.3                                                                            N                                      4-Cl                                                                               0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          CH.sub.3                                                                            CH                                     4-Cl                                                                               0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     4-Cl                                                                               0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  Cl  OCH.sub.3                                                                           CH                                     4-Cl                                                                               0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     4-Cl                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     4-Cl                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   1 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   1 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   1 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   1 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   1 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   1 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  OC.sub.2 H.sub.5                                                                   NHCH.sub.3                                                                          N                                      H   0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  OC.sub.2 H.sub.5                                                                   NHCH.sub.3                                                                          N                                      H   0 --                                                                               Q-3                                                                               -- H     -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- H     -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- H     -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-3                                                                               -- H     -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- H     -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- H     -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            N                                      H   0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-4                                                                               -- C.sub.2 H.sub.5                                                                      -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-4                                                                               -- C.sub.2 H.sub.5                                                                      -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-4                                                                               -- C.sub.2 H.sub.5                                                                      -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-4                                                                               -- C.sub.2 H.sub.5                                                                      -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-4                                                                               -- C.sub.2 H.sub.5                                                                      -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-4                                                                               -- C.sub.2 H.sub.5                                                                      -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-4                                                                               -- OCH.sub.3                                                                            -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-4                                                                               -- OCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-4                                                                               -- OCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-4                                                                               -- OCH.sub.3                                                                            -- O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-4                                                                               -- OCH.sub.3                                                                            -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-4                                                                               -- OCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-5                                                                               -- --    C.sub.2 H.sub.5                                                                   O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-6                                                                               -- --    CH.sub.3                                                                          O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-6                                                                               -- --    CH.sub.3                                                                          O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-6                                                                               -- --    CH.sub.3                                                                          O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-6                                                                               -- --    C.sub.2 H.sub.5                                                                   O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-6                                                                               -- --    C.sub.2 H.sub.5                                                                   O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-6                                                                               -- --    C.sub.2 H.sub.5                                                                   O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-7                                                                               -- --    CH.sub.3                                                                          O    H  Cl  OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-7                                                                               -- --    CH.sub.3                                                                          O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-7                                                                               -- --    CH.sub.3                                                                          O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-7                                                                               -- --    C.sub.2 H.sub.5                                                                   O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-7                                                                               -- --    C.sub.2 H.sub.5                                                                   O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-7                                                                               -- --    C.sub.2 H.sub.5                                                                   O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      4-CH.sub.3                                                                         0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      4-CH.sub.3                                                                         0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     4-CH.sub.3                                                                         0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     4-CH.sub.3                                                                         0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     4-CH.sub.3                                                                         0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  Cl  OCH.sub.3                                                                           CH                                     4-CH.sub.3                                                                         0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      4-CH.sub.3                                                                         0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      4-CH.sub.3                                                                         0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     4-CH.sub.3                                                                         0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     4-CH.sub.3                                                                         0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     4-CH.sub.3                                                                         0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  Cl  OCH.sub.3                                                                           CH                                     4-CH.sub.3                                                                         0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      4-CH.sub.3                                                                         0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      4-CH.sub.3                                                                         0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     4-CH.sub.3                                                                         0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     4-CH.sub.3                                                                         0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     4-CH.sub.3                                                                         0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  Cl  OCH.sub.3                                                                           CH                                     4-CH.sub.3                                                                         0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      4-CH.sub.3                                                                         0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      4-Cl                                                                               0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      4-Cl                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     4-Cl                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     4-Cl                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      4-Cl                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      4-Cl                                                                               0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     4-Cl                                                                               0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     4-Cl                                                                               0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     4-Cl                                                                               0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  Cl  OCH.sub.3                                                                           CH                                     4-Cl                                                                               0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      4-Cl                                                                               0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      4-Cl                                                                               0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     4-Cl                                                                               0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     4-Cl                                                                               0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     4-Cl                                                                               0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  Cl  OCH.sub.3                                                                           CH                                     4-Cl                                                                               0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      4-Cl                                                                               0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      4-Br                                                                               0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     4-Br                                                                               0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     4-Br                                                                               0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     4-Br                                                                               0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  Cl  OCH.sub.3                                                                           CH                                     4-Br                                                                               0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      4-Br                                                                               0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      4-Br                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     4-Br                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     4-Br                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     4-Br                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  Cl  OCH.sub.3                                                                           CH                                     4-Br                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      4-Br                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      4-Br                                                                               0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     4-Br                                                                               0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     4-Br                                                                               0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     4-Br                                                                               0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  Cl  OCH.sub.3                                                                           CH                                     4-Br                                                                               0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      4-Br                                                                               0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      4-Br                                                                               0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     4-Br                                                                               0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     4-Br                                                                               0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           CH.sub.3                                                                            CH                                     4-Br                                                                               0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  Cl  OCH.sub.3                                                                           CH                                     4-Br                                                                               0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  OCH.sub.3                                                                          OCH.sub.3                                                                           N                                      4-Br                                                                               0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    H  CH.sub.3                                                                           OCH.sub.3                                                                           N                                      H   0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- S    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- 0    CH.sub.3                                                                          CH.sub.3                                                                           OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- NCH.sub.3                                                                           H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- S    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- NOCH.sub.3                                                                          H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     H   0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O    CH.sub.3                                                                          CH.sub.3                                                                           CH.sub.3                                                                            CH                                     H   0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          S    H  OCH.sub.3                                                                          OCH.sub.3                                                                           CH                                     __________________________________________________________________________

                                      TABLE IX                                     __________________________________________________________________________     General Structure 9                                                            R.sub.1 n E Q  R.sub.3                                                                           R.sub.4                                                                              R.sub.5                                                                           W  R  X   Y   Z  m.p. (°C.)                  __________________________________________________________________________     H       0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    H       0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                    H       0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  Cl  OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O  H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                    H       0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O  H  Cl  OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    H       0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                    H       0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  Cl  OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    H       0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                     H       0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    H       0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O  H  Cl  OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O  H  Cl  OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    H       0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O  H  Cl  OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O  H  Cl  OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    H       0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O  H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                    H       0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N -H 0 -- Q-3 -- CH(CH.sub.3).sub                                              .2 -- O H CH.sub.3 OCH.sub.3 CH       H       0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O  H  Cl  OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O  H  Cl  OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    H       0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O  H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                     H       0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O  H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                     H       0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O  H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                    H       0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O  H  Cl  OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    H       0 --                                                                               Q-5                                                                               -- --    CH.sub. 3                                                                         O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    H       0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O  H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                    H       0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O  H  Cl  OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     4-CH.sub.3                                                                             0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    4-CH.sub.3                                                                             0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    4-CH.sub.3                                                                             0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    4-CH.sub.3                                                                             0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  Cl  OCH.sub.3                                                                          CH                                    4-CH.sub.3                                                                             0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     4-Br    0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    4-Br    0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    4-Br    0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    4-Br    0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  Cl  OCH.sub.3                                                                          CH                                    4-Cl    0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     4-Cl    0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    4-Cl    0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    4-Cl    0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  Cl  OCH.sub.3                                                                          CH                                    4-Cl    0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    4-CH.sub.3                                                                             0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    4-CH.sub.3                                                                             0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    4-CH.sub.3                                                                             0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    4-CH.sub.3                                                                             0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  Cl  OCH.sub.3                                                                          CH                                    4-CH.sub.3                                                                             0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O  H  Cl  OCH.sub.3                                                                          CH                                    4-CH.sub.3                                                                             0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    4-CH.sub.3                                                                             0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    4-CH.sub.3                                                                             0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    H       0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           N                                     H       0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    H       0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O  H  Cl  OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    H       0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    H       0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O  H  Cl  OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    H       0 --                                                                               Q-3                                                                               -- OC.sub. 2 H.sub.5                                                                    -- O  H  Cl  OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O  H  Cl  OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-6                                                                               -- --    CH.sub.3                                                                          O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-6                                                                               -- --    CH.sub.3                                                                          O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-6                                                                               -- --    CH.sub.3                                                                          O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    H       0 --                                                                               Q-6                                                                               -- --    CH.sub.3                                                                          O  H  Cl  OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-6                                                                               -- --    CH.sub.3                                                                          O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-6                                                                               -- --    CH.sub.3                                                                          O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-7                                                                               -- --    CH.sub.3                                                                          O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-7                                                                               -- --    CH.sub.3                                                                          O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-7                                                                               -- --    CH.sub.3                                                                          O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    H       0 --                                                                               Q-7                                                                               -- --    CH.sub.3                                                                          O  H  Cl  OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-7                                                                               -- --    CH.sub.3                                                                          O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-7                                                                               -- --    CH.sub.3                                                                          O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     4-CH.sub.3                                                                             0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     4-CH.sub.3                                                                             0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     4-CH.sub.3                                                                             0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     4-CH.sub.3                                                                             0 --                                                                               Q-3                                                                               -- H     -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    4-CH.sub.3                                                                             0 --                                                                               Q-3                                                                               -- H     -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    4-CH.sub.3                                                                             0 --                                                                               Q-3                                                                               -- H     -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    4-CH.sub.3                                                                             0 --                                                                               Q-3                                                                               -- H     -- O  H  Cl  OCH.sub.3                                                                          CH                                    4-CH.sub.3                                                                             0 --                                                                               Q-3                                                                               -- H     -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     4-CH.sub.3                                                                             0 --                                                                               Q-3                                                                               -- H     -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     4-CH.sub.3                                                                             0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    4-CH.sub.3                                                                             0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    4-CH.sub.3                                                                             0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    4-CH.sub.3                                                                             0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O  H  Cl  OCH.sub.3                                                                          CH                                    4-CH.sub. 3                                                                            0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     4-CH.sub.3                                                                             0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     4-Cl    0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     4-Cl    0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    4-Cl    0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    4-Cl    0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    4-Cl    0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  Cl  OCH.sub.3                                                                          CH                                    4-Cl    0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     4-Cl    0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     4-Cl    0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    4-Cl    0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    4-Cl    0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    4-Cl    0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O  H  Cl  OCH.sub.3                                                                          CH                                    4-Cl    0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     4-Cl    0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     4-Cl    0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    4-Cl    0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    4-Cl    0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    4-Cl    0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O  H  Cl  OCH.sub.3                                                                          CH                                    4-Cl    0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     4-Cl    0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     4-Br    0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    4-Br    0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     4-Br    0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    4-Br    0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    4-Br    0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    4-Br    0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  Cl  OCH.sub.3                                                                          CH                                    4-Br    0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     4-Br    0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     4-Br    0 --                                                                               Q-3                                                                               -- H     -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    4-Br    0 --                                                                               Q-3                                                                               -- H     -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    4-Br    0 --                                                                               Q-3                                                                               -- H     -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    4-Br    0 --                                                                               Q-3                                                                               -- H     -- O  H  Cl  OCH.sub.3                                                                          CH                                    4-Br    0 --                                                                               Q-3                                                                               -- H     -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     4-Br    0 --                                                                               Q-3                                                                               -- H     -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     4-Br    0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    4-Br    0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    4-Br    0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    4-Br    0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O  H  Cl  OCH.sub.3                                                                          CH                                    4-Br    0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     4-Br    0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     4-SCH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    4-SCH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    4-SCH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     4-SCH.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  Cl  OCH.sub. 3                                                                         CH                                    4-SCH.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    4-SCH.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     4-SOCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  Cl  OCH.sub.3                                                                          CH                                    4-SOCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    4-SOCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     4-SOCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    4-SOCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    4-SOCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     4-SO.sub.2 CH.sub.3                                                                    0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    4-SO.sub.2 CH.sub.3                                                                    0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  Cl  OCH.sub.3                                                                          CH                                    4-SO.sub.2 CH.sub.3                                                                    0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     4-SO.sub.2 CH.sub.3                                                                    0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    4-SO.sub.2 CH.sub.3                                                                    0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    4-SO.sub.2 CH.sub.3                                                                    0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     4-SO.sub.2 N(CH.sub.3).sub.2                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    4-SO.sub.2 N(CH.sub.3).sub.2                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    4-SO.sub.2 N(CH.sub.3).sub.2                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     4-SO.sub.2 N(CH.sub.3).sub.2                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    4-SO.sub.2 N(CH.sub.3).sub.2                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  Cl  OCH.sub.3                                                                          CH                                    4-SO.sub.2 N(CH.sub.3).sub.2                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     H       0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- S  H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  CH.sub.3                                                                          OCH.sub.3                                                                          CH.sub.3                                                                           CH                                    H       0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- S  H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    H       0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O  CH.sub.3                                                                          Cl  OCH.sub.3                                                                          CH                                    H       0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          NH H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H       1 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O  H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H       1 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O  H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    __________________________________________________________________________

                                      TABLE X                                      __________________________________________________________________________     General Structure 10                                                           R.sub.1                                                                           n E Q  R.sub.3                                                                           R.sub.4                                                                              R.sub.5                                                                           W     R  X   Y   Z  m.p. (°C.)                    __________________________________________________________________________     H  0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- 0     H  Cl  OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O     H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O     H  Cl  OCH.sub. 3                                                                         CH                                      H  0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  Cl  OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                       H  0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O     H  Cl  OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O     H  Cl  OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O     H  Cl  OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O     H  Cl  OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O     H  OCH.sub. 3                                                                         CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O     H  Cl  OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  Cl  CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O     H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                       H  0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O     H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                       H  0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O     H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O     Cl OCH.sub.3                                                                          CH                                          H  0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O     H  Cl  OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --f   -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- H     -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- H     -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- H     -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-3                                                                               -- H     -- O     H  Cl  OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- H     -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- H     -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O     H  Cl  OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O     H  CH.sub.3                                                                           CH.sub.                                                                            CH                                      H  0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O     H  Cl  OCH.sub. 3                                                                         CH                                      H  0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O     H  Cl  OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O     H  Cl  OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O     H  OCH.sub.3                                                                          OCH.sub.3                                   H  0 --                                                                               Q-4                                                                               -- C.sub.2 H.sub.5                                                                      -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-4                                                                               -- C.sub.2 H.sub.5                                                                      -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-4                                                                               -- C.sub.2 H.sub.5                                                                      -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      H  0 --                                                                               Q-4                                                                               -- C.sub.2 H.sub.5                                                                      -- O     H  Cl  OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-4                                                                               -- C.sub.2 H.sub.5                                                                      -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-4                                                                               -- C.sub.2 H.sub.5                                                                      -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       2-Cl                                                                              0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      2-Cl                                                                              0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      2-Cl                                                                              0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      2-Cl                                                                              0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  Cl  OCH.sub.3                                                                          CH                                      2-Cl                                                                              0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       2-Cl                                                                              0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       2-Cl                                                                              0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      2-Cl                                                                              0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      2-Cl                                                                              0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      2-Cl                                                                              0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  Cl  OCH.sub.3                                                                          CH                                      2-Cl                                                                              0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       2-Cl                                                                              0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       2-Cl                                                                              0 --                                                                               Q-3                                                                               -- H     -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      2-Cl                                                                              0 --                                                                               Q-3                                                                               -- H     -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      2-Cl                                                                              0 --                                                                               Q-3                                                                               -- H     -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      2-Cl                                                                              0 --                                                                               Q-3                                                                               -- H     -- O     H  Cl  OCH.sub.3                                                                          CH                                      2-Cl                                                                              0 --                                                                               Q-3                                                                               -- H     -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       2-Cl                                                                              0 --                                                                               Q-3                                                                               -- H     -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       2-Cl                                                                              0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      2-Cl                                                                              0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      2-Cl                                                                              0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      2-Cl                                                                              0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  Cl  OCH.sub.3                                                                          CH                                      2-Cl                                                                              0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       2-Cl                                                                              0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       2-Br                                                                              0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      2-Br                                                                              0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      2-Br                                                                              0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      2-Br                                                                              0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  Cl  OCH.sub.3                                                                          CH                                      2-Br                                                                              0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       2-Br                                                                              0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       2-Br                                                                              0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      2-Br                                                                              0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      2-Br                                                                              0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      2-Br                                                                              0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  Cl  OCH.sub.3                                                                          CH                                      2-Br                                                                              0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       2-Br                                                                              0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       2-Br                                                                              0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      2-Br                                                                              0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      2-Br                                                                              0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      2-Br                                                                              0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  Cl  OCH.sub.3                                                                          CH                                      2-Br                                                                              0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                       2-Br                                                                              0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O     H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                       H  0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --       S     H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --       O     CH.sub.3                                                                          CH.sub.3                                                                           OCH.sub.3                                                                          CH                                      H  0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- NNHCH.sub.3                                                                          H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                      H  1 --                                                                               Q-3                                                                               -- H     -- O     H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                      __________________________________________________________________________

                                      TABLE XI                                     __________________________________________________________________________     General Structure 11                                                           R.sub.1                                                                             n E  Q  R.sub.2                                                                              R.sub.3                                                                              R.sub.4                                                                              R.sub.5                                                                           W R  X   Y   Z  m.p. (° C.)           __________________________________________________________________________     H    O -- Q-1                                                                               C.sub.6 H.sub.5                                                                      CH.sub.3                                                                             --    H  0 H  CH.sub.3                                                                           CH.sub.3                                                                           CH                              H    0 -- Q-1                                                                               C.sub.6 H.sub.5                                                                      CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                              H    0 -- Q-1                                                                               C.sub.6 H.sub.5                                                                      CH.sub.3                                                                             --    -- O H  Cl  OCH.sub.3                                                                          CH                              H    0 -- Q-1                                                                               C.sub.6 H.sub.5                                                                      CH.sub.3                                                                             --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                               H    0 -- Q-1                                                                               C.sub.6 H.sub.5                                                                      CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                               H    0 -- Q-1                                                                               C.sub.6 H.sub.5                                                                      C.sub.2 H.sub.5                                                                      --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                              H    0 -- Q-1                                                                               C.sub.6 H.sub.5                                                                      C.sub. 2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              H    0 -- Q-1                                                                               C.sub.6 H.sub.5                                                                      C.sub.2 H.sub.5                                                                      --    -- O H  Cl  OCH.sub.3                                                                          CH                              H    0 -- Q-1                                                                               C.sub.6 H.sub.5                                                                      C.sub.2 H.sub.5                                                                      --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                              H    0 -- Q-1                                                                               C.sub.6 H.sub.5                                                                      C.sub.2 H.sub.5                                                                      --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                               H    0 -- Q-2                                                                               C.sub.6 H.sub.5                                                                      CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                               H    0 -- Q-2                                                                               C.sub.6 H.sub.5                                                                      CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              H    0 -- Q-2                                                                               C.sub.6 H.sub.5                                                                      CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                              H    0 -- Q-2                                                                               C.sub.6 H.sub.5                                                                      CH.sub.3                                                                             --    -- O H  Cl  OCH.sub.3                                                                          CH                              H    0 -- Q-2                                                                               C.sub.6 H.sub.5                                                                      CH.sub.3                                                                             --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                              H    0 -- Q-2                                                                               C.sub. 6 H.sub.5                                                                     CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                               H    0 -- Q-2                                                                               C.sub.6 H.sub.5                                                                      C.sub.2 H.sub.5                                                                      --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                               H    0 -- Q-2                                                                               C.sub.6 H.sub.5                                                                      C.sub.2 H.sub.5                                                                      --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                              H    0 -- Q-2                                                                               C.sub.6 H.sub.5                                                                      C.sub.2 H.sub.5                                                                      --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                              H    0 -- Q-2                                                                               C.sub.6 H.sub.5                                                                      C.sub.2 H.sub.5                                                                      --    -- O H  Cl  OCH.sub.3                                                                          CH                              H    0 -- Q-2                                                                               C.sub.6 H.sub.5                                                                      C.sub.2 H.sub.5                                                                      --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                               H    0 -- Q-2                                                                               C.sub.6 H.sub.5                                                                      C.sub.2 H.sub.5                                                                      --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                               H    0 -- Q-3                                                                               C.sub.6 H.sub.5                                                                      --    CH.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                              H    0 -- Q-3                                                                               C.sub.6 H.sub.5                                                                      --    CH.sub.3                                                                             -- O H  Cl  OCH.sub. 3                                                                         CH                              H    0 -- Q-3                                                                               C.sub.6 H.sub.5                                                                      --    CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              H    0 -- Q-3                                                                               C.sub.6 H.sub.5                                                                      --    CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                               H    0 -- Q-3                                                                               C.sub.6 H.sub.5                                                                      --    CH.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                               H    0 -- Q-3                                                                               C.sub.6 H.sub.5                                                                      --    C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                              H    0 -- Q-3                                                                               C.sub.6 H.sub.5                                                                      --    C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                              H    0 -- Q-3                                                                               C.sub.6 H.sub.5                                                                      --    C.sub.2 H.sub.5                                                                      -- O H  Cl  OCH.sub.3                                                                          CH                              H    0 -- Q-3                                                                               C.sub.6 H.sub.5                                                                      --    C.sub.2 H.sub.5                                                                      -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              H    0 -- Q-3                                                                               C.sub.6 H.sub.5                                                                      --    C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                               H    0 -- Q-3                                                                               C.sub.6 H.sub.5                                                                      --    CH.sub.2 Cl                                                                          -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                              H    0 -- Q-3                                                                               C.sub.6 H.sub.5                                                                      --    CH.sub.2 Cl                                                                          -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              H    0 -- Q-3                                                                               C.sub.6 H.sub.5                                                                      --    CH.sub.2 Cl                                                                          -- O H  Cl  OCH.sub.3                                                                          CH                              H    0 -- Q-3                                                                               C.sub.6 H.sub.5                                                                      --    CH.sub.2 Cl                                                                          -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                               H    0 -- Q-3                                                                               C.sub.6 H.sub.5                                                                      --    CH.sub.2 Cl                                                                          -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                               H    0 -- Q-3                                                                               C.sub.6 H.sub.5                                                                      --    CF.sub.3                                                                             -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                              H    0 -- Q-3                                                                               C.sub.6 H.sub.5                                                                      --    CF.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              H    0 -- Q-3                                                                               C.sub.6 H.sub.5                                                                      --    CF.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                              H    0 -- Q-3                                                                               C.sub.6 H.sub.5                                                                      --    CF.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                               H    0 -- Q-3                                                                               C.sub.6 H.sub.5                                                                      --    CH(CH.sub.3).sub.2                                                                   -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                              H    0 -- Q-3                                                                               C.sub.6 H.sub.5                                                                      --    CH(CH.sub.3).sub.2                                                                   -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              H    0 -- Q-3                                                                               C.sub.6 H.sub.5                                                                      --    CH(CH.sub.3).sub.2                                                                   -- O H  Cl  OCH.sub.3                                                                          CH                              H    0 -- Q-3                                                                               C.sub.6 H.sub.5                                                                      --    CH(CH.sub.3).sub.2                                                                   -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                               H    0 -- Q-3                                                                               C.sub.6 H.sub.5                                                                      --    OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              H    0 -- Q-3                                                                               C.sub.6 H.sub.5                                                                      --    OCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                              H    0 -- Q-3                                                                               C.sub.6 H.sub.5                                                                      --    OCH.sub.3                                                                            -- O H  Cl  CH.sub.3                                                                           CH                              H    0 -- Q-3                                                                               C.sub.6 H.sub.5                                                                      --    OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                               H    0 -- Q-3                                                                               C.sub.6 H.sub.5                                                                      --    SCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                              H    0 -- Q-3                                                                               C.sub.6 H.sub.5                                                                      --    SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              H    0 -- Q-3                                                                               C.sub.6 H.sub.5                                                                      --    SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                               H    0 -- Q-3                                                                               C.sub.6 H.sub.5                                                                      --    SCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                               H    0 -- Q-3                                                                               C.sub.6 H.sub.5                                                                      --    N(CH.sub.3).sub.2                                                                    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                              H    0 -- Q-3                                                                               C.sub.6 H.sub.5                                                                      --    N(CH.sub.3).sub.2                                                                    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              H    0 -- Q-3                                                                               C.sub.6 H.sub.5                                                                      --    N(CH.sub.3).sub.2                                                                    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                               H    0 -- Q-5                                                                               C.sub.6 H.sub.5                                                                      --    --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                               H    0 -- Q-5                                                                               C.sub.6 H.sub.5                                                                      --    --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                              H    0 -- Q-5                                                                               C.sub.6 H.sub.5                                                                      --    --    CH.sub.3                                                                          O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                              H    0 -- Q-5                                                                               C.sub.6 H.sub.5                                                                      --    --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              H    0 -- Q-5                                                                               C.sub.6 H.sub.5                                                                      --    --    CH.sub.3                                                                          O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                              H    0 -- Q-1                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                              H    0 -- Q-1                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                              H    0 -- Q-1                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  Cl  OCH.sub.3                                                                          CH                              H    0 -- Q-1                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                               H    0 -- Q-1                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                               H    0 -- Q-1                                                                               CH.sub.3                                                                             C.sub.2 H.sub.5                                                                      --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                              H    0 -- Q-1                                                                               CH.sub.3                                                                             C.sub.2 H.sub.5                                                                      --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              H    0 -- Q-1                                                                               CH.sub.3                                                                             C.sub.2 H.sub.5                                                                      --    -- O H  Cl  OCH.sub.3                                                                          CH                              H    0 -- Q-1                                                                               CH.sub.3                                                                             C.sub.2 H.sub.5                                                                      --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                              H    0 -- Q-1                                                                               CH.sub.3                                                                             C.sub.2 H.sub.5                                                                      --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                               H    0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                               H    0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              H    0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                              H    0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  Cl  OCH.sub.3                                                                          CH                              H    0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                              H    0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                               H    0 -- Q-2                                                                               CH.sub.3                                                                             C.sub.2 H.sub.5                                                                      --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                               H    0 -- Q-2                                                                               CH.sub.3                                                                             C.sub.2 H.sub. 5                                                                     --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                              H    0 -- Q-2                                                                               CH.sub.3                                                                             C.sub.2 H.sub.5                                                                      --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                              H    0 -- Q-2                                                                               CH.sub.3                                                                             C.sub.2 H.sub.5                                                                      --    -- O H  Cl  OCH.sub.3                                                                          CH                              H    0 -- Q-2                                                                               CH.sub.3                                                                             C.sub.2 H.sub.5                                                                      --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                               H    0 -- Q-2                                                                               CH.sub.3                                                                             C.sub.2 H.sub.5                                                                      --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                               H    0 -- Q-3                                                                               CH.sub.3                                                                             --    CH.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                              H    0 -- Q-3                                                                               CH.sub.3                                                                             --    CH.sub.3                                                                             -- O H  Cl  OCH.sub.3                                                                          CH                              H    0 -- Q-3                                                                               CH.sub.3                                                                             --    CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              H    0 -- Q-3                                                                               CH.sub.3                                                                             --    CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                               H    0 -- Q-3                                                                               CH.sub.3                                                                             --    CH.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                               H    0 -- Q-3                                                                               CH.sub.3                                                                             --    C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                              H    0 -- Q-3                                                                               CH.sub.3                                                                             --    C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                              H    0 -- Q-3                                                                               CH.sub.3                                                                             --    C.sub.2 H.sub.5                                                                      -- O H  Cl  OCH.sub.3                                                                          CH                              H    0 -- Q-3                                                                               CH.sub.3                                                                             --    C.sub.2 H.sub.5                                                                      -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              H    0 -- Q-3                                                                               CH.sub.3                                                                             --    C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                               H    0 -- Q-3                                                                               CH.sub.3                                                                             --    CH.sub.2 Cl                                                                          -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                              H    0 -- Q-3                                                                               CH.sub.3                                                                             --    CH.sub.2 Cl                                                                          -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              H    0 -- Q-3                                                                               CH.sub.3                                                                             --    CH.sub.2 Cl                                                                          -- O H  Cl  OCH.sub.3                                                                          CH                              H    0 -- Q-3                                                                               CH.sub.3                                                                             --    CH.sub.2 Cl                                                                          -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                               H    0 -- Q-3                                                                               CH.sub.3                                                                             --    CH.sub. 2 Cl                                                                         -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                               H    0 -- Q-3                                                                               CH.sub.3                                                                             --    CF.sub.3                                                                             -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                              H    0 -- Q-3                                                                               CH.sub.3                                                                             --    CF.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              H    0 -- Q-3                                                                               CH.sub.3                                                                             --    CF.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                              H    0 -- Q-3                                                                               CH.sub.3                                                                             --    CF.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                               H    0 -- Q-3                                                                               CH.sub.3                                                                             --    CH(CH.sub.3).sub.2                                                                   -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                              H    0 -- Q-3                                                                               CH.sub.3                                                                             --    CH(CH.sub.3).sub.2                                                                   -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              H    0 -- Q-3                                                                               CH.sub.3                                                                             --    CH(CH.sub.3).sub.2                                                                   -- O H  Cl  OCH.sub.3                                                                          CH                              H    0 -- Q-3                                                                               CH.sub.3                                                                             --    CH(CH.sub.3).sub.2                                                                   -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                               H    0 -- Q-3                                                                               CH.sub.3                                                                             --    OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              H    0 -- Q-3                                                                               CH.sub.3                                                                             --    OCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                              H    0 -- Q-3                                                                               CH.sub.3                                                                             --    OCH.sub.3                                                                            -- O H  Cl  CH.sub.3                                                                           CH                              H    0 -- Q-3                                                                               CH.sub.3                                                                             --    OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                               H    0 -- Q-3                                                                               CH.sub.3                                                                             --    SCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                              H    0 -- Q-3                                                                               CH.sub.3                                                                             --    SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              H    0 -- Q-3                                                                               CH.sub.3                                                                             --    SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                               H    0 -- Q-3                                                                               CH.sub.3                                                                             --    SCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                               H    0 -- Q-3                                                                               CH.sub.3                                                                             --    N(CH.sub.3).sub.2                                                                    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                              H    0 -- Q-3                                                                               CH.sub.3                                                                             --    N(CH.sub.3).sub.2                                                                    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              H    0 -- Q-3                                                                               CH.sub.3                                                                             --    N(CH.sub.3).sub.2                                                                    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                               H    0 -- Q-5                                                                               CH.sub.3                                                                             --    --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                               Cl   0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                              Cl   0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                              Cl   0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              Cl   0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  Cl  OCH.sub.3                                                                          CH                              Cl   0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                               Cl   0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                               Cl   0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O CH.sub.3                                                                          OCH.sub.3                                                                          CH.sub.3                                                                           N                               Cl   0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.2 CH.sub.3                                                                    --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                              Cl   0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.2 CH.sub.3                                                                    --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                              Cl   0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.2 CH.sub.3                                                                    --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              Cl   0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.2 CH.sub.3                                                                    --    -- O H  Cl  OCH.sub.3                                                                          CH                              Cl   0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.2 CH.sub.3                                                                    --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                               Cl   0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.2 CH.sub.3                                                                    --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                               H    0 -- Q-2                                                                               CH.sub.2 CH.sub.3                                                                    CH.sub.3                                                                             --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                              H    0 -- Q-2                                                                               CH.sub.2 CH.sub.3                                                                    CH.sub.3                                                                             --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                              H    0 -- Q-2                                                                               CH.sub.2 CH.sub.3                                                                    CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              H    0 -- Q-2                                                                               CH.sub.2 CH.sub.3                                                                    CH.sub.3                                                                             --    -- O H  Cl  OCH.sub.3                                                                          CH                              H    0 -- Q-2                                                                               CH.sub.2 CH.sub.3                                                                    CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                               H    0 -- Q-2                                                                               CH.sub.2 CH.sub.3                                                                    CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                               Cl   0 -- Q-1                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                              Cl   0 -- Q-1                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              Cl   0 -- Q-1                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                               Cl   0 -- Q-1                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                               Cl   0 -- Q-3                                                                               CH.sub.3                                                                             --    CH.sub.3                                                                             -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                              Cl   0 -- Q-3                                                                               CH.sub.3                                                                             --    CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                              Cl   0 -- Q-3                                                                               CH.sub.3                                                                             --    CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              Cl   0 -- Q-3                                                                               CH.sub.3                                                                             --    CH.sub.3                                                                             -- O H  Cl  OCH.sub.3                                                                          CH                              Cl   0 -- Q-3                                                                               CH.sub.3                                                                             --    CH.sub.3                                                                             -- O H  OCH.sub. 3                                                                         CH.sub.3                                                                           N                               Cl   0 -- Q-3                                                                               CH.sub.3                                                                             --    CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                               Br   0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                              Br   0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              Br   0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  Cl  OCH.sub.3                                                                          CH                              Br   0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                               Br   0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                               Br   0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.2 CH.sub.3                                                                    --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                              Br   0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.2 CH.sub.3                                                                    --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              Br   0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.2 CH.sub.3                                                                    --    -- O H  Cl  OCH.sub.3                                                                          CH                              Br   0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.2 CH.sub.3                                                                    --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                               Br   0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.2 CH.sub.3                                                                    --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                               Br   0 -- Q-1                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                              Br   0 -- Q-1                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              Br   0 -- Q-1                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                               Br   0 -- Q-1                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                               Br   0 -- Q-4                                                                               CH.sub.3                                                                             --    CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                              Br   0 -- Q-4                                                                               CH.sub.3                                                                             --    CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              Br   0 -- Q-4                                                                               CH.sub.3                                                                             --    CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                               Br   0 -- Q-4                                                                               CH.sub.3                                                                             --    CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                               F    0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub. 3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                              F    0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              F    0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                               F    0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                               F    0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  Cl  OCH.sub.3                                                                          CH                              F    0 -- Q-1                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                              F    0 -- Q-1                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              F    0 -- Q-1                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                               F    0 -- Q-1                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                               F    0 -- Q-3                                                                               CH.sub.3                                                                             --    CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                              F    0 -- Q-3                                                                               CH.sub.3                                                                             --    CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              F    0 -- Q-3                                                                               CH.sub.3                                                                             --    CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                               F    0 -- Q-3                                                                               CH.sub.3                                                                             --    CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                               OCH.sub.3                                                                           0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                              OCH.sub.3                                                                           0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              OCH.sub.3                                                                           0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  Cl  OCH.sub.3                                                                          CH                              OCH.sub.3                                                                           0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                               OCH.sub.3                                                                           0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                               OCH.sub.3                                                                           0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.2 CH.sub.3                                                                    --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                              OCH.sub.3                                                                           0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.2 CH.sub.3                                                                    --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              OCH.sub.3                                                                           0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.2 CH.sub.3                                                                    --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                               OCH.sub.3                                                                           0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.2 CH.sub.3                                                                    --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                               OCH.sub.3                                                                           0 -- Q-1                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                              OCH.sub.3                                                                           0 -- Q-1                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              OCH.sub.3                                                                           0 -- Q-1                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                               OCH.sub.3                                                                           0 -- Q-1                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                              OCH.sub.3                                                                           0 -- Q-1                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  Cl  OCH.sub.3                                                                          CH                              OCH.sub.3                                                                           0 -- Q-1                                                                               CH.sub.3                                                                             CH.sub.2 CH.sub.3                                                                    --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              OCH.sub.3                                                                           0 -- Q-1                                                                               CH.sub.3                                                                             CH.sub.2 CH.sub.3                                                                    --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                              OCH.sub.3                                                                           0 -- Q-1                                                                               CH.sub.3                                                                             CH.sub.2 CH.sub.3                                                                    --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                               OCH.sub.3                                                                           0 -- Q-3                                                                               CH.sub.3                                                                             --    CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              OCH.sub.3                                                                           0 -- Q-3                                                                               CH.sub.3                                                                             --    CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                              OCH.sub.3                                                                           0 -- Q-3                                                                               CH.sub.3                                                                             --    CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                               OCH.sub.3                                                                           0 -- Q-3                                                                               CH.sub.3                                                                             --    CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                               OCH.sub.3                                                                           0 -- Q-3                                                                               CH.sub.3                                                                             --    CH.sub.3                                                                             -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                              CF.sub.3                                                                            0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                              CF.sub.3                                                                            0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                               CF.sub.3                                                                            0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                               CF.sub.3                                                                            0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              CF.sub.3                                                                            0 -- Q-1                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                              CF.sub.3                                                                            0 -- Q-1                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              CF.sub.3                                                                            0 -- Q-1                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                               CF.sub.3                                                                            0 -- Q-1                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                               CF.sub.3                                                                            0 -- Q-3                                                                               CH.sub.3                                                                             --    CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                              CF.sub.3                                                                            0 -- Q-3                                                                               CH.sub.3                                                                             --    CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              CF.sub.3                                                                            0 -- Q-3                                                                               CH.sub.3                                                                             --    CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                               CF.sub.3                                                                            0 -- Q-3                                                                               CH.sub.3                                                                             --    CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                               OCF.sub.2 H                                                                         0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                              OCF.sub. 2 H                                                                        0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              OCF.sub.2 H                                                                         0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                               Cl   0 -- Q-3                                                                               CH.sub.3                                                                             --    OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                              Cl   0 -- Q-3                                                                               CH.sub.3                                                                             --    OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              Cl   0 -- Q-3                                                                               CH.sub.3                                                                             --    OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                               Cl   0 -- Q-3                                                                               CH.sub.3                                                                             --    OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                               Br   0 -- Q-3                                                                               CH.sub.3                                                                             --    OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                              Br   0 -- Q-3                                                                               CH.sub.3                                                                             --    OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              Br   0 -- Q-3                                                                               CH.sub.3                                                                             --    OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                               F    0 -- Q-3                                                                               CH.sub.3                                                                             --    OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                               F    0 -- Q-3                                                                               CH.sub.3                                                                             --    OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              F    0 -- Q-3                                                                               CH.sub.3                                                                             --    OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                              OCH.sub.3                                                                           0 -- Q-3                                                                               CH.sub.3                                                                             --    OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                              OCH.sub.3                                                                           0 -- Q-3                                                                               CH.sub.3                                                                             --    OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              OCH.sub.3                                                                           0 -- Q-3                                                                               CH.sub.3                                                                             --    OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                               OCH.sub.3                                                                           0 -- Q-3                                                                               CH.sub.3                                                                             --    OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                               CF.sub.3                                                                            0 -- Q-3                                                                               CH.sub.3                                                                             --    OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                              CF.sub.3                                                                            0 -- Q-3                                                                               CH.sub.3                                                                             --    OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              CF.sub.3                                                                            0 -- Q-3                                                                               CH.sub.3                                                                             --    OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                               CF.sub.3                                                                            0 -- Q-3                                                                               CH.sub.3                                                                             --    OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                               Cl   0 -- Q-3                                                                               CH.sub.3                                                                             --    SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                              Cl   0 -- Q-3                                                                               CH.sub.3                                                                             --    SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              Cl   0 -- Q-3                                                                               CH.sub.3                                                                             --    SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                               Br   0 -- Q-3                                                                               CH.sub.3                                                                             --    SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              Br   0 -- Q-3                                                                               CH.sub.3                                                                             --    SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                              F    0 -- Q-3                                                                               CH.sub.3                                                                             --    SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                               F    0 -- Q-3                                                                               CH.sub.3                                                                             --    SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                              OCH.sub.3                                                                           0 -- Q-3                                                                               CH.sub.3                                                                             --    SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                               OCH.sub.3                                                                           0 -- Q-3                                                                               CH.sub.3                                                                             --    SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                              OCH.sub.3                                                                           0 -- Q-3                                                                               CH.sub. 3                                                                            --    SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              CH.sub.3                                                                            0 -- Q-1                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                              CH.sub.3                                                                            0 -- Q-1                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                              CH.sub.3                                                                            0 -- Q-1                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              CH.sub.3                                                                            0 -- Q-1                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  Cl  OCH.sub.3                                                                          CH                              CH.sub.3                                                                            0 -- Q-1                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                               CH.sub.3                                                                            0 -- Q-1                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                               CH.sub.3                                                                            0 -- Q-3                                                                               CH.sub.3                                                                             --    OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                              CH.sub.3                                                                            0 -- Q-3                                                                               CH.sub.3                                                                             --    OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              CH.sub.3                                                                            0 -- Q-3                                                                               CH.sub.3                                                                             --    OCH.sub.3                                                                            -- O H  Cl  OCH.sub.3                                                                          CH                              CH.sub.3                                                                            0 -- Q-3                                                                               CH.sub.3                                                                             --    OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                               CH.sub.3                                                                            0 -- Q-3                                                                               CH.sub.3                                                                             --    OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                               Cl   0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O CH.sub.3                                                                          OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              Br   0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O CH.sub.3                                                                          OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              F    0 -- Q-2                                                                               CH.sub.3                                                                             CH.sub.3                                                                             --    -- O CH.sub.3                                                                          OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              Cl   0 -- Q-5                                                                               CH.sub.3                                                                             --    --    CH.sub.3                                                                          O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                              Cl   0 -- Q-5                                                                               CH.sub.3                                                                             --    --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              Br   0 -- Q-5                                                                               CH.sub.3                                                                             --    --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                              Br   0 -- Q-5                                                                               CH.sub.3                                                                             --    --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              F    0 -- Q-5                                                                               CH.sub.3                                                                             --    --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              F    0 -- Q-5                                                                               CH.sub.3                                                                             --    --    CH.sub.3                                                                          O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                              OCH.sub.3                                                                           0 -- Q-5                                                                               CH.sub.3                                                                             --    --    CH.sub.3                                                                          O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                              OCH.sub.3                                                                           0 -- Q-5                                                                               CH.sub.3                                                                             --    --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                              OCH.sub.3                                                                           0 -- Q-5                                                                               CH.sub.3                                                                             --    --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                               Cl   0 -- Q-5                                                                               CH.sub.3                                                                             --    --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                               Cl   0 -- Q-5                                                                               CH.sub.3                                                                             --    --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                               __________________________________________________________________________

                                      TABLE XII                                    __________________________________________________________________________     General Structure 12                                                           R.sub.1                                                                            n E Q  R.sub.2                                                                             R.sub.3                                                                             R.sub.4                                                                              R.sub.5                                                                           W R  X   Y   Z  m.p. (°C.)                __________________________________________________________________________     H   0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                  H   0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                  H   0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                  H   0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                   H   0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                   H   0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                  H   0 --                                                                               Q-1                                                                               C.sub.6 H.sub. 5                                                                    C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  H   0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  Cl  OCH.sub.3                                                                          CH                                  H   0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                  H   0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                   H   0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                   H   0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH 232-233                          H   0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH 193-195                          H   0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH 195-198                          H   0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub. 3                                                                          CH 165-170                          H   0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N  140-145                          H   0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N  195-196                          H   0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                  H   0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                  H   0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  Cl  OCH.sub.3                                                                          CH                                  H   0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                   H   0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                   H   0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                  H   0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  Cl  OCH.sub.3                                                                          CH                                  H   0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  H   0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                   H   0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                   H   0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                  H   0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                  H   0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  Cl  OCH.sub.3                                                                          CH                                  H   0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  H   0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                   H   0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                  H   0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  H   0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  Cl  OCH.sub.3                                                                          CH                                  H   0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                   H   0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                   H   0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CF.sub.3                                                                             -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                  H   0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CF.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  H   0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CF.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                  H   0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CF.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                   H   0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH(CH.sub.3).sub.2                                                                   -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                  H   0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH(CH.sub.3).sub.2                                                                   -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  H   0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH(CH.sub.3).sub.2                                                                   -- O H  Cl  OCH.sub.3                                                                          CH                                  H   0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH(CH.sub.3).sub.2                                                                   -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                   H   0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  H   0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   OCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                  H   0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   OCH.sub.3                                                                            -- O H  Cl  CH.sub.3                                                                           CH                                  H   0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                   H   0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   SCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                  H   0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  H   0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                   H   0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   SCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                   H   0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   N(CH.sub.3).sub.2                                                                    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                  H   0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   N(CH.sub.3).sub.2                                                                    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  H   0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   N(CH.sub.3).sub.2                                                                    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                   H   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH 165-167                          H   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH 125-127                          H   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH 189-191                          H   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N  166-170                          H   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N  160-172                          H   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                  H   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  H   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  Cl  OCH.sub.3                                                                          CH                                  H   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                  H   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                   H   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N  180-183                          H   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH 171-173                          H   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH 181-183                          H   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH 178-180                          H   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH 200-202                          H   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N  179-180                          H   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH 195                              H   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH 172-173                          H   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH 152-156                          H   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  Cl  OCH.sub.3                                                                          CH 170-171                          H   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N  173-174                          H   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N  168-170                          H   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                  H   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  Cl  OCH.sub.3                                                                          CH                                  H   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  H   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                   H   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                   H   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                  H   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                  H   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   C.sub.2 H.sub.5                                                                      -- O H  Cl  OCH.sub.3                                                                          CH                                  H   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   C.sub.2 H.sub.5                                                                      -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  H   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                   H   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.2 Cl                                                                          -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                  H   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.2 Cl                                                                          -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  H   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.2 Cl                                                                          -- O H  Cl  OCH.sub.3                                                                          CH                                  H   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.2 Cl                                                                          -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                   H   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.2 Cl                                                                          -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                   H   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CF.sub.3                                                                             -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                  H   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CF.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  H   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CF.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                  H   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CF.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                   H   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH(CH.sub.3).sub.2                                                                   -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                  H   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH(CH.sub.3).sub.2                                                                   -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  H   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH(CH.sub.3).sub.2                                                                   -- O H  Cl  OCH.sub.3                                                                          CH                                  H   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH(CH.sub.3).sub.2                                                                   -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                   H   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  H   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                  H   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  Cl  CH.sub.3                                                                           CH                                  H   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                   H   0 --                                                                               Q-3                                                                               CH.sub. 3                                                                           --   SCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                  H   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  H   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                   H   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                   H   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   N(CH.sub.3).sub.2                                                                    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                  H   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   N(CH.sub.3).sub.2                                                                    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  H   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   N(CH.sub.3).sub.2                                                                    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                   H   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                   H   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                  H   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  H   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  Cl  OCH.sub.3                                                                          CH                                  H   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                  Cl  0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                  Cl  0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                  Cl  0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  Cl  0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                  Cl  0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                   Cl  0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                   Cl  0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O CH.sub.3                                                                          OCH.sub.3                                                                          CH.sub.3                                                                           N                                   Cl  0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                  Cl  0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                  Cl  0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  Cl  0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  Cl  OCH.sub.3                                                                          CH                                  Cl  0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                   Cl  0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                   H   0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                  H   0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                  H   0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  H   0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                  H   0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                   H   0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                   Cl  0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                  Cl  0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  Cl  0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                   Cl  0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                   Cl  0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                  Cl  0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                  Cl  0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  Cl  0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  Cl  OCH.sub.3                                                                          CH                                  Cl  0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                   Cl  0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                   Br  0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                  Br  0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  Br  0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                  Br  0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                   Br  0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                   Br  0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                  Br  0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  Br  0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  Cl  OCH.sub.3                                                                          CH                                  Br  0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                   Br  0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                   Br  0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                  Br  0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  Br  0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                   Br  0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                   Br  0 --                                                                               Q-4                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                  Br  0 --                                                                               Q-4                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  Br  0 --                                                                               Q-4                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                   Br  0 --                                                                               Q-4                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                   F   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                  F   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  F   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                   F   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                   F   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                  F   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                  F   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  F   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                   F   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                   F   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                  F   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  F   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                   F   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                   OCH.sub.3                                                                          0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                  OCH.sub.3                                                                          0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  OCH.sub.3                                                                          0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                  OCH.sub.3                                                                          0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                   OCH.sub.3                                                                          0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                   OCH.sub.3                                                                          0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                  OCH.sub.3                                                                          0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  OCH.sub.3                                                                          0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                   OCH.sub.3                                                                          0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                   OCH.sub.3                                                                          0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                  OCH.sub.3                                                                          0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  OCH.sub.3                                                                          0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                   OCH.sub.3                                                                          0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                  OCH.sub.3                                                                          0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                  OCH.sub.3                                                                          0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  OCH.sub.3                                                                          0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                  OCH.sub.3                                                                          0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                   OCH.sub.3                                                                          0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  OCH.sub.3                                                                          0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                  OCH.sub.3                                                                          0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                   OCH.sub.3                                                                          0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                   OCH.sub.3                                                                          0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                  CF.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                  CF.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                   CF.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub. 3                                                                         OCH.sub.3                                                                          N                                   CF.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  CF.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                  CF.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  CF.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                   CF.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                   CF.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                  CF.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  CF.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                   CF.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                   OCF.sub.2 H                                                                        0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                  OCF.sub.2 H                                                                        0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  OCF.sub.2 H                                                                        0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                   Cl  0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                  Cl  0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  Cl  0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                   Cl  0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                   Br  0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                  Br  0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  Br  0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                   F   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                   F   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  F   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                  OCH.sub.3                                                                          0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                  OCH.sub.3                                                                          0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  OCH.sub.3                                                                          0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                   OCH.sub.3                                                                          0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                   CF.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                  CF.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  CF.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                   CF.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                   Cl  0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                  Cl  0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  Cl  0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                   Br  0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  Br  0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                  F   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                   F   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                  OCH.sub.3                                                                          0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                   OCH.sub.3                                                                          0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                  OCH.sub.3                                                                          0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  CH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                  CH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                  CH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  CH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                  CH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                   CH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                   CH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                  CH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  CH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  Cl  OCH.sub.3                                                                          CH                                  CH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                   CH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                   Cl  0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O CH.sub.3                                                                          OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  Br  0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O CH.sub.3                                                                          OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  F   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O CH.sub.3                                                                          OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  Cl  0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                  Cl  0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  Br  0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                  Br  0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub. 3                                                                         CH                                  F   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  F   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                  OCH.sub.3                                                                          0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                  OCH.sub.3                                                                          0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                  OCH.sub.3                                                                          0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                   Cl  0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                   Cl  0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                   CH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH 213-216                          CH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH 186-189                          CH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub. 3                                                                           --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH 207-208                          CH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH 170-173                          CH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OC.sub.2 H.sub.5                                                                   NHCH.sub.3                                                                         N  186-191                          CH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N  141-144                          CH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N  191-193                          H   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OC.sub.2 H.sub.5                                                                   NHCH.sub.3                                                                         N  179-183                          H   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH 165-167                          __________________________________________________________________________

                                      TABLE XIII                                   __________________________________________________________________________     General Structure 13                                                           R.sub.1                                                                             n E Q  R.sub.2                                                                             R.sub.3                                                                             R.sub.4                                                                              R.sub.5                                                                           W R  X   Y   Z  m.p. (°C.)               __________________________________________________________________________     H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub. 5                                                                    --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub. 5                                                                    CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CF.sub.3                                                                             -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CF.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CF.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CF.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH(CH.sub.3 ).sub.2                                                                  -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH(CH.sub.3).sub.2                                                                   -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH(CH.sub.3).sub.2                                                                   -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH(CH.sub.3).sub.2                                                                   -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   OCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   OCH.sub.3                                                                            -- O H  Cl  CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   SCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   SCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   N(CH.sub.3).sub.2                                                                    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   N(CH.sub.3).sub.2                                                                    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   N(CH.sub.3).sub.2                                                                    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  H    0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O CH.sub.3                                                                          OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  Cl  OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  H    0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Cl   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Cl   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  Cl  OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub. 3                                                                           --    -- O H  Cl  OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  Cl  OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Br   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Br   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Br   0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Br   0 --                                                                               Q-4                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Br   0 --                                                                               Q-4                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-4                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Br   0 --                                                                               Q-4                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 F    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  F    0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  OCH.sub.3                                                                           0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 CF.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 CF.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                  CF.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  CF.sub.3                                                                            0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 CF.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 CF.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 CF.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  CF.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCF.sub.2 H                                                                         0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCF.sub.2 H                                                                         0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCF.sub.2 H                                                                         0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Br   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Br   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  CF.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Br   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  F    0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 OCH.sub.3                                                                           0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                 CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                 CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  CH.sub.3                                                                            0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  CH.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 CH.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 CH.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  Cl  OCH.sub.3                                                                          CH                                 CH.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  CH.sub.3                                                                            0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O CH.sub.3                                                                          OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub. 3                                                                           --    -- O CH.sub.3                                                                          OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O CH.sub.3                                                                          OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 Cl   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 Br   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                 Br   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 F    0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                 OCH.sub.3                                                                           0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  Cl   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                  Cl   0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                  __________________________________________________________________________

                                      TABLE XIV                                    __________________________________________________________________________     General Structure 14                                                           R.sub.1                                                                          n E  Q  R.sub.3                                                                           R.sub.4                                                                          W R X   Y   Z  m.p. (°C.)                                __________________________________________________________________________     H 0 -- Q-1                                                                               CH.sub.3                                                                          - O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                                  H 0 -- Q-1                                                                               CH.sub.3                                                                          --                                                                               O H OCH.sub.3                                                                          CH.sub.3                                                                           CH                                                  H 0 -- Q-1                                                                               CH.sub.3                                                                          --                                                                               O H Cl  OCH.sub.3                                                                          CH                                                  H 0 -- Q-1                                                                               CH.sub.3                                                                          --                                                                               O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                                   H 0 -- Q-1                                                                               CH.sub.3                                                                          --                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                   H 0 -- Q-1                                                                               C.sub.2 H.sub.5                                                                   --                                                                               O H OCH.sub.3                                                                          CH.sub.3                                                                           CH                                                  H 0 -- Q-1                                                                               C.sub.2 H.sub.5                                                                   --                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                                  H 0 -- Q-1                                                                               C.sub.2 H.sub.5                                                                   --                                                                               O H Cl  OCH.sub.3                                                                          CH                                                  H 0 -- Q-1                                                                               C.sub.2 H.sub.5                                                                   --                                                                               O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                                  H 0 -- Q-1                                                                               C.sub.2 H.sub.5                                                                   --                                                                               O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                                   H 0 -- Q-2                                                                               CH.sub.3                                                                          --                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                   H 0 -- Q-2                                                                               CH.sub.2                                                                          --                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                                  H 0 -- Q-2                                                                               CH.sub.3                                                                          --                                                                               O H OCH.sub.3                                                                          CH.sub.3                                                                           CH                                                  H 0 -- Q-2                                                                               CH.sub.3                                                                          --                                                                               O H Cl  OCH.sub.3                                                                          CH                                                  H 0 -- Q-2                                                                               CH.sub.3                                                                          --                                                                               O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                                  H 0 -- Q-2                                                                               CH.sub.3                                                                          --                                                                               O H OCH.sub.3                                                                          CH.sub.3                                                                           N                                                   H 0 -- Q-2                                                                               C.sub.2 H.sub.5                                                                   --                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                   H 0 -- Q-2                                                                               C.sub.2 H.sub.5                                                                   --                                                                               O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                                  H 0 -- Q-2                                                                               C.sub.2 H.sub.5                                                                   --                                                                               O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                                  H 0 -- Q-2                                                                               C.sub.2 H.sub.5                                                                   --                                                                               O H Cl  OCH.sub.3                                                                          CH                                                  H 0 -- Q-2                                                                               C.sub.2 H.sub.5                                                                   --                                                                               O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                                   H 0 -- Q-2                                                                               C.sub.2 H.sub.5                                                                   --                                                                               O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                   __________________________________________________________________________

                                      TABLE XV                                     __________________________________________________________________________     General Structure 15                                                           R.sub.1                                                                          n E Q  R.sub.3                                                                           R.sub.4                                                                              R.sub.5                                                                           W R   X   Y   Z  m.p. (°C.)                        __________________________________________________________________________     H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O H   CH.sub.3                                                                           CH.sub.3                                                                           CH                                          H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O H   OCH.sub.3                                                                          CH.sub.3                                                                           CH                                          H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O H   Cl  OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O H   CH.sub.3                                                                           OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O H   OCH.sub.3                                                                          OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O H   OCH.sub.3                                                                          CH.sub.3                                                                           CH                                          H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O H   OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O H   Cl  OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O H   CH.sub.3                                                                           CH.sub.3                                                                           CH                                          H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O H   CH.sub.3                                                                           OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O H   OCH.sub.3                                                                          OCH.sub.3                                                                          CH 138-143                                  H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O H   OCH.sub.3                                                                          CH.sub.3                                                                           CH 155-159                                  H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O H   Cl  OCH.sub.3                                                                          CH 157-158                                  H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O H   CH.sub.3                                                                           CH.sub.3                                                                           CH 135-140                                  H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O H   OCH.sub.3                                                                          CH.sub.3                                                                           N                                           H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --    -- O H   OCH.sub.3                                                                          OCH.sub.3                                                                          N  75-78                                    H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O H   CH.sub.3                                                                           CH.sub.3                                                                           CH                                          H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O H   CH.sub.3                                                                           OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O H   Cl  OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O H   CH.sub.3                                                                           OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O H   OCH.sub.3                                                                          OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O H   CH.sub.3                                                                           OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O H   Cl  OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O H   OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O H   OCH.sub.3                                                                          OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O H   CH.sub.3                                                                           OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O H   CH.sub.3                                                                           CH.sub.3                                                                           CH                                          H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O H   CH.sub.3                                                                           OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O H   Cl  OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O H   OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                      -- O H   CH.sub.3                                                                           OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O H   CH.sub.3                                                                           OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O H   OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O H   Cl  OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O H   CH.sub.3                                                                           OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O H   OCH.sub.3                                                                          OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O H   CH.sub.3                                                                           CH.sub.3                                                                           CH                                          H 0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O H   OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- CF.sub.3 --                                                                               O   H   OCH.sub.3                                                                          CH.sub.                                                                           CH                                       H 0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O H   CH.sub.3                                                                           OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O H   CH.sub.3                                                                           OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O H   OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O H   Cl  OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O H   CH.sub.3                                                                           OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O H   OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O H   CH.sub.3                                                                           OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O H   Cl  OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O H   OCH.sub.3                                                                          OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O H   CH.sub.3                                                                           OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O H   OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O H   OCH.sub.3                                                                          OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O H   CH.sub.3                                                                           OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O H   CH  CH.sub.3                                                                           CH                                          H 0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O H   OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O H   OCH.sub.3                                                                          CH  N                                           H 0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O H   OCH.sub.3                                                                          CH.sub.3                                                                           N                                           H 0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O H   OCH.sub.3                                                                          CH.sub.3                                                                           CH                                          H 0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O H   OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O H   Cl  OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O H   CH.sub.3                                                                           CH.sub.3                                                                           CH                                          H 0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O H   CH.sub.3                                                                           CH.sub.3                                                                           CH                                          H 0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O H   OCH.sub.3                                                                          CH.sub.3                                                                           CH                                          H 0 --Q-5                                                                            -- -- CH.sub.3                                                                             O  H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O H   Cl  OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --    -- O H   OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --    -- O H   OCH.sub.3                                                                          OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --    -- O H   OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- H     -- O H   OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- H     -- O H   CH.sub.3                                                                           OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- H     -- O H   CH.sub.3                                                                           CH.sub.3                                                                           CH                                          H 0 --                                                                               Q-3                                                                               -- H     -- O H   Cl  OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- H     -- O H   OCH.sub.3                                                                          OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-3                                                                               -- H     -- O H   CH.sub.3                                                                           OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                             -- O H   CH.sub.3                                                                           CH.sub.3                                                                           CH                                          H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub. 5                                                                     -- O H   OCH.sub.3                                                                          OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-3                                                                               -- CH.sub.2 Cl                                                                          -- O H   CH.sub.3                                                                           CH.sub.3                                                                           CH                                          H 0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O H   Cl  OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- CF.sub.3                                                                             -- O H   OCH.sub.3                                                                          OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O H   CH.sub.3                                                                           CH.sub.3                                                                           CH                                          H 0 --                                                                               Q-3                                                                               -- CH(CH.sub.3).sub.2                                                                   -- O H   OCH.sub.3                                                                          OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O H   CH.sub.3                                                                           CH.sub.3                                                                           CH                                          H 0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                            -- O H   CH.sub.3                                                                           OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O H   OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O H   CH.sub.3                                                                           OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O H   CH.sub.3                                                                           CH.sub.3                                                                           CH                                          H 0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O H   Cl  OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O H   OCH.sub.3                                                                          OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-3                                                                               -- OC.sub.2 H.sub.5                                                                     -- O H   CH.sub.3                                                                           OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O H   CH.sub.3                                                                           CH.sub.3                                                                           CH                                          H 0 --                                                                               Q-3                                                                               -- SCH.sub.3                                                                            -- O H   Cl  OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O H   CH.sub.3                                                                           OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O H   Cl  OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-3                                                                               -- N(CH.sub.3).sub.2                                                                    -- O H   OCH.sub.3                                                                          OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                             -- O H   OCH.sub.3                                                                          OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O H   OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-5                                                                               -- --    CH.sub.3                                                                          O H   CH.sub.3                                                                           OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-5                                                                               -- --    C.sub.2L H.sub.5                                                                  O H   OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-5                                                                               -- --    C.sub.2 H.sub.5                                                                   O H   CH.sub.3                                                                           OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-5                                                                               -- --    C.sub.2 H.sub.5                                                                   O H   CH.sub.3                                                                           CH.sub.3                                                                           CH                                          H 0 --                                                                               Q-5                                                                               -- --    C.sub.2 H.sub.5                                                                   O H   Cl  OCH.sub.3                                                                          CH                                          H 0 --                                                                               Q-5                                                                               -- --    C.sub.2 H.sub.5                                                                   O H   OCH.sub.3                                                                          OCH.sub.3                                                                          N                                           H 0 --                                                                               Q-5                                                                               -- --    C.sub.2 H.sub.5                                                                   O H   CH.sub.3                                                                           OCH.sub.3                                                                          N                                           __________________________________________________________________________

                                      TABLE XVI                                    __________________________________________________________________________     General Structure 16                                                           R.sub.1                                                                          n E Q  R.sub.3                                                                           R.sub.4                                                                            R.sub.5                                                                           W R X   Y   Z  m.p. (°C.)                            __________________________________________________________________________     H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                           CH.sub.                                                                            CH                                              H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H Cl  OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --  -- O H OCH.sub.3                                                                          CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --  -- O H Cl  OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --  -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --  -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H Cl  OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          CH.sub.3                                                                           N                                               H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --  -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --  -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --  -- O H Cl  OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --  -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H Cl  OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                    -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                    -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                    -- O H Cl  OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H Cl  OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H OCH.sub.3                                                                          CH.sub.3                                                                           N                                               H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- H OCH.sub.3                                                                        OCH.sub.3                                                                          CH                                                  H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                    -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                    -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                    -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H Cl  OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                           -- O H Cl  OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-4                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               __________________________________________________________________________

                                      TABLE XVII                                   __________________________________________________________________________     General Structure 17                                                           R.sub.1                                                                            E Q  G  n R.sub.3                                                                           W R X   Y   Z  m.p. (°C.)                              __________________________________________________________________________     H   --                                                                               Q-1                                                                               O  0 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                                H   --                                                                               Q-1                                                                               S  0 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                                H   --                                                                               Q-1                                                                               SO 0 CH.sub.3                                                                          O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                                H   --                                                                               Q-1                                                                               SO.sub.2                                                                          0 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                 H   --                                                                               Q-1                                                                               O  1 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                                 H   --                                                                               Q-1                                                                               S  1 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                                H   --                                                                               Q-1                                                                               SO 1 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                                H   --                                                                               Q-1                                                                               SO.sub.2                                                                          1 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                                H   --                                                                               Q-1                                                                               O  2 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                                 H   --                                                                               Q-1                                                                               S  2 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                 H   --                                                                               Q-1                                                                               SO 2 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                                H   --                                                                               Q-1                                                                               SO.sub.2                                                                          2 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                                6-CH.sub.3                                                                         --                                                                               Q-1                                                                               O  0 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                                6-CH.sub.3                                                                         --                                                                               Q-1                                                                               S  1 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                                6-CH.sub.3                                                                         --                                                                               Q-1                                                                               SO 2 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                 6-CH.sub.3                                                                         --                                                                               Q-1                                                                               SO.sub.2                                                                          1 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                                 5-Cl                                                                               --                                                                               Q-1                                                                               O  1 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                                5-Cl                                                                               --                                                                               Q-1                                                                               S  2 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                                5-Cl                                                                               --                                                                               Q-1                                                                               SO 1 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                 5-Cl                                                                               --                                                                               Q-1                                                                               SO.sub.2                                                                          2 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                                 H   --                                                                               Q-2                                                                               O  0 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                                H   --                                                                               Q-2                                                                               S  0 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                                H   --                                                                               Q-2                                                                               SO 0 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                                 H   --                                                                               Q-2                                                                               SO.sub.2                                                                          0 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                 H   --                                                                               Q-2                                                                               O  1 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                                H   --                                                                               Q-2                                                                               S  1 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                                H   --                                                                               Q-2                                                                               SO 1 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                                 H   --                                                                               Q-2                                                                               SO.sub.2                                                                          1 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                 H   --                                                                               Q-2                                                                               O  2 CH.sub.3                                                                          O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                                H   --                                                                               Q-2                                                                               S  2 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                                H   --                                                                               Q-2                                                                               SO 2 CH.sub.3                                                                          O H CH.sub.3                                                                           CH.sub.3                                                                           N                                                 H   --                                                                               Q-2                                                                               SO.sub.2                                                                          2 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                 __________________________________________________________________________

                                      TABLE XVIIa                                  __________________________________________________________________________     General Structure 17                                                           R.sub.1                                                                          E Q  G  n R.sub.4                                                                           W R X   Y   Z  m.p. (°C.)                                __________________________________________________________________________     H --                                                                               Q-3                                                                               O  1 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                                   H --                                                                               Q-3                                                                               S  1 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                                  H --                                                                               Q-3                                                                               SO 1 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                                  H --                                                                               Q-3                                                                               SO.sub.2                                                                          1 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                   H --                                                                               Q-3                                                                               O  2 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                                  H --                                                                               Q-3                                                                               S  2 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                   H --                                                                               Q-3                                                                               SO 2 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                                   H --                                                                               Q-3                                                                               SO.sub.2                                                                          2 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                                  H --                                                                               Q-4                                                                               O  1 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                                   H --                                                                               Q-4                                                                               S  1 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                                  H --                                                                               Q-4                                                                               SO 1 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                                  H --                                                                               Q-4                                                                               SO.sub.2                                                                          1 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                   H --                                                                               Q-4                                                                               O  2 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                                   H --                                                                               Q-4                                                                               S  2 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                                  H --                                                                               Q-4                                                                               SO 2 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                                  H --                                                                               Q-4                                                                               SO.sub.2                                                                          2 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                   __________________________________________________________________________

                                      TABLE XVIIb                                  __________________________________________________________________________     General Structure 17                                                           R.sub.1                                                                          E Q  G  n R.sub.5                                                                           W R X   Y   Z  m.p. (°C.)                                __________________________________________________________________________     H --                                                                               Q-5                                                                               O  1 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                                  H --                                                                               Q-5                                                                               S  1 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                   H --                                                                               Q-5                                                                               SO 1 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                                   H --                                                                               Q-5                                                                               SO.sub.2                                                                          1 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                                  H --                                                                               Q-5                                                                               O  2 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                                   H --                                                                               Q-5                                                                               S  2 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                                  H --                                                                               Q-5                                                                               SO 2 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                                  H --                                                                               Q-5                                                                               SO.sub.2                                                                          2 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                   H --                                                                               Q-6                                                                               O  1 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                                   H --                                                                               Q-6                                                                               S  1 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                                  H --                                                                               Q-6                                                                               SO 1 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                                  H --                                                                               Q-6                                                                               SO.sub.2                                                                          1 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                   H --                                                                               Q-6                                                                               O  2 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                                  H --                                                                               Q-6                                                                               S  2 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                   H --                                                                               Q-6                                                                               SO 2 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                                   H --                                                                               Q-6                                                                               SO.sub.2                                                                          2 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                                  H --                                                                               Q-7                                                                               O  1 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                                  H --                                                                               Q-7                                                                               S  1 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                   H --                                                                               Q-7                                                                               SO 1 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                                   H --                                                                               Q-7                                                                               SO.sub.2                                                                          1 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                                  H --                                                                               Q-7                                                                               O  2 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                                  H --                                                                               Q-7                                                                               S  2 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                   H --                                                                               Q-7                                                                               SO 2 CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                                   H --                                                                               Q-7                                                                               SO.sub.2                                                                          2 CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                                  __________________________________________________________________________

                                      TABLE XVIII                                  __________________________________________________________________________     General Structure 18                                                           R.sub.1                                                                          n E Q  R.sub.2                                                                             R.sub.3                                                                             R.sub.4                                                                              R.sub.5                                                                           W R  X   Y   Z  m.p. (°C.)                  __________________________________________________________________________     H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    H 0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                    H 0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     H 0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H 0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                    H 0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  Cl  OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    H 0 --                                                                               Q-1                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     H 0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H 0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                    H 0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    H 0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH  N                                     H 0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H 0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    H 0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  Cl  OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     H 0 --                                                                               Q-2                                                                               C.sub.6 H.sub.5                                                                     C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H 0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  Cl  OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H 0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     H 0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    H 0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  Cl  OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     H 0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  CH.sub. 3                                                                          OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  Cl  OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     H 0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH.sub.2 Cl                                                                          -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H 0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CF.sub.3                                                                             -- O H  CH.sub.3                                                                           CH.sub.                                                                            CH                                    H 0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CF.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CF.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                    H 0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CF.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     H 0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH(CH.sub.3).sub.2                                                                   -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH(CH.sub.3).sub.2                                                                   -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH(CH.sub.3).sub.2                                                                   -- O H  Cl  OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   CH(CH.sub.3).sub.2                                                                   -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     H 0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   OCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   OCH.sub.3                                                                            -- O H  Cl  OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H 0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   SCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H 0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   SCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     H 0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   N(CH.sub.3).sub.2                                                                    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    H 0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   N(CH.sub.3).sub.2                                                                    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-3                                                                               C.sub.6 H.sub.5                                                                     --   N(CH.sub.3).sub.2                                                                    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                     H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                    H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub. 3                                                                          OCH.sub.3                                                                          N                                     H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                    H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  Cl  OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                    H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                     H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  Cl  OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                            C.sub.2 H.sub.5                                                                     --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H 0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  Cl  OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H 0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     H 0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    H 0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   C.sub.2 H.sub.5                                                                      -- O H  Cl  OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   C.sub.2 H.sub.5                                                                      -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   C.sub.2 H.sub.5                                                                      -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     H 0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.2 Cl                                                                          -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.2 Cl                                                                          -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.2 Cl                                                                          -- O H  Cl  OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.2 Cl                                                                          -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     H 0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.2 Cl                                                                          -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H 0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CF.sub.3                                                                             -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    H 0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CF.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CF.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                    H 0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CF.sub.3                                                                             -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     H 0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH(CH.sub.3).sub.2                                                                   -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH(CH.sub.3).sub.2                                                                   -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH(CH.sub.3).sub.2                                                                   -- O H  Cl  OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH(CH.sub.3).sub.2                                                                   -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     H 0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  Cl  CH.sub.3                                                                           CH                                    H 0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H 0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub. 3                                                                         N                                     H 0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     H 0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   N(CH.sub.3).sub.2                                                                    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    H 0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   N(CH.sub.3).sub.2                                                                    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   N(CH.sub.3).sub.2                                                                    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                     H 0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                     H 0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                    H 0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  Cl  OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    Cl                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    Cl                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    Cl                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    Cl                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                    Cl                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     Cl                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     Cl                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O CH.sub.3                                                                          OCH.sub.3                                                                          CH.sub.3                                                                           N                                     Cl                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    Cl                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    Cl                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    Cl                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  Cl  OCH.sub.3                                                                          CH                                    Cl                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                     Cl                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     H 0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    H 0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                    H 0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH  N                                     H 0 --                                                                               Q-2                                                                               CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     Cl                                                                               0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                    Cl                                                                               0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    Cl                                                                               0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                     Cl                                                                               0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     Cl                                                                               0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    Cl                                                                               0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                    Cl                                                                               0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    Cl                                                                               0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  Cl  OCH.sub.3                                                                          CH                                    Cl                                                                               0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                     Cl                                                                               0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     Br                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    Br                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    Br                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                    Br                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                     Br                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     Br                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    Br                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    Br                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  Cl  OCH.sub.3                                                                          CH                                    Br                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     Br                                                                               0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                     Br                                                                               0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                    Br                                                                               0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    Br                                                                               0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     Br                                                                               0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                     Br                                                                               0 --                                                                               Q-4                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                    Br                                                                               0 --                                                                               Q-4                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    Br                                                                               0 --                                                                               Q-4                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     Br                                                                               0 --                                                                               Q-4                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                     F 0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                    F 0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    F 0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                     F 0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     F 0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                    F 0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                    F 0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    F 0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     F 0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                     F 0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                    F 0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    F 0 --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                     F 0 --                                                                               Q-3                                                                               CH.sub. 3                                                                           --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     OCH.sub.3                                                                        0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    OCH.sub.3                                                                        0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    OCH.sub.3                                                                        0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                    OCH.sub.3                                                                        0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                     OCH.sub.3                                                                        0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     OCH.sub.3                                                                        0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                    OCH.sub.3                                                                        0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    OCH.sub.3                                                                        0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                     OCH.sub.3                                                                        0 --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     OCH.sub.3                                                                        0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                    OCH.sub.3                                                                        O --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    OCH.sub.3                                                                        O --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     OCH.sub.3                                                                        O --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                    OCH.sub.3                                                                        0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                    OCH.sub.3                                                                        0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    OCH.sub.3                                                                        O --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                    OCH.sub.3                                                                        O --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.2 CH.sub.3                                                                   --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     OCH.sub.3                                                                        O --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    OCH.sub.3                                                                        O --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                    OCH.sub.3                                                                        O --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                     OCH.sub.3                                                                        O --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     OCH.sub.3                                                                        O --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    CF.sub.3                                                                         O --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    CF.sub.3                                                                         O --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          N                                     CF.sub.3                                                                         O --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     CF.sub.3                                                                         O --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    CF.sub.3                                                                         O --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    CF.sub.3                                                                         O --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    CF.sub.3                                                                         O --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     CF.sub.3                                                                         O --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                     CF.sub.3                                                                         O --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                    CF.sub.3                                                                         O --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    CF.sub.3                                                                         O --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                     CF.sub.3                                                                         O --                                                                               Q-3                                                                               CH.sub.3                                                                            --   CH.sub.3                                                                             -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     OCF.sub.2                                                                        O --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --       O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                    OCF.sub.2 H                                                                      O --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --       O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    OCF.sub.2 H                                                                      O --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     Cl                                                                               O --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                    Cl                                                                               O --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    Cl                                                                               O --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     Cl                                                                               O --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                     Br                                                                               O --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                    Br                                                                               O --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    Br                                                                               O --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     F O --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     F O --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    F O --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                    OCH.sub.3                                                                        O --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                    OCH.sub.3                                                                        O --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    OCH.sub.3                                                                        O --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     OCH.sub.3                                                                        O --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                     CF.sub.3                                                                         O --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                    CF.sub.3                                                                         O --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    CF.sub.3                                                                         O --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                     CF.sub.3                                                                         O --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     Cl                                                                               O --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                    Cl                                                                               O --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    Cl                                                                               O --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     Br                                                                               O --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    Br                                                                               O --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                    F O --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     F O --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                    OCH.sub.3                                                                        O --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     OCH.sub.3                                                                        O --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                    OCH.sub.3                                                                        O --                                                                               Q-3                                                                               CH.sub.3                                                                            --   SCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    CH.sub.3                                                                         O --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  CH.sub.3                                                                           CH.sub.3                                                                           CH                                    CH.sub.3                                                                         O --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                    CH.sub.3                                                                         0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    O  H OCH.sub.3                                                                         OCH.sub.3                                                                          CH                                        CH.sub.3                                                                         O --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  Cl  OCH.sub.3                                                                          CH                                    CH.sub.3                                                                         0 --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                     CH.sub.3                                                                         O --                                                                               Q-1                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     CH.sub.3                                                                         O --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                    CH.sub.3                                                                         O --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    CH.sub.3                                                                         O --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  Cl  OCH.sub.3                                                                          CH                                    CH.sub.3                                                                         O --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                     CH.sub.3                                                                         O --                                                                               Q-3                                                                               CH.sub.3                                                                            --   OCH.sub.3                                                                            -- O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     Cl                                                                               O --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O CH.sub.3                                                                          OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    Br                                                                               O --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O CH.sub.3                                                                          OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    F O --                                                                               Q-2                                                                               CH.sub.3                                                                            CH.sub.3                                                                            --    -- O CH.sub.3                                                                          OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    Cl                                                                               O --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    Cl                                                                               O --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    Br                                                                               O --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          CH.sub.3                                                                           CH                                    Br                                                                               O --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    F O --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    F O --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    OCH.sub.3                                                                        O --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  CH.sub.3                                                                           OCH.sub.3                                                                          CH                                    OCH.sub.3                                                                        O --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                    OCH.sub.3                                                                        O --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub. 3                                                                         OCH.sub.3                                                                          N                                     Cl                                                                               O --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          CH.sub.3                                                                           N                                     Cl                                                                               O --                                                                               Q-5                                                                               CH.sub.3                                                                            --   --    CH.sub.3                                                                          O H  OCH.sub.3                                                                          OCH.sub.3                                                                          N                                     __________________________________________________________________________

                                      TABLE XIX                                    __________________________________________________________________________     General Structure 19                                                           .sup.R 1                                                                         n E Q   R.sub.3                                                                           R.sub.4                                                                            R.sub.5                                                                          W R X   Y   Z  m.p. (°C.)                            __________________________________________________________________________     H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H Cl  OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --  -- O H OCH.sub.3                                                                          CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --  -- O H Cl  OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --  -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --  -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H Cl  OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-2                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          CH.sub.3                                                                           N                                               H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --  -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --  -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --  -- O H Cl  OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --  -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H Cl  OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                    -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                    -- O H CH.sub.3 OCH.sub.3                                                                 CH                                                  H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                    -- O H Cl  OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H Cl  OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H OCH.sub.3                                                                          CH.sub.3                                                                           N                                               H 0 --                                                                               Q-1                                                                               CH.sub.3                                                                          --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   --  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H 0 --                                                                               Q-3                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                    -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H 0 --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                    -- O H OCH.sub.3                                                                          OCH.sub. 3                                                                         N                                               H O --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                    -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                               H O --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H O --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                              H O --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H O --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H Cl  OCH.sub.3                                                                          CH                                              H O --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H O --                                                                               Q-3                                                                               -- OCH.sub.3                                                                          -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                               H O --                                                                               Q-4                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                              H O --                                                                               Q-4                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                              H O --                                                                               Q-4                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                              H O --                                                                               Q-4                                                                               -- CH.sub.3                                                                           -- O H Cl  OCH.sub.3                                                                          CH                                              H O --                                                                               Q-4                                                                               -- CH.sub.3                                                                           -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               H O --                                                                               Q-4                                                                               -- CH.sub.3                                                                           -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                               H O --                                                                               Q-5                                                                               -- --  CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                               __________________________________________________________________________

                                      TABLE XX                                     __________________________________________________________________________     General structure 20                                                           R.sub.1                                                                          n E Q  R.sub.3                                                                           R.sub.4                                                                           R.sub.5                                                                           W R X   Y   Z  m.p. (°C.)                             __________________________________________________________________________     H O --                                                                               Q-1                                                                               CH.sub.3                                                                          -- -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                               H O --                                                                               Q-1                                                                               CH.sub.3                                                                          -- -- O H OCH.sub.3                                                                          CH.sub.3                                                                           CH                                               H O --                                                                               Q-1                                                                               CH.sub.3                                                                          -- -- O H Cl  OCH.sub.3                                                                          CH                                               H O --                                                                               Q-1                                                                               CH.sub.3                                                                          -- -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                                H O --                                                                               Q-1                                                                               CH.sub.3                                                                          -- -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                H O --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   -- -- O H OCH.sub.3                                                                          CH.sub.2                                                                           CH                                               H O --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   -- -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                               H O --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   -- -- O H Cl  OCH.sub.3                                                                          CH                                               H O --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   -- -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                               H O --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   -- -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                                H O --                                                                               Q-2                                                                               CH.sub.3                                                                          -- -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                H O --                                                                               Q-2                                                                               CH.sub.3                                                                          -- -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                               H O --                                                                               Q-2                                                                               CH.sub.3                                                                          -- -- O H OCH.sub.3                                                                          CH.sub.3                                                                           CH                                               H O --                                                                               Q-2                                                                               CH.sub.3                                                                          -- -- O H Cl  OCH.sub.3                                                                          CH                                               H O --                                                                               Q-2                                                                               CH.sub.3                                                                          -- -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                               H O --                                                                               Q-2                                                                               CH.sub.3                                                                          -- -- O H OCH.sub.3                                                                          CH.sub.3                                                                           N                                                H O --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   -- -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                               H O --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   -- -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                               H O --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   -- -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                               H O --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   -- -- O H Cl  OCH.sub.3                                                                          CH                                               H O --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   -- -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                                H O --                                                                               Q-2                                                                               C.sub.2 H.sub.5                                                                   -- -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                H O --                                                                               Q-3                                                                               -- CH.sub.3                                                                          -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                               H O --                                                                               Q-3                                                                               -- CH.sub.3                                                                          -- O H Cl  OCH.sub.3                                                                          CH                                               H O --                                                                               Q-3                                                                               -- CH.sub.3                                                                          -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                               H O --                                                                               Q-3                                                                               -- CH.sub.3                                                                          -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                H O --                                                                               Q-3                                                                               -- CH.sub.3                                                                          -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                                H O --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                   -- O H CH.sub. 3                                                                          CH.sub.3                                                                           CH                                               H O --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                   -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                               H O --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                   -- O H Cl  OCH.sub.3                                                                          CH                                               H O --                                                                               Q-5                                                                               -- -- CH.sub.3                                                                          O H Cl  OCH.sub.3                                                                          CH                                               H O --                                                                               Q-5                                                                               -- -- CH.sub.3                                                                          O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                               H O --                                                                               Q-5                                                                               -- -- CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                               H O --                                                                               Q-5                                                                               -- -- CH.sub.3                                                                          O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                               H O --                                                                               Q-5                                                                               -- -- CH.sub.3                                                                          O H OCH.sub.3                                                                          CH.sub.3                                                                           N                                                H O --                                                                               Q-1                                                                               CH.sub.3                                                                          -- -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                               H O --                                                                               Q-1                                                                               C.sub.2 H.sub.5                                                                   -- -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                H O --                                                                               Q-3                                                                               -- CH.sub.3                                                                          -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                               H O --                                                                               Q-3                                                                               -- C.sub.2 H.sub. 5                                                                  -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                               H O --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                   -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                H O --                                                                               Q-3                                                                               -- C.sub.2 H.sub.5                                                                   -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                                H O --                                                                               Q-3                                                                               -- OCH.sub.3                                                                         -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                               H O --                                                                               Q-3                                                                               -- OCH.sub.3                                                                         -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                               H O --                                                                               Q-3                                                                               -- OCH.sub.3                                                                         -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                               H O --                                                                               Q-3                                                                               -- OCH.sub.3                                                                         -- O H Cl  OCH.sub.3                                                                          CH                                               H O --                                                                               Q-3                                                                               -- OCH.sub.3                                                                         -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                H O --                                                                               Q-3                                                                               -- OCH.sub.3                                                                         -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                                H O --                                                                               Q-4                                                                               -- CH.sub.3                                                                          -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          CH                                               H O --                                                                               Q-4                                                                               -- CH.sub.3                                                                          -- O H CH.sub.3                                                                           OCH.sub.3                                                                          CH                                               H O --                                                                               Q-4                                                                               -- CH.sub.3                                                                          -- O H CH.sub.3                                                                           CH.sub.3                                                                           CH                                               H O --                                                                               Q-4                                                                               -- CH.sub.3                                                                          -- O H Cl  OCH.sub.3                                                                          CH                                               H O --                                                                               Q-4                                                                               -- CH.sub.3                                                                          -- O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                H O --                                                                               Q-4                                                                               -- CH.sub.3                                                                          -- O H CH.sub.3                                                                           OCH.sub.3                                                                          N                                                H O --                                                                               Q-5                                                                               -- -- CH.sub.3                                                                          O H OCH.sub.3                                                                          OCH.sub.3                                                                          N                                                __________________________________________________________________________

Formulations

Useful formulations of the compounds of Formula I can be prepared in conventional ways. They include dusts, granules, pellets, solutions, suspensions, emulsions, wettable powders, emulsifiable concentrates and the like. Many of these may be applied directly. Sprayable formulations can be extended in suitable media and used at spray volumes of from a few liters to several hundred liters per hectare. High strength compositions are primarily used as intermediates for further formulation. The formulations, broadly, contain about 0.1% to 99% by weight of active ingredient(s) and at least one of (a) about 0.1% to 20% surfactant(s) and (b) 1% to 99.9% solid or liquid inert diluent(s). More specifically, they will contain these ingredients in the following approximate proportions:

    ______________________________________                                                     Active  Weight Percent*                                                        Ingredient                                                                             Diluent(s)                                                                               Surfactant(s)                                    ______________________________________                                         Wettable Powders                                                                             20-90     0-74      1-10                                         Oil Suspensions,                                                                             3-50      40-95     0-15                                         Emulsions, Solutions,                                                          (including Emulsifiable                                                        Concentrates)                                                                  Aqueous Suspension                                                                           10-50     40-84     1-20                                         Dusts         1-25      70-99     0-5                                          Granules and Pellets                                                                         0.1-95    5-99.9    0-15                                         High Strength 90-99     0-10      0-2                                          Compositions                                                                   ______________________________________                                          *Active ingredient plus at least one of a Surfactant or a Diluent equals       100 weight percent.                                                      

Lower or higher levels of active ingredient can, of course, be present depending on the intended use and the physical properties of the compound. Higher ratios of surfactant to active ingredient are somtimes desirable, and are achieved by incorporation into the formulation or by tank mixing.

Typical solid diluents are described in Watkins, et al., "Handbook of Insecticide Dust Diluents and Carriers", 2nd Ed., Dorland Books, Caldwell, N.J., but other solids, either mined or manufactured, may be used. The more absorptive diluents are preferred for wettable powders and the denser ones for dusts. Typical liquid diluents and solvents are described in Marsden, "Solvents Guide," 2nd Ed., Interscience, New York, 1950. Solubility under 0.1% is preferred for suspension concentrates; solution concentrates are preferably stable against phase separation at 0° C. "McCutcheon's Detergents and Emulsifiers Annual", MC Publishing Corp., Ridgewood, N.J., as well as Sisely and Wood, "Encyclopedia of Surface Active Agents", Chemical Publishing Co., Inc., N.Y., 1964, list surfactants and recommended uses. All formulations can contain minor amounts of additives to reduce foaming, caking, corrosion, microbiological growth, etc.

The methods of making such compositions are well known. Solutions are prepared by simply mixing the ingredients. Fine solid compositions are made by blending and, usually, grinding as in a hammer or fluid energy mill. Suspensions are prepared by wet milling (see, for example, Littler, U.S. Pat. No. 3,060,084). Granules and pellets may be made by spraying the active material upon preformed granular carriers or by agglomeration techniques. See J. E. Browning, "Agglomeration", Chemical Engineering, Dec. 4, 1967, pp. 147ff. and "Perry's Chemical Engineer's Handbook", 5th Ed., McGraw-Hill, New York, 1973, pp. 8-57ff.

For further information regarding the art of formulation, see for example:

H.M. Loux, U.S. Pat. No. 3,235,361, Feb. 15, 1966, Col. 6, line 16 through Col. 7, line 19 and Examples 10 through 41;

R. W. Luckenbaugh, U.S. Pat. No. 3,309,192, Mar. 14, 1967, Col. 5, line 43 through Col. 7, line 62 and Examples 8, 12, 15, 39, 41, 52, 53, 58, 132, 138-140, 162-164, 166, 167 and 169-182;

H. Gysin and E. Knusli, U.S. Pat. No. 2,891,855, June 23, 1959, Col. 3, line 66 through Col. 5, line 17 and Examples 1-4;

G. C. Klingman, "Weed Control as a Science", John Wiley & Sons, Inc., New York, 1961, pp. 81-96; and

J. D. Fryer and S. A. Evans, "Weed Control Handbook", 5th Ed., Blackwell Scientific Publications, Oxford, 1968, pp. 101-103.

In the following examples, all parts are by weight unless otherwise indicated.

EXAMPLE 16

Wettable Powder

    ______________________________________                                         N-[(4,6,dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(1-                                                       80%                                                methyl-1H-tetrazol-5-yl)benzenesulfonamide                                     sodium alkylnaphthalenesulfonate                                                                           2%                                                 sodium ligninsulfonate      2%                                                 synthetic amorphous silica  3%                                                 kaolinite                   13%                                                ______________________________________                                    

The ingredients are blended, hammer-milled until all the solids are essentially under 50 microns, reblended, and packaged.

EXAMPLE 17

Wettable Powder

    ______________________________________                                         N-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(5-                                                       50%                                                methyl-1H-tetrazol-1-yl)benzenesulfonamide                                     sodium alkylnaphthalenesulfonate                                                                           2%                                                 low viscosity methyl cellulose                                                                             2%                                                 diatomaceous earth          46%                                                ______________________________________                                    

The ingredients are blended, coarsely hammer-milled and then air-milled to produce particles essentially all below 10 microns in diameter. The product is reblended before packaging.

EXAMPLE 18

Granule

    ______________________________________                                         Wettable Powder of Example 17 (above)                                                                    5%                                                   attapulgite granules      95%                                                  (U.S.S. 20-40 mesh; 0.84-0.42 mm)                                              ______________________________________                                    

A slurry of wettable powder containing 25% solids is sprayed on the surface of attapulgite granules while tumbling in a double-cone blender. The granules are dried and packaged.

EXAMPLE 19

Extruded Pellet

    ______________________________________                                         N-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(5-                                                       25%                                                methyl-1H-tetrazol-1-yl)benzenesulfonamide                                     anhydrous sodium sulfate    10%                                                crude calcium ligninsulfonate                                                                              5%                                                 sodium alkylnaphthalenesulfonate                                                                           1%                                                 calcium/magnesium bentonite 59%                                                ______________________________________                                    

The ingredients are blended, hammer-milled and then moistened with about 12% water. The mixture is extruded as cylinders about 3 mm diameter which are cut to produce pellets about 3 mm long. These may be used directly after drying, or the dried pellets may be crushed to pass a U.S. Ser. No. 20 sieve (0.84 mm openings). The granules held on a U.S. Ser. No. 40 sieve (0.42 mm openings) may be packaged for use and the fines recycled.

EXAMPLE 20

Oil Suspension

    ______________________________________                                         N-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(1-                                                       25%                                                methyl-1H-tetrazol-5-yl)benzenesulfonamide                                     Polyoxyethylene sorbitol hexaoleate                                                                        5%                                                 highly aliphatic hydrocarbon oil                                                                           70%                                                ______________________________________                                    

The ingredients are ground together in a sand mill until the solid particles have been reduced to under about 5 microns. The resulting thick suspension may be applied directly, but preferably after being extended with oils or emulsified in water.

EXAMPLE 21

Wettable Powder

    ______________________________________                                         N-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(5-                                                       20%                                                methyl-1H-tetrazol-1-yl)benzenesulfonamide                                     sodium alkylnaphthalenesulfonate                                                                           4%                                                 sodium ligninsulfonate      4%                                                 low viscosity methyl cellulose                                                                             3%                                                 attapulgite                 69%                                                ______________________________________                                    

The ingredients are thoroughly blended. After grinding in a hammern-mill to produce particles essentially all below 100 microns, the material is reblended and sifted through a U.S. Ser. No. 50 sieve (0.3 mm opening) and packaged.

EXAMPLE 22

Low Strength Granule

    ______________________________________                                         N-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(1-                                                       1%                                                 methyl-1H-tetrazol-5-yl)benezenesulfonamide                                    N,N-dimethylformamide       9%                                                 attapulgite granules        90%                                                (U.S.S. 20-40 sieve)                                                           ______________________________________                                    

The active ingredient is dissolved in the solvent and the solution is sprayed upon dedusted granules in a double cone blender. After spraying of the solution has been completed, the blender is allowed to run for a short period and then the granules are packaged.

EXAMPLE 23

Aqueous Suspension

    ______________________________________                                         N-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(1-                                                       40%                                                methyl-1H-tetrazol-5-yl)benzenesulfonamide                                     polyacrylic acid thickener  0.3%                                               dodecylphenol polyethylene glycol ether                                                                    0.5%                                               disodium phosphate          1%                                                 monosodium phosphate        0.5%                                               polyvinyl alcohol           1.0%                                               water                       56.7%                                              ______________________________________                                    

The ingredients are blended and grond together in a sand mill to produce particles essentially all under 5 microns in size.

EXAMPLE 24

Solution

    ______________________________________                                         N-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(1-                                                       5%                                                 methyl-1H-tetrazol-5-yl)benzenesulfonamide, Sodium                             Salt                                                                           water                       95%                                                ______________________________________                                    

The salt is added directly to the water with stirring to produce the solution, which may then be packaged for use.

EXAMPLE 25

Low Strength Granule

    ______________________________________                                         N-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(1-                                                       0.1%                                               methyl-1H-tetrazol-5-yl)benzenesulfonamide                                     attapulgite granules        99.9%                                              (U.S.S. 20-40 mesh)                                                            ______________________________________                                    

The active ingredient is dissolved in a solvent and the solution is sprayed upon dedusted granules in a double-cone blender. After spraying of the solution has been completed, the material is warmed to evaporate the solvent. The material is allowed to cool and then packaged.

EXAMPLE 26

Granule

    ______________________________________                                         N-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(1-                                                       80%                                                methyl-1H-tetrazol-5-yl)benzenesulfonamide                                     wetting agent               1%                                                 crude ligninsulfonate salt (containing                                                                     10%                                                5-20% of the natural sugars)                                                   attapulgite clay            9%                                                 ______________________________________                                    

The ingredients are blended and milled to pass through a 100 mesh screen. This material is then added to a fluid bed granulator, the air flow is adjusted to gently fluidize the material, and a fine spray of water is sprayed onto the fluidized material. The fluidization and spraying are continued until granules of the desired size range are made. The spraying is stopped, but fluidization is continued, optionally with heat, until the water content is reduced to the desired level, generally less than 1%. The material is then discharged, screened to the desired size range, generally 14-100 mesh (1410-149 microns), and packaged for use.

EXAMLE 27

High Strength Concentrate

    ______________________________________                                         N-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(1-                                                       99%                                                methyl-1H-tetrazol-5-yl)benzenesulfonamide                                     silica aerogel              0.5%                                               synthetic amorphous silica  0.5%                                               ______________________________________                                    

The ingredients are blended and ground in a hammer-mill to produce a material essentially all passing a U.S. Ser. No. 50 screen (0.3 mm opening). The concentrate may be formulated further if necessary.

EXAMPLE 28

Wettable Powder

    ______________________________________                                         N-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(1-                                                       90%                                                methyl-1H-tetrazol-5-yl)benzenesulfonamide                                     dioctyl sodium sulfosuccinate                                                                              0.1%                                               synthetic fine silica       9.9%                                               ______________________________________                                    

The ingredients are blended and ground in a hammer-mill to produce particles essentially all below 100 microns. The material is sifted through a U.S.S. No. 50 screen and then packaged.

EXAMPLE 29

Wettable Powder

    ______________________________________                                         N-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(1-                                                       40%                                                methyl-1H-tetrazol-5-yl)benzenesulfonamide                                     sodium ligninsulfonate      20%                                                montmorillonite clay        40%                                                ______________________________________                                    

The ingredients are thoroughly blended, coarsely hammer-milled and then air-milled to produce particles essentially all below 10 microns in size. The material is reblended and then packaged.

EXAMPLE 30

Oil Suspension

    ______________________________________                                         N (4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(1-                                                        35%                                                methyl-1H-tetrazol-5-yl)benzenesulfonamide                                     blend of polyalcohol carboxylic                                                                            6%                                                 esters and oil soluble petroleum                                               sulfonates                                                                     xylene                      59%                                                ______________________________________                                    

The ingredients are combined and ground together in a sand mill to produce particles essentially all below 5 microns. The product can be used directly, extended with oils, or emulsified in water.

EXAMPLE 31

Dust

    ______________________________________                                         N-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(1-                                                       10%                                                methyl-1H-tetrazol-5-yl)benzenesulfonamide                                     attapulgite                 10%                                                Pyrophyllite                80%                                                ______________________________________                                    

The active ingredient is blended with attapulgite and then passed through a hammer-mill to produce particles substantially all below 200 microns. The ground concentrate is then blended with powdered pyrophyllite until homogeneous.

EXAMPLE 32

Wettable Powder

    ______________________________________                                         N-[[N-(4,6-dimethoxy-1,3,5-triazin-2-yl)-N-methyl-                                                         50%                                                amino]carbonyl]-2-(5-methyl-1H-tetrazol-1-yl)-                                 benzenesulfonamide                                                             sodium alkylnaphthalenesulfonate                                                                           2%                                                 low viscosity methyl cellulose                                                                             2%                                                 diatomaceous earth          46%                                                ______________________________________                                    

The ingredients are blended, coarsely hammer-milled and then air-milled to produce particles essentially all below 10 microns in diameter. The product is reblended before packaging.

EXAMPLE 33

Granule

    ______________________________________                                         Wettable Powder of Example 32 (above)                                                                     5%                                                  attapulgite granules       95%                                                 (U.S.S. 20-40 mesh; 0.84-0.42 mm)                                              ______________________________________                                    

A slurry of wettable powder containing 25% solids is sprayed on the surface of attapulgite granules while tumbling in a double-cone blender. The granules are dried and packaged.

EXAMPLE 34

Extruded Pellet

    ______________________________________                                         N-[[N-(4,6-dimethoxy-1,3,5-triazin-2-yl)-N-methyl-                                                         25%                                                amino]carbonyl]-2-(5-methyl-1H-tetrazol-1-yl)-                                 benzenesulfonamide                                                             anhydrous sodium sulfate    10%                                                crude calcium ligninsulfonate                                                                              5%                                                 sodium alkyulnaphthalenesulfonate                                                                          1%                                                 calcium/magnesium bentonite 59%                                                ______________________________________                                    

The ingredients are blended, hammer-milled and then moistened with about 12% water. The mixture is extruded as cylinders about 3 mm diameter which are cut to produce pellets about 3 mm long. These may be used directly after drying, or the dried pellets may be crushed to pass a U.S.S. No. 20 sieve (0.84 mm openings). The granules held on a U.S.S. No. 40 sieve (0.42 mm openings) may be packaged for use and the fines recycled.

EXAMPLE 35

Oil Suspension

    ______________________________________                                         N-[[N-(4,6-dimethoxy-1,3,5-triazin-2-yl)-N-methyl-                                                         25%                                                amino]carbonyl]-2-(5-methyl-1H-tetrazol-1-yl)-                                 benzenesulfonamide                                                             polyoxyethylene sorbitol hexaoleate                                                                        5%                                                 highly aliphatic hydrocarbon oil                                                                           70%                                                ______________________________________                                    

The ingredients are ground together in a sand mill until the solid particles have been reduced to under about 5 microns. The resulting thick suspension may be applied directly, but preferably after being extended with oils or emulsified in water.

EXAMPLE 36

Wettable Powder

    ______________________________________                                         N-[[N-(4,6-dimethoxy-1,3,5-triazin-2-yl)-N-methyl-                                                         20%                                                amino]carbonyl]-2-(5-methyl-1H-tetrazol-1-yl)-                                 benzenesulfonamide                                                             sodium alkylnaphthalenesulfonate                                                                           4%                                                 sodium ligninsulfonate      4%                                                 low viscosity methyl cellulose                                                                             3%                                                 attapulgite                 69%                                                ______________________________________                                    

The ingredients are thoroughly blended. After grinding in a hammer-mill to produce particles essentially all below 100 microns, the material is reblended and sifted through a U.S.S. No. 50 sieve (0.3 mm opening) and packaged.

EXAMPLE 37

Low Strength Granule

    ______________________________________                                         N-[[N-(4,6-dimethoxy-1,3,5-triazin-2-yl)-N-methyl-                                                         1%                                                 amino]carbonyl]-2-(5 methyl-1H-tetrazol-1-yl)-                                 benzenesulfonamide                                                             N,N-dimethylformamide       9%                                                 attapulgite granules        90%                                                ______________________________________                                    

The active ingredient is dissolved in the solvent and the solution is sprayed upon dedusted granules in a double cone blender. After spraying of the solution has been completed, the blender is allowed to run for a short period and then the granules are packaged.

EXAMPLE 38

Aqueous Suspension

    ______________________________________                                         N-[[N-(4,6-dimethoxy-1,3,5-triazin-2-yl)-N--methyl-                                                        40%                                                amino]carbonyl]-2-(5-methyl-lH-tetrazol-1-yl)-                                 benzenesulfonamide                                                             polyacrylic acid thickener  0.3%                                               dodecylphenol polyethylene glycol ether                                                                    0.5%                                               disodium phosphate          1%                                                 monosodium phosphate        0.5%                                               polyvinyl alcohol           1.0%                                               water                       56.7%                                              ______________________________________                                    

The ingredients are blended and ground together in a sand mill to produce particles essentially all under 5 microns in size.

EXAMPLE 39

Solution

    ______________________________________                                         N-[[N-(4,6-dimethoxy-1,3,5-triazin-2-yl)-N-methyl-                                                         5%                                                 amino]carbonyl]-2-(5-methyl-1H-tetrazol-l-yl)-                                 benzenesulfonamide, sodium salt                                                water                       95%                                                ______________________________________                                    

The salt is added directly to the water with stirring to produce the solution, which may then be packaged for use.

EXAMPLE 40

Low Strength Granule

    ______________________________________                                         N-[[N-(4,6-dimethoxy-1,3,5-triazin-2-yl)-N--methyl-                                                        0.1%                                               amino]carbonyl]-2-(5-methyl-lH-tetrazol-1-yl)-                                 benzenesulfonamide                                                             attapulite granules         99.9%                                              (U.S.S. 20-40 mesh)                                                            ______________________________________                                    

The active ingredient is dissolved in a solvent and the solution is sprayed upon dedusted granules in a double-cone blender. After spraying of the solution has been completed, the material is warmed to evaporate the solvent. The material is allowed to cool and then packaged.

EXAMPLE 41

Granule

    ______________________________________                                         N-[[N-(4,6-dimethoxy-1,3,5-triazin-2-yl)-N-methyl-                                                         80%                                                amino]carbonyl]-2-(5-methyl-lH-tetrazol-1-yl)-                                 benzenesulfonamide                                                             wetting agent               1%                                                 crude ligninsulfonate salt (containing                                                                     10%                                                5-20% of the natural sugars)                                                   attapulgite clay            9%                                                 ______________________________________                                    

The ingredients are blended and milled to pass through a 100 mesh screen. This material is then added to a fluid bed granulator, the air flow is adjusted to gently fluidize the material, and a fine spray of water is sprayed onto the fluidized material. The fluidization and spraying are continued until granules of the desired size range are made. The spraying is stopped, but fluidization is continued, optionally with heat, until the water content is reduced to the desired level, generally less than 1%. The material is then discharged, screened to the desired size range, generally 14-100 mesh (1410-149 microns), and packaged for use.

EXAMPLE 42

High Strength Concentrate

    ______________________________________                                         N-[[N-(4,6-dimethoxy-1,3,5-triazin-2-yl)-N-methyl-                                                         99%                                                amino]carbonyl]-2-(5-methyl-lH-tetrazol-1-yl)-                                 benzenesulfonamide                                                             silica aerogel              0.5%                                               synthetic amorphous silica  0.5%                                               ______________________________________                                    

The ingredients are blended and ground in a hammer mill to produce a material essentially all passing a U.S.S. No. 50 screen (0.3 mm opening). The concentrate may be formulated further if necessary.

EXAMPLE 43

Wettable Powder

    ______________________________________                                         N-[[N-(4,6-dimethoxy-1,3,5-triazin-2-yl)-N-methyl-                                                         90%                                                amino]carbonyl]-2-(5-methyl-lH-tetrazol-1-yl)-                                 benzenesulfonamide                                                             dioctyl sodium sulfosuccinate                                                                              0.1%                                               synthetic fine silica       9.9%                                               ______________________________________                                    

The ingredients are blended and ground in a hammer-mill to produce particles essentially all below 100 microns. The material is sifted through a U.S.S. No. 50 screen and then packaged.

EXAMPLE 44

Wettable Powder

    ______________________________________                                         N-[[N-(4,6-dimethoxy-1,3,5-triazin-2-yl)-N-methyl-                                                         40%                                                amino]carbonyl]-2-(5-methyl-lH-tetrazol-1-yl)-                                 benzenesulfonamide                                                             sodium ligninsulfonate      20%                                                montmorillonite clay        40%                                                ______________________________________                                    

The ingredients are thoroughly blended, coarsely hammer-milled and then air-milled to produce particles essentially all below 10 microns in size. The material is reblended and then packaged.

EXAMPLE 45

Oil Suspension

    ______________________________________                                         N-[[N-(4,6-dimethoxy-1,3,5-triazin-2-yl)-N-methyl-                                                         35%                                                amino]carbonyl]-2-(5-methyl-lH-tetrazol-1-yl)-                                 benzenesulfonamide                                                             blend of polyalcohol carboxylic                                                                            6%                                                 esters and oil soluble petroleum                                               sulfonates                                                                     xylene                      59%                                                ______________________________________                                    

The ingredients are combined and ground together in a sand mill to produce particles essentially all below 5 microns. The product can be used directly, extended with oils, or emulsified in water.

EXAMPLE 46

Dust

    ______________________________________                                         N-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(1-                                                       10%                                                methyl-lH-tetrazol-5-yl)benzenesulfonamide                                     attapulgite                 10%                                                Pyrophyllite                80%                                                ______________________________________                                    

The active ingredient is blended with attapulgite and then passed through a hammer-mill to produce particles substantially all below 200 microns. The ground concentrate is then blended with powdered pyrophyllite until homogeneous.

Utility

Test results indicate that the compounds of the present invention are highly active preemergent or postemergent herbicides or plant growth regulants. They have utility for broad-spectrum pre- and/or post-emergence weed control in areas where complete control of all vegetation is desired, such as around fuel storage tanks, industrial storage areas, parking lots, drive-in theaters, around billboards, highway and railroad structures. Some of the compounds have utility for selective weed control in crops such as corn, rice, wheat, barley, soybean and rape. Alternatively, many of the subject compounds are useful to modify plant growth.

The rates of application for the compounds of the invention are determined by a number of factors, including their use as plant growth modifiers or as herbicides, the crop species involved, the types of weeds to be controlled, weather and climate, formulations selected, mode of application, amount of foliage present, etc. In general terms, the subject compounds should be applied at levels of about 0.001 to 10 kg/ha, the lower rates being suggested for use on lighter soils and/or those having a low organic matter content, for plant growth modification or for situations where only short-term persistence is required.

The compounds of the invention may be used in combination with any other commercial herbicide, examples of which are those of the triazine, triazole, uracil, urea, amide, diphenylether, carbamate, phenoxyacetic acid and bipyridylium types, as well as other sulfonylureas. They are particularly useful in combination with the following herbicides.

    ______________________________________                                         Common Name                                                                              Chemical Name                                                        ______________________________________                                         alachlor  2-chloro-2',6'-diethyl-N-(methoxymethyl)-                                      acetanillde                                                          atrazine  2-chloro-4-(ethylamino)-6-(isopropyl-                                          amino)- .sub.-s-triazine                                             butylate  S-ethyl-diisobutylthiocarbamate                                      cyanazine 2-[[4-chloro-6-(ethylamino)- .sub.-s-triazin-2-                                yl]amino]-2-methylpropionitrile                                      dicamba   3,6-dichloro- -o-anisic acid                                         EPTC      S--ethyl dipropylthiocarbamate                                       glyphosate                                                                               N-(phosphonomethyl)glycine                                           linuron   3-(3,4-dichlorophenyl)-1-methoxy-1-                                            methylurea                                                           metolachlor                                                                              2-chloro-N-(2-ethyl-6-methylphenyl)-N-                                         (2-methoxy-1-methylethyl)acetamide                                   metribuzin                                                                               4-amino-6-tert-butyl-3-(methylthio)-as-                                        triazine-5(4H)-one                                                   tridiphane                                                                               2-(3,5-dichlorophenyl)-2-(2,2,2-tri-                                           chloroethyl)oxirane                                                  2,4-D     (2,4-dichlorophenoxy)acetic acid                                     thiobencarb                                                                              S-4-chlorobenzyldiethylthiocarbamate                                 molinate  S- ethyl N,N- hexamethylenethiocarbamate                             butachlor N-(butoxymethyl)-2-chloro-2',6'-di-                                            ethylacetanilide                                                     naproanilide                                                                             N- phenyl-2-(1-naphthyloxy)propionamide                              paraquat  1,1'-dimethyl-4,4'-bipyridinium ion                                  pyrazolate                                                                               4-(2,4-dichlorobenzoyl)-1,3-dimethyl-                                          pyrazol-5-yl-4-toluenesulfonate                                      pretilachlor                                                                             2-chloro-2',6'-diethyl-N-(n-propoxy-                                           ethyl)acetanilide                                                    oxidiazon 3-[2,4-dichloro-5-(1-methylethoxy)-                                            phenyl[5-(1,1-dimethylethyl)-1,3,4-                                            oxadiazol-2(3H)-one                                                  ______________________________________                                         Trade Name or                                                                  Code Number                                                                              Chemical Name                                                        ______________________________________                                         Harmony ®                                                                            3-[[(4-methoxy-6-methyl-1,3.5-triazin-                                         2-yl)aminocarbonyl]aminosulfonyl]-2-                                           thiophenecarboxylic acid, methyl ester                               Cinch ®                                                                              exo-1-methyl-4-(1-methylethyl)-2-[(2-                                          methylphenyl)methoxy]-7-oxabicyclo-                                            [2.2.1]heptane                                                       MY-93     S-(1-methyl-1-phenethyl)piperidine-1-                                          carbothioate                                                         CH-83     S-(2-methylpropyl)-hexanhydro-lH-aze-                                          pine-1-carbothioic acid, ester                                       X-52      2,4-dichlorophenyl-3-methoxy-4-nitro-                                          phenyl ether                                                         SC-2957   S- benzyl-N--ethyl-N--propylthiocarbamate                            HW-52     N-(2,3-dichlorophenyl)-4-(ethoxy-                                              methoxy)benzamide                                                    NTN-801   2-(benzothiazol-2-yl)-N--methyl-N-                                             phenylacetamide                                                      SL-49     2-[4-[(2,4,dichlorophenyl)carbonyl]-                                           1,3-dimethyl-1H-pyrazol-5-yloxy]-1-                                            phenylethanone                                                       BAS-514   3,7-dichloro-8-quinoline carboxylic                                            acid                                                                 Assure ®                                                                             ethyl 2-[4-(6-chloro-2-quinoxalinyloxy)-                                       phenoxy]-propionate                                                  DPX-L5300 2-[[N-(4-methoxy-6-methyl-1,3,5-tria-                                (Express ®)                                                                          zine-2-yl)-N- methylaminocarbonyl]-                                            aminosulfonyl]benzoic acid, methyl                                             ester                                                                ______________________________________                                    

Some of the compounds of this invention may particularly be useful in combination with the following herbicides for use as pre- or post-emergent treatments for control of weeds of soybeans:

    ______________________________________                                         Common Name                                                                               Tradename  Chemical Name                                            ______________________________________                                         acifluorfen                                                                               Blazer ®                                                                              5-[2-chloro-4-(trifluoro-                                                      methyl)phenoxy]-2-ni-                                                          trobenzoic acid                                          alachlor   Lasso ®                                                                               2-chloro-2',6'-diethyl-                                                        N-(methoxymethyl)acet-                                                         anilide                                                  bentazon   Basagran ®                                                                            3-isopropyl-1H-2,1,3-                                                          benzothiadiazin-4(3H)-                                                         one 2,2-dioxide                                          chloramben Amiben ®                                                                              3-amino-2,5-dichloro-                                                          benzoic acid                                             fluazifop- Fusilade ®                                                                            butyl 2-[4-[5-(trifluoro-                                butyl                 methyl)-2-pyridinyl-                                                           oxy]phenoxy]propanoate                                   linuron    Lorox ®                                                                               3-(3,4-dichlorophenyl)-1-                                                      methoxy-1-methylurea                                     metolachlor                                                                               Dual ® 2-chloro-N-(2-ethyl-6-                                                         methylphenyl)-N-(2-                                                            methoxy-1-methylethyl)-                                                        acetamide                                                metribuzin Lexone ®                                                                              4-amino-6-tert-butyl-3-                                                        (methylthio)-as-tri-                                                           azin-5(4H)one                                            pendimethalin                                                                             Prowl ®                                                                               N-(1-ethylpropyl)-3,4-                                                         dimethyl-2,6-dinitro-                                                          benzeneamine                                             sethoxydim Poast ®                                                                               2-[1-(ethoxyimino)butyl]-                                                      5-[2-(ethylthio)-                                                              propyl]-3-hydroxy-2-                                                           cyclohexene-1-one                                        trifluralin                                                                               Treflan ®                                                                             α,α,α-trifluoro-2,6-di-                                      nitro-N,N- dipropyl-p-                                                         toluidine                                                AC 252,214 --         2-(4,5-dihydro-4-methyl-                                                       4-(1-methylethyl)-5-                                                           oxo-lH-imidazol-2-yl)-                                                         3-quinolinecarboxylic                                                          acid                                                     FMC 57020  --         2-(2'-chlorophenyl)-                                                           methyl-4,4-dimethyl-                                                           3-isoxazolidinone                                        fomesafen  Flex ® 5-(2-chloro-4-trifluoro-                                                       methylphenoxy)-N-                                                              methylsulfonyl-2-nitro-                                                        benzamide                                                lactofen   --         1'-(carboethoxy)ethyl-5-                                                       (2-chloro-4-(trifluoro                                                         methyl)phenoxy)-2-                                                             nitrobenzoate                                            DOWCO 453 ME          2-(4-(3-chloro-5-tri-                                                          fluoromethylpyridin-2-                                                         yloxy)phenoxy)propanoic                                                        acid, methyl ester                                       fenoxaprop ethyl                                                                          Whip ® ethyl 2-(4-(6-chloro-2-                                                        benzoxazolyloxy)phen-                                                          oxy)propanoate                                           CGA 82725  Topik ®                                                                               2-(4-(3,5-dichloropyri-                                                        din-2-yloxy)phenoxy-                                                           propanoic acid, propyn-                                                        yl ester                                                 chlorimuron ethyl                                                                         Classic ®                                                                             2-[[(4-chloro-6-methoxy-                                                       pyrimidin-2-yl)amino-                                                          carbonyl]aminosul-                                                             fonyl]benzoic acid                                                             ethyl ester                                              cinmethylin                                                                               Cinch ®                                                                               exo-1-methyl-4-(1-methyl-                                                      ethyl)-2-[(2-methyl-                                                           phenyl)methoxy]-7-oxa-                                                         bicyclo[2.2.1]heptane                                    AC 263,499 Pursuit ®                                                                             2-[4,5-dihydro-4-methyl-                                                       4-(1-methylethyl)-5-                                                           oxo-lH-imidazol-2-yl)]-                                                        5-ethyl-3-pyridine-                                                            carboxylic acid                                          AC 252,214 Scepter ®                                                                             2-[4,5-dihydro-4-methyl-                                                       4-(1-methylethyl)-5-                                                           oxo-lH-imidazol-2-yl]-                                                         3-quinolinecarboxylic                                                          acid                                                     ______________________________________                                    

The herbicidal properties of the subject compounds were discovered in a number of greenhouse tests. The test procedures and results follow.

    __________________________________________________________________________     COMPOUNDS                                                                      __________________________________________________________________________     General Structures for Compounds 1-58                                           ##STR49##                                                                      ##STR50##                                                                     Compound                                                                               Q   R.sub.1                                                                             R.sub.3                                                                               R.sub.4                                                                              R.sub.5                                                                            X     Y      Z                               __________________________________________________________________________     1       Q-3 H    --     CH.sub.3                                                                             --  OCH.sub.3                                                                            CH.sub.3                                                                              N                               2       Q-3 H    --     CH.sub.3                                                                             --  OCH.sub.3                                                                            OCH.sub.3                                                                             CH                              3       Q-1 H    CH.sub.3                                                                              --    --  OCH.sub.3                                                                            OCH.sub.3                                                                             CH                              4       Q-3 H    --     CH.sub.3                                                                             --  CH.sub.3                                                                             OCH.sub.3                                                                             CH                              5       Q-3 H    --     CH.sub.3                                                                             --  Cl    OCH.sub.3                                                                             CH                              6       Q-3 H    --     CH.sub.3                                                                             --  OCH.sub.3                                                                            OCH.sub.3                                                                             N                               7       Q-3 H    --     CH.sub.3                                                                             --  NHCH.sub.3                                                                           OCH.sub.2 CH.sub.3                                                                    N                               8       Q-3 H    --     H     --  OCH.sub.3                                                                            OCH.sub.3                                                                             N                               9       Q-3 H    --     H     --  Cl    OCH.sub.3                                                                             CH                              10      Q-3 H    --     H     --  CH.sub.3                                                                             OCH.sub.3                                                                             CH                              11      Q-3 H    --     H     --  CH.sub.3                                                                             CH.sub.3                                                                              CH                              12      Q-3 H    --     H     --  CH.sub.3                                                                             OCH.sub.3                                                                             N                               13      Q-3 H    --     H     --  OCH.sub.3                                                                            OCH.sub.3                                                                             CH                              14      Q-3 5-CH.sub.3                                                                          --     CH.sub.3                                                                             --  OCH.sub.3                                                                            OCH.sub. 3                                                                            CH                              15      Q-3 5-CH.sub.3                                                                          --     CH.sub.3                                                                             --  CH.sub.3                                                                             OCH.sub.3                                                                             N                               16      Q-3 5-CH.sub.3                                                                          --     CH.sub.3                                                                             --  Cl    OCH.sub.3                                                                             CH                              17      Q-3 H    --     CH.sub.2 CH.sub.3                                                                    --  CH.sub.3                                                                             OCH.sub.3                                                                             CH                              18      Q-3 H    --     CH.sub.2 CH.sub.3                                                                    --  OCH.sub.3                                                                            OCH.sub.3                                                                             CH                              19      Q-3 H    --     CH.sub.2 CH.sub.3                                                                    --  CH.sub.3                                                                             CH.sub.3                                                                              CH                              20      Q-3 H    --     CH.sub.2 CH.sub.3                                                                    --  Cl    OCH.sub.3                                                                             CH                              21      Q-3 H    --     CH.sub.2 CH.sub.3                                                                    --  OCH.sub.3                                                                            OCH.sub.3                                                                             N                               22      Q-3 H    --     CH.sub.2 CH.sub.3                                                                    --  CH.sub.3                                                                             OCH.sub.3                                                                             N                               23      Q-3 5-Cl --     CH.sub.3                                                                             --  OCH.sub.3                                                                            OCH.sub.3                                                                             CH                              24      Q-3 5-Cl --     CH.sub.3                                                                             --  CH.sub.3                                                                             OCH.sub.3                                                                             CH                              25      Q-3 5-Cl --     CH.sub.3                                                                             --  OCH.sub.3                                                                            OCH.sub.3                                                                             N                               26      Q-3 5-Cl --     CH.sub.3                                                                             --  CH.sub.3                                                                             OCH.sub.3                                                                             N                               27      Q-3 5-Cl --     CH.sub.3                                                                             --  CH.sub.3                                                                             CH.sub.3                                                                              CH                              28      Q-3 5-Cl --     CH.sub.3                                                                             --  Cl    OCH.sub.3                                                                             CH                              29      Q-3 5-Cl --     CH.sub.3                                                                             --  NHCH.sub.3                                                                           OCH.sub.2 CH.sub.3                                                                    N                               30      Q-1 H    CH.sub.2 CH.sub.3                                                                     --    --  OCH.sub.3                                                                            OCH.sub.3                                                                             N                               31      Q-1 H    CH.sub.2 CH.sub.3                                                                     --    --  CH.sub.3                                                                             OCH.sub.3                                                                             N                               32      Q-1 H    CH.sub.2 CH.sub.3                                                                     --    --  OCH.sub.3                                                                            OCH.sub.3                                                                             CH                              33      Q-1 H    CH.sub.2 CH.sub.3                                                                     --    --  CH.sub.3                                                                             OCH.sub.3                                                                             CH                              34      Q-1 H    CH.sub.2 CH.sub.3                                                                     --    --  CH.sub.3                                                                             CH.sub.3                                                                              CH                              35      Q-1 H    CH.sub.2 CH.sub.3                                                                     --    --  Cl    OCH.sub.3                                                                             CH                              36      Q-1 H    CH.sub.2 CH.sub.3                                                                     --    --  NHCH.sub.3                                                                           OCH.sub.2 CH.sub.3                                                                    N                               37      Q-1 3-CH.sub.3                                                                          CH.sub.3                                                                              --    --  OCH.sub.3                                                                            OCH.sub.3                                                                             N                               38      Q-1 3-CH.sub.3                                                                          CH.sub.3                                                                              --    --  CH.sub.3                                                                             OCH.sub.3                                                                             N                               39      Q-1 3-CH.sub.3                                                                          CH.sub.3                                                                              --    --  OCH.sub.3                                                                            OCH.sub.3                                                                             CH                              40      Q-1 3-CH.sub.3                                                                          CH.sub.3                                                                              --    --  CH.sub.3                                                                             OCH.sub.3                                                                             CH                              41      Q-1 3-CH.sub.3                                                                          CH.sub.3                                                                              --    --  CH.sub.3                                                                             CH.sub.3                                                                              CH                              42      Q-1 3-CH.sub.3                                                                          CH.sub.3                                                                              --    --  Cl    OCH.sub.3                                                                             CH                              43      Q-1 3-CH.sub.3                                                                          CH.sub.3                                                                              --    --  NHCH.sub.3                                                                           OCH.sub.2 CH.sub.3                                                                    N                               44      Q-1 4-CH.sub.3                                                                          CH.sub.3                                                                              --    --  OCH.sub.3                                                                            OCH.sub.3                                                                             N                               45      Q-1 4-CH.sub.3                                                                          CH.sub.3                                                                              --    --  CH.sub.3                                                                             OCH.sub.3                                                                             N                               46      Q-1 4-CH.sub.3                                                                          CH.sub.3                                                                              --    --  OCH.sub.3                                                                            OCH.sub.3                                                                             CH                              47      Q-1 4-CH.sub.3                                                                          CH.sub.3                                                                              --    --  CH.sub.3                                                                             OCH.sub.3                                                                             CH                              48      Q-1 4-CH.sub.3                                                                          CH.sub.3                                                                              --    --  CH.sub.3                                                                             CH.sub.3                                                                              CH                              49      Q-1 4-CH.sub.3                                                                          CH.sub.3                                                                              --    --  Cl    OCH.sub.3                                                                             CH                              50      Q-1 4-CH.sub.3                                                                          CH.sub.3                                                                              --    --  NHCH.sub.3                                                                           OCH.sub.2 CH.sub.3                                                                    N                               51      Q-1 6-CH.sub.3                                                                          CH.sub.3                                                                              --    --  OCH.sub.3                                                                            OCH.sub.3                                                                             N                               52      Q-1 6-CH.sub.3                                                                          CH.sub.3                                                                              --    --  CH.sub.3                                                                             OCH.sub.3                                                                             N                               53      Q-1 6-CH.sub.3                                                                          CH.sub.3                                                                              --    --  OCH.sub.3                                                                            OCH.sub.3                                                                             CH                              54      Q-1 6-CH.sub.3                                                                          CH.sub. 3                                                                             --    --  CH.sub.3                                                                             OCH.sub.3                                                                             CH                              55      Q-1 6-CH.sub.3                                                                          CH.sub.3                                                                              --    --  CH.sub.3                                                                             CH.sub.3                                                                              CH                              56      Q-1 6-CH.sub.3                                                                          CH.sub.3                                                                              --    --  Cl    OCH.sub.3                                                                             CH                              57      Q-5 H    --     --    CH.sub.3                                                                           OCH.sub.3                                                                            OCH.sub.3                                                                             CH                              58      Q-5 H    --     --    CH.sub.3                                                                           CH.sub.3                                                                             OCH.sub.3                                                                             N                               __________________________________________________________________________     General Structures for Compounds 59-63                                          ##STR51##                                                                     Compound            X          Y          Z                                    __________________________________________________________________________     59                  OCH.sub.3  OCH.sub.3  CH                                   60                  CH.sub.3   OCH.sub.3  CH                                   61                  CH.sub.3   CH.sub.3   CH                                   62                  OCH.sub.3  OCH.sub.3  N                                    63                  Cl         OCH.sub.3  CH                                   __________________________________________________________________________     General Structures for Compounds 64-179                                         ##STR52##                                                                      ##STR53##                                                                     Compound                                                                             Q  R  R.sub.1                                                                             R.sub.3                                                                             R.sub.4 R.sub.5                                                                             X      Y       Z                            __________________________________________________________________________     64    Q-1                                                                               H  6-Cl CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.3                                                                              N                            65    Q-1                                                                               H  6-Cl CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.3                                                                              N                            66    Q-1                                                                               H  6-Cl CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.3                                                                              CH                           67    Q-1                                                                               H  6-Cl CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.3                                                                              CH                           68    Q-1                                                                               H  6-Cl CH.sub.3                                                                            --      --   CH.sub.3                                                                              CH.sub.3                                                                               CH                           69    Q-1                                                                               H  6-Cl CH.sub.3                                                                            --      --   Cl     OCH.sub.3                                                                              CH                           70    Q-1                                                                               H  3-Cl CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.3                                                                              N                            71    Q-1                                                                               H  3-Cl CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.3                                                                              N                            72    Q-1                                                                               H  3-Cl CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.3                                                                              CH                           73    Q-1                                                                               H  3-Cl CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.3                                                                              CH                           74    Q-1                                                                               H  3-Cl CH.sub.3                                                                            --      --   CH.sub.3                                                                              CH.sub.3                                                                               CH                           75    Q-1                                                                               H  3-Cl CH.sub.3                                                                            --      --   Cl     OCH.sub.3                                                                              CH                           76    Q-3                                                                               H  H    --   OCH.sub.2 CH.sub.3                                                                     --   OCH.sub.3                                                                             OCH.sub.3                                                                              CH                           77    Q-3                                                                               H  H    --   OCH.sub.2 CH.sub.3                                                                     --   CH.sub.3                                                                              OCH.sub.3                                                                              CH                           78    Q-3                                                                               H  H    --   OCH.sub.2 CH.sub.3                                                                     --   CH.sub.3                                                                              CH.sub.3                                                                               CH                           79    Q-3                                                                               H  H    --   OCH.sub.2 CH.sub.3                                                                     --   Cl     OCH.sub.3                                                                              CH                           80    Q-3                                                                               H  H    --   OCH.sub.2 CH.sub.3                                                                     --   OCH.sub.3                                                                             OCH.sub.3                                                                              N                            81    Q-3                                                                               H  H    --   OCH.sub.2 CH.sub.3                                                                     --   CH.sub.3                                                                              OCH.sub.3                                                                              N                            82    Q-3                                                                               H  H    --   OCH.sub.3                                                                              --   OCH.sub.3                                                                             OCH.sub.3                                                                              CH                           83    Q-3                                                                               H  H    --   OCH.sub.3                                                                              --   CH.sub.3                                                                              OCH.sub.3                                                                              CH                           84    Q-3                                                                               H  H    --   OCH.sub.3                                                                              --   CH.sub.3                                                                              CH.sub.3                                                                               CH                           85    Q-3                                                                               H  H    --   OCH.sub.3                                                                              --   Cl     OCH.sub.3                                                                              CH                           86    Q-3                                                                               H  H    --   OCH.sub.3                                                                              --   OCH.sub.3                                                                             OCH.sub.3                                                                              N                            87    Q-3                                                                               H  H    --   OCH.sub.3                                                                              --   CH.sub.3                                                                              OCH.sub.3                                                                              N                            88    Q-3                                                                               H  H    --   OCH.sub.2 CH.sub.2 CH.sub.3                                                            --   OCH.sub.3                                                                             OCH.sub.3                                                                              CH                           89    Q-3                                                                               H  H    --   OCH.sub. 2 CH.sub.2 CH.sub.3                                                           --   CH.sub.3                                                                              OCH.sub.3                                                                              CH                           90    Q-3                                                                               H  H    --   OCH.sub.2 CH.sub.2 CH.sub.3                                                            --   CH.sub.3                                                                              CH.sub.3                                                                               CH                           91    Q-3                                                                               H  H    --   OCH.sub.2 CH.sub.2 CH.sub.3                                                            --   Cl     OCH.sub.3                                                                              CH                           92    Q-3                                                                               H  H    --   OCH.sub.2 CH.sub.2 CH.sub.3                                                            --   OCH.sub.3                                                                             OCH.sub.3                                                                              N                            93    Q-3                                                                               H  H    --   OCH.sub.2 CH.sub.2 CH.sub.3                                                            --   CH.sub.3                                                                              OCH.sub.3                                                                              N                            94    Q-1                                                                               H  6-Cl CH.sub.3                                                                            --      --   OCF.sub.2 H                                                                           OCH.sub.3                                                                              CH                           95    Q-1                                                                               H  6-Cl CH.sub.3                                                                            --      --   OCF.sub.2 H                                                                           CH.sub.3                                                                               CH                           96    Q-1                                                                               H  H    CH.sub.2 CH.sub.3                                                                   --      --   OCF.sub.2 H                                                                           OCH.sub.3                                                                              CH                           97    Q-1                                                                               H  5-F  CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.3                                                                              CH                           98    Q-1                                                                               H  5-F  CH.sub.3                                                                            --      --   Cl     OCH.sub.3                                                                              CH                           99    Q-5                                                                               H  5-CH.sub.3                                                                          --   --      CH.sub.2 CH.sub.3                                                                   OCH.sub.3                                                                             OCH.sub.3                                                                              CH                           100   Q-5                                                                               H  5-CH.sub.3                                                                          --   --      CH.sub.2 CH.sub.3                                                                   Cl     OCH.sub.3                                                                              CH                           101   Q-5                                                                               H  5-CH.sub.3                                                                          --   --      CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                              CH.sub.3                                                                               CH                           102   Q-5                                                                               H  5-CH.sub.3                                                                          --   --      CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                              OCH.sub.3                                                                              CH                           103   Q-1                                                                               H  5-OCH.sub.3                                                                         CH.sub.3                                                                            --      --   Cl     OCH.sub.3                                                                              CH                           104   Q-1                                                                               H  5-OCH.sub.3                                                                         CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.3                                                                              CH                           105   Q-1                                                                               H  5-OCH.sub.3                                                                         CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.3                                                                              CH                           106   Q-1                                                                               H  5-OCH.sub.3                                                                         CH.sub.3                                                                            --      --   CH.sub.3                                                                              CH.sub.3                                                                               CH                           107   Q-3                                                                               H  5-CH.sub.3                                                                          --   OCH.sub.3                                                                              --   OCH.sub.3                                                                             OCH.sub.3                                                                              CH                           108   Q-3                                                                               H  5-CH.sub.3                                                                          --   OCH.sub.3                                                                              --   CH.sub.3                                                                              OCH.sub.3                                                                              CH                           109   Q-3                                                                               H  5-CH.sub.3                                                                          --   OCH.sub.3                                                                              --   CH.sub.3                                                                              CH.sub.3                                                                               CH                           110   Q-3                                                                               H  5-CH.sub.3                                                                          --   OCH.sub.3                                                                              --   Cl     OCH.sub.3                                                                              CH                           111   Q-3                                                                               H  5-CH.sub.3                                                                          --   OCH.sub.3                                                                              --   OCH.sub.3                                                                             OCH.sub.3                                                                              N                            112   Q-3                                                                               H  5-CH.sub.3                                                                          --   OCH.sub.3                                                                              --   CH.sub.3                                                                              OCH.sub.3                                                                              N                            113   Q-1                                                                               H  5-F  CH.sub. 3                                                                           --      --   OCH.sub.3                                                                             OCH.sub.3                                                                              N                            114   Q-1                                                                               H  5-F  CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.3                                                                              N                            115   Q-1                                                                               H  5-F  CH.sub.3                                                                            --      --   CH.sub.3                                                                              CH.sub.3                                                                               CH                           116   Q-1                                                                               H  5-F  CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.3                                                                              CH                           117   Q-5                                                                               H  5-CH.sub.3                                                                          --   --      CH.sub.2 CH.sub.3                                                                   OCH.sub.3                                                                             OCH.sub.3                                                                              N                            118   Q-5                                                                               H  5-CH.sub.3                                                                          --   --      CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                              OCH.sub.3                                                                              N                            119   Q-1                                                                               H  6-OCH.sub.3                                                                         CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.3                                                                              CH                           120   Q-1                                                                               H  6-OCH.sub.3                                                                         CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.3                                                                              N                            121   Q-1                                                                               H  6-OCH.sub.3                                                                         CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.3                                                                              CH                           122   Q-1                                                                               H  6-OCH.sub.3                                                                         CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.3                                                                              N                            123   Q-1                                                                               H  6-OCH.sub.3                                                                         CH.sub.3                                                                            --      --   Cl     OCH.sub.3                                                                              CH                           124   Q-1                                                                               H  6-OCH.sub.3                                                                         CH.sub.3                                                                            --      --   CH.sub.3                                                                              CH.sub.3                                                                               CH                           125   Q-5                                                                               H  H    --   --      CH.sub.2 CH.sub.3                                                                   OCH.sub.3                                                                             OCH.sub.3                                                                              CH                           126   Q-5                                                                               H  H    --   --      CH.sub.2 CH.sub.3                                                                   OCH.sub.3                                                                             OCH.sub.3                                                                              N                            127   Q-5                                                                               H  H    --   --      CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                              OCH.sub.3                                                                              CH                           128   Q-5                                                                               H  H    --   --      CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                              OCH.sub.3                                                                              N                            129   Q-5                                                                               H  H    --   --      CH.sub.2 CH.sub.3                                                                   Cl     OCH.sub.3                                                                              CH                           130   Q-5                                                                               H  H    --   --      CH.sub.2 CH.sub.3                                                                   CH.sub.3                                                                              CH.sub.3                                                                               CH                           131   Q-3                                                                               H  5-OCH.sub.3                                                                         --   OCH.sub.3                                                                              --   OCH.sub.3                                                                             OCH.sub.3                                                                              CH                           132   Q-3                                                                               H  5-OCH.sub.3                                                                         --   OCH.sub.3                                                                              --   CH.sub.3                                                                              OCH.sub.3                                                                              CH                           133   Q-3                                                                               H  5-OCH.sub.3                                                                         --   OCH.sub.3                                                                              --   CH.sub.3                                                                              CH.sub.3                                                                               CH                           134   Q-3                                                                               H  5-OCH.sub.3                                                                         --   OCH.sub.3                                                                              --   Cl     OCH.sub.3                                                                              CH                           135   Q-3                                                                               H  5-OCH.sub.3                                                                         --   OCH.sub.3                                                                              --   OCH.sub.3                                                                             OCH.sub.3                                                                              N                            136   Q-3                                                                               H  5-OCH.sub.3                                                                         --   OCH.sub.3                                                                              --   CH.sub.3                                                                              OCH.sub.3                                                                              N                            137   Q-1                                                                               H  6-CH.sub.3                                                                          CH.sub.3                                                                            --      --   Br     OCH.sub.3                                                                              CH                           138   Q-1                                                                               CH.sub. 3                                                                         6-CH.sub.3                                                                          CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.3                                                                              CH                           139   Q-1                                                                               CH.sub.3                                                                          6-CH.sub.3                                                                          CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.3                                                                              N                            140   Q-1                                                                               H  6-CH.sub.3                                                                          CH.sub.3                                                                            --      --   CH.sub.3                                                                              H       CH                           141   Q-1                                                                               H  6-CH.sub.3                                                                          CH.sub.3                                                                            --      --   OCH.sub.3                                                                             H       CH                           142   Q-1                                                                               H  6-CH.sub.3                                                                          CH.sub.3                                                                            --      --   CH.sub.2 CH.sub.3                                                                     OCH.sub.3                                                                              CH                           143   Q-1                                                                               H  6-CH.sub.3                                                                          CH.sub.3                                                                            --      --   CH.sub.2 CH.sub.3                                                                     OCH.sub.3                                                                              N                            144   Q-1                                                                               CH.sub.3                                                                          6-CH.sub.3                                                                          CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.3                                                                              N                            145   Q-1                                                                               H  6-CH.sub.3                                                                          CH.sub.3                                                                            --      --   cyclopropyl                                                                           OCH.sub.3                                                                              N                            146   Q-1                                                                               H  6-CH.sub.3                                                                          CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.2 CH.sub.3                                                                     CH                           147   Q-1                                                                               H  6-CH.sub.3                                                                          CH.sub.3                                                                            --      --   OCH.sub.3                                                                             CH.sub.2 OCH.sub.2 CH.sub.3                                                            CH                           148   Q-1                                                                               H  6-CH.sub.3                                                                          CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.2 CF.sub.3                                                                     N                            149   Q-1                                                                               H  6-CH.sub.3                                                                          CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.2 CH.sub.3                                                                     N                            150   Q-1                                                                               H  5-Cl CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.3                                                                              N                            151   Q-1                                                                               H  5-Cl CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.3                                                                              N                            152   Q-1                                                                               H  5-Cl CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.3                                                                              CH                           153   Q-1                                                                               H  5-Cl CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.3                                                                              CH                           154   Q-1                                                                               H  5-Cl CH.sub.3                                                                            --      --   CH.sub.3                                                                              CH.sub.3                                                                               CH                           155   Q-1                                                                               H  5-Cl CH.sub.3                                                                            --      --   Cl     OCH.sub.3                                                                              CH                           156   Q-1                                                                               H  5-Cl CH.sub.3                                                                            --      --   OCH.sub.2 CH.sub.3                                                                    NHCH.sub.3                                                                             N                            157   Q-1                                                                               H  5-Cl CH.sub.3                                                                            --      --   OCH.sub.3                                                                             CH(OCH.sub.3).sub.2                                                                    CH                           158   Q-5                                                                               H  5-Cl --   --      CH.sub.3                                                                            OCH.sub.3                                                                             OCH.sub.3                                                                              CH                           159   Q-5                                                                               H  5-Cl --   --      CH.sub.3                                                                            CH.sub.3                                                                              OCH.sub.3                                                                              CH                           160   Q-5                                                                               H  5-Cl --   --      CH.sub.3                                                                            CH.sub.3                                                                              OCH.sub.3                                                                              N                            161   Q-1                                                                               H  6-CH.sub.3                                                                          CH.sub.3                                                                            --      --   OCF.sub.2 H                                                                           OCH.sub.3                                                                              CH                           162   Q-1                                                                               H  6-CH.sub.3                                                                          CH.sub.3                                                                            --      --   OCF.sub. 2 H                                                                          CH.sub.3                                                                               CH                           163   Q-1                                                                               H  H    CH.sub.3                                                                            --      --   CH.sub.3                                                                              CH.sub.3                                                                               CH                           164   Q-1                                                                               H  H    CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.3                                                                              CH                           165   Q-1                                                                               H  H    CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.3                                                                              CH                           166   Q-1                                                                               H  H    CH.sub.3                                                                            --      --   Cl     OCH.sub.3                                                                              CH                           167   Q-1                                                                               H  H    CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.3                                                                              N                            168   Q-1                                                                               H  H    CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.3                                                                              N                            169   Q-1                                                                               H  H    CH.sub.3                                                                            --      --   OCH.sub.2 CH.sub.3                                                                    NHCH.sub.3                                                                             N                            170   Q-1                                                                               H  H    CH.sub.3                                                                            --      --   OCF.sub.2 H                                                                           OCH.sub.3                                                                              CH                           171   Q-5                                                                               H  H    --           CH.sub.3                                                                            OCF.sub.2 H                                                                           OCH.sub.3                                                                              CH                           172   Q-5                                                                               H  H    --   --      CH.sub.3                                                                            OCF.sub.2 H                                                                           CH.sub.3                                                                               CH                           173   Q-1                                                                               H  H    CH.sub.3                                                                            --      --   OCF.sub.2 H                                                                           CH.sub.3                                                                               CH                           174   Q-1                                                                               H  5-CH.sub.3                                                                          CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.3                                                                              N                            175   Q-1                                                                               H  5-CH.sub.3                                                                          CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.3                                                                              N                            176   Q-1                                                                               H  5-CH.sub.3                                                                          CH.sub.3                                                                            --      --   OCH.sub.3                                                                             OCH.sub.3                                                                              CH                           177   Q-1                                                                               H  5-CH.sub.3                                                                          CH.sub.3                                                                            --      --   CH.sub.3                                                                              OCH.sub.3                                                                              CH                           178   Q-1                                                                               H  5-CH.sub.3                                                                          CH.sub.3                                                                            --      --   CH.sub.3                                                                              CH.sub.3                                                                               CH                           179   Q-1                                                                               H  5-CH.sub.3                                                                          CH.sub.3                                                                            --      --   Cl     OCH.sub.3                                                                              CH                           __________________________________________________________________________     General Structure for Compounds 180-205                                         ##STR54##                                                                      ##STR55##                                                                     Compound    Q     R.sub.1                                                                              R.sub.3                                                                              X      Y       Z                                 __________________________________________________________________________     180         Q-2   CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                              CH.sub.3                                                                               CH                                181         Q-2   CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                              OCH.sub.3                                                                              CH                                182         Q-2   CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                183         Q-2   CH.sub.3                                                                             CH.sub.3                                                                             Cl     OCH.sub.3                                                                              CH                                184         Q-2   CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.2 CH.sub.3                                                                    NHCH.sub.3                                                                             N                                 185         Q-2   CH.sub.3                                                                             CH.sub.3                                                                             CH.sub.3                                                                              OCH.sub.3                                                                              N                                 186         Q-2   CH.sub.3                                                                             CH.sub.3                                                                             OCH.sub.3                                                                             OCH.sub.3                                                                              N                                 187         Q-2   H     CH.sub.3                                                                             CH.sub.3                                                                              CH.sub.3                                                                               CH                                188         Q-2   H     CH.sub.3                                                                             CH.sub.3                                                                              OCH.sub.3                                                                              CH                                189         Q-2   H     CH.sub.3                                                                             OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                190         Q-2   H     CH.sub.3                                                                             Cl     OCH.sub.3                                                                              CH                                191         Q-2   H     CH.sub.3                                                                             CH.sub.3                                                                              OCH.sub.3                                                                              N                                 192         Q-2   H     CH.sub.3                                                                             OCH.sub.3                                                                             OCH.sub.3                                                                              N                                 193         Q-2   H     CH.sub.3                                                                             OCH.sub.2 CH.sub.3                                                                    NHCH.sub.3                                                                             N                                 194         Q-1   H     CH.sub.3                                                                             CH.sub.3                                                                              OCH.sub.3                                                                              CH                                195         Q-1   H     CH.sub.3                                                                             OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                196         Q-1   H     CH.sub.3                                                                             CH.sub.3                                                                              CH.sub.3                                                                               CH                                197         Q-1   H     CH.sub.3                                                                             Cl     OCH.sub.3                                                                              CH                                198         Q-1   H     CH.sub.3                                                                             CH.sub.3                                                                              OCH.sub.3                                                                              N                                 199         Q-1   H     CH.sub.3                                                                             OCH.sub.3                                                                             OCH.sub.3                                                                              N                                 200         Q-2   H     CH.sub.2 CH.sub.3                                                                    CH.sub.3                                                                              CH.sub.3                                                                               CH                                201         Q-2   H     CH.sub.2 CH.sub.3                                                                    CH.sub.3                                                                              OCH.sub.3                                                                              CH                                202         Q-2   H     CH.sub.2 CH.sub.3                                                                    OCH.sub.3                                                                             OCH.sub.3                                                                              CH                                203         Q-2   H     CH.sub.2 CH.sub.3                                                                    Cl     OCH.sub.3                                                                              CH                                204         Q-2   H     CH.sub.2 CH.sub.3                                                                    CH.sub.3                                                                              OCH.sub.3                                                                              N                                 205         Q-2   H     CH.sub.2 CH.sub.3                                                                    OCH.sub.3                                                                             OCH.sub.3                                                                              N                                 __________________________________________________________________________     General Structure for Compounds 206-207                                        Compound                                                                       __________________________________________________________________________     206                                                                                                   ##STR56##                                               207                   sodium salt of compound 206                              __________________________________________________________________________          TEST A

Seeds of crabgrass (Digitaria spp.), giant foxtail (Setaria faberii) (in some cases), barnyardgrass (Echinochloa crus-galli), cheatgrass (Bromus secalinus), wild oats, (Avena fatua), velvetleaf (Abutilon theo-phrasti), morningglory (Ipomoea spp.), cocklebur (Xanthium pensylvanicum), sorghum, corn, soybean, sugarbeet, cotton, rice, barley (in some cases), wheat and purple nutsedge (Cyperus rotundus) tubers were planted and treated preemergence with the test chemicals dissolved in a non-phytotoxic solvent. At the same time, these crops and weed species were treated with a soil/foliage application. At the time of treatment, the plants ranged in height from 2 to 18 cm. Treated plants and controls were maintained in a greenhouse for sixteen days, after which all species were compared to controls and visually rated for response to treatment. The ratings, summarized in Table A, are based on a numerical scale extending from 0=no injury, to 10=complete kill. The accompanying description symbols have the following meanings:

C=chlorosis/necrosis;

B=burn;

D=defoliation;

E=emergence inhibition;

G=growth retardation;

H=formative effect;

U=unusual pigmentation;

X=axillary stimulation;

S=albinism; and

6Y=abscised buds or flowers.

    TABLE A       Cmpd. 1 Cmpd. 2 Cmpd. 3 Compound 4 Compound 5 Compound 6 Compound 7      Compound 8 Compound 9 Compound 10 Compound 11 Rate kg/ha 0.05 0.05 0.05      0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.05 0.01 0.05 0.01 0.05      0.01 0.05 0.01        POSTEMERGENCE                      Morningglory 3C,8G 10C 10C 10C 10C      10C 9C 1C,1H 1C 6C,9G 4C,9H 1H 3H 0 5C,9G 2C,5G 10C 9C 2C,6G 2H Cocklebur       3C,7H 9C 9C 9C 9C 10C 9C 1H 0 8G 2G 0 2H 0 9C 3C,9H 9C 9C 9C 5C,9G      Velvetleaf 2C,4G 10C 9C 9C 9C 9C 4C,9H 0 0 4C,8H 3C,5G 2G 0 0 4C,8G 1C      9C 4C,8G 5C,9H 4C,9H Nutsedge 8G 9C 9C 4C,9G 3C,9G 9C 4C,9G 0 0 6G 0 0 0      0 4C,9G 3C,9G 9C 9C 4C,9G 3C,9G Crabgrass 5G 5C,9G 9C 5C,9G 3C,8G 4C,8G      3C,5G 0 0 4C,8G 2C,5G 0 0 0 2G 0 3C,7G 2H 3C,5G 1H Giant Foxtail    --      -- -- -- -- -- -- -- 0 -- -- -- -- -- -- -- -- Barnyardgrass 5C,9G 9C      5C,9G 9C 9C 9C 9C 4C,9H 0 5C,9H 3C,9H 1H 2H 0 9H 2C,5H 9H 3C,7H 5C,9H      2C,3H Cheatgrass 0 7G 9C 3C,9G 6G 4G 0 0 0 6G 2G 0 0 0 7G 0 9C 3C,9G 9C      8G Wild Oats 3C,8G 9C 9C 5C,9G 5C,9G 4C,9G 3C,9G 2G 0 5C,9G 4C,9G 0 0 0      0 0 5C,9G 2C,7H 9C 9H Wheat 4C,9G 9C 9C 5C,9G 2C,9G 4C,9H 8G 3G 0 4C,9G      2C,9G 0 0 0 0 0 9G 3G 9G 5G Corn 9C 9C 9C 5C,9G 3C,9H 5C,9G 9H 4C,9H      3C,7H 6C,9G 4C,9H 5H 5H 2G 7H 1C,3G 9C 3C,9H 5C,9G 3C,9H Barley    -- --      -- -- -- -- -- -- 0 -- -- -- -- -- -- -- -- Soybean 5C,9G 9C 9C 5C,9G      5C,9G 4C,9G 4C,9H 4C,8H 1C,1H 3C,7G 3G 2G 3H 0 5G 0 5C,9G 3C,8H 3C,7H 2H      Rice 6C,9G 9C 9C 9C 9C 6C,9G 9C 5C,9G 5G 9C 9C 2G 2G 0 4C,8G 0 9C 2C,7G      9C 5C,9G Sorghum 6C,9H 9C 9C 5C,9G 6C,9G 9C 9C 4C,8H 3G 5C,9G 4C,9H 5G 0      0 5C,9H 3C,8H 9C 3C,9H 9C 4C,9H Sugar Beets 6C,9H 9C 9C 8G 10C 9C 9C      4C,6G 0 5C,9H 4C,6H 2C,3H 3C,5H 0 10C 4C,9H 10C 10C 9C 9C Cotton 6C,9H      9C 9C 9C 9C 9C 4C,9G 4C,6G 3C,4G 3C,5G 3C,5G 2G 0 0 9C 3C,8H 9C 9C 9C 9H P      REEEMERGENCE                      Morningglory 3G 9H 9G 9G 9G 9G 9G 0 0      9G 7G 0 0 0 9G 4C,8H 9G 8G 8G 3C,5H Cocklebur 0 9H 9H 9H 9H 9H 9H 0 0 8G      7G 0 0 0 8H 2C,5G -- 9H 9H 8H Velvetleaf 0 10C 10C 9C 9C 9C 4C,8G 0 0      4C,9G 0 0 0 0 7H 4G 9C 6C,9G 9C 3C,7H Nutsedge 0 10E 10E 10E 4C,8G 10E      10E 0 0 0 0 0 0 0 10E 3G 10E 9G 10E 4G Crabgrass 0 3C,8G 8G 5C,9G 5C,9G      4C,9G 7G 0 0 4C,8G 0 0 0 0 2C 0 4C,7G 2C,4G 2C,3G 0 Giant Foxtail    --      -- -- -- -- -- -- -- 0 -- -- -- -- -- -- -- -- Barnyardgrass 0 4C,9H 9H      5C,9H 5C,9H 4C,9H 4C,9H 0 0 9H 3G 0 0 0 3C,7G 0 4C,9H 2C,6G 3C,5G 0      Cheatgrass 0 7G 9H 9G 7G 5G 3G 0 0 5G 0 0 0 0 3C,7H 4G 10E 4C,9H 5C,9H      5G Wild Oats 0 5C,9G 5C,9G 6C,9H 4C,8H 5C,9G 3C,7G 0 0 5C,9H 3C,6G 0 1C      0 2C,7G 0 9C 4C,9G 9C 3C,7G Wheat 5G 10E 10E 10E 5C,9H 4C,9H 9G 4G 0      4C,9H 2C,6G 0 0 0 6G 0 4C,9G 7G 9G 5G Corn 3C,8G 4C,9G 3C,9H 9H 5C,9H      3C,9G 8G 2G 0 9G 3C,7G 0 4G 0 3C,8H 0 9H 4C,9H 2C,9H 3C,7H Barley    --      -- -- -- -- -- -- -- 0 -- -- -- -- -- -- -- -- Soybean 5G 9H 9H 9H 4C,7G      3C,8H 4C,6G 0 0 2G 0 0 2G 0 3G 0 9H 4C,8H 2C,7G 2C,3G Rice 1C 10E 10E      10E 10E 10E 10E 3G 0 10E 4C,8H 0 5G 0 10E 7G 10E 4C,9H 10E 3C,8G Sorghum      3C,6G 5C,9H 10H 10E 5C,9H 10E 9H 0 0 10E 4C,9H 0 0 0 4C,9H 4C,8G 10E      5C,9H 9H 3C,8H Sugar Beets 0 5C,9G 9C 5C,9G 5C,9G 5C,9G 5C,9G 0 0 5C,9G      4C,8G 0 4G 3H 9C 4C,8G 5C,9G 5C,9G 9C 5C,9G Cotton 0 3C,9G 9C 3C,9G      3C,9G 3C,9G 3C,9G 0 0 2C,5G 0 0 0 0 9G 8G 9C 9G 9G 9G        Cmpd. 12 Cmpd. 13 Compound 14 Compound 15 Compound 16 Compound 17      Compound 18 Compound 19 Compound 20  Compound 21 Compound 22 Rate kg/ha      0.01 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01      0.05 0.01 0.05 0.01 0.05 0.01        POSTEMERGENCE                      Morningglory 2G 10C 5C,9G 4G 3C,8H      0 10C 5C,9G 10C 10C 10C 9C 10C 4C,9G 10C 9C 4C,9G 3C,7H 4C,8H 3C,7H      Cocklebur 0 10C 10C 10C 2C,4G 0 10C 8G 10C 10C 10C 10C 9C 7G 10C 9C      5C,9H 5H 5C,9G 3C,7H Velvetleaf 0 9C 10C 10C 2C,4H 0 9C 3C,8G 9C 9C 10C      9C 9C 9C 9C 2C,7G 3C,6G 1H 3C,7H 3C,5H Nutsedge 0 9C 9C 5C,9G 0 0 5C,9G      2C,8G 5C,9G 3C,9G 10C 10C 5C,9G 3C,8G 5C,9G 4C,9G 4G 3C,8G 5G 0 Crabgrass       0 4G 2C,7G 1C 0 0 5G 0 3C,8G 3C,5G 9C 3C,7G 4C,8G 3C,4G 3C,7G 3C,3G      3C,5G 2G 3C,7H 3C,6G Giant Foxtail -- -- -- -- -- -- -- -- 9C 9C 9C      5C,9H 9C 5C,9G 5C,9H 4C,8G 9C 4C,9G 9C 4C,9H Barnyardgrass 0 5C,9H 9C 9C      3C,8H 3G 9C 3C,8H 9C 9C 9C 9C 9C 9C 9C 9C 9C 9C 9C 9C Cheatgrass 0 4C,9G      3G 0 0 0 0 0 5C,9G 3C,8G 9C 2C,8G 3C,7G 5G 5G 2G 0 0 2C 0 Wild Oats 0      3C,5G 5C,9G 3C,9G 2C,9G 2C,2G 3C,9G 2C,5G 9C 5C,9G 5C,9G 4C,9G 9C 9C      3C,9G 3C,7G 2C 0 2C,6G 0 Wheat 0 0 5C,9G 2C,9G 0 0 8G 5G 4C,9G 9G 9C      3C,9G 9C 5C,9G 3C,9G 9G 5G 0 8G 0 Corn 0 9H 9C 5C,9H 1C,5G 2G 4G 2G 9C      5C,9G 10C 3C,9H 9C 4C,9H 4C,9H 3C,9H 10C 9C 10C 9C Barley -- -- -- -- --      -- -- -- 5C,9G 3C,8H 6C,9G 3C,8G 9C 4C,9G 2C,8G 3C,7G 0 0 2G 0 Soybean      1H 9C 9C 9C 4C,9G 3H 3C,9G 2H,7G 9C 9C 9C 9C 9C 4C,9G 9C 4C,9G 5C,9G      4C,9G 9C 5C,9G Rice 0 2C,8G 9C 9C 5G 0 5C,9G 7G 9C 9C 9C 9C 9C 9C 9C      5C,9G 5C,9G 7G 9C 6G Sorghum 0 9H 9C 5C,9H 3C,9H 0 9C 3C,9H 9C 9C 9C 9C      10C 9C 9C 9C 9C 4C,9G 9C 9C Sugar Beets 1C,1H 5C,9G 5C,9G 9C 3C,6G 2C,3G      9C 4C,8G 10C 5C,9G 10C 9C 10C 4C,8G 9C 4C,9G 3C,6H 3C,5G 9C 3C,8G Cotton      1C 9C 9C 5C,9G 3C,9H 1H 2C,9G 8G 9C 5C,9G 9C 10C 9C 4C,9G 5C,9G 9C 4C,9H      4C,9H 4C,9H 3C,8H PREEEMERGENCE                      Morningglory 0 9G      9G 8G 5H 3H 9C 9H 9C 7H 9G 8G 8H 3C,7G 9G 7H 5H 0 3C,8H 2H Cocklebur 0      9H 9H 9H 7H 0 9H 9H 9H 9H 9H 9H 8H -- 9H 9H 9H -- 9H 2C Velvetleaf 0      5C,9G 10C 9C 6G 0 9C 2C,4G 9C 3C,8G 9C 9C 9C 3C,7H 5C,9G 7G 7G 0 8H 5G      Nutsedge 0 10E 10E 4C,9G 0 0 10E 3C,9G 10E 10E 10E 10E 9G 7G 10E 9G 0 0      0 0 Crabgrass 0 3G 2C,7G 3G 0 0 4G 2G 4C,8G 3C,7G 8G 4G 5G 0 9C 2G 2C,5G      0 2C,5G 4G Giant Foxtail -- -- -- -- -- -- -- -- 4C,9H 3C,8H 9H 3C,6G 9H      5G 4C,8G 4G 2C,5G 2G 3C,7G 3G Barnyardgrass 0 3C,8H 5C,9H 3C,8H 1C 0      3C,9H 3C,3G 5C,9H 4C,9H 5C,9H 3C,9H 3C,8H 3C,6G 9H 3C,8H 3C,6G 0 3C,8G 0      Cheatgrass 0 8G 6G 2G 0 0 0 0 4C,8H 3G 7H 6G 2G 0 3G 0 0 0 0 0 Wild Oats      0 5G 9C 5C,9G 2C,5G 0 5C,9G 3C,6G 5C,9G 4C,9G 5C,9G 2C,9G 5C,9G 3C,8H      3C,9H 2C,5G 2G 0 2C 0 Wheat 0 0 4C,9G 3C,8G 0 0 8G 3G 10H 3C,8G 10H 9G      5C,9G 3C,8H 3C,9H 7G 0 0 3G 0 Corn 2G 8G 3C,9G 7G 6G 0 6G 2G 10H 4C,9H      4C,9H 8G 4C,9H 3C,7H 3C,9H 9H 4C,9H 2C,6G 9H 3C,8H Barley -- -- -- -- --      -- -- -- 9G 3C,9G 3C,9G 9G 4C,9G 9G 3C,9G 8G 0 0 7G 0 Soybean 2C 3C,8H      3C,9H 2C,7G 2C,2H 1C 3C,7G 3C,3H 9H 4C,8H 9H 4C,8H 9H 3C,6H 3C,8H 3C,5G      3C,7H 0 3C,7H 2C,3G Rice 0 2C,9H 10E 3C,8G 5G 1C 10E 2C,8G 10E 9H 10E      10E 10E 4C,8H 10E 9H 8G 2G 9H 0 Sorghum 1C 3C,9H 10E 3C,9H 3C,6G 0 10H      3C,9H 10H 6C,9H 10H 10H 5C,9H 6C,9H 10H 10H 5C,9H 3C,6G 4C,9H 3C,8H      Sugar Beets 3H 10C 5C,9G 5C,9G 3C,7H 0 10E 5C,9G 10E 9C 5C,9G 5C,9G 9C      5G 9C 5C,9G 5G 3G 4C,7H 5G Cotton 0 9G 9G 9G 2C 0 9G 2C,5G 9C 2C,9G      4C,9G 4C,9G 9G 2C,8G 9G 8G 5G 0 2C,5G 1C                  Com-  Com-         pound Compound 23 pound 24 Compound 25      Compound 26 Compound 27 Compound 28 Compound 29 Compound 30 Compound 31      Compound 32 33 Rate kg/ha 0.05 0.01 0.01 0.05 0.01 0.05 0.01 0.05 0.01      0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01  0.05        POSTEMERGENCE                      Morningglory 10C 8G 5G 0 0 3C,5G 0      2C,6G 2G 10C 3C,8G 3C,9G 3C,7H 10C 4C,8H 10C 3C,8H 10C 10C 10C Cocklebur      10C 10C 10C 3H 2H 4C,8H 2H 10C 5C,9G 10C 9C 3H 0 9C 4C,9G 10C 9C 10C 10C      10C Velvetleaf 10C 5C,9G 5C,9G 0 0 2C,5G 0 9C 3C,7G 4C,9G 3C,9G 3C,7G 0      9C 7G 9C 4C,8H 10C 10C 10C Nutsedge 10C 10C 5C,9G 0 0 3C,6G 0 10C 3C,8G      10C 4C,9G 0 0 4C,8G 4G 7G 0 10C 9C 9C Crabgrass 5G 3G 0 0 0 3C,4H 0 2G      2G 3G 0 3C,5G 0 6C,9H 4C,6G 9C 3C,8G 5C,8G 7G 3C,7G Giant Foxtail 5C,9G      3C,8G 3C,7G 3C,8H 2H 4C,9H 3C,5G 4C,9G 4G 7G 2G 5C,9G 3C,7G 9C 10C 10C      9C 9C 9C 9C Barnyardgrass 9C 3C,9H 3C,7G 5C,9H 0 5C,9H 2C,6G 4C,9H 4C,8H      3C,7H 1C,4G 3C,8H 2H 10C 9C 10C 9C 9C 9C 10C Cheatgrass 5G 2G 2G 0 0 3G      0 4G 0 0 0 0 0 3G 0 3G 0 7G 5G 7G Wild Oats 5G 2G 0 4C,8G 0 4C,9G 3C,4G      9G 3C,6G 2G 0 4C,9G 7G 4G 3G 7G 4G 4C,9G 9G 5C,9G Wheat 8G 6G 5G 5C,9G 0      3C,9G 7G 5C,9G 2C,6G 4G 0 9G 7G 4G 0 2C,6G 3G 10C 6C,9G 9C Corn 9H 6H 0      3C,9H 2H 9H 0 2G 0 0 0 4C,8H 5H 10C 10C 10C 9C 10C 2C,7H 3C,9H Barley      3C,9H 6G 3G 9G 2G 8G 0 9G 3G 2G 0 9C 9G 0 0 1C,4G 0 9C 8G 3C,9G Soybean      9C 9C 9C 2H,4G 0 3C,8G 2H 5C,9G 4C,9H 3H,8G 3H,8G 3C,7H 4H 9C 5C,9G 9C      4C,9G 9C 9C 10C Rice 9C 4C,9G 3C,7G 9C 2G 9C 8G 9C 5C,9G 2C,8G 6G 9C      3C,8G 5C,9G 4C,9G 9C 4C,9G 9C 9C 9C Sorghum 9C 9C 4C,9H 4C,9H 3G 5C,9G      3C,7H 9C 4C,9G 4C,9H 4C,9G 5C,9G 4C,9G 9C 9C 10C 9C 10C 9C 10C Sugar      Beets 10C 10C 10C 5G 0 9C 2H 10C 9C 9C 9C 3C,7H 4H 10C 5C,9G 10C 9C 10C      10C 9C Cotton 9C 9C 4C,9G 0 0 3C,7G 0 9C 9H 9H 9G 5H 0 9C 9H 9C 9C 9C      10C 9C PREEEMERGENCE                      Morningglory 9H 7H 7H 0 0 2H      1H 6G 0 3C,9G 5H 5H 1C 9C 4C,4H 4C,8H 3C,5H 9C 8H 9C Cocklebur 9H 9H 9H      0 0 2C 0 8H 6H 9H 3C,4H 0 0 9H 3C 9H 2C,5G 9H 8H 9H Velvetleaf 10C 9G 9C      3G 0 0 0 3C,8H 7G 5C,9H 2G 0 0 9C 9C 9C 0 10C 10C 4C,9G Nutsedge 10E 9G      3C,7G 0 0 0 0 5G 0 10E 0 0 0 4G 0 4G 0 10E 10E 10E Crabgrass 0 0 2G 0 0      0 0 0 0 0 0 0 0 3C,7G 3C,4G 3C,5G 0 7G 4G 3C,7G Giant Foxtail 4C,9H 1C      3C,5G 3G 0 0 0 3C,6G 3C 3C,3H 3G 5G 0 9H 3G 3C,6G 1C 5C,9G 4C,7G 4C,8H      Barnyardgrass 5C,9H 3C,8H 3C,6G 0 0 2C 0 4C,9H 3C,3G 5C,9H 3C,3G 3C,5G 0      5C,9H 3C,7G 9C 3C,4H 9C 9H 4C,9H Cheatgrass 4G 0 0 0 0 0 0 0 0 3G 3G 0 0      3G 0 2G 0 7G 0 8G Wild Oats 6G 0 2C 0 0 0 0 3C,7G 2C 2C 0 3C,6G 0 2C 0      2C,4G 0 5C,9G 3C,8G 4C,9H Wheat 4C,9G 4G 5G 0 0 0 0 7G 2G 6G 0 9H 2G 2G      0 2G 0 10E 4C,9G 9C Corn 3C,8G 2C,5G 0 3G 0 0 0 2C 0 2G 0 2C,5G 0 5C,9H      9H 9H 0 3C,9H 3C,7G 3C,8H Barley 3C,9G 2C,8G 2C,8G 5G 0 5G 3G 9G 6G 8G      5G 2C,8G 2G 5G 0 5G 0 5C9G 4C9G 5C,9G Soybean 3C,8H 3C,8H 3C,7H 0 0 0 0      2C,7G 2C,2H 3C,5G 3C,4G 2C,3H 0 3C,8H 3C,7H 3C,8H 2H 9H 3C,7H 9H Rice 9H      4C,9G 3C,6H 5G 0 3C,5G 2C 9H 3C,7H 5C,9H 4C,8H 3C,8H 2C 9H 3C,6H 4C,9H      2C,4G 10E 10E 10E Sorghum 10E 3C,9H 4C,8H 2C 0 3C,5G 2G 9H 2C,6G 5C,9H      5C,9H 3C,8H 1C 6C,9H 4C,8H 10H 4C,7G 6C,9H 9C 10H Sugar Beets 5C,9G      5C,9G 5C,9G 0 0 2H 3G 4C,8G 3C,7H 10C 3C,7G 3G 4H 10E 5H 5C,9G 5H 4C,8G      9C 9C Cotton 10C 9C 2C,7H -- 0 1C 0 4C,8G 2C,3G 3C,7G 2C,4G 0 2H 4C,9G      2C,2H 4C,8H 2C 9C 9G 9G                  Com- Com-          pound pound 33 Compound 34 Compound 35      Compound 36 Compound 37 Compound 38 Compound 39 Compound 40 Compound 41      Compound 42 43 Rate kg/ha 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01      0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05        POSTEMERGENCE                      Morningglory 10C 10C 5C,9G 10C 10C      9C 10C 3C,8H 3C,5H 3C,8H 1C 10C 10C 10C 9C 4C,8H 2C,4G 2C,8G 2C,7G 3C,8H      Cocklebur 9C 10C 5C,9G 10C 10C 9C 3C,8H 2C,2G 0 3C,7H 0 9C 9C 9C 9C      5C,9H 2C,4G 5C,9H 3C,8G 3G Velvetleaf 9C 10C 5C,9G 10C 4C,9G 9C 9C 2C,4G      0 2C,5G 1C 9C 10C 10C 5C,9H 4C,8H 3C,5H 4C,8H 5G 7G Nutsedge 5C,9G 5C,9G      5C,9G 10C 4C,9G 3C,7G 3G 0 0 0 0 9C 5C,9G 2C,8G 5G 0 0 3G 4G 0 Crabgrass      2G 2C,9G 2C,4G 3C,7H 3G 9C 3C,7G 2C,3G 0 2G 0 5C,9G 3C,7G 3C,7G 4G 2G 0      0 0 3G Giant Foxtail 4C,9H 10C 9C 9C 4C,9G 9C 9C 4C,8G 4G 3C,8H 2G 5C,9G      3C,7G 3C,7G 2G 5G 0 4G 0 2G Barnyardgrass 9C 10C 4C,9H 10C 10C 9C 10C 9C      3C,7H 5C,9G 4H 9C 9C 9C 3C,7H 2C,7H 3H 4C,9H 4G 4G Cheatgrass 5G 6G 2G      6G 2G 7G 3G 2C,6G 2G 2G 0 10C 9C 9C 4C,9G 3C,8G 4G 7G 0 8G Wild Oats      3C,7G 9C 4C,9G 3C,9G 3C,6G 9C 9C 2C,6G 0 2C,5G 0 5C,9G 9G 4C,9G 3C,6G 7G      3G 2C,7G 0 4C,9G Wheat 4C,9G 9C 3C,9G 5C,9G 2C,8G 9C 5C,9G 0 0 4G 0      3C,9G 9G 9G 9G 4G 2G 2G 0 9G Corn 3C,7H 4C,9H 1H 4G 0 9C 9C 4C,9G 3C,8H      3C,9H 3C,7H 3C,9G 2U,9G 3C,8H 1C,3G 0 0 2G 0 0 Barley 4C,9G 9C 2C,8G 9C      6G 9C 4C,9G 0 0 0 0 4C,9G 9G 5G 2G 0 0 0 0 9G Soybean 5C,9G 9C 4C,9G      4C,9G 4C,9G 5C,9G 4C,9G 4C,9G 3C,3G 3C,8G 2C,4H 6C,9G 5C,9G 9C 4C,9G      4C,8H 3C,5H 2C,7G 1H 3H,8G Rice 9C 9C 9C 9C 5C,9G 9C 9C 5C,9G 4C,9G      5C,9G 5G 9C 5C,9G 9C 4C,9G 5C,9G 3C,5G 2C,9G 5G 4C,9G Sorghum 10C 9C      4C,9H 9C 9C 9C 9C 4C,9G 4C,9G 4C,9G 2C,6G 3U,9G 9G 4C,9H 3C,8G 2C,6G      2C,4G 9G 7G 4C,8G Sugar Beets 5C9G 10C 9C 10C 10C 9C 10C 3C,7H 2H 3C,7H      3C,4H 10C 9C 10C 3C,8H 3C,6H 2C,3G 3C,8G 2C,6G 3C,7G Cotton 9C 10C 9C      10C 10C 9C 9C 3C,8H 2C,3G 3C,7H 2C,2G 9C 4C,9G 4C,9G 4C,9H 4C,9H 2C,3G      2C,8G 5G 5G PREEEMERGENCE                      Morningglory 9G 9H 8H 9C      8H 2C,9H 3C,7H 0 0 1C 0 9C 8G 3C,8H 2C,3H 1C 2G 2C,4H 1H 3H Cocklebur --      8H 9H 9H 7H 9H 3H -- 0 0 0 9H 8H 3C,7H 2C,3H 3C,3G -- 3C,7H 7H 8G      Velvetleaf 9G 9H 3C,9G 9G 8G 9G 3C,5H 5G 0 0 0 3C,9G 4C,9G 3C,8H 3C,5H      1H 0 0 2G 0 Nutsedge 3C,5G 4C,8G 2C,3G 10E 9G 5G 0 2G 0 3G 0 10E 8G 4G 0      0 0 0 0 0 Crabgrass 2C,4G 3C,5G 1C 2C,5G 3C,4G 4C,9G 3C,6G 0 0 -- 0      3C,3G 2G 2C,5G 0 0 0 6G 0 0 Giant Foxtail 3C,4G 4C,8G 2G 3C,6G 4G 4C,9H      3C,5G 0 0 0 0 4C,9H 3C,6G 3C,7G 2G 0 0 2C,7G 0 5G Barnyardgrass 2C,2H      3C,7H 0 4C,9H 3C,7G 3C,9H 3C,7H 1C 0 3G 0 5C,9H 4C,9H 3C,8H 2C,3G 0 0 9H      6G 0 Cheatgrass 2G 6G 0 0 0 8G 0 0 0 2G 0 5C,9H 9H 9H 3C,6G 0 0 8G 4G 7G      Wild Oats 6C,9G 4C,9H 4C,8G 3C,8G 3C,5G 6C,9H 3C,8G 0 0 0 0 4C,9H 3C,8H      3C,8G 3C,5G 0 0 2G 0 2C,6G Wheat 4C,9G 4C,8G 8G 5C,9H 7G 6C,9H 5G 0 0 0      0 5C,9H 3C,9G 3C,8G 5G 0 0 2G 0 6G Corn 1C,5G 4C,8H 2G 2C,8G 4G 10H      4C,9H 3C,7H 2C 2C,5G 0 3C,9H 2C,8G 3C,5G 2C,2G 2G 0 2G 0 2C,6G Barley 9G      5C,9G 9G 9G 9G 9C 5C,9G 0 0 0 0 9G 9G 3C,9G 8G 2G 0 5G 0 9G Soybean 9H      9H 3C,7H 3C,8H 3C,7H 9H 3C,7H 3C,3H 1C 3C,3H 0 9H 3C,6H 4C,6H 3C,4H      3C,3H 1C 7G 0 1C Rice 10E 10E 3C,8H 10E 10E 10E 3C,9H 3C,6H 3C,3G 2C,7G      2G 10E 5C,9H 4C,9H 2C,6G 0 0 8H 7G 9H Sorghum 7C,9H 6C,9H 4C,8H 10H 10H      10H 6C,9H 3C,8G 3C,4G 3C,8G 2C 4C,9G 4C,8H 4C,9G 3C,6G 3C,3G 0 8G 2C,7G      3C,6H Sugar Beets 9C 9C 4C,8H 4C,9G 3C,8G 10C 4C,9G 3C,5G 7G 5H 3G 9G 8G      5C,9G 4C,8G 6G 3H 8G 0 9G Cotton 8G 4C,8G 2G 9G 4C,9G 8G 1C 2C,4G 1C 2G      0 9G 9G 8G 2C,6G 2C,3G 0 5G 2G 0

      Com-          Com- pound 43 Compound 44 Compound 45 Compound 46      Compound 47 Compound 48 Compound 49 Compound 50 Compound 51 Compound 52      pound 53 Rate kg/ha 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05      0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05        POSTEMERGENCE                      Morningglory 3C,7H 3C,7H 3C,3H      4C,9H 2C,5G 10C 10C 9C 4C,9H 4C,9H 2C,2H 4C,8G 2C,5G 2C,5H 0 4C,8H 1C      5C,9G 4C,9H 9C Cocklebur 0 2C,5G 2C 4C,9H 1C 10C 8H 7H 2G 1H 1H 4C,9H 5G      0 0 3C,6G 0 4C,9H 3C,4G 9C Velvetleaf 2C,5G 3C,6H 0 3C,7H 3C,3G 10C 9C      5C,9G 3C,8G 3C,7H 3G 3C,8H 3H 2C,5G 0 2G 0 3C,8H 3C,4G 9C Nutsedge 0 0 0      3G 0 2C,9G 4C,8G 7G 3G 4G 0 5G 0 0 0 8G 0 9G 2C,7G 9C Crabgrass 0 0 0 2G      0 7G 5G 4G 0 0 0 0 0 0 0 2C,2G 0 3C,7G 2C 8G Giant Foxatil 0 1C 0 2G 0      5C,9G 3C,8G 5G 2G 0 0 3C,6G 0 2C,4G 0 6C,9H 3C,7H 9C 4C,8G 9C Barnyardgra      ss 3G 3C,7H 2C,4G 3C,9H 2C,5H 10C 5C,9G 3C,9H 3C,8H 3C,7H 1H 3C,8H 3H      3C,7H 0 9C 3C,8H 9C 9H 9C Cheatgrass 7G 0 0 3G 0 9G 8G 2C,6G 4G 2G 0 0 0      0 0 8G 0 3C,8G 5G 9C Wild Oats 5C,9G 0 0 2G 0 2C,9G 9G 3C,8G 3G 2G 0 0 0      0 0 4C,9G 0 4C,9G 3C,7G 2G Wheat 9G 0 0 2G 0 5C,9G 9G 8G 2G 2G 0 2G 0 0      0 8G 2G 8G 4G 9G Corn 0 3C,7G 0 2C,6G 0 2C,9G 9H 3C,8H 2G 1H 0 1H 0 2G 0      4C,9H 2C,5G 3C,8H 0 3H Barley 9G 2C 0 0 0 3C,9G 9G 3C,8G 4G 2G 0 1C 0 0      0 3G 0 3C,7G 2G 3C,9G Soybean 2H,5G 2C,7H 3H 3C,8G 2C,6H 9C 5C,9G 4C,9G      3C,8G 2C,7G 2H 2H 1H 0 0 3C,7H 2C,5G 4C,9G 2C,8H 9C Rice 4C,9G 4C,9G 4G      5C,9G 5G 9C 9C 4C,9G 4C,9G 4C,9G 2G 4C,9G 4C,9G 6G 0 9C 5C,9G 9C 4C,9G      9C Sorghum 2C,5G 5C,9H 5G 4C,9H 2C,8G 9C 5C,9G 4C,9G 4C,9G 4C,8G 6G      4C,9G 4C,9H 8G 4G 9C 4C,9H 9C 5C,9G 9C Sugar beet 2C,5G 3C,7H 3C,6G      5C,9G 3C,7H 10C 9C 9C 9C 4C,8H 2C,6G 3C,8H 2C,5G 3C,7G 0 9C 3C,7H 9C      4C,8H 9C Cotton 0 3C,6G 1C 3C,8H 2C,4G 10C 2C,8G 8H 3C,8G 6H 0 7G 3G 2G      0 8H 7H 4C,9G 3C,8H 9C PREEMERGENCE                      Morningglory 0      2C 5G 4H 4H 9G 9G 9G 7G 2G 3G 8G 7G 0 0 5G 7G 8G 0 9C Cocklebur 0 1H 0      6H 4H 9H 8G 8H -- 0 -- 9H 7H 8G -- 4H -- 7H 0 9H Velvetleaf 0 7G 0 2G 3G      9C 9G 4C,9G 7H 0 -- 3H 0 7G -- 0 5G 5G 0 9C Nutsedge 0 0 0 0 0 4C,9G 0      4G 0 0 0 4G 0 0 0 0 0 5G 0 10E Crabgrass 0 0 0 0 0 3G 0 2G 0 0 0 0 0 0 0      0 0 0 0 2G Giant Foxatil 0 3G 0 0 0 9H 7G 8G 2C 0 0 3C,4G 2G 0 0 4G 2G      6G 2G 9H Barnyardgrass 0 3G 0 4G 0 9H 3C,9H 8H 2C 0 0 3C,8H 2G 0 0 2G 2G      5G 0 9H Cheatgrass 3G 0 0 0 0 7G 3G 6G 0 0 0 0 0 0 0 2G 0 5G 0 10H Wild      Oats 0 0 0 0 0 4C,9H 8H 2C,8G 2G 0 0 2G 0 0 0 0 0 2G 0 0 Wheat 0 0 0 0 0      10H 3C,9H 8G 3G 0 0 3G 0 0 0 2G 0 7G 0 9H Corn 0 3C,7H 0 3C,8H 0 10H      3C,9H 2C,9G 2C,6G 0 0 4G 0 0 0 2C,8G 0 3C,8H 2G 2C,7G Barley 7G 0 0 0 0      9G 9H 9G 2C,7G 2G 0 8G 0 0 0 6G 0 8G 3G 9G Soybean 0 0 0 2C,2H 0 9H 8H      3C,7H 7H 2C 0 4G 0 0 0 2C,5G 1H 8H 5H 9H Rice 4G 3C,8H 2C,4G 3C,7H 0 10E      10E 5C,9H 6G 0 3G 3C,8H 4G 2C 0 9H 2G 9H 5H 10E Sorghum 0 3C,8H 2C 3C,8G      2C,4G 10H 5C,9H 5C,9H 2C,8G 2C -- 10H 3C,8H 2C,5G 0 2C,9H 2C,5G 3C,9H      3C,8G 5C,9H Sugar beet 2G 7G 5G 4G 4G 5C,9G 5C,9G 4C,9G 7G -- 2G 3C,8G      8G 4G 0 5G 5G 9G 8G 9C Cotton 0 2C 0 5G 2C 9G 9G 9G 2C,5G 2G -- 2C,7G 1C      0 0 7G 0 2C,7G 2G 9G        Com-          Com- pound 53 Compound 54 Compound 55 Compound 56      Compound 57 Compound 58 Compound 59 Compound 60 Compound 61 Compound 62      pound 63 Rate kg/ha 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05      0.01 0.05  0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05        POSTEMERGENCE                      Morningglory 10C 10C 10C 10C 8C 10C      10C 10C 2C,8G 1C,7G 0 10C 10C 3C,8G 1C,1H 1C,1H 0 0 0 10C Cocklebur 9C      10C 10C 10C 9C 10C 4C,9G 10C 10C 0 0 10C 10C 2C,8G 2H 3H 0 0 0 4C,9H      Velvetleaf 9C 10C 9C 10C 9C 10C 3C,8G 10C 2C,9H 2G 0 10C 9C 3C,9G 4G 4H      0 0 0 4C,8H Nutsedge 9C 9C 5C,9G 9C 9G 5C,9G 4C,9G 5C,9G 2C,9G 0 0 10C      10C 2C,5G 0 0 0 0 0 9G Crabgrass 3G 6G 3G 3C,6G 2C,5G 6G 2G 7G 0 0 0      3C,9G 7G 0 0 0 0 0 0 3C,6G Giant Foxatil 3C,8G 5C,9G 3C,9G 9C 3C,8G      4C,9G 7G 3C,9G 2C,7G 0 0 9C 9C 3C,8G 4G 5G 2G 2G 0 9C Barnyardgrass 9C      10C 9C 9C 10C 9C 9H 2C,9G 2C,5H 0 0 9C 9C 3C,7H 2H 2C,5G 3G 2C,5G 0 9C      Cheatgrass 9G 9C 4C,9G 9C 5C,9G 4C,9G 9G 8C 2C,9G 2G 0 9C 10C 9G 3G 6G 0      6G 0 5C,9G Wild Oats 0 3C,5G 0 5C,9G 3C,3G 3G 0 2C,9G 2C,6G 0 0 9C 5C,9G      2C,7G 0 2C,5G 2G 2C,5G 0 3C,8G Wheat 7G 3C,9G 9G 9G 9G 8G 3G 1C,6G 0 0 0      9C 4C,9G 9G 0 9G 8G 6G 0 9G Corn 0 2H 0 2H 0 0 0 1C,8H 3C,8H 0 0 9C 10C      3C,8H 0 2C,7G 3G 3G 0 5C,9G Barley 2C,6G 8G 5G 9G 3C,7G 2G 0 5C,9G 3C,9G      0 0 9C 5C,9G 2C,4G 0 2C,5G 3G 4G 0 9G Soybean 5C,9G 9C 4C,9G 5C,9G 4C,8G      3C,8G 3C,5H 5C,8H 2C,6H 0 0 9C 9C 3G 2H 2C,6H 3H 0 0 3C,8H Rice 5C,9G 9C      9C 5C,9G 5C,9G 9C 5C,9G 5C,9G 2C,8G 3C 0 9C 9C 5C,9G 0 3C,9G 3G 7G 0      6C,9G Sorghum 10C 9C 9C 5C,9G 5C,9G 9C 5C,9G 3C,9G 3C,9G 1C,5G 0 9C 9C      2C,9G 5G 4G 2G 7G 0 3C,9G Sugar beet 10C 10C 9C 9C 9C 10C 9C 9C 10C      2C,4H 0 9C 9C 9C 3G 2C,4G 0 2C 0 9C Cotton 9C 9C 5C,9G 9G 9G 10C 3C,8G      10C 2C,8H 2G 0 10C 9C 3C,8G 0 0 0 0 0 4C,9G PREEMERGENCE           Morningglory 9G 9G 9G 9G 8G 9G 9G 8H 3C,7H 0 0 9G 9G 0 0 0 0 0 0 3H      Cocklebur -- 9H 9H 9H 9H 9H 5H 2C,8H 2C,7H 0 0 9H 9H 2H 0 0 0 0 0 4G      Velvetleaf 9C 5C,9G 5C,9G 4C,9G 8G 8H 6H 2C,7H 2C,5H 0 0 9C 3C,9G 0 0 0      0 0 0 0 Nutsedge 10E 10E 10E 10E 9G 10E 4G 10E 9G 0 0 10E 10E 0 0 0 0 0      0 7G Crabgrass 0 3G 0 2G 0 2G 0 1C,5G 2C,4G 0 0 3C,7G 3G 0 0 0 0 0 0 3G      Giant Foxatil 8H 9H 3C,8H 9H 3C,8G 3C,7G 6G 2C,7H 2C,6G 0 0 5C,9H 3C,7G      0 0 0 0 0 0 3G Barnyardgrass 9H 9H 9H 9H 3C,8H 9H 8H 2C,6H 2C,4H 0 0      5C,9H 4C,9H 0 0 0 0 0 0 4G Cheatgrass 9H 9H 10E 9H 8G 8H 6G 3C,9H 2C,9H      0 0 10E 9H 0 0 0 0 0 0 5G Wild Oats 0 8G 2C,5G 8G 0 0 0 2C,6G 2C,6G 0 0      4C,9H 3C,6G 0 0 0 0 0 0 2C Wheat 7H 10H 4C,9H 9G 2G 8G 5G 4G 0 0 0 10H      4C,9H 0 0 0 0 0 0 3G Corn 4G 7G 6G 3G 1C,2G 1C 0 2C,7G 3C,4G 0 0 5C,9H      4C,9H 0 0 0 0 0 0 3C,3G Barley 9G 9G 9G 9G 8G 4C,8G 5G 6G 6G 0 0 4C,9G      3C,9G 0 0 0 0 0 0 3C,9G Soybean 9H 9H 3C,8H 3C,8H 2C,6G 7H 2H 2C,5G      1C,2G 0 0 9H 9H 0 0 0 0 0 0 1C Rice 10E 10E 10E 10E 9H 10E 8H 3C,9H      2C,8H 0 0 10E 10E 0 0 0 0 0 0 4C,8H Sorghum 9H 10H 5C,9H 10H 9H 9H 5C,9H      2C,9H 2C,8H 0 0 10H 4C,9H 0 0 0 0 0 0 4C,9H Sugar beet 9C 9C 5C,9G 9G 9G      4C,9G 8G 9C 4C,8G 1C 0 5C,9G 4C,9G 0 0 0 0 0 0 7G Cotton 9G 4C,9G 9G 9G      9G 9G 7G 2C,8G 2C,8G 0 0 9G 9G 0 0 0 0 0 0 3C,6G        Com-          CMPD pound 63 CMPD 64* CMPD 65* CMPD 66 CMPD 67 CMPD 68      CMPD 69 CMPD 70 CMPD 71 CMPD 72 73 Rate kg/ha 0.01 0.05 0.01 0.05 0.01      0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01      0.05        POSTEMERGENCE                      Morningglory 4C,8G 0 0 0 0 10C 10C      10C 10C 9C 5C,9G 10C 4C,9H 3C,8G 3C,7G 4C,9H 3C,8H 10C 4C,9G 10C      Cocklebur 3C,7H 0 0 0 0 10C 10C 10C 9C 10C 5C,9G 9C 4C,9H 2G 0 4C,9H      2C,2H 10C 5C,9G 10C Velvetleaf 3C,7H 0 0 0 0 10C 9C 10C 4C,9H 9C 5C,9G      3C,7H 2C 0 0 4C,6H 0 10C 10C 10C Nutsedge 2C,8G 0 0 0 0 6C,9G 5C,9G      5C,9G 4C,8G 5C,9G 7G 2C,8G 5G 0 0 4G 0 5C,9G 5C,9G 5C,9G Crabgrass 5G 0      0 0 0 2C,6G 4G 4G 3H 6G 3G 3H 2H 0 0 0 0 2H 0 0 Giant Foxatil 2C,8G 0 0      0 0 9C 4C,9G 9C 5C,9G 9C 5C,9G 5C,9G 7G 4C,9H 3G 4C,9H 3C,7G 3C,8G 3G      3C,7H Barnyardgrass 3C,9G 0 0 0 0 9C 9C 9C 9C 9C 5C,9H 9C 4C,9H 5C,9H 5G      5C,9H 9C 10C 9C 4C,9H Cheatgrass 9G 0 0 0 0 9C 4C,9G 9C 4C,9G 10C 4C,9G      4C,9G 4C,9G 3C,8G 2C,5G 3C,6G 4G 9C 9C 9C Wild Oats 2C,5G 0 0 0 0 2G 0      2C,6G 2G 4C,9G 2C,3G 3G 0 4C,8G 2G 3C,8G 3G 5C,9G 3C,7G 6C,9G Wheat 7G 0      0 0 0 9G 8G 9G 7G 9G 9G 6G 0 3C,8G 3G 3G 0 5C,9G 8G 4C,9G Corn 3C,9G 0 0      0 0 4G 2G 0 0 2H 0 0 0 5C,9G 6G 6G 3G 4C,9G 4G 3C,5G Barley 8G 0 0 0 0      7G 3G 3G 0 2G 0 0 0 2G 0 5G 0 9G 4G 3G Soybean 3C,4H 0 0 0 0 9C 9C 9C      5C,9G 4C,9G 5C,9G 5C,9G 3C,7H 4C,9G 3C,7H 4C,9G 3C,8G 9C 5C,9G 5C,9G      Rice 4C,9G 0 0 0 0 9C 9C 9C 9C 9C 9C 9C 4C,9G 4C,9G 5G 8G 2C,5G 9C 5C,9G      5C,9G Sorghum 4C,9G 0 0 0 0 9C 9C 9C 5C,9G 9C 4C,9G 9C 4C,9G 3C,9H 4C,8H      5C,9H 3C,9H 10C 9C 9C Sugar beet 5C,9G 0 0 0 0 9C 10C 10C 9C 10C 9C 9C      5C,9G 3C,7H 2C,2H 4C,8H 3C,6H 10C 10C 10C Cotton 3C,8H 0 0 0 0 10C 4C,9G      9C 4C,9H 4C,9G 4C,9H 4C,8G 4C,9H 3C,8H 0 4C,9H 3C,8H 9C 4C,9G 4C,9H      PREEMERGENCE                      Morningglory 0 0 0 0 0 9H 2C,9H 8H      2C,6H 9G 3H 8G 2C,2H 2G 0 3H 0 7H 4H 2G Cocklebur 1H 0 0 0 0 9H 7H 3C,7H      2C,5G 3C,7H 1C 3C,7H 2C 0 0 0 -- 8H 2C 0 Velvetleaf 0 0 0 0 0 5C,9G      2C,7G 3C,7H 0 3C,5H 1C 2H 2C,2G 1C 0 0 0 5H 0 2G Nutsedge 0 0 0 0 0 10E      9G 5G 5G 10E 0 2C,5G 3G 0 0 0 0 10E 3C,7G 5G Crabgrass 0 0 0 0 0 4G 0 0      0 2G 0 2G 0 0 0 0 0 0 0 0 Giant Foxatil 2G 0 0 0 0 9H 2C,8H 3C,8G 3G      3C,9H 2C,5G 9H 3C,5G 2C,2G 0 2G 0 3C,8H 2C,2G 3C,3G Barnyardgrass 2G 0 0      0 0 9H 3C,9H 3C,9H 2G 3C,9H 1C 3C,7H 0 2C,5G 0 0 0 9H 2C,5G 3C,7G      Cheatgrass 0 0 0 0 0 9H 8G 9G 8G 3C,9G 8G 9H 8G 5G 0 0 0 9H 3C,9H 9H      Wild Oats 0 0 0 0 0 2G 0 2C 0 2C,4G 0 0 0 0 0 0 0 3C,7G 2G 3C,5G Wheat 0      0 0 0 0 4C,9H 2C,8H 3C,8H 5G 8G 6G 5G 0 0 0 0 0 8G 2G 7G Corn 0 0 0 0 0      4C,8H 6G 4G 0 2G 2G 0 0 3G 0 2C,4G 0 3C,8H 3G 2G Barley 4G 0 0 0 0 9G      2C,6G 2G 2G 3C,7G 0 2G 0 0 0 0 0 8G 5G 2G Soybean 0 0 0 0 0 9H 9H 9H      3C,7H 3C,9H 3C,6H 3C,7H 2C,4G 0 0 0 0 7H 3C,5H 3C,4H Rice 3G 0 0 0 0 9H      9H 3C,9H 3C,7G 5C,9H 3C,7G 9H 7G 6G 0 0 0 10E 9H 9H Sorghum 3C,5G 0 0 0      0 10H 5C,9H 3C,9H 3C,9H 5C,9H 3C,7H 3C,9H 2C,8H 2G 0 3C,5G 0 10H 9H 9H      Sugar beet 3C,5G 0 0 0 0 5C,9G 4C,9G 9G 7G 4C,8H 3C,8G 3C,7H 2C,5G 2G 0      3G 0 9G 9G 7G Cotton 5G 0 0 0 0 4C,9G 2C,8G 3C,7H 6G 3C,8H 2C 2C,6G 2C 0      0 0 0 8G 3G 2G      *It is noted that Compounds 64 and 65 were inactive at the levels tested.      However, it is believed that at higher levels, herbicidal activity would      be present.     CMPD          CMPD 73 CMPD 74 CMPD 75 CMPD 76 CMPD 77 CMPD 78 CMPD 79      CMPD 80 CMPD 81 CMPD 82 83 Rate kg/ha 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0      .05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05        POSTEMERGENCE                      Cotton 4C,9H 9G 9G 9G 9G 9C 9C 9C      5C,9G 3C,9G 9G 10C 9C 9C 2C,8H 9C 2C,8H 9C 5C,9G 9C Morningglory 9C      4C,9G 3C,8H 9C 2C,9G 10C 7G 10C 10C 10C 3C,8H 10C 9C 3C,8H 4C,8H 10C      4C,8H 10C 10C 10C Cocklebur 4C,9G 4C,9G 3C,8H 5C,9G 3C,8H 10C 10C 10C      10C 9C 3C,8H 10C 9C 5C,9H 4C,8H 10C 10C 10C 10C 10C Nutsedge 3C,9G 4C,9G      2C,5G 3C,9G 5C,9G 10C 10C 10C 5C,9G 4C,9G 2C,9G 10C 4C,9G 8G 6G 3C,8G 0      9C 9C 9C Crabgrass 2H 0 0 0 0 2C,7G 7G 2C,6G 3G 6G 0 6G 2G 5G 0 2C,5G 0      6C,9G 4C,6G 4C,8G Barnyardgrass 3C,7H 3C,8H 4G 3C,8H 3C,5G 10C 9C 9C 9C      9C 4C,9H 3C,9G 2C,8G 9C 2C,9H 10C 3C,9G 9C 9C 9C Wild Oats 2C,2G 9C      3C,7G 2C,3G 0 2C,9G 2C,6G 3C,9G 2C,7G 3C,9G 3C,9G 6G 2C,6G 3C,7G 2C,5G      5C,9G 3C,8G 9C 3C,9G 5C,9G Wheat 2C,5G 4C,8G 3G 2C,3G 0 4C,9G 10C 2C,9G      9C 3C,9G 9G 2C,9G 9G 4G 0 2G 0 9C 3C,9G 6C,9G Corn 3G 1C 0 0 0 6U,9C      3U,8G 4U,9G 2C,9G 3C,8H 1C,4G 3C,9G 2C,7H 6U,9C 3U,9G 6U,9C 3U,9C 10C      3C,9G 9C Soybean 4C,9G 4C,9G 4C,9G 3C,8G 4H 10C 9C 6C,9G 5C,9G 5C,9G      3C,9G 3C,8H 2H,7G 5C,9H 4C,8H 4C,9G 3C,9G 5C,9G 5C,9G 9C Rice 3G 5C,9G      2C,8G 3C,8G 2G 6C,9G 9C 9C 5C,9G 9C 3C,9G 5C,9G 2C,9G 9C 8G 4C,9G 8G      6C,9G 9C 9C Sorghum 4C,9H 9H 2C,5G 10C 9G 9C 3U,9G 9C 9C 10C 2C,9G 5C,9G      5C,9G 9C 2C,9G 9C 9C 9C 9C 9C Cheatgrass 4C,9G 4C,9G 2C,7G 3C,8G 2C,5G      10C 10C 10C 9C 10C 5C,9G 9C 9G 9G 5G 3C,9G 6G 9C 9C 9C Sugar beet 3C,8H      3C,8H 3C,8G 4C,9G 1C,2G 10C 10C 10C 10C 10C 10C 10C 10C 10C 5C,9H 10C      3C,9H 9C 10C 10C Velvetleaf 4C,9H 9C 3C,7H 5C,9G 3C,5G 10C 10C 10C 9C      10C 5C,9H 10C 5C,9H 5C,9H 3C,6H 9C 3C,8H 10C 9C 10C Giant Foxatil 2G 3G      2G 1C 0 4C,9G 2C,9G 9C 4C,9G 10C 3C,9G 9G 6G 9C 2C,8G 10C 9C 10C 9C 10C      Barley 0 3C,7G 0 0 0 3C,9G 9G 9C 9G 4C,9G 9G 9G 9G 2C,6G 5G 6G 2G 4C,9G      4C,9G 5C,9G PREEMERGENCE                      Cotton 0 1C 0 2G 0 9G 9G      3C,9G 8G 9G 5G 9G 8G 9G 0 3C,9G 0 9G 9G 9G Morningglory 0 0 0 3C,8H 6G      9G 8G 9G 9G 9G 2C,7H 9G 9G 2C,8H 2C,6H 9G 2C,4H 9G 9G 9G Cocklebur 0 0 0      2C,2H 1C 9H 9H 9H 8H 9H 2C,3H 9H -- 8H 2C,4G 9H 1C,2G 9G 9H 9H Nutsedge      0 10E 0 3C,8G 0 10E 10E 10E 9G 9G 6G 10E 9G 4C,9G 4G 9G 2G 10E 10E 10E      Crabgrass 0 0 0 0 0 7G 6G 3C,8G 2C,7G 10E 0 5G 0 3C,7H 0 3C,7H 0 8G 7G      4C,8G Barnyardgrass 0 2G 0 3C,8H 0 9H 9H 9H 3C,9H 3C,9H 3G 3C,8H 2C,7H      5C,9H 5G 9H 0 9H 9H 9H Wild Oats 0 0 0 0 0 7G 7G 3C,8G 2C,7G 2C,8H 2C,7G      2C,8G 0 7G 4G 8G 2C,4G 3C,9G 4C,8G 6C,9H Wheat 0 0 0 0 0 3C,9G 2C,9G 10C      4C,9H 10H 8H 3C,9H 7G 5G 0 6G 0 4C,9H 3C,9G 5C,9H Corn 0 0 0 0 0 9G 9G      10C 9G 9G 2C,7G 9G 2C,7G 9G 8G 9G 9G 2U,9G 2U,9G 9H Soybean 1C,1H 1H 0      2C 0 9H 9H 9H 8H 9H 2C,6G 3C,8H 2C,7G 4C,8H 3C,7H 9H 2C,6G 9H 9H 9H Rice      3G 7H 0 7H 6H 10E 10E 10E 10H 10E 9H 10E 10E 9H 3C,8H 10E 2C,8H 10E 10E      10E Sorghum 3C,3G 3C,7G 0 9H 3C,7G 10C 10C 10E 10E 9H 9H 10H 10H 10H 9H      10E 3C,8H 9H 4C,9H 10E Cheatgrass 0 5G 0 8H 0 10E 10H 10H 9H 9H 8H 9H 9H      9H 1C,4G 9H 4G 9H 9H 9H Sugar beet 1H 5H 0 5H 2G 9G 9G 5C,9G 5C,9G 4C,9G      3C,8G 3C,9G 2C,6G 4C,9G 5G 9G 2C,6G 9G 9G 9G Velvetleaf 0 2G 0 2G 4G 9G      9G 3C,9G 3C,9G 2C,8G 2C,7H 9G 9G 2C,7H 3C 3C,8H 2C 4C,9G 8G 5C,9G Giant      Foxatil 0 0 0 2C 0 9H 8G 3C,9H 3C,9H 2C,9H 2C,5H 8G 5G 7G 2G 9H 5G 9H 9H      9H Barley 0 0 0 0 0 9G 9G 10C 9G 9C 8G 9G 9G 7G 6G 9G 6G 3C,9G 2C,9G      4C,9H

      CMPD          CMPD 83 CMPD 84 CMPD 85 CMPD 86 CMPD 87 CMPD 88 CMPD 89      CMPD 90 CMPD 91 CMPD 92 93 Rate kg/ha 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0      .05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05        POSTEMERGENCE                      Cotton 9C 9C 4C,9G 9C 4C,9G 4C,9H      3C,4G 4C,9H 4C,8H -- -- -- -- -- -- -- -- -- -- -- Morningglory 10C 10C      10C 10C 10C 3C,8H 3C,6H 5C,9G 3C,9G 2C 0 3C,8H 2C,7G 2C,4H 0 2C,4G 2G      2C,7G 2H 3C,8H Cocklebur 10C 10C 10C 10C 10C 4G 0 9C 3C,8H 4C,9H 3C,8H      5C,9H 4C,8H 4C,9H 0 3C,8H 1C,5G 4C,8H 2C,7H 3C,8H Nutsedge 4C,8G 9C 9C      9C 5C,9G 3C,5G 0 4C,9G 3C,5G 2C,6G 6G 2C,8G 3G 0 0 0 0 0 0 0 Crabgrass      4G 4C,9G 7G 3C,6G 2G 3C,5G 0 5,9G 4G 0 0 0 0 0 0 0 0 0 0 0 Barnyardgrass      9C 9C 9C 10C 9C 9C 5C,9H 9C 9C 3C,6G 4G 3C,8H 0 2G 0 0 0 3C,6H 0 2C,7G      Wild Oats 4C,9G 9C 4C,9G 5C,9G 4C,9G 5C,9G 5C,9G 6C,9G 4C,9G 2C,2G 2G      2C,5G 2C,3G 3C,5G 2G 0 0 0 0 4G Wheat 4C,9G 9C 4C,9G 4C,9G 8G 5C,9G      4C,9G 3C,9G 3C,7G 6G 3G 3C,9G 2C,7G 2C,4G 2G 0 0 0 0 2G Corn 9C 6C,9G      3C,9G 5C,9G 9G 9C 9G 9C 9C 2C,6H 2G 3C,8H 3G 0 0 0 0 3C,7H 0 2C,7H      Soybean 4C,9G 6C,9G 4C,9G 5C,9G 3C,9G 4C,9G 4C,9G 5C,9G 4C,9G 4C,9G      4C,8G 5C,9G 3C,9H 3C,7H 0 0 0 3C,9G 2C,6H 3C,8H Rice 9C 9C 9C 9C 5C,9G      5C,9G 3C,8G 4C,9G 4C,9G 3C,8G 7G 2C,8G 2C,5G 4G 0 2G 0 4G 0 4G Sorghum      9C 9C 5C,9G 9C 9C 5C,9G 3C,8H 9C 9C 3C,8H 6G 3C,9H 2C,8H 2C,7H 0 3G 0      2C,8H 1C,5G 2C,8H Cheatgrass 9C 9C 9C 9C 3C,9G 4C,8G 4C,8G 6C,9G 2C,9G      2C,9G 2C,8G 9G 2C,9G 9G 4G 0 0 7G 0 5G Sugar beet 10C 10C 10C 10C 9C 10C      3C,7H 10C 5C,9G 10C 1C,3G 3C,9G 0 2C,5G 0 0 0 4C,8G 2C,7G 5C,8G Velvetlea      f 9C 10C 10C 10C 9C 3C,5H 1C 9C 3C,4H 3C,9H 2C,7G 4C,9G 2C,7G 2C,7G 5G 0      0 2C,4H 2G 3C,7H Giant Foxtail 10C 9C 9C 9C 9C 9C 3C,7H 10C 9C 4G 0 5G      2G 2G 0 0 0 4G 0 6G Barley 3C,9G 9C 4C,9G 4C,9G 3C,7G 2C 0 3C,6G 0 5G 0      5G 5G 3G 0 0 0 2G 0 0 PREEMERGENCE                      Cotton 9G 9G 9G      9G 9G 4C,8G 7G 5G 4G 0 0 0 0 0 0 0 0 0 0 2G Morningglory 9G 9G 9G 9G 9G      8H 2H 9G 8H 0 0 2C,3G 0 0 0 0 0 0 0 0 Cocklebur 9H 9H -- 9H 9H 4G -- 8H      8G -- 2G 3C,8H 0 0 0 0 -- 2C 0 0 Nutsedge 10E 10E 10E 10E 10E 3G 5G 7G      4G 4G 0 2G 0 0 0 0 0 0 0 0 Crabgrass 4C,8H 10E 2G 8H 0 9G 0 5G -- 2G 0      2G 0 0 0 0 0 9G 8G 0 Barnyardgrass 9H 9H 9H 9H 9H 3C,9H 3G 9H 7H 0 0 2G      0 0 0 0 0 0 0 0 Wild Oats 4C,8G 6C,9H 4C,9G 3C,9H 3C,5G 2C,3G 0 2C,4G 0      0 0 2G 0 0 0 0 0 0 0 0 Wheat 8G 10H 4C,8G 2C,9H 3C,8H 3G 0 5G 0 7G 0 4G      0 0 0 0 0 0 0 0 Corn 9G 9H 9H 9H 9H 3C,9H 4C,8G 9H 3C,9G 2C,3H 0 3C,6G      2G 0 0 0 0 0 0 1C Soybean 9H 9H 9H 9H 9H 9H 2H 9H 3C,6H 2C,3G 0 3C,5G      1C,3G 0 0 0 0 1C,2G 0 2C,4G Rice 10E 10E 10E 10E 10E 9H 7H 9H 5G 3C,8H 0      2C,3H 0 0 0 0 0 0 0 0 Sorghum 10H 10E 10E 10E 10H 3C,9H 4C,9G 10H 4C,9H      2C,9H 0 3C,7H 2C,3H 0 0 0 0 2C,5G 1C 3C,7H Cheatgrass 9H 9H 9H 9H 8H 7G      6G 9H 5G 8G 2G 8H 3G 0 0 0 0 0 0 0 Sugar beet 9C 9C 9G 3C,9G 9G 4C,8G 4H      4C,9G 3G 6G 0 2C,4G 4G 0 0 0 0 4G 2G 2H Velvetleaf 8G 4C,9G 4C,9G 9C 7H      2C 2G 7H 3G 0 0 2C,3H 0 0 0 0 0 0 0 2G Giant Foxtail 9H 9H 9H 9H 10H      3C,8H 3G 4C,9H 4C,8G 0 0 3G 0 0 0 0 0 0 0 0 Barley 4C,9H 9H 9H 3C,9H      4C,9H 4C,8G 0 9G 0 8G 0 2C,7H 2G 0 0 0 0 0 0 0        CMPD          CMPD 93 CMPD 94 CMPD 95 CMPD 96 CMPD 97 CMPD 98 CMPD 99      CMPD 100 CMPD 101 CMPD 102 103 Rate kg/ha 0.01 0.05 0.01 0.05 0.01 0.05      0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01      0.05      POSTEMERGENCE                      Cotton -- 4C,9G 1C,5G 0 0      4C,9G 4C,9G 9C 4C,9H 4C,9G 3C,9H 9C 3C,9G 4C,9H 2C,7G 3C,9G 2C,4G 4C,9H      3C,8H 9C Morningglory 2C,6H 5C,9G 5C,9G 0 0 10C 10C 10C 10C 9C 9C 10C      10C 3C,5G 2H 4C,9G 3C,8H 10C 5C,9G 10C Cocklebur 2C 4C,9H 3C,8H 4G 3G      10C 10C 10C 4G 10C 5C,9G 10C 10C 3C,9H 6G 5C,9G 3C,8H 9C 4C,9G 10C      Nutsedge 0 6G 0 0 0 5C,9G 3C,8G 10C 9C 4C,9G 4C,8G 10C 9C 3C,9G 3G 3C,8G      0 5C,9G 4C,9G 9C Crabgrass 0 0 0 0 0 7G 2G 4C,8G 5G 1C 0 2G 0 0 0 2G 0 0      0 0 Barnyardgrass 3G 4C,9H 2C,7H 0 0 10C 10C 10C 10C 9C 3C,8H 3C,9H      1C,4H 2H 0 2C,5H 0 3C,8H 1H 3C,9H Wild Oats 0 2G 0 0 0 9G 2C,5G 4C,9G      3C,6G 5G 0 3C,7G 0 0 0 2C,5G 0 3C,6G 3G 2C,5G Wheat 0 4G 3G 0 0 9G 2C,6G      3C,9G 8G 2C,7G 3G 2C,8G 7G 0 0 2C,7G 3G 5C,9G 7G 7G Corn 0 0 0 0 0 2G 0      2C,7G 2G 0 0 10C 10C 3G 0 3C,9H 4G 4C,9H 2C,7G 1H Soybean 2C,7H 4C,9G      3C,7H 0 0 4C,9G 4C,9G 9C 9C 4C,9G 4C,9G 9C 4C,9G 3H 0 3C,7H 2C,5H 5C,9G      4C,9G 3C,9G Rice 3G 2C,5G 0 0 0 9C 4C,8G 9C 5C,9G 4C,9G 5G 4C,9G 8G 2G 0      7G 0 8G 0 5C,9G Sorghum 2C,7G 4C,9G 3C,9G 0 0 9C 9C 10C 10C 10C 9C 5C,9G      10C 4C,9G 7H 2C,9G 3C,8H 9C 4C,9H 9C Cheatgrass 0 10C 4G 0 0 2C,5G 0      4C,9G 6G 3C,7G 0 9C 3C,8G 2C,5G 0 8G 2G 4C,9G 3C,7G 8G Sugar beet 3C,7G      9C 2C,3H 0 0 4C,9G 2C,3G 10C 10C 10C 4C,8G 10C 9C 3C,5G 1C 10C 3C,7G 9C      3C,7G 10C Velvetleaf 2C,2H 4C,9H 2C,4H 3G 2G 10C 5C,9G 10C 10C 4C,9H      4C,8H 10C 10C 3C,8H 3C,7G 4C,8H 3C,7H 9C 4C,9G 10C Giant Foxtail 2G      2C,7G 2G 0 0 4C,9G 3C,9G 5C,9G 6G 3C,8G 2C,6G 2C,7G 3G 2G 0 2C,7G 2G      4C,9G 4G 6G Barley 0 2G 0 0 0 9G 6G 9G 5G 2C,2G 0 9C 8G 2G 0 2C,6G 0      2C,9G 2C,6G 7G PREEMERGENCE                      Cotton 0 5G 0 0 0 2C,8G      6G 9G 9G 3C,8G 2C,4G 7H 6G 1C 0 0 0 8G 2C,3G 9G Morningglory 0 3C,8G 5G      0 0 9G 8G 9G 9G 9H 4H 9G 6H 2G 0 3C,4H 0 8H 3C,4H 9G Cocklebur -- 2C,4H      0 0 -- 9H 3C,8H 3G 5G 2C,7G 0 8H 8H 5G 0 2C,2G 0 8H 3C,3H 9G Nutsedge 0      0 0 10E 4G 10E 3C,9G 10E 10E 10E 10E 10E 9G 9G 0 3G 0 10E 0 10E Crabgrass       0 2C,5G 2G 0 0 2C,7G 5G 10E 2C,5G 2C,3G 2G 10E 6G 5G 0 0 0 0 0 2G      Barnyardgrass 0 4C,9H 5G 0 0 9H 2C,7H 9H 9H 9H 3C,7H 7H 0 0 0 0 0 6H 2G      8H Wild Oats 0 0 0 0 0 7G 0 3C,8G 2C,6G 2C 0 7G 5G 0 0 0 0 3C,8G 0 5G      Wheat 0 7G 0 0 0 9G 9G 10H 9H 7G 0 9G 8G 0 0 5G 0 9H 3C,8G 7G Corn 0      2C,3G 0 0 0 4C,7G 1C,3G 3C,8G 3G 0 0 3C,9G 7G 0 0 0 0 3C,9H 3C,6G 0      Soybean 0 2C,3G 0 0 0 9G 3C,7H 9H 9H 3C,8H 3C,4G 3C,8H 6H 2C 0 2C 0      3C,6H 3C,5H 8H Rice 0 5G 0 6G 0 10E 8G 10E 9H 10H 3C,7G 9H 9H 6G 0 4G 0      8H 0 10H Sorghum 0 4C,9H 3C,8H 4G 0 10E 6C,9G 10E 5C,9H 10H 10H 10H 9H      3C,8G 2G 2C,6G 0 10H 4C,8H 10E Cheatgrass 0 8G 0 0 0 7G 7G 9G 7G 9G 2G      9G 8H 0 0 5G 0 8G 7G 8G Sugar beet 0 4C,8G 5G 6G 0 4C,9G 8G 9G 9G 4C,9G      8H 4C,9G 6H 2H 2G 7G 0 4C,9G 4C,8H 9G Velvetleaf 0 3G 0 0 0 4C,9G 2C,8G      5C,9G 7H 2C,7H 2C,3H 4C,9G 8G 3H 0 3C,5G 0 4C,8H 1H 7H Giant Foxtail 0      3C,8H 4G 0 0 2C,9G 8G 2C,7G 2C,5G 2C,9H 3G 4G 0 0 0 3G 0 8G 2G 7G Barley      0 3G 0 0 0 9G 7G 9G 9G 2C,8G 7G 9G 8G 0 0 5G 0 9G 3C,7G 9G        CMPD          CMPD 103 CMPD 104 CMPD 105 CMPD 106 CMPD 107 CMPD 108      CMPD 109 CMPD 110 CMPD 111 CMPD 112 113 Rate kg/ha 0.01 0.05 0.01 0.05      0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05      0.01 0.05        POSTEMERGENCE                      Cotton 4C,9H 9C 4C,9G 5C,9G 4C,9H      4C,9G 4C,9H 10C 5C,9G 5C,9G 10C 9C 5C,9G 6C,9G 3C,9G 4C,8H 3C,7H 4C,9H      4C,8G 1H Morningglory 4C,9G 10C 10C 10C 3C,8G 10C 0 10C 2H 10C 9C 2C,7G      5G 10C 10C 4C,8H 3C,7G 10C 4C,9G 0 Cocklebur 10C 10C 10C 9C 10C 10C 10C      10C 10C 10C 10C 10C 10C 10C 10C 4C,9H 2C,4G 10C 4C,8H 1H Nutsedge 5C,9G      9C 9C 5C,9G 8G 9C 4C,8G 5C,9G 3C,8G 3C,8G 2C,7G 4C,9G 6C,9G 5C,9G 3C,8G      2C,4G 0 3C,9G 0 0 Crabgrass 0 3G 0 3G 0 5G 0 3C,7G 2G 3C,7G 5G 3C,6G 5G      3C,5G 3G 0 0 2G 0 2G Barnyardgrass 7H 10C 9C 9C 3C,8H 10C 5C,9H 10C 9C      9C 9C 10C 9C 9C 4C,9H 3C,7H 2C,5H 9C 3C,7G 5C,9H Wild Oats 2G 3C,9G      3C,7G 3C,7G 3C,5G 3C,9G 3C,8G 3C,9G 3C,8G 4C,9G 3C,7G 4C,9G 4C,9G 3C,9G      2C,3G 0 0 3C,5G 0 3C,5G Wheat 2G 2C,9G 3C,9G 6C,9G 2C,8G 3C,9G 5C,9G      5C,9G 3C,9G 9C 5C,9G 9C 2C,9G 3C,9G 3G 0 0 4G 0 9C Corn 0 0 0 0 0 0 0 9C      3C,9G 4C,9G 4C,9H 3C,8H 3C,7H 3C,8H 2G 3C,7G 0 9G 3C,6G 2C,9G Soybean 8H      9C 9C 9C 5C,9G 5C,9G 5C,9G 9C 5C,9G 5C,9G 9C 9C 4C,9G 4C,9G 3C,6G 4C,9G      3C,8G 4C,9G 4C,8G 2G Rice 7G 9C 3C,9G 5C,9G 4C,9G 5C,9G 5C,9G 9C 5C,9G      9C 9C 9C 9C 9C 4C,9G 3G 0 4G 0 9C Sorghum 9C 9C 9C 9C 5C,9G 10C 3C,9H 9C      9C 10C 9C 9C 9C 9C 4C,9H 3C,7H 0 3C,9G 3C,8H 4C,9G Cheatgrass 3G 7G 3G      7G 5G 5C,9G 5C,9H 10C 2C,8G 5C,9G 3C,8G 5C,9G 8G 4C,8G 6G 0 0 0 0 3C,9G      Sugar beet 10C 10C 10C 10C 4C,9H 10C 10C 10C 9C 10C 10C 10C 9C 9C 9C      3C,5H 3C,8H 10C 4C,8H 3C,8G Velvetleaf 5C,9G 10C 10C 10C 4C,8G 9C 4C,9H      10C 9C 9C 10C 9C 4C,8H 9C 9C 3C,7H 0 4C,9G 3C,6H 4G Giant Foxtail 3G      3C,7H 3C,6G 4C,8G 7G 4C,8G 3C,8G 5C,9G 3C,8G 5C,9G 4C,8G 4C,8G 2C,6G      3C,8G 3G 2G 0 3C,7G 2C,2G 3C,8H Barley 2G 3C,9G 3C,8G 8G 6G 2C,9G 3C,8G      4C,9G 9G 3C,9G 8G 4C,9G 2C,8G 9G 5G 0 0 3G 0 2C,9G PREEMERGENCE                  Cotton 2G 9H 5G 2C,8H 0 2C,4G 2G 9G 9G 3C,8G 7G 8H 3G 8G 7G      0 0 2G 0 0 Morningglory 6H 9G 2C,5G 3H 0 2C,5G 0 5G 2G 9H 3G 5G 1H 9G 7H      2C,3H 0 8G 0 0 Cocklebur 9H -- 1H 8H 2H 2C,5G 3C,7H 9H 9H 9H 9H -- 3C,8H      9H 8H 0 -- 7H 2C,5G 0 Nutsedge 10E 9G 10E 9G 0 8G 0 10E 10E 10E 4C,9G      10E 10E 10E 10E 10E 0 10E 0 0 Crabgrass 0 4G 0 0 0 10H 0 8G 2C,5G 4C,8G      3C,7G 4C,8G 2C,2G 3C,5G 3G 2G 0 2G 0 2G Barnyardgrass 4G 9H 2G 4C,9H 0 0      0 5C,9H 9H 9H 3C,9H 5C,9H 2C,7H 9H 3C,9H 7H 0 9H 6H 4G Wild Oats 0 7G 0      2C,6G 0 0 2G 8G 5G 5C,9G 3C,8G 4C,8H 3C,7G 3C,8G 3G 0 0 0 0 0 Wheat 2G      9H 5G 8H 0 5G 5G 9H 7G 9H 3C,9G 3C,9H 6G 3C,7G 3G 0 0 0 0 2G Corn 0 3G 0      0 3G 0 0 9G 7G 3C,9H 3C,8G 3C,7G 2C,3G 3C,7G 2C,2G 3C,3G 0 2G 3G 2G      Soybean 3C,7H 9H 6H 3C,7H 3C,3H 9H 3C,4H 9H 3C,6H 3C,8H 3C,7H 9H 3C,6G      4C,8H 3C,6H 2C,4H 0 3C,7G 3C,4G 0 Rice 3C,7G 9H 7G 10H 0 8H 3C,6G 10E 9H      10E 4C,9H 10E 10H 10E 9H 2C,5G 0 3C,7H 3G 2C,5G Sorghum 9H 6C,9H 9H 9H      2C 4C,9H 3C,8H 10H 9H 10E 4C,9H 10H 9H 5C,9H 5C,9H 3C,6G 0 8H 3C,5G      3C,5G Cheatgrass 5G 8G 0 8G 0 8G 5G 10E 4C,9G 10E 3C,8G 5C,9G 8H 9G      3C,7G 0 0 4G 0 0 Sugar beet 9G 5C,9G 8G 5C,9G 7G 3C,8G 7H 9C 10C 10C      4C,9G 9C 9G 9C 9C 5G 2G 3C,9H 7H 1H Velvetleaf 1H 4C,8G 3G 6H 2G 2C,2H      2H 5C,9G 8H 5C,9G 3C,5H 5C,9G 3C,7G 4C,8H 5H 2G 0 2C,2H 0 2G Giant      Foxtail 1C 3G 0 3G 0 0 0 9H 3C,7G 9H 3C,7G 3C,8G 3C,5G 3C,8G 3C,6G 1H 0      7G 0 2G Barley 6G 8G 4G 8G 3G 9G 3C,7H -- -- -- 2C,8G 8G 7G -- 2C,5G 0 0      0 3G 9G        CMPD          CMPD 113 CMPD 114 CMPD 115 CMPD 116 CMPD 117 CMPD 118      CMPD 119 CMPD 120 CMPD 121 CMPD 122 123 Rate kg/ha  0.01 0.05 0.01 0.05      0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05      0.01 0.05        POSTEMERGENCE                      Cotton 0 2C,3H 2G 4C,9G 9H 5C,9G      10C 5C,9G 4C,8G 9H 8H 9C 9C 1C 0 10C 4C,9G 0 -- 4C,9H Morningglory 0 1H      0 10C 5C,9G 10C 10C 5C,9G 4C,9H 9C 3C,8H 10C 10C 3H 0 10C 10C 0 -- 10C      Cocklebur 0 2H 2H 8G 2G 10C 2C,3H 4C,9H 3C,5H 4C,9G 3C,7H 10C 10C 1H 0      10C 9C 2H -- 9C Nutsedge 0 4C,9G 0 10C 4C,8G 9C 3C,8G 9G 8G 9C 4C,8G      5C,9G 4C,9G 0 0 9G 8G 0 -- 3C,8G Crabgrass 0 3C,6G 3G 6G 2G 3C,6G 2C 0 0      0 0 3C,5G 2G 0 0 3C,5G 2G 0 -- 2C,5G Barnyardgrass 3C,6G 9C 3C,8H 9C      5C,9G 9C 9C 2H 0 4H 0 9C 9C 4H 0 9C 9C 1H -- 9C Wild Oats 2G 9C 3C,6H      5C,9G 3G 3C,7G 3G 0 0 0 0 4C,8G 3C,5G 3C,7G 0 4C,9G 3C,5G 2C,5G -- 4C,9G      Wheat 8G 9C 3C,7H 9G 2C,9G 5C,9G 9G 2G 0 0 0 9C 4C,9G 8G 0 5C,9G 8G 6G      -- 9G Corn 2C,5H 4H 0 2G 0 6H 0 0 0 0 0 2C,7H 3H 0 0 0 0 0 -- 0 Soybean      0 3C,8G 0 5C,9G 4C,9G 9C 5C,9G 4C,9G 3C,7H 3C,7H 3C,7H 5C,9G 5C,9G 3C,4G      0 5C,9G 4C,9G 2G -- 4C,9G Rice 8G 5C,9G 9G 9C 9C 9C 3C,8G 2G 0 2G 0 9C      9C 8G 0 9C 9C 3G -- 9C Sorghum 3C,7H 9C 4C,9G 9C 9C 9C 9C 3C,3H 0 6H 0      9C 9C 4C,9H 0 9C 4C,9G 2C,5G -- 9C Cheatgrass 0 9C 3C,7G 8G 6G 3C,8G      3C,6G 0 0 0 0 5C,9G 4C,8G 3C,8G 0 4C,9G 4C,9G 3C,8G -- 9C Sugar beet 3G      3C,7H 3C,6G 9C 9C 10C 9C 9C 3C,7G 9C 3C,7H 10C 9C 1H 0 10C 10C 0 -- 10C      Velvetleaf 0 2H 0 9C 9C 10C 9C 3C,8H 3C,4H 4C,8H 3C,6H 10C 9C 1C 0 10C      9C 1C -- 9C Giant Foxtail 2G 9C 3C,8H 9C 4C,9G 4C,9H 3C,7G 0 0 1C 2G 9C      9C 2C,5G 0 9C 4C,9G 0 -- 5C,9G Barley 9G 10C 2C,8G 3C,8G 3C,6G 3C,8G 3G      0 0 0 0 5C,9G 4C,9G 7G 0 4C,9G 3C,8G 8G -- 3C,8G PREEMERGENCE                Cotton 0 2H 0 3C,5G 6G 3C,5G 0 2G 0 2G 0 4C,8G 6G 0 0 3C,7H 0      0 -- 5G Morningglory 0 0 0 7H 0 2C,6G 0 7H 0 8H 0 9G 3C,7H 0 0 3C,7H      3C,3H 0 -- 3C,8H Cocklebur -- 0 0 3G 0 -- 3G 3C,5G 1C 3C,3H 0 9H 2C,2H 0      0 3C,8H 3C,3G 0 -- 3C,6H Nutsedge 0 0 0 9G 0 8G 0 4G 0 9G 0 10E 3C,9G 0      0 4C,8G 0 0 -- 9G Crabgrass 0 7G 3G 4G 0 9G 0 0 0 0 0 3C,4G 3C,5G 0 0      3C,6G 3G 0 -- 7G Barnyardgrass 0 6G 0 8H 2G 3C,9H 2G 0 0 3G 0 4C,9H      3C,7H 0 0 4C,9H 4G 0 -- 3C,9H Wild Oats 0 0 0 2C 0 1C 0 0 0 0 0 3C,6G 0      0 0 2G 0 0 -- 3G Wheat 0 7G 0 2G 0 3C,7H 0 0 0 0 0 3C,9H 3G 0 0 8G 6G 0      -- 8G Corn 0 0 0 0 0 3G 0 0 0 7G 0 3C,6H 0 0 0 2H 0 0 -- 1H Soybean 0 0      0 3C,6H 2C 8H 3C,6H 3C,5G 2C 2C,6H 0 4C,8H 3C,6H 0 0 3C,7H 0 0 -- 3C,5H      Rice 0 2C,5G 0 9H 3C,5G 10H 5G 0 0 4G 0 10E 3C,8H 0 0 3C,8H 4G 0 -- 9H      Sorghum 0 3C,7G 0 9H 3C,7G 10E 8G 0 0 3G 0 5C,9H 3C,8H 0 0 4C,9H 2C,6G 0      -- 5C,9H Cheatgrass 0 0 0 7G 0 9H 2G 0 0 0 0 5C,9G 3C,9G 0 0 9H 7G 0 --      5C,9G Sugar beet 0 4H 0 4C,9G 7H 4C,9G 6H 3C,7G 2H 7G 0 9C 9C 3G 0 9C      4C,8H 2G -- 9C Velvetleaf 0 0 0 3C,5H 0 3C,8H 1C 2C 0 3C,4G 0 4C,8H      3C,6H 0 0 3C,7H 1C 0 -- 5G Giant Foxtail 0 3G 0 7G 0 3C,8G 0 0 0 0 0      4C,9H 3C,8G 0 0 3C,8H 0 0 -- 9H Barley 0 9G 2G 2C,9G 3G 9G 0 0 0 4G 0      3C,9G 3C,8G 0 0 8G 0 0 -- 7G

      CMPD          CMPD 123 CMPD 124 CMPD 125 CMPD 126 CMPD 127 CMPD 128      CMPD 129 CMPD 130 CMPD 131 CMPD 132 133 Rate kg/ha 0.010.05 0.01 0.05      0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05      0.01 0.05        POSTEMERGENCE                      Cotton 4C,9H 4C,9H 3C,8H 5C,9G 9C      9H -- 10C 3C,9G 2C,9H 2C,5H 3C,9H 2C,8H 2C,8H 3C,6H 10C 5C,9G 9C 10C 9C      Morningglory 9C 4C,9G 4C,9H 10C 10C 4C,9G -- 10C 9C 6C,9G 4C,8H 3C,8H      2C,8G 6C,9G 4C,8H 10C 4C,9G 10C 9C 9C Cocklebur 4C,9H 5C,9G 4C,9H 10C      10C 4C,9G -- 10C 5C,9H 3C,9H 3C,4H 9C 4C,9H 10C 2C,3H 10C 10C 10C 10C      10C Nutsedge 2C,5G 9G 3C,9G 10C 5C,9G 8G -- 2C,8G 8G 2C,6G 0 6G 2C,7G      3C,8G 2C,4G 9C 3C,8G 4C,9G 2C,9G 9C Crabgrass 2G 3C,4G 2G 3C,8G 5G 0 --      0 0 0 0 0 0 0 0 4C,8G 2G 4C,8G 3G 5C,9G Barnyardgrass 4C,9H 5C,9H 4C,8H      5C,9H 3C,6H 0 -- 3C,9H 2C,7H 2C,5H 0 2G 3G 2C,6H 2C,6G 9C 9C 10C 9C 10C      Wild Oats 5G 4C,9G 7G 8G 4G 0 -- 2C,6G 2C 2C 0 2G 0 2C,5G 3G 3C,9G 5G      4C,9G 3C,6G 4C,9G Wheat 8G 3C,9G 9G 8G 4G 0 -- 9G 9G 2C 0 2G 0 2C,9G 2G      3C,9G 9G 3C,9G 9G 4C,9G Corn 0 0 0 3C,9G 9G 2H -- 3C,9G 3C,7H 2C,8H      2C,3G 2C 0 3C,8H 2C,2H 10C 3C,9G 5C,9G 4G 3C,9H Soybean 3C,8G 5C,9G      4C,9G 4C,9G 4C,9G 3C,5G -- 3C,8H 3C,8G 3C,8H 2C,3H 2H 0 4C,8H 3C,4H 9C      9C 5C,9G 9C 9C Rice 5C,9G 9C 5C,9G 5C,9G 3C,9G 0 -- 2C,9G 6G 4G 0 2C,5G      0 3C,9G 2C,4G 9C 9C 9C 9C 9C Sorghum 4C,9G 5C,9G 3C,9G 5C,9G 3C,9G 3C,6G      -- 5C,9G 2C,9G 9H 2C,7H 9G 3C,8H 2C,9G 2C,7H 10C 9C 9C 9C 10C Cheatgrass      9G 6C,9G 3C,9G 9C 9C 5G -- 10C 3C,9G 5G 3G 2C,8G 5G 8G 8G 9C 9C 10C 9C      10C Sugar beet 4C,8H 9C 4C,9H 10C 10C 3C,8G -- 10C 6C,9G 3C,9H 2C,3G      3C,6G 2C,7G 3C,9G 3C,5H 9C 10C 10C 10C 10C Velvetleaf 3C,7H 9C 4C,8H 10C      10C 3C,6G -- 9C 9C 3C,7H 2C,4G 2C,8G 2C,7G 5C,9H 3C,7G 10C 10C 10C 5C,9G      10C Giant Foxtail 3C,7H 6C,9G 4C,8G 3C,7G 5G 0 -- 2C,9G 6G 3G 2G 2G 3G      2C,7G 3G 9C 4C,9G 9C 3C,8G 9C Barley 3C,6G 5C,9G 2C,9G 8G 5G 0 -- 9G 6G      4G 0 0 0 7G 0 4C,9G 5G 9C 7G 4C,9G PREEMERGENCE      Cotton 0 2G 0 9G 8G 0 -- 2C,8G 4G 0 0 2G 0 4G 0 9G 6G 8G 3H 9G Morningglo      ry 2C,6H 7H 1H 9G 9G 1H -- 9G 3C,9H 2C,3H 0 2C,6H 0 0 0 9G 3G 2C,3G 2G      7G Cocklebur -- 2H 1H 9H 9H 7G -- 3C,8H 3C,7H 2H 0 3C,8H 0 0 0 8H 9H 9H      2C,2H 8H Nutsedge 10E 3G 0 10E 10E 0 -- 10E 2C,9G 8G 0 9G 0 0 0 10E 10E      9G 3C,9G 10E Crabgrass 0 0 0 5G 0 0 -- 2C 0 2G 0 2G 0 0 0 5G 0 3C,9G 5G      8G Barnyardgrass 3C,8H 5G 0 9H 3C,7G 0 -- 4C,8H 2C,3G 5G 0 6G 0 3G 0 9H      5G 3C,9H 3C,7G 9H Wild Oats 0 2G 0 6G 3G 0 -- 4C,7G 3G 0 0 2G 0 0 0      3C,6G 0 3C,5G 0 3C,7G Wheat 0 3G 0 7G 2G 0 -- 8G 3G 0 0 0 0 0 0 9H 0      3C,9H 0 3C,9H Corn 0 0 0 9H 2C,9G 0 -- 4C,8H 2C,3G 0 0 3G 0 0 0 3C,9H 2G      3C,8H 3G 3C,9H Soybean 2C,3H 3C,6G 0 2C,7H 3C,2H 2G -- 3C,5G 2C 2C 0 2C      0 0 0 9H 3C,4G 3C,7G 3C,5H 9H Rice 3C,8G 3C,6G 0 9H 9H 4G -- 9H 3C 0 0      2C,8H 0 5G 0 10E 8G 10E 9H 10E Sorghum 3C,9H 3C,7G 2C 9H 5C,9H 2C --      5C,9H 3C,8H 2C,3G 0 3C,9H 0 2C,5G 2G 5C,9H 3C,8G 5C,9H 3C,9H 10H      Cheatgrass 8G 8G 0 9H 8G 0 -- 4C,9H 3C,8H 0 0 4G 0 3C,7G 2G 9H 8G 8G 8H      9H Sugar beet 5G 9G 4G 10C 9C 8G -- 3C,9G 3C,9G 0 0 3C,8G 0 9C 0 5C,9G      9C 5C,9G 7H 4C,9G Velvetleaf 0 2C,3G 2H 5C,9G 4C,8H 0 -- 4C,8H 3C,6G 0 0      3G 0 0 0 8H 7G 2C,6H 2C,2H 7H Giant Foxtail 2G 0 0 8G 2C,5G 0 -- 3C,8H      6G 0 0 3G 0 2G 0 9H 6G 3C,9H 4G 9H Barley 3C,7G 7G -- 8G 8G 0 -- 8G 2G 0      0 2G 0 7G 0 9G 2C,4G 3C,8G 2C,8G 9G        CMPD          CMPD 133 CMPD 134 CMPD 135 CMPD 136 CMPD 137 CMPD 138      CMPD 139 CMPD 140 CMPD 141 CMPD 142 143 Rate kg/ha 0.01 0.05  0.01 0.05      0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05      0.01 0.05        POSTEMERGENCE                      Cotton 7G 9C 3C,8H 2C,3G 1C 8H      2C,2G 10C 4C,9G 3C,7G 0 4C,9G 3C,8G 9C 3C,9G 5C,9H 4C,8H 10C 5G 5C,9G      Morningglory 7G 10C 9C 4C,8H 3C,4H 4C,8H 3C,8H 10C 4C,8G 10C 3C,7H 4C,9G      4C,8G 9C 5C,9G 9C 4C,8H 10C 5C,9G 10C Cocklebur 5C,9G 10C 10C 3C,5H 3G      4C,8H 3C,5G 10C 10C 2H 0 4C,9G 4C,9G 10C 8H 10C 4C,9H 9C 3C,7H 10C      Nutsedge 3C,9G 9C 9G 0 2C,4G 3C,7G 3C,5G 3C,9G 3C,8G 0 0 3C,5G 2C,4G      4C,9G 9G 2C,5G 3G 4C,9G 4C,9G 4C,8G Crabgrass 6G 3G 0 2G 0 3G 0 4G 0 0 0      5G 0 5G 0 0 0 3G 0 3G Barnyardgrass 10C 9C 5C,9H 3C,8H 3C,7H 9C 4C,9H 9C      3C,9H 9H 4C,9H 9C 3C,8H 9C 5C,9H 4C,9H 3C,7H 4C,9H 3C,7H 9C Wild Oats      4C,9G 4C,9G 2G 0 0 2C,3G 2G 0 0 0 0 2C 0 1C 0 1C 0 0 0 2C,5G Wheat 9C 9G      4G 2G 0 0 0 2G 0 7G 0 9G 3G 5G 0 2G 0 4G 0 7G Corn 2H 0 3G 3C,9G 3C,7H      9C 3C,8H 0 0 0 0 0 0 3G 0 0 0 1C 0 3C,7G Soybean 4C,9G 4C,9G 3C,8H 3C,8G      4H 4C,9G 4C,8H 3C,9G 1H 3C,5H 2H 4C,9G 4C,8G 5C,9G 3C,5H 4C,9G 1H 4C,9G      5C,9G 5C,9G Rice 5C,9G 9C 7G 3G 0 2C,3G 0 5C,9G 3C,6G 3C,7G 3G 5C,9G      2C,5G 6C,9G 6G 5G 0 5C,9G 8G 9C Sorghum 5C,9G 9C 3C,8H 3C,9H 3C,7H 9C      3C,9G 9C 9G 5C,9G 4C,9H 4C,9G 2C,5G 6C,9G 4C,9H 5C,9H 3C,6G 5C,9H 3C,9H      9C Cheatgrass 9C 9C 9G 8G 6G 5C,9G 7G 8G 5G 3C,8G 6G 5G 0 9C 3C,9G 9G 8G      3C,9G 8G 3C,9G Sugar beet 9C 9C 9C 8H 5H 9C 3C,7G 9C 3C,8G 3C,4H 2H      5C,9H 4C,9H 10C 9C 9C 9C 9C 9G 10C Velvetleaf 10C 9C 5C,9G 2G 2G 3C,7G      1C 10C 3C,8G 3C,7H 2G 10C 3C,8H 10C 9C 9C 4C,7G 10C 9C 10C Giant Foxtail      4C,8G 5C,9G 3C,7G 2C,8G 7G 9C 3C,7G 3C,9G 3C,7G 3C,7G 5G 5C,9G 3C,5G      3C,8G 3C,5G 3C,7G 3G 3C,7G 3C,5G 9C Barley 8G 7G 0 0 0 2G 0 0 0 0 0 2G 0      0 0 0 0 2C,3G 0 8G PREEMERGENCE                      Cotton 2G 7H 1H 0 0      0 0 6G 0 0 0 0 0 2C 0 1C 0 2C 0 3C,5G Morningglory 0 9G 7G 1H 0 3C,7H 0      9G 4G 0 0 0 0 8H 0 3C,3H 0 2C,2H 0 8G Cocklebur 2C,8H 8H -- 4H -- 3C,5G      2C 3C,5H 2C,5G -- 0 0 0 8G 0 2C 0 2C 0 3C,3H Nutsedge 10E 10E 9G 10E 0      7G 0 9G 0 0 0 0 0 9G 0 0 0 10E 0 0 Crabgrass 0 3G 0 0 -- 3C,7G 0 3G 0 0      0 0 0 4G 0 0 0 2G 0 0 Barnyardgrass 8G 9H 7H 5G 0 4C,8H 0 9H 0 0 0 0 0      3C,7G 0 1C 0 3C,7H 0 7G Wild Oats 2C,3G 6G 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0      1C 0 0 Wheat 5G 7G 0 0 0 0 0 3G 0 0 0 0 0 0 0 0 0 6G 0 6G Corn 3C,5G      3C,7G 5G 6H 0 3C,8H 2C 2G 0 0 0 0 0 0 0 0 0 2C,3G 0 3C,7G Soybean 3C,6H      3C,7H 3C,4H 0 0 3C,3G 0 3C,3H 2G 0 0 0 0 3C,3H 0 2G 0 3C,5H 0 3C,7G Rice      9H 10E 9H 2G 0 4G 0 9G 9G 0 0 0 0 9H 0 0 0 3C,9H 0 10E Sorghum 3C,9H 10H      5C,9H 3C,7G 0 5C,9H 3C,6G 10H 9H 0 0 0 0 4C,8G 3C 4C,7G 0 3C,9H 0 9H      Cheatgrass 8H 9H 8G 6G 0 8H 0 9G 0 0 0 0 0 8G 0 2G 0 9H 0 4G Sugar beet      4C,9G 9G 8G 7G 2H 4C,8H 1H 9H 8H 4G 0 0 0 9G 4G 4C,7H 0 9G 0 4C,9G      Velvetleaf 3G 7H 5G 0 2G 0 0 5H 0 0 0 0 0 7H 0 2C 0 2H 0 3C,6H Giant      Foxtail 6G 9H 6G 2G 2G 3C,8G 0 9H 0 0 0 0 0 3C,4G 0 3G 0 2C,5G 0 8G      Barley 9G 9G 7G 0 0 4G 0 2C,3G 0 0 0 0 0 0 0 0 0 2C,3G 0 2C,4G        CMPD          CMPD 143 CMPD 144 CMPD 145 CMPD 146 CMPD 147 CMPD 148      CMPD 149 CMPD 150 CMPD 151 CMPD 152 153 Rate kg/ha 0.01 0.05 0.01 0.05      0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05      0.01 0.05        POSTEMERGENCE                      Cotton 4C,8H 3C,7G 2C,2G 4C,9H      4C,9H 10C 4C,8G 3C,8H 0 8H 0 9G 4C,8H 0 0 3C,7G 0 10C 9C 10C Morningglory       5C,9G 3C,8G 3C,6G 9C 5C,9H 10C 4C,8G 3C,5G 0 3C,4H 0 4C,9G 3C,8H 2C,3G      0 4C,8H 0 10C 10C 10C Cocklebur 9C 4C,8H 2H 10C 3C,9G 10C 4C,9H 5C,9G 2H      3C,3H 0 4C,9G 3C,3H 2C 0 4C,8H 0 10C 10C 10C Nutsedge 2C,5G 0 -- -- --      4C,9G 4C,9G -- -- -- 0 -- 2G 0 0 0 0 4C,9G 4C,9G 4C,9G Crabgrass 3G 0 0      5G 0 5G 4G 2G 0 3G 0 5G 3G 0 0 3C,5G 3G 3C,7G 3C,6G 3C,7G Barnyardgrass      3C,8H 3C,6H 0 5C,9H 3C,7H 9C 4C,8H 4C,8H 2H 5C,9H 3C,7H 9C 3C,8H 3C,9H      5G 9C 3C,9H 9C 9C 9C Wild Oats 0 0 0 2G 0 0 0 1C 0 3C,7G 0 3C,8G 2G      2C,9G 3C,4G 5C,9G 3C,8G 4C,9G 2C,6G 3C,7G Wheat 3G 0 0 -- -- 7G -- 3G 0      -- 0 -- -- 9G 9G 9G 9G 2C,9G 9G 4C,9G Corn 2G 0 0 3C,9H 2C,5G 3C,7H 1H      2H 0 5C,9G 3C,3G 9C 3C,8H 3G 0 0 0 0 0 0 Soybean 4C,9G 3C,6H 2C,2H 5C,9G      3C,9H 5C,9G 4C,8G 3C,8G 0 3C,7G 2G 5C,9G 3C,7G 3C,7H 1H 3C,8G 3C,6G      5C,9G 9C 9C Rice 6C,9G 2C 0 9C 3C,8G 5C,9G 3C,5G 4C,9G 0 8G 2G 9C 5C,9G      3C,9G 5G 4C,9G 6G 5C,9G 5C,9G 5C,9G Sorghum 6C,9G 3C,7G 2G 9C 5C,9G 9C      4C,9H 4C,9G 3G 4C,9H 3C,6G 9C 4C,9G 3C,8H 3G 5C,9G 3C,9G 9C 9C 9C      Cheatgrass 2G 0 0 3C,7G 2G 9C 9G 3C,5G 0 5C,9G 6G 8G 6G 5G 0 8G 2C,5G 9G      8G 4C,9G Sugar beet 9C 3C,8G 0 9C 9C 10C 5C,9H 3C,7G 3G 3C,7H 2H 9C      4C,8H 3C,7H 5H 4C,8G 4C,6G 10C 9C 9C Velvetleaf 4C,8H 3C,7G 0 6C,9G      3C,6G 10C 5C,9H 3C,6G 0 0 -- 4C,8G 2C 3G 0 1C 0 10C 5C,9G 10C Giant      Foxtail 5C,9G 3G 0 5C,9G 5C,9G 5C,9G 3C,8G 3C,7G 0 4C,8G 3G 5C,9G      3C,8G2G 0 5C,9G 2C,5G 4C,8G 3C,7G 4C,8G Barley 0 0 0 7G 0 5G 0 3C,7G 0 0      0 6G 0 8G 7G 8G 6G 8G 8G 8G PREEMERGENCE                       Cotton 0      0 0 1C 0 2G 0 0 0 0 0 2C,2G 0 0 0 1C 0 9G 8G 8G Morningglory 0 0 0 3C,3H      0 0 0 0 0 0 0 3C,5H 0 0 0 0 0 9G 6G 8H Cocklebur 0 0 0 1C 0 0 0 0 -- 0      -- 2C 0 0 0 6G 2H 9H -- -- Nutsedge 0 0 0 0 0 8G 0 0 0 0 0 2G 0 0 0 0 0      10E 9G 10E Crabgrass 0 0 0 0 0 1C 0 0 0 0 0 0 0 0 0 0 0 8G 6G 7G      Barnyardgrass 0 0 0 5G 0 3C,8H 0 2C 0 0 0 3C,7G 0 0 0 2H 0 9H 8H 3C,8H      Wild Oats 0 0 0 0 0 1C 0 0 0 0 0 0 0 0 0 2C,5G 0 7G 3G 4C,8G Wheat 0 0 0      0 0 5G 0 0 0 0 0 2G 0 8G 0 3C,9H 0 9H 9G 4C,9H Corn 0 0 0 3C,5G 0 3C,4G      1C 0 0 0 0 3C,6G 1C 1C,1H 0 0 0 3G 0 0 Soybean 3C,4H 0 0 3C,5G 0 2C,2H 0      0 0 0 0 3C,2H 2C 0 0 0 0 9H 8H 9H Rice 2C,5G 0 0 4C,9H 0 9H 0 2C 0 0 0      3C,9H 2C,3G 7H 0 10H 0 10E 9H 9H Sorghum 3C,9H 0 0 4C,9H 3C,7G 3C,9H      3C,5G 3C,3G 0 3C,6G 0 3C,9H 3C,8H 3C,4C 0 9H 0 10H 9H 10H Cheatgrass 0 0      0 0 0 2C,8G 0 0 0 0 0 0 0 0 0 0 0 8G 6G 9H Sugar beet 7H 0 0 4C 6H 9G 2H      4H 0 3G 4G 5H 3H 5G 0 5G 1H 9C 3C,7G 9G Velvetleaf 0 0 0 2C 0 0 0 0 0 0      0 2C 0 0 0 0 0 5C,9G 4C,6H 4C,8H Giant Foxtail 0 0 0 3G 0 4C,9H 0 0 0 0      0 4C,8G 0 0 0 5G 0 6G 2G 6G Barley 2G 0 0 2C 0 2C 0 2C 0 0 0 2G 0 7H 0      4C,9G 0 9G 8G 9G        CMPD          CMPD 153 CMPD 154 CMPD 155 CMPD 156 CMPD 157 CMPD 158      CMPD 159 CMPD 160 CMPD 161 CMPD 162 163 Rate kg/ha 0.01 0.05 0.01 0.05      0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05      0.01 0.05        POSTEMERGENCE                      Cotton 10C 10C 3C,8H 10C 9C 2G 2H      2G 0 10C 10C 10C 4C,9G 3C,7H 1C 9C 3C,8G 6G 0 9C Morningglory 9C 4C,9H      2C,6G 10C 10C 4C,9G 3C,7H 2C,5G 0 9C 10C 9C 9C 4C,8H 1H 10C 9C 1C 0 10C      Cocklebur 10C 9C 4C,9H 10C 10C 7H 2H 3C,8H 2C,3H 10C 10C 10C 10C 1H 1H      10C 10C 7H 0 9C Nutsedge 9G 9G 2C,9G 9G 9G 0 0 0 0 9C 2C,9G 3C,8G 2C,9G      4G 0 2C,9G 9G 0 0 5C,9G Crabgrass 3G 5G 3G 3C,6G 5G 3C,6G 2C,4G 5G 0 1H      0 4G 0 4G 0 5G 0 0 0 4C,9G Barnyardgrass 4C,8H 4C,8H 3C,7H 3C,7H 3C,8H      6C,9H 3C,8H 3C,4G 2C,3H 9C 4C,9H 3C,8H 9C 4C,9H 3C,7H 9C 4C,9H 3C,5H 0      9C Wild Oats 2C,3G 3C,8G 2C,5G 3C,5G 0 9C 4C,9G 2C,5G 0 3C,6G 2C,2H      3C,8G 2C,5G 2C,9G 4C,9G 4G 0 0 0 6C,9G Wheat 8G 8G 4G 7G 3G 3C,9G 9G 7G      4G 9G 5G 9G 2C,9G 7G 3G 5G 0 0 0 9C Corn 0 2G 2G 0 0 0 0 0 0 5G 2G 3C,8H      3G 2C,5H 0 2G 0 0 0 1H Soybean 9C 4C,9G 4C,9G 4C,9G 3C,9G 8G 3C,7G 3C,8G      2C,3H 9C 5C,9G 9C 4C,9G 3C,6G 2H 9C 9C 3H 0 4C,9G Rice 6C,9H 5C,9G 5C,9G      4C,9G 2C,8G 6C,9G 4C,9G 6G 4G 9G 3C,8G 2C,8G 4G 4C,9G 4G 2C,9G 7G 2G 0      5C,9G Sorghum 6C,9G 4C,9G 5C,9H 5C,9G 5C,9H 5C,9G 3C,8H 3C,6G 2C,4G      2C,9G 5C,9G 4C,9G 4C,9G 3C,9H 2C,5G 9C 5C,9G 7G 0 10C Cheatgrass 7G 8G      3C,5G 2C,5G 2G 3C,8G 2C,7G 3C,4G 2G 5C,9G 3C,6G 9C 5C,9G 4C,9G 3C,8G      3C,9G 2C,8G 5G 0 5C,9G Sugar beet 6C,9G 9C 4C,9G 5C,9G 3C,7H 3C,7H 3C,7H      3C,3G 0 10C 9C 9C 5C,9G 3C,7H 4H 4C,9G 3C,7H 2C,5G 0 9C Velvetleaf 9C      4C,9H 3C,7H 4C,8H 3C,6H 2C,5G 3C,3G 2G 3G 10C 10C 10C 10C 2C,2G 0 10C      6C,9G 2C,5G 0 10C Giant Foxtail 5G 3C,7G 3G 3C,7G 2C,5G 4C,9G 3C,8G      2C,7G 3G 2C,8G 4G 4C,9G 7G 4C,9G 3C,6G 3C,9G 3C,8G 3C,6G 0 9C Barley 5G      7G 5G 8G 5G 7G 4C,9G 4C,9G 5G 9G 3C,4G 2C,9G 3G 4C,9G 2C,5G 3C,9G 2C,5G      2C,5G 0 3C,9G PREEMERGENCE                      Cotton 3G 2G 4G 3C,7G 1C      0 0 0 0 5C,9G 4C,8G 8G 2C,4G 0 0 8G 2C,3G 2G 0 3C,8H Morningglory 7H 7H      0 4C,8H 5H 2C 1H 0 0 7H 6H 9H 5H 2C,3G 0 9G 3C,8H 5G 0 8H Cocklebur --      8H 8H 3C,8H 3C,5H 3H 3H 0 0 -- -- 9H 3C,3H 2H 0 3C,8H 3C,3H 2C,4G 0 0      Nutsedge 9G 3C,8G 0 10E 9G 0 0 0 0 9G 9G 10E 5G 0 0 7G 3C,8G 0 0 10E      Crabgrass 2G 3G 0 7G 3G 3G 0 3G 0 0 0 4G 0 0 0 5G 0 0 0 4C,8G Barnyardgra      ss 0 3C,7H 0 6H 3G 4G 0 2G 0 8G 6C 3C,8H 0 2C 0 4C,9H 4C,9H 3G 0 3C,8H      Wild Oats 2C,3G 2C,3G 0 0 0 3C,6G 3G 0 0 2C,3G 2G 4C,8H 2C,4G 6G 0 0 2G      0 0 3C,9H Wheat 8G 2C,6G 0 8G 0 2C,8H 5G 0 0 2C,8G 6G 4C,9H 8H 4G 0 8G      2G 0 0 3C,9H Corn 0 0 0 0 0 0 0 0 0 3C,3G 0 3C,7H 2G 0 0 3C,7G 2C,5G 0 0      0 Soybean 3C,6H 3C,6H 2C,2H 3C,8H 3C,4H 1C,1H 0 0 0 3C,6H 5G 3C,7H 3C,3H      0 0 4C,8H 3C,6H 0 0 8H Rice 9H 9H 8G 10E 9H 9H 0 2G 0 5C,9H 8H 10E 7G      3C,6G 0 5C,9H 4C,9H 6G 0 10E Sorghum 9H 9H 3C,5G 9H 4C,9H 3C,9G 2C,5G 2G      0 5C,9H 9H 4C,9H 3C,7H 3C,6G 0 9H 4C,9H 3G 0 5C,9H Cheatgrass 3C,7G 7G 0      5G 0 4G 0 0 0 9G 6G 9H 8G 6G 0 3C,9G 8G 0 0 9H Sugar beet 3C,8H 4G 5G 7H      3H 5H 6G 0 0 9C 4C,9G 5C,9G 3C,8G 6H 0 9G 3C,7G 3G 0 5C,9G Velvetleaf      3C,4H 3C,5H 1C 3C,5H 3G 2H 1H 0 0 9G 8H 8H 3G 2H 0 3C,7G 2H 2G 0 8H      Giant Foxtail 0 5G 0 6G 2G 2C,5H 0 2H 0 7G 0 4C,8H 5G 2C,5G 0 4C,9G      3C,9H 2G 0 4C,9H Barley 6G 8G 2G 8G 4G 9G 2G 2G 0 9H 6G 3C,9G 2G 2C,8G 0      3C,9G 4G 0 0 9G

      CMPD          CMPD 163 CMPD 164 CMPD 165 CMPD 166 CMPD 167 CMPD 168      CMPD 169 CMPD 170 CMPD 171 CMPD 172 173 Rate kg/ha 0.01 0.05 0.01 0.05      0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05      0.01 0.05        POSTEMERGENCE Cotton 5C,9G 10C 10C 10C 10C 10C 9C 4C,9H 3C,8G 3C,6G 0      10C 3C,7H 9C 4C,9G 5C,9H 4C,9H 0 -- 3C,9G Morningglory 10C 10C 10C 10C      10C 10C 10C 4C,8H 4C,8H 4C,8H 3C,7H 9C 4C,8H 10C 9C 5C,9H 3C,6G 0 -- 0      Cocklebur 2G 10C 9H 9C 6H 10C 10C 5C,9H 1H 1H 0 1H 0 10C 10C 10C 4C,9H      2G -- 8G Nutsedge 5C,9G 5C,9G 4C,9G 9C 5C,9G 9C 2C,9G 5G 0 0 0 3G 0 10C      4C,9G 8G 3C,7G 3G -- 0 Crabgrass 3C,6G 3C,7H 2C,5G 6C,9G 2C,8G 3C,7G 3G      3C,7G 2C,5G 4G 0 4C,9H 2C,8G 4C,8G 2C,6G 2G 0 0 -- 0 Barnyardgrass 9C 9C      9C 10C 9C 9C 9C 9C 4C,8G 10C 0 9C 9C 9C 9C 4G 2H 0 -- 2C,5H Wild Oats      5C,9G 9C 3C,8G 5C,9G 4C,9G 4C,9G 2C,6G 3C,6G 2C 3G 0 5C,9G 5C,9G 5C,9G      3C,8G 2C,5G 0 0 -- 0 Wheat 9G 9C 3C,9G 9C 4C,9G 2C,9G 6G 4C,9G 2G 3G 0      9G 9G 9G 6G 4G 0 0 -- 5G Corn 0 3C,7H 1H 3H,7G 3G 0 0 2C,4H 2H 10C 5H      2C,8H 3H 3C,7H 0 0 0 0 -- 0 Soybean 6C,9G 9C 9C 9C 9C 5C,9G 4C,9G 5C,9G      4C,9G 5C,9G 2C,7G 3C,8H 5H 9C 9C 3C,9G 4C,8G 0 -- 0 Rice 9C 9C 9C 9C 9C      9C 9C 9C 3C,6G 4C,9G 3G 9C 9C 9C 4C,9G 4C,9G 2C,6G 0 -- 0 Sorghum 9C 10C      9C 10C 9C 9C 9C 9C 4C,9H 4C,9G 2C,3G 9C 4C,9G 9C 9C 4C,9H 3C,8G 0 -- 3G      Cheatgrass 2C,9G 9C 4C,9G 9C 4C,9G 3C,9G 6G 2C,8G 2C,5G 4G 0 4C,9G 9G 9C      3C,9G 2C,8G 8G 0 -- 3G Sugar Beets 9C 9C 9C 10C 10C 9C 10C 10C 9C 9C      2C,5G 9C 3C,7H 10C 5C,9G 9C 5C,9H 3G -- 3H Velvetleaf 10C 10C 10C 10C      10C 10C 10C 5C,8H 3C,5H 2C,4G 0 9C 4C,8H 10C 10C 5C,9H 4C,8H 0 -- 3G      Giant Foxtail 9C 9C 9C 9C 6C,9G 9C 9C 9C 4C,8H 9C 0 9C 9C 9C 4C,9G 5G 2H      0 -- 2C,6G Barley 9G 4C,9G 3C,8G 3C,9G 9G 9G 7G 2G 0 0 0 9C 4C,9G 3C,8G      7G 2C,4G 0 0 -- 0 PREEMERGENCE Cotton 2G 4C,9G 2C,5G 5C,9G 9G 2C,8H 5G      3G 0 0 0 3G 0 4C,8H 3C,8G 2C,6G 0 0 -- 2G Morningglory 5H 9C 3C,9H 9C 9C      9G 3C,8H 2H 1H 0 0 8H 0 9H 8H 8H 3C,3H 0 -- 0 Cocklebur 0 5G 0 6G 3G 7H      3H 2G 1H 0 0 0 0 9H 8H -- 2C,2H 0 -- 3G Nutsedge 8G 9G 10E 10E 10E 10E      10E 0 0 0 0 0 0 10E 8G 0 0 0 -- 0 Crabgrass 2C,8G 4C,7G 3C,6G 4C,9G      3C,6G 2C,6G 3C,6G 0 0 0 0 4C,8G 0 3C,7G 0 0 0 0 -- 0 Barnyardgrass 2C,4G      9H 4C,8H 9H 9H 9H 3C,9H 2C,6G 3G 0 0 4C,9H 3G 9H 6H 3G 0 0 -- 0 Wild      Oats 2C,3G 4C,9H 2C 4C,8G 2C,6G 2C,8G 1C 0 0 0 0 2C,8H 2G 3C,9G 3G 1C 0      0 -- 0 Wheat 8G 4C,9H 2C,8H 4C,9H 2C,8H 9H 7H 7G 0 0 0 9H 4G 3C,9G 5G 0      0 0 -- 0 Corn 0 3C,9H 0 4C,9H 4G 2G 0 6H 0 2C,3G 0 4C,9H 0 3C,8H 2G      1C,2G 0 0 -- 0 Soybean 7H 9H 7H 9H 9H 9H 3C,8H 2C,6H 2C,2H 2G 0 3G 0 9H      8H 2C,6G 0 0 -- 0 Rice 9H 10E 9H 10E 10E 10E 10E 8H 2C,5G 0 0 10E 9H      5C,9H 2C,8G 4G 2G 0 -- 2G Sorghum 9H 10E 5C,9H 10H 4C,9H 10E 10E 4C,9H      2C,4G 2C,5G 0 10H 9H 5C,9H 9H 3C,9G 3G 0 -- 4G Cheatgrass 8G 9H 9H 9H 9H      9G 7G 3G 0 0 0 9H 0 5C,9G 8G 5G 0 0 -- 0 Sugar Beets 8G 5C,9G 8H 5C,9G      9G 4C,9G 9G 6G 0 0 0 0 0 5C,9G 4C,9G 5C,9G 5G 0 -- 7G Velvetleaf 3C,5H      5C,9H 2C,5H 5C,9G 2C,8H 5C,9G 3G 0 0 0 0 2G 0 5C,9G 5G 3C,7H 2C,2G 0 --      0 Giant Foxtail 2C,5G 4C,9H 3C,8H 9H 4C,9H 9H 2C,6G 2C,5G 0 0 0 9H 3C,8G      5C,9H 4C,8H 3G 0 0 -- 2G Barley 2C,7G 3C,9G 4G 9G 9G 9G 2C,8G 7G 0 0 0      2C,9H 2C 3C,9G 8G 5G 0 0 -- 5G        CMPD          CMPD 173 CMPD 174 CMPD 175 CMPD 176 CMPD 177 CMPD 178      CMPD 179 CMPD 180 CMPD 181 CMPD 182 183 Rate kg/ha 0.01 0.05 0.01 0.05      0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05      0.01 0.05        POSTEMERGENCE Cotton 10C 5C,9G 3G 9C 4C,9G 9C 10C 9C 10C 9C 4C,9H 10C      4C,9H 10C 4C,8H 10C 9C 10C 10C 10C Morningglory 0 3C,8H 2C,4H 5C,9G      4C,8H 10C 9C 10C 5C,9G 10C 2C,7G 10C 5C,9G 3C,8H 6C,9G 10C 10C 10C 10C      10C Cocklebur 2C,6G 4C,9G 2G 10C 4C,8H 10C 10C 10C 10C 10C 9C 10C 10C 9C      5C,9H 10C 10C 10C 10C 10C Nutsedge 0 0 0 2C,8G 0 9G 9G 9G 3C,9G 8G 2C,4G      9C 3C,9G 5C,9G 2C,9G 9C 6C,8G 10C 9C 9C Crabgrass 0 0 0 3G 0 3C,8G 5G      3C,7G 2G 3G 0 5G 0 6G 4G 2C,7G 4G 2C,9G 5G 2C,4G Barnyardgrass 0 7H 3G      9H 5G 9C 4C,9H 5C,9H 3C,9H 9H 3C,7H 4C,9H 3C,7H 10C 3C,7H 9C 4C,9G 10C      10C 9C Wild Oats 0 0 0 3C,8G 5G 4C,9G 9G 5C,9G 3C,7G 4C,9G 4C,9G 3C,5G      2C,3G 3C,8G 2C,7G 2C,8G 7G 2C,6G 2G 2C,8G Wheat 0 0 0 3G 0 9G 9G 9G 9G      9G 9G 9G 5G 2C,9G 9G 9G 8G 3C,9G 7G 2C,9G Corn 0 2G 0 0 0 2H 0 1H 0 0 0      1H 0 4U,8G 2C,7G 6U,9G 3U,8G 10C 6U,9G 6U,9G Soybean 0 4C,9G 7H 5C,9G      4C,9G 9C 9C 9C 5C,9G 5C,9G 4C,9G 3C,8H 2C,5H 5C,9G 5C,8H 6C,9G 6C,9G      6C,9G 9C 4C,8H Rice 0 7G 0 9G 4G 9C 9C 9C 5C,9G 4C,9G 4C,9G 4C,9G 4C,9G      5C,9G 6C,8G 3C,7G 3G 5C,8G 2C,8G 3C,8G Sorghum 0 2G 0 3C,9G 3C,7G 5C,9G      4C,9G 5C,9G 3C,9G 3C,9G 3C,8G 3C,9G 4C,9H 10C 4U,8G 6C,9G 3C,8G 6C,9G      5C,9G 6C,9G Cheatgrass 0 0 0 3G 0 6G 4G 8G 0 0 0 3G 0 5C,9G 4C,8G 10C 9C      10C 9C 9C Sugar Beets 2G 9C 4C,8H 9C 10C 10C 10C 10C 9C 10C 10C 10C 9C      9C 9C 10C 10C 10C 9C 6C,9G Velvetleaf 2C,3G 3C,7H 0 4C,9H 3C,6H 10C 10C      10C 6C,9G 10C 4C,9H 10C 4C,9G 9C 6C,9H 10C 10C 10C 10C 10C Giant Foxtail      0 2G 0 3C,6G 3G 4C,9G 3C,7G 4C,9G 3C,6G 2C,4G 3G 3C,7H 3C,6G 10C 3C,9G      9C 4C,9G 10C 6C,9G 3C,9G Barley 0 0 0 6G 0 3C,9G 9G 3C,9G 3C,9G 9G 7G 9G      5G 6C,9G 3C,8G 2C,8G 7G 8G 5G 8G PREEMERGENCE Cotton 0 3G 0 2G 0 2C,9G      8G 3C,6G 1C  2G 0 9G 2C,6G 2C,6G 0 3C,7G 3G 3C,9G 3C,8G 2C,8G Morningglor      y 0 5H 0 6H 1H 9H 4G 7G 0 2H 0 3C,8G 3C,7H 7H 3G 9G 6G 9H 9C 9H Cocklebur       0 2C,6H 0 2C,5G 0 9H 7H -- 3C,4G 2C,3H 0 9H 8H -- 3C 8H 2G 2C,9H -- 8H      Nutsedge 0 0 0 0 0 9G 5G 8G 3G 2C,5G 0 10E 10E 7G 0 9G 0 10E 9G 10E      Crabgrass 0 0 0 0 0 9G 0 2C 0 0 0 2G 0 0 2G 0 3G 2C,4G 6G 2C Barnyardgras      s 0 2H 0 0 0 9G 1H 3H 0 1C 0 8H 7H 0 0 3C,7G 0 9H 2C,7H 9H Wild Oats 0 0      0 0 0 3C,7G 2C,5G 3C,5G 0 3C,4G 0 2C,5G 0 2C,4G 0 2C,6G 0 2C,7G 3G 2C,4G      Wheat 0 0 0 0 0 9H 9H 9H 0 6G 0 8H 3G 2C,8H 4G 2C,8G 7G 2C,8H 7G 2C,8H      Corn 0 6G 0 0 0 5G 0 0 0 0 0 0 0 9H 0 2C,9H 3C,7H 9H 2C,9H 9H Soybean 0      2C,5G 0 3C,6H 1C,1H 9H 3C,6H 3C,7H 2C,4G 2C,5G 0 3C,7H 5G 2C,8H 5G 3C,8H      2C,4G 2C,8H 3C,8H 2C,7H Rice 0 8H 0 8G 2G 10E 10H 9H 1C 2C,3G 0 10E 9H      3C,9H 2C 2C,7G 0 3C,8H 2C,6G 2C,9H Sorghum 0 2G 0 2C,8H 2G 4C,9H 9H 9H      3C,5G 3C,7G 0 9H 9H 3C,9H 3C,6G 3C,7H 3C,7G 10H 2C,9H 10H Cheatgrass 0 0      0 0 0 5G 0 4G 0 0 0 0 0 2C,8H 2G 3C,9H 3G 9H 2C,9H 2C,9H Sugar Beets 5G      4G 0 7H 2G 9G 9G 9G 7G 4C,9G 3C,6H 9G 9G 4C,8G 3G 4C,9G 2C,8G 3C,9G      4C,9G 4C,8G Velvetleaf 0 2G 0 0 0 4C,9G 3H 6G 3C,3H 3C,3H 0 3C,7H 3C,3H      4C,7H 2H 4C,8H 7G 4C,9H 2C,8H 4C,8H Giant Foxtail 0 0 0 0 0 2C,5G 0 4G      1C 0 0 5G 3G 0 2G 3G 3G 2C,9H 3C,9H 2C,7G Barley 0 0 0 8G 0 9G 2C,6H      3C,9G 0 2C,8G 0 9G 4G 2C,9H 4G 2C,8G 2C,5G 8G 8G 8G        CMPD          CMPD 183 CMPD 184 CMPD 185 CMPD 186 CMPD 187 CMPD 188      CMPD 189 CMPD 190 CMPD 191 CMPD 192 193 Rate kg/ha 0.01 0.05 0.01 0.05      0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05      0.01 0.05        POSTEMERGENCE Cotton 4C,8H 4C,8H 3C,7H 3C,8H 2C,8H 2C,8H 3C,8H 2C,7H      2C,6H 9C 5C,9H 10C 5C,9G 3C,9H 8H 6H 0 1H 0 7H Morningglory 2C,8H 10C      5C,9H 5C,9G 4C,8H 4C,9G 3C,8H 4C,9H 4C,8H 10C 10C 10C 10C 4C,9G 3C,5G      3C,6H 0 8H 5G 4C,9H Cocklebur 3C,7H 2C,9H 7G 5C,9G 5C,9H 4C,9H 4C,8H      3C,8H 2C,7H 10C 10C 10C 10C 3C,8G 6H 3C,7H 0 7H 0 5G Nutsedge 9G 3G 2G      2C,8G 3G 6G 3C 2C,9G 2C,7G 9C 9C 10C 9C 9G 3C,9G 7G 0 0 0 0 Crabgrass 2G      6G 2G 2G 0 0 0 0 0 2G 0 5G 0 0 0 0 0 0 0 3C,5G Barnyardgrass 5C,8G 9C      5C,9G 10C 10C 10C 3C,8H 2C,7G 3G 9C 4C,9H 10C 4C,9H 3C,5G 1H 9H 3H 5C,9H      4H 9C Wild Oats 0 3C,9G 2C,8G 3C,9G 2C,5G 2C,7G 2C,8G 0 0 2C,4G 0 2G 0 0      0 0 0 0 0 4C,8G Wheat 3G 3C,9G 2C,8G 9G 2C,6G 9G 9G 0 0 2C,5G 0 8G 0 0 0      0 0 0 0 9G Corn 3C,7G 4U,9C 2U,9G 5U,9C 2U,9G 10C 4U,9C 3C,7G 3C,3G 9C      5C,9G 9C 4C,9G 2C,5G 1H 2C,9G 3C,8H 3C,9G 5H 4U,9G Soybean 2C,6H 5C,8H      4C,9H 4C,9H 4C,7H 4C,9H 3C,8H 2C,8G 7H 5C,9G 4C,9G 4C,9G 3C,9G 1H 0      3C,7H 0 3C,5H 1H 5C,9G Rice 3G 9C 9C 9C 4C,9G 9C 4C,9G 4G 0 7G 0 4C,9G      2G 0 0 6G 5G 5C,9G 7G 9C Sorghum 2C,8G 10C 5C,9G 9C 3C,9G 5C,9G 4C,9G      2C,8G 2C,6G 9C 3C,9G 5C,9G 9G 9G 3C,6G 3C,9H 4G 3C,8H 2G 9C Cheatgrass      3C,8G 5C,9G 3C,9G 5C,9G 5C,9G 9C 4C,9G 2C,8G 7G 9C 4C,8G 5C,9G 9C 7G 0      8G 2G 7G 0 5C,9G Sugar Beets 5C,9G 2C,7G 0 4C,9G 5C,9H 9H 5C,9G 9C 3C,7H      9C 10C 9C 10C 9C 3C,7G 7H 3G 3C,8H 4H 6G Velvetleaf 6C,9H 5C,9G 4C,8H      4C,9H 3C,8H 4C,8H 3C,5H 4C,8H 4C,7H 10C 10C 10C 9C 3C,8G 0 0 0 1C 0      4C,7H Giant Foxtail 2C,7G 9C 5C,9G 10C 5C,9G 9C 3C,9G 6G 2G 3C,8G 3G      4C,9G 6G 0 0 0 0 0 0 5C,9G Barley 2C,4G 4C,9G 3C,9G 4C,9G 2C,8G 3C,9G      2C,8G 2C,6G 3G 2G 0 7G 0 0 0 0 0 0 0 2G PREEMERGENCE Cotton 4G 1C,3G 0      1C,3G 2G 1C,4G 0 0 0 1C 0 9G 9G 2C,7H 3G 0 0 0 0 1C Morningglory 3C,8H      9G 2C,7G 2C,8H 2C,5G 3C,8H 2G 0 0 2C,2H 0 9G 8G 3H 0 2H 4H 0 0 3H      Cocklebur 4C,8G 8G 0 3C,7G -- 8H 0 0 0 2C,5G 1C 9H 9H 2C 0 0 0 0 0 1C      Nutsedge 3C,8G 0 0 5G 0 0 0 0 0 0 0 10E 9G 5G 0 0 0 0 0 0 Crabgrass 0 2C      0 0 0 0 0 0 0 0 0 3G 0 0 0 0 0 0 0 0 Barnyardgrass 7G 3C,9H 0 2C,4G 0      2C,4G 0 0 0 0 0 3C,9H 5G 7H 0 0 0 0 0 0 Wild Oats 0 2C,8G 2C 2C,4G 3G      2C,7G 3G 0 0 0 0 3C,4G 0 2G 0 0 0 0 0 2C,4G Wheat 4G 2C,9H 7G 2C,8H 6G      8H 5G 0 0 0 0 5G 0 0 0 0 0 0 0 3C,8G Corn 9H 9H 3C,8G 9H 2C,8G 9H 3C,9G      0 0 3C,4G 0 5C,9H 3C,7G 3C,6G 0 2C,6G 0 5G 0 3C,8H Soybean 3H 3C,7H      2C,5G 1C,6G 4G 2C,8H 1C,3G 2G 0 5G 2C,2H 9H 6H 3H 0 0 0 0 0 3C,8H Rice      3C,8H 10E 7G 10E 2C,7G 10H 2C,4G 2C 0 0 2G 8H 0 7G 0 0 0 5G 0 8G Sorghum      10H 9C 3C,9H 10C 3C,9H 10C 4C,9G 0 0 3C,7G 3C,3G 9G 9H 2C,8G 3C,5G 6G 0      3C,3G 0 9H Cheatgrass 9H 9H 2C,9H 9H 6G 9H 6G 0 0 7G 0 9H 7G 7G 0 0 0 0      0 6G Sugar Beets 4C,8H 5G 5G 5G 0 3C,7G 1C,3G 0 0 7H 2H 9H 9G 7H 0 0 0      2H 0 3H Velvetleaf 2C,4G 3C,7H 0 0 0 4G 0 4G 2H 2C 2G 4C,9G 3G 0 0 0 0 0      0 0 Giant Foxtail 2C 2C,8H 0 2C,5G 0 2C,5G 0 0 0 0 0 9G 0 2G 0 0 0 0 0 0      Barley 5G 9H 7G 9G 2C,8H 4C,9G 2C,8G 0 0 0 0 3C,9G 2G 0 0 0 0 0 0      7H       CMPD          CMPD 193 CMPD 194 CMPD 195 CMPD 196 CMPD 197 CMPD      198* CMPD 199 CMPD 200 CMPD 201 CMPD 202 203 Rate kg/ha 0.01 0.05 0.01      0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01 0.05 0.01      0.05 0.01 0.05        POSTEMERGENCE Cotton 3G 4C,8H 2C,4H 4G,9G 2C,9G 0 0 5H 0 0 0 0 0 3C,9G 3      C,8H 5C,9G 5C,9G 9C 10C 9C Morningglory 3C,7H 4C,9G 4C,8H 9C 3C,8H 1H 0      0 0 0 0 0 0 4C,9G 4C,9G 10C 10C 10C 10C 4C,9G Cocklebur 2G 4C,9H 3C,5G      5C,9G 4C,9H 2C,3G 0 0 0 0 0 0 0 5C,9G 4C,9G 10C 10C 10C 10C 5C,9G      Nutsedge 0 2G 0 8G 3C,5G 0 -- 0 0 0 0 0 0 0 0 3C,9G 3C,7G 9C 10C 2C,8G      Crabgrass 4G 0 0 0 3G 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 Barnyardgrass 3C,8H      3H 0 5H 3C,5H 0 0 0 0 0 0 0 0 2G 0 3C,9H 6H 3C,9H 6H 1C,2H Wild Oats      3C,6G 0 0 0 0 0 0 0 0 0 0 0 0 0 0 1C 0 0 0 0 Wheat 3C,7G 2G 0 0 0 0 0 0      0 0 0 0 0 0 0 2G 0 2G 0 0 Corn 3C,9G 9G 7H 1C 1C 0 0 0 0 0 0 0 0 2G 0      4C,9G 3C,9H 10C 4C,9G 2C,4G Soybean 4C,8G 8H 4H 4C,9G 3C,7H 0 0 0 0 0 0      0 0 3C,8G 3C,4H 4C,8G 3C,8H 5C,9G 4C,9G 3H Rice 9C 7G 4G 3G 2G 4G 0 0 0      0 0 0 0 0 0 3G 0 7G 2G 0 Sorghum 3C,9G 3C,8H 2G 4C,9G 4C,9H 0 0 0 0 0 0      0 0 3C,6G 3G 9G 4C,9G 4C,9G 4C,9G 3C,8G Cheatgrass 9G 5C,9G 5G 2C,8G 8G      0 0 0 0 0 0 0 0 6G 3G 4C,9G 7G 9C 9G 6G Sugar Beets 3H 4C,8G 2C,3G 9C      5C,8H 0 0 0 0 0 0 2G 0 9C 5C,9G 10C 10C 10C 9C 3C,9H Velvetleaf 6G 1C 0      3C,7H 3C,3G 0 0 0 0 0 0 0 0 9C 3C,8H 10C 10C 10C 10C 5C,9H Giant Foxtail      3C,7G 1H 0 0 1H 0 0 0 0 0 0 0 0 0 0 3G 0 3G 2G 1C Barley 0 2G 0 0 0 0 0      0 0 0 0 0 0 0 02C,2G 0 0 0 0 PREEMERGENCE Cotton 0 0 0 3C,5G 0 0 0 0 0 0 0       0 0 2G 0 3C,6G 0 3C,9G 7H 6G Morningglory 0 0 0 6H 0 0 0 0 0 0 0 0 0 0      0 3C,8G 2C 9G 7H 2C,2H Cocklebur -- 0 0 0 2C 0 0 0 0 0 0 0 0 0 0 3C,6H      2C,6H 8H 7H 2C,2H Nutsedge 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 9G 5G 10E 10E      7G Crabgrass 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 Barnyardgrass 0 0 0      1C 0 0 0 0 0 0 0 0 0 0 0 3C,7H 3C,2G 3C,8H 1H 1C Wild Oats 0 0 0 0 0 0 0      0 0 0 0 0 0 2G 0 2G 0 3G 0 0 Wheat 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 4G      0 0 Corn 0 0 0 0 0 0 0 0 0 0 0 0 0 0 04C,8G 3C,5G 3C,9G 3C,8G 2C,3G      Soybean 2G 0 0 3C,5G 1C 0 0 0 0 0 0 0 0 0 0 2C,3H 1C,2H 4C,8H 3H 1C Rice      0 0 0 2C,4G 0 0 0 0 0 0 0 0 0 0 0 5G 0 8G 2G 2G Sorghum 3C,3G 0 0 3C,7G      3G 0 0 0 0 0 0 0 0 2C,3G 0 4C,9H 3C,6G 3C,9H 3C,8H 2C,6G Cheatgrass 0 0      0 7G 3G 0 0 0 0 0 0 0 0 5G 0 8G 3C,5G 9G 6G 3G Sugar Beets 2H 0 0 4C,8G      5G 0 0 0 0 0 0 0 0 3C,8G 0 5C,9G 3C,8G 5C,9G 8G 3C,8G Velvetleaf 0 0 0      2C 0 0 0 0 0 0 0 0 0 0 0 3C,5H 3C 3C,8G 3C,3G 2G Giant Foxtail 0 0 0 0 0      0 0 0 0 0 0 0 0 0 0 2G 0 2G 0 0 Barley 0 0 0 0 0 0 0 0 0 0 0 0 0 0 0 2G      0 2C,4G 0 2G        CMPD 203 CMPD 204 CMPD 205 CMPD 206 Rate kg/ha 0.01 0.05 0.01 0.05      0.01 0.05 0.01        POSTEMERGENCE Cotton 9H 3C,8G 3C,5G 4C,9H 3C,9H 9C 4C,9H Morningglory      3C,8H 5C,9G 3C,8G 4C,9G 3C,8H 10C 9C Cocklebur3C,8G 5C,9G 3C,8H 4C,9H      3C,8H 10C 4C,9G Nutsedge 8G 0 0 5G 0 Purple nutsedge      2C,8G --      Crabgrass 0 0 0 2G 0 Large crabgrass      2C,8G 4G Barnyardgrass 0 2C,8H      5H 3C,8H 2C,7H 4C,9G 3C,7H Wild Oats 0 2G 0 1C 0 4G 0 Wheat 0 0 0 0 0 5G      0 Corn 0 3G 0 0 0 4C,9G 3C,7H Soybean 1H 4C,9G 3C,8G 4C,9G 3C,5G 3C,4H      1C,1H Rice 0 6G 1C 9G 2C,4G Rice dry seeded      7G 3G Sorghum 2G 3C,7G      1C 3C,9H 3G 3C,7G 5G Cheatgrass 0 8G 5G 5C,9G 7G 0 0 Sugar Beets 4C,9G      4C,9G 9C 9C 3C,8H 10C 9C Velvetleaf3C,8H 4C,8H 3C,6H 3C,8H 3C,5H 10C      4C,8H Giant Foxtail 0 2C,5G 0 3C,4G 0 5C,9G 4C,9G Barley 0 0 0 0 0 0 0      PREEMERGENCE Cotton 0 1C 0 2G 0 9G 2C,4G Morningglory 0 0 0 3C,6H 0 7G      6H Cocklebur 0 0 0 2C 6G 3C,6H 6G Nutsedge 0 0 0 0 0 Purple nutsedge       7G -- Crabgrass 0 0 0 0 0 Large crabgrass      2C 0 Barnyardgrass 0 3G      0 3C,4G 0 5G 2G Wild Oats 0 0 0 0 0 0 0 Wheat 0 0 0 0 0 0 0 Corn 0 3C,5G      0 3C,7G 1C 3C,6G 2G Soybean 0 1C 0 2C,2H 1H 0 0 Rice 0 6G 0 9H 3G Rice      dry seeded      2C,7G 0 Sorghum 0 3C,9H 3C,3G 4C,9G 3C,3G 2C,3G 0      Cheatgrass0 4G 0 8H 0 0 0 Sugar Beets 3H 3C,8H 2H 4C,9G 3H 4C,9G 3C,7G      Velvetleaf 0 0 0 1C 0 3C,6H 3C,3H Giant Foxtail0 2G 0 0 0 2C,8G 3G      Barley 0 0 0 2C,2G 0 0 0      *It is noted that Compound 198 was inactive at the levels tested. However      it is believed that at higher levels, herbicidal activity would be      present.

Test B

Postemergence

Two round pans (25 cm diameter by 12.5 cm deep) were filled with Sassafras sandy loam soil. One pan was planted with blackgrass. (Alopecurus myosuroides), sugar beets, nutsedge (Cyperus rotundus) tubers, rape (Brassica napus), crabgrass (Digitaria sanquinalis), sicklepod (Cassia obtusifolia), teaweed (Sida spinosa), jimsonweed (Datura stramonium), velvetleaf (Abutilon theophrasti), and giant foxtail (Setaria faberil). The other pan was planted with wheat, barley, cotton, rice, corn, soybean, wild oats, (Avena fatua), cocklebur (Xanthium pensylvanicum), morningglory (Ipomoea hederacea), johnsongrass (Sorghum halepense) and barnyardgrass (Echinochloa crusgalli). The plants were grown for approximately fourteen days, then sprayed post-emergence with the chemicals dissolved in a non-phytotoxic solvent.

Preemergence

Two round pans (25 cm diameter by 12.5 cm deep) were filled with Sassafras sandy loam soil. One pan was planted with blackgrass, sugar beets, nutsedge, rape, crabgrass, sicklepod, teaweed, jimsonweed, velvetleaf, and giant foxtail. The other pan was planted with wheat, barley, cotton, rice, corn, soybeans, wild oats, cocklebur, morningglory, johnsongrass, and barnyardgrass. The two pans were sprayed preemergence with the chemicals dissolved in a non-phytotoxic solvent.

Treated plants and controls were maintained in the greenhouse for 28 days, then all treated plants were compared to controls and visually rated for plant response. Response ratings are based on a scale of 0 to 100 where 0=no effect, and 100=complete control. A dash (-) response means no test.

Response ratings are contained in Table B.

    TABLE B       Compound 2 Compound 3 Compound 4 Compound 5 Compound 8 POSTEMERGENCE      Rate g/ha 62 16 16 4 4 1 25 52 16 16 16 4 4 4 1 1 .25 .25 62 16 4 1 62      16 4 1 62 16        Corn 100 100 100 100 100 60 40 100 100 100 100 100 0 100 80 70 60 0      100 100 80 40 100 90 60 40 100 80 Wheat 100 100 100 60 100 40 0 100 100      30 70 40 0 20 0 0 0 0 100 100 40 0 70 40 0 0 30 0 Barley -- -- -- -- --      -- -- -- -- -- -- -- -- -- -- -- -- -- -- -- -- -- -- -- -- -- -- --      Rice 100 100 100 90 70 50 30 100 100 80 100 90 60 100 50 30 30 0 100 100      60 30 100 90 30 0 90 70 Soybean 100 100 100 100 90 90 60 100 100 100 100      100 90 90 80 70 80 0 100 100 100 60 90 90 60 40 100 80 Cotton 100 100 60      70 20 40 0 100 100 100 100 100 80 100 70 40 30 0 100 90 70 30 100 90 60      30 100 90 Sugar beet 100 100 100 100 100 100 100 100 100 100 100 100 100      100 100 100 100 0 100 100 100 100 100 100 100 90 100 100 Rape 100 100      100 100 100 100 100 100 100 100 100 100 100 100 100 100 100 0 100 100      100 100 100 100 100 100 100 100 Crabgrass 100 80 100 50 60 40 0 100 90      50 70 70 30 30 50 0 30 0 100 80 50 30 70 50 40 30 90 50 Johnsongrass 100      100 100 100 90 60 40 100 100 100 100 100 70 90 70 30 30 0 100 100 70 30      100 100 80 40 90 50 Blackgrass 100 100 100 100 90 50 30 100 100 100 100      100 60 100 80 30 70 0 100 100 60 30 100 100 60 30 100 90 Barnyardgrass      100 100 100 100 100 60 40 100 100 100 100 100 70 100 100 30 40 0 100 100      60 30 100 100 80 40 90 50 Nutsedge 100 100 100 100 80 90 80 100 100 100      100 100 100 100 100 100 100 0 100 90 50 30 100 100 80 70 100 70 Giant      Foxtail 100 100 100 90 90 50 30 100 100 80 60 60 30 30 30 0 0 0 100 90      60 30 100 80 30 0 90 50 Wild Oats 90 100 80 60 70 40 0 100 100 50 100 40      0 80 0 0 0 0 100 90 30 0 70 40 0 0 30 0 Cocklebur 100 100 90 70 60 30 0      100 100 90 100 100 70 90 60 60 30 0 100 90 50 30 100 100 60 30 100 90      Morningglory 100 100 90 100 70 90 60 100 100 100 100 100 100 100 100 80      70 0 100 100 80 50 100 90 80 60 100 90 Teaweed 100 100 90 70 30 40 0 100      100 60 90 80 30 60 50 0 30 0 100 80 60 40 90 70 50 30 100 90 Sicklepod      100 100 100 90 70 60 0 100 100 100 100 100 100 100 90 100 80 0 100 80 60      30 70 60 40 30 90 50 Jimsonweed 100 100 100 90 70 70 40 100 100 90 100      90 60 100 70 30 40 0 100 100 70 40 100 90 60 30 100 100 Velvetleaf 100      100 100 100 80 80 50 100 100 90 100 100 80 100 90 50 50 0 100 100 100 60      100 100 60 30 100 100        PREEMERGENCE Rate g/ha 250 62 62 16 16 4 1 250 62 62 16 16 16 4 4 1 1      250 62 16 4 250 62 16 4 250 62        Corn 100 100 100 80 90 20 0 100 100 100 70 70 100 20 40 0 0 100 100 90      60 100 100 90 30 100 90 Wheat 100 90 100 80 100 30 0 100 100 100 20 0 40      0 0 0 0 100 100 90 70 100 100 50 0 80 30 Barley -- -- -- -- -- -- -- --      -- -- -- -- -- -- -- -- -- -- -- -- -- -- -- -- -- -- -- Rice 100 100      100 100 100 90 70 100 100 100 100 100 100 100 100 90 0 100 100 100 100      100 100 100 100 100 100 Soybean 100 100 100 80 100 40 20 100 100 100 70      70 90 40 40 0 0 100 100 90 60 100 90 80 60 100 80 Cotton 100 80 100 80      80 30 0 100 100 100 70 70 100 30 0 0 0 100 90 60 30 100 80 50 30 100 60      Sugar beet 100 100 100 100 100 100 30 100 100 100 100 100 100 100 90 80      0 100 100 100 90 100 100 100 80 100 100 Rape 100 100 100 90 100 20 0 100      100 100 90 90 100 90 80 20 0 100 100 100 50 100 100 80 60 100 100      Crabgrass 100 100 100 90 90 30 0 100 90 100 60 30 80 30 0 0 0 100 90 50      30 90 70 50 30 80 70 Johnsongrass 100 100 100 100 100 90 30 100 100 100      90 70 100 80 30 50 0 100 100 100 70 100 100 100 100 100 90 Blackgrass      100 90 100 100 100 70 20 100 100 100 100 90 100 100 70 50 0 100 100 100      90 100 100 100 90 100 90 Barnyardgrass 100 100 100 90 100 80 20 100 100      100 80 50 100 30 0 0 0 100 100 100 60 100 100 90 70 100 90 Nutsedge 100      100 100 100 100 70 20 100 100 100 100 90 100 90 50 50 0 100 90 80 60 100      100 100 90 100 100 Giant Foxtail 100 100 100 90 100 80 50 100 100 100 80      30 100 50 0 0 0 100 100 100 60 100 100 90 60 100 90 Wild Oats 100 90 100      90 90 20 0 100 100 100 70 90 80 0 40 0 0 100 90 70 70 90 80 50 30 100 90      Cocklebur 100 90 100 80 90 20 0 100 100 100 50 80 80 50 40 20 0 100 100      80 50 100 90 70 50 100 80 Morningglory 100 50 100 40 70 0 0 100 100 100      40 80 100 30 40 0 0 100 90 50 30 100 80 70 30 100 60 Teaweed 100 100 100      80 90 50 20 100 100 100 80 70 90 70 30 0 0 100 90 70 30 90 70 50 30 100      90 Sicklepod 100 90 100 80 80 60 20 100 90 100 90 50 90 80 30 20 0 100      90 60 30 90 70 50 50 100 90 Jimsonweed 100 100 100 90 90 60 20 100 100      100 100 80 100 80 30 50 0 100 90 80 50 100 90 60 30 100 100 Velvetleaf      100 100 100 100 100 60 0 100 100 100 100 80 100 90 30 60 0 100 100 80 50      100 90 60 30 100 100        Com-        Com- pound 8 Compound 13 Compound 14 Compound 16 Compound      20 Compound 21 Compound 22 Compound 23 pound 24 POSTEMERGENCE Rate g/ha      4 1 62 16 4 1 16 4 1 .25 52 16 4 1 62 16 4 62 15 4 62 16 4 62 16 4 1      62    Corn 50 30 100 100 70 40 100 80 60 40 0 0 0 0 100 90 40 100 90 70      100 100 70 50 30 0 0 0 Wheat 0 0 30 0 0 0 30 0 0 0 0 0 0 0 90 60 20 0 0      0 70 20 0 40 0 0 0 30 Barley -- -- -- -- -- -- -- -- -- -- -- -- -- --      -- -- -- 0 0 0 0 0 0 -- -- -- -- -- Rice 0 0 90 30 0 0 60 30 0 0 60 0 0      0 95 90 85 80 20 0 90 50 20 70 40 0 0 30 Soybean 70 0 100 100 100 70 100      100 70 50 100 70 430 0 95 90 80 100 90 50 100 100 80 100 100 80 60 100      Cotton 60 40 100 100 90 50 100 70 50 30 90 70 50 30 100 100 90 60 0 0 80      70 20 100 100 70 40 100 Sugar beet 100 90 100 100 100 100 100 100 90 70      100 100 90 70 95 90 90 80 0 100 90 70 100 100 100 100 100 100 Rape 100      90 100 100 100 100 100 100 90 69 100 100 90 60 100 100 100 100 90 30 100      100 70 100 100 100 100 100 Crabgrass 30 0 90 60 50 30 30 0 0 0 30 0 0 0      60 30 20 40 0 0 60 30 0 60 40 30 0 30 Johnsongrass 0 0 100 90 60 30 100      80 60 30 90 70 30 0 100 100 85 100 70 20 100 100 70 100 100 80 60 100      Blackgrass 30 0 100 70 40 0 70 30 0 0 70 30 0 0 100 95 85 80 60 0 100 70      50 100 70 30 0 100 Barnyardgrass 0 0 100 90 60 30 100 80 50 30 90 50 0 0      100 95 80 100 70 30 100 100 50 100 100 80 60 80 Nutsedge 70 40 100 100      90 80 90 70 50 30 90 70 60 40 100 80 60 0 0 0 0 0 0 100 100 70 50 100      Giant Foxtail 0 0 100 80 30 0 70 30 0 0 0 0 0 0 90 85 60 100 60 20 100      100 50 70 50 30 0 70 Wild Oats 0 0 60 30 0 0 40 0 0 0 0 0 0 0 85 70 30 0      0 0 60 20 0 40 0 0 0 30 Cocklebur 50 30 100 70 50 30 100 90 60 30 90 80      50 30 100 95 85 60 0 0 100 60 20 100 100 100 100 100 Morningglory 60 30      100 100 100 50 90 70 50 30 90 80 60 30 100 100 90 50 0 50 70 60 20 100      80 60 30 100 Teaweed 30 30 100 90 60 40 90 50 30 0 70 30 30 0 90 95 90      40 20 0 70 50 20 90 70 50 30 70 Sicklepod 30 0 100 100 80 40 80 50 0 0      50 30 0 0 70 25 30 50 0 0 80 50 20 100 70 50 30 70 Jimsonweed 60 30 100      100 60 30 90 90 50 30 100 80 50 30 95 90 30 80 70 20 90 70 50 100 100 70      50 100 Velvetleaf 70 50 100 100 100 70 100 90 50 30 100 80 30 0 100 100      90 30 0 0 70 30 20 100 100 100 90 100 Green Foxtail                  70      20 0 100 80 50 Cheatgrass                  0 0 0 0 0 0 Wild Buckwheat                    100 80 0 80 80 50 Viola                  40 20 0 80 -- 20      Lambsquarter                  90 50 0 80 60 50        PREEMERGENCE Rate g/ha 16 4 250 62 16 4 62 16 4 1 250 62 16 4 250 62      16 250 62 16 250 62 16 250 62 16 4 250        Corn 30 0 100 90 90 20 90 70 50 30 80 50 30 0 100 95 90 90 60 20 90 80      0 70 50 30 0 30 Wheat 0 0 30 0 0 0 80 40 0 0 90 40 0 0 95 95 80 40 0 0      50 0 0 80 60 40 0 70 Barley -- -- -- --  -- -- -- -- -- -- -- -- -- --      -- -- -- 0 0 0 60 20 0 -- -- -- -- -- Rice 100 20 100 100 100 70 100 100      70 40 100 100 90 60 100 100 100 -- -- -- -- -- -- 100 100 80 50 90      Soybean 40 0 100 100 90 70 100 90 70 60 100 80 60 30 95 95 85 80 80 30      90 80 30 100 80 60 40 90 Cotton 20 0 100 80 80 20 80 70 50 30 90 70 50      30 95 90 80 90 20 0 90 80 200 90 70 40 0 70 Sugar beet 100 50 100 100      100 90 100 100 100 80 100 100 100 100 100 95 90 90 70 50 80 70 80 100      100 100 80 100 Rape 90 40 100 100 90 90 100 100 60 60 100 90 60 0 100 95      80 80 60 0 90 80 70 100 90 70 50 100 Crabgrass 40 20 90 70 50 0 90 70 50      30 90 70 50 40 90 30 10 90 0 0 70 70 20 90 70 50 30 90 Johnsongrass 60      20 100 100 100 60 100 80 50 30 100 80 50 30 95 95 90 100 80 0 100 90 80      100 90 80 60 90 Blackgrass 70 30 100 90 80 50 100 90 60 30 100 90 60 30      100 95 80 100 50 0 90 70 70 100 100 80 50 90 Barnyardgrass 20 0 100 100      90 60 100 70 50 0 100 80 40 0 100 95 80 100 50 0 100 90 50 100 80 60 40      90 Nutsedge 80 60 100 100 100 90 100 100 90 80 100 100 100 90 100 100      100 0 0 0 0 0 0 100 100 80 60 100 Giant Foxtail -- 0 100 90 70 50 100 60      40 0 80 60 30 0 100 95 90 90 70 0 100 90 70 100 100 90 70 100 Wild Oats      80 0 -- -- -- -- 80 40 0 0 90 40 0 0 90 85 65 60 20 0 50 50 20 70 50 30      0 70 Cocklebur 20 0 100 70 80 20 100 90 70 50 100 80 70 30 95 90 90 30      20 0 -- 30 0 90 80 70 50 90 Morningglory 20 0 100 90 80 30 90 70 50 30      100 80 50 30 95 90 80 70 20 0 80 60 20 70 50 30 0 80 Teaweed 90 20 100      90 90 20 90 80 50 30 90 80 50 30 90 80 50 80 30 0 70 30 0 90 70 50 -- 90      Sicklepod 30 0 100 100 80 20 90 70 50 30 90 70 50 30 90 50 10 50 0 0 70      30 0 90 70 40 0 90 Jimsonweed 80 30 100 100 90 50 90 70 50 30 90 70 50      30 100 90 60 60 0 0 70 30 0 100 80 60 40 90 Velvetleaf 60 20 100 100 90      80 90 70 50 30 90 70 50 30 100 95 70 30 0 0 60 30 0 100 80 60 40 90      Green Foxtail                  90 90 30 100 90 50 Cheatgrass           50 0 0 60 0 0 Wild Buckwheat                  100 50 50 90 60 20      Viola                  100 -- 20 90 50 30 Lambsquarter      90 70 0 90 60 0

      Compound 24 compound 27 compound 28 compound 31 Compound 32 Compound 33 C      ompound 34 Compound 35 Rate g/ha 16 4 1 250 62 16 4 250 62 16 62 16 4 1      62 16 4 1 62 16 4 62 16 14 1 62 116        Corn 0 0 0 0 0 0 0 0 0 0 100 70 50 30 80 40 0 0 80 40 30 70 30 0 0 30      0 Wheat 0 0 0 40 20 0 0 30 0 0 0 0 0 0 80 650 40 20 90 70 30 60 30 0 0      40 0 Barley -- -- -- -- -- -- --    -- -- -- -- -- -- -- -- -- -- -- --      -- -- -- -- -- Rice 0 0 0 90 70 50 30 50 30 0 70 30 0 0 100 70 50 30 80      70 30 90 70 50 30 100 70 Soybean 100 80 60 90 80 70 50 80 60 40 100 90      70 100 100 90 70 90 90 70 90 90 80 60 90 80 Cotton 90 70 40 100 90 609      30 100 70 30 80 60 30 0 100 100 100 80 90 90 50 90 80 50 30 100 80 Sugar      beet 100 100 90 100 100 100 100 100 100 100 100 100 60 30 100 100 70 50      100 100 80 100 100 70 50 100 100 Rape 100 100 100 100 100 100 100 100      100 100 100 100 100 100 100 100 100 100 100 100 100 100 100 100 100 100      100 Crabgrass 0 0 0 70 50 30 0 50 30 0 90 70 50 30 90 70 50 30 60 30 0      80 50 30 0 60 30 Johnsongrass 70 50 30 100 90 70 50 90 70 50 100 100 60      30 100 100 100 80 100 100 60 100 90 70 30 100 100 Blackgrass 100 70 40      90 60 30 0 100 90 70 100 100 60 30 100 100 90 70 90 70 30 100 70 30 0      100 80 Barnyardgrass 60 30 0 100 90 70 50 90 60 30 100 100 70 30 100 100      100 90 100 70 50 100 70 50 0 100 100 Nutsedge 90 70 50 100 100 70 50 70      50 30 30 0 0 0 100 100 100 90 100 60 50 90 70 50 30 90 70 Giant Foxtail      30 0 0 70 50 30 0 80 60 30 100 100 70 40 100 90 70 50 90 70 50 90 70 60      0 90 80 Wild Oats 0 0 0 60 40 20 0 30 0 0 70 40 20 0 80 60 40 20 80 40      30 70 50 30 0 50 0 Cocklebur 100 100 90 100 90 70 50 90 70 50 90 70 50      30 100 100 100 70 100 80 60 90 70 30 0 100 90 Morningglory 90 70 50 90      80 70 50 100 100 70 90 70 50 30 100 100 90 70 100 100 50 90 80 60 40 100      90 Teaweed 50 30 0 80 60 40 20 80 60 40 80 60 30 0 100 80 60 30 80 50 30      80 50 30 0 90 60 Sicklepod 50 30 0 80 60 30 0 50 30 0 80 60 30 0 100 100      90 80 90 50 30 90 50 30 0 90 40 Jimsonweed 70 50 30 100 70 50 30 100 80      60 100 80 60 40 100 90 80 70 90 80 60 100 80 70 50 100 80 Velvetleaf 100      70 50 100 100 80 50 100 80 50 100 80 60 40 100 100 100 90 100 100 90 100      100 80 50 100 100        tc,1 PREEMERGENCE Rate g/ha 62 16 4 250 62 16 4 250 62 16 4 250 62 16      4 250 62 16 4 250 62 16 250 62 16 4 250 62        Corn 0 0 0 0 0 0 0 0 0 0 0 90 60 0 0 90 80 70 40 40 0 0 60 0 0 0 30 0      Wheat 30 0 0 70 50 30 0 70 30 0 0 60 30 0 0 80 60 40 20 90 40 0 70 30 0      0 80 60 Barley -- -- -- -- -- -- -- 70 30 0 0 -- -- -- -- -- -- -- -- --      -- -- -- -- -- -- -- Rice 70 50 30 100 90 70 50 100 90 60 30 100 100 90      70 100 100 100 100 100 100 30 100 100 40 0 100 100 Soybean 70 50 30 70      50 30 0 90 60 30 0 90 70 50 30 100 80 60 40 90 60 30 90 50 0 0 90 80      Cotton 50 30 0 50 30 0 0 70 30 0 0 80 40 0 0 90 70 50 30 80 60 30 60 30      0 0 90 70 Sugar beet 100 90 80 100 90 70 50 90 70 50 30 100 90 70 50 100      100 90 70 100 80 40 100 90 70 50 100 100 Rape 90 70 50 90 70 50 30 90 70      50 30 90 70 50 20 100 90 70 50 90 70 50 90 70 40 0 100 90 Crabgrass 60      30 0 80 70 60 30 70 50 30 0 90 60 30 0 90 80 70 60 70 50 30 70 50 40 30      80 60 Johnsongrass 80 70 50 90 80 70 40 100 90 70 50 100 80 60 40 100      100 90 70 100 90 70 90 70 40 0 100 100 Blackgrass 80 70 40 90 70 50 30      90 70 50 30 100 90 70 50 90 80 70 50 90 70 30 100 80 40 0 100 100      Barnyardgrass 80 60 30 90 6030 0 90 70 50 30 90 80 60 30 100 90 70 40      100 70 30 90 40 0 0 100 90 Nutsedge 80 60 40 90 70 50 30 100 70 50 30 80      60 40 20 100 90 80 70 90 70 50 90 70 50 30 100 100 Giant Foxtail 90 70      40 90 60 40 0 90 70 50 30 100 80 50 30 100 100 80 50 100 80 50 90 50 0 0      100 90 Wild Oats 40 30 0 80 60 30 0 30 0 0 0 60 30 0 0 90 70 50 30 80 30      0 70 30 0 0 80 60 Cocklebur 70 50 30 80 60 40 0 90 70 50 30 90 70 50 30      90 70 50 30 90 60 30 90 50 30 0 90 80 Morningglory 60 40 20 30 0 0 0 90      60 30 0 80 60 40 20 100 90 60 30 90 60 30 80 50 30 0 90 80 Teaweed 70 50      30 90 70 50 30     70 50 30 0 100 80 60 40 60 30 0 80 50 30 0 90 70      Sicklepod 70 40 0 90 70 40 0 40 0 0 0 80 60 40 0 100 80 40 0 90 60 30 70      30 0 0 50 30 Jimsonweed 70 50 30 90 70 50 30 90 70 50 30 90 70 50 30 90      80 70 50 90 70 50 90 70 50 30 100 80 Velvetleaf 70 50 30 90 70 50 30 90      70 50 30 90 70 50 30 90 80 70 50 80 60 40 80 70 50 30 90 80 Green      Foxtail        90 70 50 30 Cheatgrass        60 30 0 0 Wild Buckwheat          90 70 50 30 Viola        90 70 50 30 Lambsquarter        100 70 50      30  Com-        pound 35 Compound 36 Compound 39 Compound 40 Compound 41 C      ompound 53 Compound 54 Compound 55 Rate g/ha 4 1 62 16 4 1 62 16 4 1 62      16 4 1 62 16 4 1 62 16 4 1 62 16 4 1 62 16        Corn 0 0 70 30 0 0 100 80 70 20 80 20 0 0 90 80 0 0 0 0 0 0 0 0 0 0 0      0 Wheat 0 0 80 50 30 0 100 100 80 50 90 80 20 0 80 70 20 0 60 30 0 0 80      60 30 0 0 70 Barley -- -- -- -- -- -- 100 80 40 0 20 0 0 0 90 80 50 0 60      30 0 0 60 30 0 0 70 40 Rice 30 0 90 70 50 30 100 100 80 30 90 60 30 0      100 100 70 20 90 60 30 0 90 60 30 0 90 60 Soybean 60 50 100 80 60 40 100      100 90 70 100 80 80 50 100 90 80 60 100 90 80 70 100 90 70 50 90 80      Cotton 40 0 90 70 40 0 780 30 30 0 70 60 30 0 100 70 50  90 60 20 0 90      70 20 0 90 60 Sugar beet 100 70 100 100 100 70 100 90 40 20 70 50 0 0      100 100 60 20 100 100 100 90 100 100 90 70 100 100 Rape 100 100 0 0 0 0      100 100 100 80 100 100 70 50 100 100 90 50 100 100 100 100 100 100 100      90 100 100 Crabgrass 0 0 90 60 30 0 90 50 20 0 40 0 0 0 60 30 0 0 70 50      30 0 60 30 0 0 80 60 Johnsongrass 70 40 100 90 60 30 100 100 70 50 80 50      20 0 90 100 80 20 100 90 70 50 100 90 70 50 100 90 Blackgrass 30 0 100      100 70 30 90 100 70 60 80 50 20 0 100 90 60 0 100 90 60 30 100 90 70 50      100 90 Barnyardgrass 70 30 100 90 70 30 100 100 90 60 90 60 20 0 100 100      80 20 100 100 90 60 100 90 70 50 100 100 Nutsedge 50 30 0 0 0 0 70 80 30      0 50 0 0 0 30 -- -- 0 -- -- -- -- -- -- -- -- -- -- Giant Foxtail 50 30      90 70 50 30 90 40 20 0 60 30 0 0 100 80 40 0 100 90 70 50 90 70 50 30 90      80 Wild Oats 0 0 90 60 30 0 100 100 90 40 100 40 0 0 90 90 30 0 30 0 0 0      30 0 0 0 70 30 Cocklebur 50 30 30 0 0 0 100 100 100 30 100 90 80 0 100      70 20 0 100 90 70 50 100 90 70 50 100 90 Morningglory 50 30 100 90 70 50      100 100 90 30 100 100 70 30 100 100 80 60 100 100 90 60 100 70 50 30 100      80 Teaweed 30 0 70 50 30 0 90 50 20 0 60 50 30 0 80 60 40 0 90 70 50 30      90 70 50 30 90 70 Sicklepod 0 0 90 60 30 0 100 100 50 0 100 30 30 20 100      90 70 0 100 100 70 50 100 70 50 30 100 70 Jimsonweed 50 30 80 60 40 0      100 100 70 50 90 70 50 0 100 90 80 20 100 90 70 50 100 90 70 50 90 80      Velvetleaf 70 30 80 60 40 0 100 90 60 20 100 80 60 0 100 90 60 20 100      100 80 60 100 90 70 50 100 90 Green Foxtail       100 70 50 0 60 30 20 0      100 80 60 0 90 70 50 30 90 70 50 30 90 70 Cheatgrass       100 100 60 50      80 70 50 0 40 20 0 0 100 90 70 50 100 70 50 30 100 90 Wild Buckwheat        100 90 70 0 70 0 0 0 100 100 80 0 100 90 70 50 90 70 50 30 100 90      Viola       70 80 80 30 80 -- -- -- 90 70 30 30 100 90 70 50 90 70 50 30      100 90 Lambsquarter       100 90 50 20 90 70 20 0 100 100 80 50 100 90      70 50 100 90 70 50 100 90        PREEMERGENCE Rate g/ha 16 4 250 62 16 4 250 62 16 4 250 62 16 4 250 62 1      6 4 250 62 16 4 250 62 16 4 250 62        Corn 0 0 70 30 0 0 100 80 70 20 80 20 0 0 90 80 0 0 0 0 0 0 0 0 0 0 0      0 Wheat 30 0 60 30 0 0 90 70 60 0 80 60 0 0 90 70 40 20 70 40 20 0 80 50      30 0 80 40 Barley -- -- -- -- -- -- 90 80 20 0 0 0 0 0 90 90 50 0 60 40      20 0 50 30 0 0 80 30 Rice 100 70 100 100 100 90 100 100 90 60 100 80 50      0 100 100 90 80 90 80 70 30 90 70 50 30 100 70 Soybean 70 30 80 40 0 0      100 100 60 60 100 50 30 0 90 80 40 0 90 80 60 30 80 60 30 0 90 70 Cotton      50 30 40 0 0 0 80 70 20 0 30 0 0 0 90 70 40 0 60 50 30 0 80 40 0 0 90 60      Sugar beet 90 70 100 90 70 50 100 100 60 20 90 80 60 0 100 90 70 50 100      90 80 70 100 90 80 70 100 90 Rape 60 30 80 60 40 0 100 100 90 20 100 90      40 0 100 100 80 50 100 90 70 50 90 80 70 50 90 80 Crabgrass 50 30 100 70      50 30 100 90 70 20 100 80 20 0 90 50 30 0 90 70 50 30 70 50 30 0 70 50      Johnsongrass 90 70 100 90 70 40 100 100 90 80 100 100 90 80 100 70 50 30      90 80 70 30 90 70 50 30 90 80 Blackgrass 90 50 100 100 80 60 100 90 90      50 100 90 70 50 90 90 50 30 100 70 50 30 90 80 70 50 100 100 Barnyardgras      s 80 50 100 80 40 0 100 90 70 30 10 90 80 0 90 70 40 0 90 80 70 30 90 80      70 40 90 80 Nutsedge 70 50 70 50 30 0 100 -- -- -- -- -- 0 -- 90 70 50      30 90 80 70 50 100 90 70 50 90 80 Giant Foxtail 80 50 100 90 70 40 100      90 70 30 100 90 70 0 90 80 50 30 90 80 70 30 90 80 70 40 90 80 Wild Oats      30 0 70 40 0 0 90 90 60 20 90 30 0 0 70 60 30 0 40 20 0 0 40 0 0 0 50 30      Cocklebur 50 40 -- 0 0 0 100 80 70 0 90 -- -- -- 40 0 0 0 90 70 50 30 90      70 50 30 100 70 Morningglory 60 30 80 60 30 0 100 90 40 0 90 70 20 0 90      80 70 50 90 80 70 60 90 80 70 50 100 90 Teaweed 40 0 90 70 50 20 100 90      60 30 90 90 50 0 90 70 50 30 90 70 50 30 90 70 50 30 90 70 Sicklepod 0 0      90 70 50 30 100 80 30 0 80 0 0 0 50 30 0 0 90 80 70 60 90 70 50 30 90 70      Jimsonweed 50 30 90 70 40 20 100 90 70 50 100 40 20 0 90 70 50 30 90 80      70 50 100 70 50 30 90 70 Velvetleaf 50 30 90 70 50 20 100 90 50 20 90 30      0 0 90 70 50 30 90 70 50 30 90 70 50 30 90 70 Green Foxtail       100 90      80 70 100 100 40 0 90 80 50 30 90 70 50 30 90 80 70 50 90 80 Cheatgrass           100 100 90 70 100 90 70 60 90 80 30 20 90 80 70 30 90 80 70 50 90      80 Wild Buckwheat       100 90 80 70 100 70 60 20 100 80 60 30 90 80 70      50 90 80 70 50 90 80 Viola       100 100 90 20 90 80 20 0 100 100 100 90      100 90 70 50 100 100 90 70 100 100 Lambsquarter       100 100 90 60 100      100 80 70 100 100 70 50 90 70 50 30 90 80 70 50 90 70        Compound 55  Compound 56 Compound 206 POSTEMERGENCE Rate g/ha 4 1 62      16 4 1 62 16 4 1        Corn 0 0 0 0 0 0 60 30 0 0 Wheat 30 0 40 20 0 09 30 0 0 0 Barley 0 0      20 0 0 0 0 0 0 0 Rice 30 0 80 60 30 0 Soybean 70 50 70 30 0 0 30 0 0 0      Cotton 0 0 40 0 0 0 80 70 60 30 Sugar beet 90 70 100 90 70 50 100 100 90      70 Rape 100 80 100 100 90 80 100 100 90 70 Crabgrass 40 20 50 30 0 0      Johnsongrass 70 50 90 70 50 30 50 30 0 0 Blackgrass 70 50 90 70 50 30 70      50 30 0 Barnyardgrass 70 50 90 70 50 30 100 60 30 0 Nutsedge -- -- -- --      -- -- Giant Foxtail 70 30 90 60 30 0 50 30 0 0 Green Foxtail 50 30 90 70      50 30 80 50 30 0 Cheatgrass 70 50 90 70 50 30 0 0 0 0 Wild Oats 0 0 0 0      0 0 0 0 0 0 Wild Buckwheat 80 60 90 70 50 30 70 50 30 0 Viola 70 50 --      70 50 30 Lambsquarter 70 50 90 70 50 30 100 90 70 50 Cocklebur 70 50 90      70 50 30 90 60 30 0 Morningglory 60 30 100 60 30 0 Teaweed 50 30 90 70      50 30 Sicklepod 50 30 70 50 30 0 70 50 30 0 Jimsonweed 60 30 90 70 50 30      100 70 50 30 Velvetleaf 70 40 100 70 50 30 100 100 90 70 Large crabgrass            50 30 0 0 Prikley sida       80 70 50 30 Rice dry seeded       70      50 30 0 Ivy morningglory       90 80 70 50 Purple nutsedge       70 30 0      0 Chickweed spp.       100 90 60 30        PREEMERGENCE Rate g/ha 16 4 250 62 16 4 250 62 16  4        Corn 0 0 0 0 0 0 100 30 0 0 Wheat 0 0 80 40 0 0 0 0 0 0 Barley 0 0 0 0      0 0 0 0 0 -- Rice 50 30 90 80 70 40 Soybean 30 0 80 60 30 0 0 0 0 0      Cotton 30 0 70 0 0 0 30 0 0 0 Sugar beet 80 70 100 90 80 70 90 70 50 --      Rape 70 40 100 90 80 70 90 90 60 -- Crabgrass 30 0 70 50 30 0 Johnsongras      s 70 50 100 90 80 60 80 50 30 0 Blackgrass 90 80 90 80 70 50 60 30 0 --      Barnyardgrass 70 40 100 80 70 50 70 30 0 0 Nutsedge 70 50 90 80 70 50      Giant Foxtail 60 30 90 80 70 40 80 70 50 30 Green Foxtail 70 50 90 80 70      50 100 50 30 0 Cheatgrass 70 40 90 80 70 50 0 0 0 -- Wild Oats 0 0 30 0      0 0 0 0 0 -- Wild Buckwheat 70 50 90 70 60 40 80 50 30 -- Viola 90 70      100 100 90 80 Lambsquarter 50 30 90 70 50 30 90 70 50 30 Cocklebur 50 30      100 70 50 30 40 20 0 0 Morningglory 60 30 90 70 50 30 Teaweed 50 30 90      70 50 30 Sicklepod 50 30 100 70 50 30 30 20 0 0 Jimsonweed 50 30 90 70      50 30 70 50 30 0 Velvetleaf 50 30 90 70 60 50 90 70 50 -- Large crabgrass             60 30 0 0 Prikley sida       70 50 30 20 Rice dry seeded       80      60 40 20 Ivy morningglory       80 50 30 0 Purple nutsedge       30 0 0      0 Chickweed spp.       60 30 0 --

Test C

The Corn and Sorghum Herbicide Test included the following species in both the preemergence and postemergence evaluations:

    ______________________________________                                                 SPECIES                                                                Category  Common Name  Scientific Name                                         ______________________________________                                         Crops     Corn         Zea mays                                                          Soybean      Glycine max                                                       Sorghum      Sorghum bicolor                                         Grasses   Green foxtail                                                                               Setaria viridis                                                   Giant foxtail                                                                               Setaria faberii                                                   Johnsongrass Sorghum halepense                                                 Barnyardgrass                                                                               Echinochloa crus-galli                                            Fall panicum panicum dichotomiflorum                                           Crabgrass    Digiraria sanguinalis                                             Nutsedge     Cyperus rotundus                                        Broadleaves                                                                              Cocklebur    Xanthium pensylvanicum                                            Morningglory Ipomoea hederacea                                                 Velvetleaf   Abutilon theophrasti                                              Jimsonweed   Datura stramonium                                                 Lambsquarters                                                                               Chenopodium album                                                 Pigweed      Amaranthus retroflexus                                            Smartweed    Polygonum persicaris                                    ______________________________________                                    

Postemergence

Postemergence plants were grown in Sassafras sandy loam soil. Corn and soybeans were grown in separate 25 cm diameter containers. Sorghum and the seven grass weed species were grown in two 18 cm diameter containers, 4 species per container. The seven broadleaf weed species were also grown in two 18 cm diameter containers, 4 species in one container, 3 species in the second container. One additional planting of corn in an 18 cm diameter container was made. The soil surface of this additional container of corn was covered with the absorbent, perlite, before spray treatment so that test chemicals would enter the plant only via the foliage. The plants were grown 10-21 days, dependent upon the species and then sprayed postemergence with the test chemicals dissolved in a non-phytotoxic solvent.

PREEMERGENCE

Preemergence plantings were grown in fertilized Tama silt loam soil. These plants are identical to those described in the postemergence section, with the exception of the corn planting having perlite covering the soil surface. These plantings were made the day of or the day before spraying the test chemicals dissolved in a non-phytotoxic solvent.

EVALUATION

Treated plants and controls were maintained in the greenhouse for 2 to 4 weeks. Visual planting response ratings were made on a percentage scale of 0 to 100 in comparison with a control where 0=no injury, and 100=death.

                  TABLE C                                                          ______________________________________                                         RATE RATE GM                                                                               0004   0008   0016 0031 0062 0125 0250                             ______________________________________                                         Compound 35                                                                    POSTEMERGENCE                                                                  CORN        0      0      0    0    25   45   --                               SOYBEAN     45     70     85   100  100  100  --                               GREEN FXTL  45     55     70   85   95   100  --                               GIANT FXTL  40     45     60   75   95   100  --                               PANICUM     90     100    100  100  100  100  --                               CRABGRASS   0      0      0    30   45   55   --                               BARNYARD-   85     95     100  100  100  100  --                               GRASS                                                                          JOHNSONGRASS                                                                               100    100    100  100  100  100  --                               SORGHUM     100    100    100  100  100  100  --                               NUTSEDGE    30     50     85   90   100  100  --                               VELVETLEAF  25     55     75   90   100  100  --                               COCKLEBUR   100    100    100  100  100  100  --                               SMARTWEED   60     80     85   90   100  100  --                               LAMBSQUARTER                                                                               0      30     60   75   85   100  --                               PIGWEED     50     85     100  100  100  100  --                               MORNING-    60     75     95   100  100  100  --                               GLORY                                                                          JIMSONWEED  65     100    100  100  100  100  --                               PREEMERGENCE                                                                   CORN         --    --     0    0    0    0    35                               SOYBEAN     --     --     0    20   30   45   65                               GREEN FXTL  --     --     55   85   95   95   100                              GIANT FXTL  --     --     55   85   95   100  100                              PANICUM     --     --     80   100  100  100  100                              CRABGRASS   --     --     0    20   25   60   70                               BARNYARD-   --     --     85   100  100  100  100                              GRASS                                                                          JOHNSONGRASS                                                                               --     --     100  100  100  100  100                              SORGHUM     --     --     100  100  100  100  100                              NUTSEDGE    --     --     60   95   100  100  100                              VELVETLEAF  --     --     0    0    0    35   60                               COCKLEBUR   --     --     0    0    0    30   65                               SMARTWEED   --     --     0    0    30   80   100                              LAMBSQUARTER                                                                               --     --     0    50   80   100  100                              PIGWEED     --     --     0    35   70   95   100                              MORNING-    --     --     0    0    0    30   55                               GLORY                                                                          JIMSONWEED  --     --     0    30   45   70   100                              Compound 53                                                                    POSTEMERGENCE                                                                  CORN        0      0      0    0    25   45   --                               SOYBEAN     100    100    100  100  100  100  --                               GREEN FXTL  30     40     55   75   85   95   --                               GIANT FXTL  35     50     75   90   100  100  --                               PANICUM     80     100    100  100  100  100  --                               CRABGRASS   0      0      0    30   45   60   --                               BARNYARD-   75     100    100  100  100  100  --                               GRASS                                                                          JOHNSONGRASS                                                                               95     100    100  100  100  100  --                               SORGHUM     95     100    100  100  100  100  --                               NUTSEDGE    70     95     100  100  100  100  --                               VELVETLEAF  65     95     100  100  100  100  --                               COCKLEBUR   75     90     100  100  100  100  --                               SMARTWEED   55     75     90   100  100  100  --                               LAMBSQUARTER                                                                               25     50     70   90   95   100  --                               PIGWEED     70     95     100  100  100  100  --                               MORNING-    60     80     90   100  100  100  --                               GLORY                                                                          JIMSONWEED  70     95     100  100  100  100  --                               PREEMERGENCE                                                                   CORN        --     --     0    0    0    20   40                               SOYBEAN     --     --     0    35   60   80   100                              GREEN FXTL  --     --     35   50   70   90   95                               GIANT FXTL  --     --     35   50   65   85   95                               PANICUM     --     --     65   85   100  100  100                              CRABGRASS   --     --     0    0    0    30   40                               BARNYARD-   --     --     30   70   85   100  100                              GRASS                                                                          JOHNSONGRASS                                                                               --     --     70   100  100  100  100                              SORGHUM     --     --     80   100  100  100  100                              NUTSEDGE    --     --     70   85   100  100  --                               VELVETLEAF  --     --     0    0    30   45   --                               COCKLEBUR   --     --     0    0    0    0    --                               SMARTWEED   --     --     30   60   80   100  --                               LAMBSQUARTER                                                                               --     --     25   60   85   100  --                               PIGWEED     --     --     0    40   75   95   --                               MORNING-    --     --     0    0    25   35   --                               GLORY                                                                          JIMSONWEED  --     --     0    30   55   80   --                               Compound 163                                                                   POSTEMERGENCE                                                                  CORN        0      0      0    20   55   65   --                               SOYBEAN     100    100    100  100  100  100  --                               GREEN FXTL  60     80     90   100  100  100  --                               GIANT FXTL  60     80     95   100  100  100  --                               PANICUM     90     100    100  100  100  100  --                               CRABGRASS   0      25     40   85   100  100  --                               BARNYARD-   80     100    100  100  100  100  --                               GRASS                                                                          JOHNSONGRASS                                                                               100    100    100  100  100  100  --                               SORGHUM     100    100    100  100  100  100  --                               NUTSEDGE    60     75     90   100  100  100  --                               VELVETLEAF  100    100    100  100  100  100  --                               COCKLEBUR   0      30     60   80   100  100  --                               SMARTWEED   60     80     100  100  100  100  --                               LAMBSQUARTER                                                                               65     80     100  100  100  100  --                               PIGWEED     65     95     100  100  100  100  --                               MORNING-    85     95     100  100  100  100  --                               GLORY                                                                          JIMSONWEED  90     100    100  100  100  100  --                               PREEMERGENCE                                                                   CORN        --     --     0    0    0    0    20                               SOYBEAN     --     --     20   30   40   60   80                               GREEN FXTL  --     --     25   60   75   100  100                              GIANT FXTL  --     --     20   40   70   100  100                              PANICUM     --     --     30   70   95   100  100                              CRABGRASS   --     --     0    25   55   70   100                              BARNYARD-   --     --     0    35   65   100  100                              GRASS                                                                          JOHNSONGRASS                                                                               --     --     40   95   100  100  100                              SORGHUM     --     --     70   95   100  100  100                              NUTSEDGE    --     --     60   80   95   100  100                              VELVETLEAF  --     --     0    0    25   45   80                               COCKLEBUR   --     --     0    0    30   55   70                               SMARTWEED   --     --     0    35   60   85   100                              LAMBSQUARTER                                                                               --     --     20   60   95   100  100                              PIGWEED     --     --     30   70   100  100  100                              MORNING-    --     --     0    0    20   35   70                               GLORY                                                                          JIMSONWEED  --     --     0    30   70   90   100                              Compound 165                                                                   POSTEMERGENCE                                                                  CORN        0      20     45   85   100  --   --                               SOYBEAN     100    100    100  100  100  --   --                               GREEN FXTL  25     70     75   95   95   --   --                               GIANT FXTL  40     90     95   100  100  --   --                               PANICUM     100    100    100  70   100  --   --                               CRABGRASS   20     40     60   70   100  --   --                               BARNYARD-   100    100    100  100  100  --   --                               GRASS                                                                          JOHNSONGRASS                                                                               100    100    100  70   100  --   --                               SORGHUM     100    100    100  100  100  --   --                               NUTSEDGE    100    100    100  100  100  --   --                               VELVETLEAF  90     100    100  100  100  --   --                               COCKLEBUR   25     50     80   100  100  --   --                               SMARTWEED   65     80     90   100  100  --   --                               LAMBSQUARTER                                                                               40     70     85   100  100  --   --                               PIGWEED     95     100    100  100  100  --   --                               MORNING-    80     95     100  100  100  --   --                               GLORY                                                                          JIMSONWEED  80     95     100  100  100  --   --                               PREEMERGENCE                                                                   CORN        --     0      0    0    0    15   --                               SOYBEAN     --     20     35   60   85   100  --                               GREEN FXTL  --     20     50   85   100  100  --                               GIANT FXTL  --     30     70   90   100  100  --                               PANICUM     --     50     85   100  100  100  --                               CRABGRASS   --     0      30   65   90   100  --                               BARNYARD-   --     0      20   50   90   100  --                               GRASS                                                                          JOHNSONGRASS                                                                               --     40     85   100  100  100  --                               SORGHUM     --     40     75   100  100  100  --                               NUTSEDGE    --     30     60   80   100  100  --                               VELVETLEAF  --     0      0    25   50   85   --                               COCKLEBUR   --     0      0    0    35   70   --                               SMARTWEED   --     25     50   75   95   100  --                               LAMBSQUARTER                                                                               --     20     55   70   90   100  --                               PIGWEED     --     30     65   90   100  100  --                               MORNING-    --     0      0    20   40   85   --                               GLORY                                                                          JIMSONWEED  --     0      0    30   70   90   --                               Compound 166                                                                   POSTEMERGENCE                                                                  CORN        0      0      0    0    0    25   60                               SOYBEAN     95     100    100  100  100  100  100                              GREEN FXTL  70     80     85   90   95   100  100                              GIANT FXTL  70     85     95   100  100  100  100                              PANICUM     90     95     100  100  100  100  100                              CRABGRASS   0      0      20   40   50   65   80                               BARNYARD-   95     100    100  100  100  100  100                              GRASS                                                                          JOHNSONGRASS                                                                               100    100    100  100  100  100  100                              SORGHUM     100    100    100  100  100  100  100                              NUTSEDGE    85     100    100  100  109  100  100                              VELVETLEAF  80     90     100  100  100  100  100                              COCKLEBUR   95     100    100  100  100  100  100                              SMARTWEED   45     80     90   95   100  100  100                              LAMBSQUARTER                                                                               65     65     85   95   95   100  100                              PIGWEED     90     70     100  100  100  100  100                              MORNING-    95     100    100  100  100  100  100                              GLORY                                                                          JIMSONWEED  85     95     100  100  100  100  100                              PREEMERGENCE                                                                   CORN        --     0      0    0    0    0    45                               SOYBEAN     --     0      0    30   50   65   70                               GREEN FXTL  --     0      65   85   100  100  100                              GIANT FXTL  --     0      45   85   100  100  100                              PANICUM     --     20     75   100  100  100  100                              CRABGRASS   --     0      20   35   50   65   70                               BARNYARD-   --     0      75   100  100  100  100                              GRASS                                                                          JOHNSONGRASS                                                                               --     70     100  100  100  100  100                              SORGHUM     --     70     100  100  100  100  100                              NUTSEDGE    --     25     85   100  100  100  100                              VELVETLEAF  --     0      0    0    35   60   80                               COCKLEBUR   --     0      0    0    0    30   65                               SMARTWEED   --     30     0    20   30   50   100                              LAMBSQUARTER                                                                               --     25     25   75   100  100  100                              PIGWEED     --     45     30   80   100  100  100                              MORNING-    --     0      0    0    20   65   75                               GLORY                                                                          JIMSONWEED  --     0      25   50   75   95   100                              ______________________________________                                    

Test D

Sixteen cm diameter Wagner pots, equipped with a stoppered drain opening near the bottom of the side wall, were partially filled with Woodstown sandy loam. About 1500 mls of water were added to each pot to bring the water level to a point 3 cm above the soil surface. Japonica and Indica rice seedlings were hand transplanted into the pots. Also, a number of barnyardgrass (Echinochloa crus-galli) seeds were added to each pot. At the same time, seedlings or tubers of the following species were transplanted into the muddy soil: water plantain (Alisma trivale), Scirpus (Scirpus mucranatus), and Cyperus (Cyperus difformis). The weed species selected for this test are of economic importance in major rice-growing areas. The chemical treatments were applied directly to the paddy water after being formulated in a non-phytotoxic solvent within hours after transplanting of two additional species: water chestnut (Eleocharis spp.) and arrowhead (Sagittaria latifolia). Shortly after treatment, the drain hole was opened to drop the water level by two cm. Water was then added to restore the water level to its original height. The following day the draining and refilling process was repeated. The pots were then maintained in the greenhouse.

Rates of application and plant response ratings made 21 days after treatment are summarized in Table D. Response ratings are based on a scale of 0 to 100 where 0=no effect and 100=complete control.

                  TABLE D                                                          ______________________________________                                                  Compound 188 Compound 189                                             Rate g/ha  0016    0008   0004  0016  0008 0004                                ______________________________________                                         Japonica Rice                                                                              0       0      0    15    15    0                                  Indica Rice                                                                                0       0      0    15     0    0                                  Barnyardgrass                                                                             77      22      0    95    77   30                                  Water Chestnut                                                                            82      87     85    90    85   70                                  Arrowhead  95      90     80    92    95   87                                  Scirpus    77      80     60    87    85   67                                  Cyperus    82      55     32    95    95   92                                  Water Plantain                                                                            75      75     60    85    72   67                                  ______________________________________                                    

Test E

The weed species used in this test are all of major economic importance in soybean-growing regions. The following species are included in the screen:

    __________________________________________________________________________                              GROWTH STAGE AT APPLICA-                              Plant Species                                                                              Scientific Name                                                                             TION (POSTEMERGENCE PHASE)                            __________________________________________________________________________     Grass Weeds:                                                                   barnyardgrass                                                                              Echinochloa crus-galli                                                                      2-3     leaves                                        giant foxtail                                                                              Setaria faberi                                                                              2-3     leaves                                        green foxtail                                                                              Setaria viridis                                                                             2-3     leaves                                        johnsongrass                                                                               Sorghum halepense                                                                           2-3     leaves                                        fall panicum                                                                               Panicum dichotomiflorum                                                                     2-3     leaves                                        broadleaf signalgrass                                                                      Brachiaria platyphylla                                                                      2-3     leaves                                        large crabgrass                                                                            Digitaria sanguinalis                                                                       2-3     leaves                                        Broadleaf Weeds:                                                               velvetleaf  Abutilon theophrasti                                                                        2-3     leaves                                        jimsonweed  Datura stramonium                                                                           1-2     true leaves                                   hemp sesbania                                                                              Sesbania exaltata                                                                           1st     true leaf                                     sicklepod   Cassia obtusifolia                                                                          1st     true leaf                                     cocklebur   Xanthium pensylvanicum                                                                      2nd     true leaf                                     morningglory                                                                               Ipomoea hederacea                                                                           1-2     true leaves                                   ladysthumb smartweed                                                                       Polygonum persicaria                                                                        3-4     leaves                                        pigweed     Amaranthus retroflexus                                                                      4-5     leaves                                        lambsquarters                                                                              Chenopodium album                                                                           4-5     leaves                                        teaweed     Sida spinosa 2-3     leaves                                        black nightshade                                                                           Solanum nigrum                                                                              2nd     true leaf                                     purple nutsedge                                                                            Cyperus rotundus                                                                            5-6     leaves                                        corn        Zea mays     2-3     leaves                                        soybeans    Glycine max  1st     trifoliate                                    __________________________________________________________________________

For the preemergence phase of the test, crop and weed species are planted in a Tama silt loam soil (approximately 3% organic matter). Approximate planting depths are: corn and soybeans--3 to 4 cm; morningglory, cocklebur, and nutsedge--2.5 to 3 cm; velvetleaf, sicklepod, and sesbania--2 cm; all other species--0.5 cm.

For the postemergence phase of the test, crop and weed species are planted in a Sassafras sandy loam soil (approximately 1% organic matter) one to three weeks before application so that they will be present as young plants at the time of treatment. Alternatively, for postemergence tests, plants are grown in a 50:50 mixture of commercially available potting mix and Sassafras soil. Approximate planting depths are: corn and soybeans--3 to 4 cm; morningglory, cocklebur, and nutsedge--2.5 to 3 cm; velvetleaf, sicklepod, and sesbania--2 cm; all other species--0.5 cm.

Treated plants and controls were maintained in a greenhouse for 3 to 4 weeks, after which all species were compared to controls and visually rated for response to treatment. The ratings, summarized in Table E, are based on a numerical scale extending from 0=no injury to 100=complete kill.

                  TABLE E                                                          ______________________________________                                                  Rate = gm/h                                                           Postemergence                                                                             0004   0008    0016  0032  0064  0125                               Soil type  Mix    Mix     Mix   Mix   Mix   Mix                                ______________________________________                                         CMPD 206                                                                       Soybeans   0      0       10    15    20    25                                 Corn       40     70      90    100   100   100                                Velvetleaf 50     75      100   100   100   100                                Jimsonweed 30     40      40    50    85    95                                 Sicklepod  10     20      30    40    40    50                                 Hemp sesbania                                                                             20     40      50    75    85    95                                 Cocklebur  50     60      80    100   100   100                                Ivy morningglory                                                                          75     85      90    95    100   100                                Redroot pigweed                                                                           20     40      45    50    50    60                                 Lambsquarter                                                                              50     50      60    90    90    90                                 Prickly sida                                                                              30     45      50    65    75    85                                 Barnyardgrass                                                                             20     30      50    75    95    100                                Giant foxtail                                                                             0      0       20    30    50    80                                 Green foxtail                                                                             0      30      40    50    60    70                                 Johnsongrass                                                                              20     30      40    50    60    70                                 Fall panicum                                                                              0      0       20    30    40    50                                 Large crabgrass                                                                           0      0       0     0     0     0                                  Brdlf sgnlgrass                                                                           20     30      40    50    50    70                                 Purple nutsedge                                                                           0      20      30    40    50    80                                 Lady smartweed                                                                            0      0       0     20    30    50                                 Black nightshad                                                                           50     60      70    95    100   100                                CMPD 207                                                                       Soybeans   0      0       0     0     10    15                                 Corn       10     20      50    75    80    80                                 Velvetleaf 50     75      95    100   100   100                                Jimsonweed 30     40      50    60    80    100                                Sicklepod  0      20      30    40    50    80                                 Hemp sesbania                                                                             20     40      50    60    70    80                                 Cocklebur  50     60      70    100   100   100                                Ivy morningglory                                                                          50     75      80    80    95    95                                 Redroot pigweed                                                                           20     30      50    60    70    95                                 Lambsquarter                                                                              50     50      70    80    80    95                                 Prickly sida                                                                              30     40      50    60    75    90                                 Barnyardgrass                                                                             0      0       20    40    65    100                                Giant foxtail                                                                             0      30      40    50    60    80                                 Green foxtail                                                                             0      30      30    40    50    60                                 Johnsongrass                                                                              20     30      40    50    60    70                                 Fall panicum                                                                              0      0       0     0     0     0                                  Large crabgrass                                                                           0      0       0     0     0     0                                  Brdlf sgnlgrass                                                                           0      0       20    50    60    70                                 Purple nutsedge                                                                           0      20      30    40    100   80                                 Lady smartweed                                                                            0      20      30    40    50    65                                 Black nightshad                                                                           50     80      100   100   100   100                                ______________________________________                                     

What is claimed is:
 1. A compound of the formula: ##STR57## wherein J is ##STR58## W is O or NH_(X) ; R_(X) is H, OH, C₁ -C₃ alkyl, C₁ -C₃ alkoxy, allyloxy, propargyloxy, C₁ -C₃ haloalkyl, C₁ -C₃ haloalkoxy or NR_(Y) R_(Z) ;R_(Y) is H or C₁ -C₃ alkyl; R_(Z) is C₁ -C₃ alkyl; G is O, S, SO or SO₂ ; m is 0 or 1; n is 0, 1 or 2; R is H or CH₃ ; E is a single bond, CH₂ or O; Q is ##STR59## R₁ is H, C₁ -C₃ alkyl, C₁ -C₃ haloalkyl, halogen, nitro, C₁ -C₃ alkoxy, SO₂ NR_(a) R_(b), C₁ -C₃ alkylthio, C₁ -C₃ alkylsulfinyl, C₁ -C₃ alkylsulfonyl, CN, SCN, CO₂ R_(c), C₁ -C₃ haloalkoxy, C₁ -C₃ haloalkylthio, amino, C₁ -C₃ alkylamino, di(C₁ -C₃ alkyl)amino or C₁ -C₂ alkyl substituted with C₁ -C₂ alkoxy, C₁ -C₂ haloalkoxy, C₁ -C₂ alkylthio, C₁ -C₂ haloalkylthio or CN; R₂ is H, C₁ -C₃ alkyl, allyl or phenyl; R₃ is H, C₁ -C₆ alkyl, C₃ -C₆ cycloalkyl, C₁ -C₆ haloalkyl, CH₂ --(C₂ -C₅ alkenyl), CH₂ (C₂ -C₅ haloalkenyl), CH₂ (C₂ -C₅ alkynyl), CH₂ (C₂ -C₅ haloalkynyl), C₆ H₅ or C₁ -C₄ alkyl substituted with C₁ -C₂ alkoxy, C₁ -C₂ alkylthio, C₁ -C₂ alkylsulfinyl or C₁ -C₂ alkylsulfonyl; R₄ is H, halogen, C₁ -C₆ alkyl, C₃ -C₆ cycloalkyl, C₁ -C₆ haloalkyl, C₂ -C₆ alkenyl, C₂ -C₆ haloalkenyl, C₂ -C₆ alkynyl, C₃ -C₆ haloalkynyl, C₆ H₅, C₁ -C₄ alkoxy, C₁ -C₄ haloalkoxy, C₁ -C₄ alkylthio, C₁ -C₄ alkylsulfinyl, C₁ -C₄ alkylsulfonyl, OCH₂ CH₂ O--(C₁ -C₂ alkyl) or di(C₁ -C₃ alkyl)amino; R₅ is H, C₁ -C₃ alkyl, C₁ -C₃ haloalkyl, allyl or propargyl; R_(a) is H, C₁ -C₄ alkyl, C₂ -C₃ cyanoalkyl, methoxy or ethoxy; R_(b) is H, C₁ -C₄ alkyl or C₃ -C₄ alkenyl; or R_(a) and R_(b) may be taken together as --(CH₂)₃ --, --(CH₂)₄ --, --(CH₂)₅ -- or --CH₂ CH₂ OCH₂ CH₂ --; R_(c) is C₁ -C₄ alkyl, C₃ -C₄ alkenyl, C₃ -C₄ alkynyl, C₂ -C₄ haloalkyl, C₁ -C₂ cyanoalkyl, C₅ -C₆ cycloalkyl, C₄ -C₇ cycloalkylalkyl or C₂ -C₄ alkoxyalkyl; A is ##STR60## X₄ is CH₃, OCH₃, OC₂ H₅, CH₂ OCH₃ or OCl; and Y₄ is CH₃, OCH₃ ; OC₂ H₅ or Cl.and their agriculturally suitable salts; provided that (a) when J is J-9 and n is 0, then Q is Q-1 or Q-2; (b) when E is 0, then J is J-1; (c) X₄ and Y₄ cannot simultaneously be Cl; (d) when J is J-1 and m is 0, then n is 0; and (e) when n is 0 and m is 1, then Q is Q-1 or Q2.
 2. A compound of claim 1 where E is a single bond.
 3. A compound of claim 1 wherein E is CH₂.
 4. A compound of claim 1 where E is
 0. 5. A compound of claim 2 where m is
 0. 6. A compound of claim 3 wherem is 0; n is 0; J is J-1, J-2, J-3, J-8, J-10 or J-11; R is H; R₁ is H, CH₃, F, Cl, Br, OCH₃, SCH₃, CH₂ CN, CH₂ OCH₃, CF₃ or OCF₂ H; R₃ is H, C₁ -C₃ alkyl, CH₂ CH₂ OCH₃, CH₂ CH₂ Cl, CH₂ CH₂ F, CH₂ CHF₂, CH₂ CF₃, allyl or propargyl; and R₄ is H or C₁ -C₃ alkyl.
 7. A compound of claim 4 wherem is 0; R is H; R₁ is H; R₃ is H or C₁ -C₃ alkyl; and R₄ is H or C₁ -C₃ alkyl.
 8. A compound of claim 5 whereR₁ is H, CH₃, F, Cl, Br, OCH₃, SCH₃, CH₂ CN, CH₂ OCH₃, CF₃ or OCF₂ H; and n is
 0. 9. A compound of claim 8 whereR₃ is H, C₁ -C₃ alkyl, C₁ -C₂ alkyl substituted with C₁ -C₂ alkoxy, CH₂ CH₂ Cl, CH₂ CH₂ F, CH₂ CHF₂, CH₂ CF₃, allyl or propargyl; and R₄ is H, C₁ -C₃ alkyl, C₁ -C₂ alkoxy, C₁ -C₂ alkylthio, N(CH₃)₂, allyl, propargyl or C₁ -C₂ alkyl substituted with 1-3 atoms of F, Cl or Br.
 10. A compound of claim 9 where J is J-1.
 11. A compound of claim 9 where Q is Q₁.
 12. A compound of claim 9 where Q is Q₂.
 13. A compound of claim 9 where Q is Q₃.
 14. A compound of claim 9 where Q is Q₄.
 15. A compound of claim 9 where Q is Q₅.
 16. A compound of claim 9 where Q is Q₆.
 17. A compound of claim 9 where Q is Q₇.
 18. A compound of claim 8 where J is J-2.
 19. A compound of claim 18 where Q is Q₁.
 20. A compound of claim 9 where J is J-3.
 21. A compound of claim 20 where Q is Q₁.
 22. A compound of claim 9 where J is J-4.
 23. A compound of claim 22 where Q is Q₁.
 24. A compound of claim 9 where J is J-5.
 25. A compound of claim 24 where Q is Q₁.
 26. A compound of claim 9 where J is J-6.
 27. A compound of claim 26 where Q is Q₁.
 28. A compound of claim 9 where J is J-7.
 29. A compound of claim 28 where Q is Q₁.
 30. A compound of claim 9 where J is J-8.
 31. A compound of claim 30 where Q is Q₁.
 32. A compound of claim 30 where Q is Q₂.
 33. A compound of claim 30 where Q is Q₃.
 34. A compound of claim 30 where Q is Q₄.
 35. A compound of claim 30 where Q is Q₅.
 36. A compound of claim 30 where Q is Q₆.
 37. A compound of claim 30 where Q is Q₇.
 38. A compound of claim 9 where J is J-9.
 39. A compound of claim 38 where Q is Q₁.
 40. A compound of claim 9 where J is J-10.
 41. A compound of claim 40 where Q is Q₁.
 42. A compound of claim 9 where J is J-11.
 43. A compound of claim 42 where Q is Q₁.
 44. A compound of claim 9 where J is J-12.
 45. A compound of claim 44 where Q is Q₁.
 46. A compound of claim 9 where J is J-13.
 47. A compound of claim 46 where Q is Q₁.
 48. A composition suitable for controlling the growth of undesired vegetation which comprises an effective amount of a compound of claim 1 and at least one of the following: surfactant, solid or liquid diluent.
 49. A composition suitable for controlling the growth of undesired vegetation which comprises an effective amount of a compound of claim 2 and at least one of the following: surfactant, solid or liquid diluent.
 50. A composition suitable for controlling the growth of undesired vegetation which comprises an effective amount of a compound of claim 3 and at least one of the following: surfactant, solid or liquid diluent.
 51. A composition suitable for controlling the growth of undesired vegetation which comprises an effective amount of a compound of claim 4 and at least one of the following: surfactant, solid or liquid diluent.
 52. A composition suitable for controlling the growth of undesired vegetation which comprises an effective amount of a compound of claim 5 and at least one of the following: surfactant, solid or liquid diluent.
 53. A method for controlling the growth of undesired vegetation which comprises applying to the locus to be protected an effective amount of a compound of claim
 1. 54. A method for controlling the growth of undesired vegetation which comprises applying to the locus to be protected an effective amount of a compound of claim
 2. 55. A method for controlling the growth of undesired vegetation which comprises applying to the locus to be protected an effective amount of a compound of claim
 3. 56. A method for controlling the growth of undesired vegetation which comprises applying to the locus to be protected an effective amount of a compound of claim
 4. 57. A method for controlling the growth of undesired vegetation which comprises applying to the locus to be protected an effective amount of a compound of claim
 5. 